![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_613bd559e314252ec76ed0cdf79b77e9.svg) | 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide | IC50 | 2450.0 [1], 11760.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_8716d1379fc9fcdaef8beabc3dd79da1.svg) | N-[[5-[1-(2-Imidazol-1-ylethyl)indazol-3-yl]-1,2,4-oxadiazol-3-yl]methyl]benzamide | IC50 | 22000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f51b049765c4fb65e756372294890310.svg) | N-[[5-[2-(2-Imidazol-1-ylethyl)indazol-3-yl]-1,2,4-oxadiazol-3-yl]methyl]-3-(trifluoromethoxy)benzamide | IC50 | 4760.0 [1], 97000.0 [2], 100000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_d33ec2b41b84fafe803d97bde6190274.svg) | N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]piperidin-1-yl]-1,3,5-triazin-2-yl]amino]phenyl]acetamide | IC50 | 300.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_25d9b33026565fc9b2cb6059f4773987.svg) | 2,2-Diphenyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]acetamide | IC50 | 17.0 [1], 20.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_15c98b90510aa98184a5de8633598a6c.svg) | Tert-butyl 2-amino-4-[3-(1H-indole-2-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 26000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_0af7015f8a6d51bb5a2a6f819cd52c8e.svg) | 4-[(5-Chloro-1,3-thiazol-2-yl)sulfamoyl]-N-[[4-chloro-3-(trifluoromethyl)phenyl]methyl]benzamide | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_b26fba70cd18ad7e9496180cfa287d08.svg) | Tert-butyl 2-amino-4-[4-[[(2R)-pyrrolidine-2-carbonyl]amino]phenyl]imidazole-1-carboxylate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_da0a7f0903fb44ea1644f38fcae8a8cc.svg) | Tert-butyl 4-[3-(furan-2-carbonylamino)phenyl]-2-(methylamino)imidazole-1-carboxylate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_508b897cf1cd2dc5f3b3b15d78938288.svg) | Tert-butyl 2-amino-4-[4-(1H-indole-2-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 22000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_c4ef4d8d86c1407074db717ee4e79b07.svg) | N-[3-[2-Amino-1-(1H-pyrrole-2-carbonyl)imidazol-4-yl]phenyl]-1H-pyrrole-2-carboxamide | IC50 | 25000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_694930826fd577333231eabfb9daa343.svg) | Tert-butyl 2-amino-4-[3-[[(2R)-pyrrolidine-2-carbonyl]amino]phenyl]imidazole-1-carboxylate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_b86da05b0fc44715c3b6bc7ed44789bb.svg) | Tert-butyl 2-amino-4-[3-(1H-indole-3-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 27000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_31562dfa9cb74a2404b8b216676dec58.svg) | Tert-butyl 2-amino-4-[3-(1H-pyrrole-3-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 23000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_e3c5d43be33ed236f49f82c3bcbaceea.svg) | Tert-butyl 2-amino-4-[3-(1H-pyrrole-2-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 25000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_63c8e2e8763cf1aaa500bdaa701dc3a2.svg) | Tert-butyl 4-[3-(1H-indole-2-carbonylamino)phenyl]-2-(methylamino)imidazole-1-carboxylate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_1fdbca44903ef51063cee5964663ba39.svg) | Tert-butyl 2-amino-4-[3-(1H-pyrrole-3-carbonylamino)phenyl]imidazole-1-carboxylate;hydrochloride | IC50 | 12000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7de504fc673a4c3ce1245de740bc48aa.svg) | Tert-butyl 2-amino-4-[4-(furan-2-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 27000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_20246adf3cfad06e6bee363818872656.svg) | Tert-butyl 2-amino-4-[4-[[(2S)-pyrrolidine-2-carbonyl]amino]phenyl]imidazole-1-carboxylate | IC50 | 25000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_1bb90bfd0c700cc281e6f9a9c486911b.svg) | Tert-butyl 2-amino-4-[4-(1H-pyrrole-2-carbonylamino)phenyl]imidazole-1-carboxylate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f6de79fc4e43ad95cc082dff3379d7d4.svg) | N-[3-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-indole-3-carboxamide | IC50 | 12000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_26f6a90ff4a4e6b49a5ef51bb234ebff.svg) | N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-pyrrole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_888d1cdbe9885fec6c5a3c4f8500c603.svg) | N-[3-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-indole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_b1aecbe717c2784fbaa6cd5fea933870.svg) | N-[3-[2-(Methylamino)-1H-imidazol-5-yl]phenyl]-1H-indole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7fc2b8579488f7cd6d2af758e1bb70ff.svg) | N-[3-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-pyrrole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_9e493a2164ceb41e1345f315a13c14fe.svg) | N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]-1H-indole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_ae9ec39b91fb9ee556a7ddd9e0037789.svg) | (2R)-N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]pyrrolidine-2-carboxamide | IC50 | 8000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_2267ee993803e1e4dc0321b5104a7af2.svg) | (2S)-N-[4-(2-Amino-1H-imidazol-5-yl)phenyl]pyrrolidine-2-carboxamide | IC50 | 13000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_dc3b519ae4da383d84a5502ee939a5d0.svg) | Lidocaine | IC50 | 10500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_71450bda5f550ba3db0463b13d3782d9.svg) | Tetrodotoxin | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_d807cd36eea3bdcc2c2c3e9b5d13b932.svg) | Lamotrigine | IC50 | 17000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_c7416e1543ca26168b769dc25d1f2310.svg) | Tetracaine | IC50 | 740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_a62cbe90f5af57b0f55ccaee19647f69.svg) | Senicapoc | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_55892479c77cb8cbec69941708da1cce.svg) | CID 46840946 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_29c7c51dd7c16d8e9004503d08bade20.svg) | 6-Amino-N-methyl-5-(2,3,5-trichlorophenyl)picolinamide | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_0655a0f80832be04b0950c13a7240f1c.svg) | 1-[2-Methoxy-4-[3-(trifluoromethyl)phenyl]phenyl]-2-oxo-N-pyrimidin-2-ylquinoline-6-sulfonamide | IC50 | 42500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_0b83c38cc47733eab66fd9a3b08ba037.svg) | CID 118734430 | IC50 | 20.3 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_e8ce2804376e26e1cfa13691a3d4be4a.svg) | N-[6-Amino-5-[2-(trifluoromethoxy)phenyl]pyridin-2-yl]-3-methyl-1,2-oxazole-4-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_42e8e96aab4c8e3ece5dee1b2eaa9ac5.svg) | 4-[4-Chloro-2-[2-(1-ethylazetidin-3-yl)pyrazol-3-yl]phenoxy]-3-cyano-N-(1,3-thiazol-4-yl)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_526071f5d6a907983935b8ce39e33166.svg) | 5-Chloro-2-fluoro-4-[2-pyridazin-4-yl-4-(trifluoromethyl)phenoxy]-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_de119abfff9f20abb9a096724bb462f5.svg) | 4-[2-(2-Amino-3H-benzimidazol-5-yl)-4-chlorophenoxy]-2,5-difluoro-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 9330.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_da41649d64ca27df34964228f23b8832.svg) | 4-[4-Chloro-2-(2-methylpyrazol-3-yl)phenoxy]-3-fluoro-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 292.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_6062e2101bd51941236f348cea3c774a.svg) | 4-[4-Chloro-2-(2-methylpyrazol-3-yl)phenoxy]-3-cyano-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_faa36e96c7388d397cc321fecb2a83aa.svg) | N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-1H-indole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_6cda3f7d1010e2185573b3761bf2c591.svg) | N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-4,5-dibromo-1H-pyrrole-2-carboxamide | IC50 | 26000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_c810f8ea8796703c08f529ffed231d4e.svg) | N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-4,5-dibromo-1H-pyrrole-2-carboxamide | IC50 | 18000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_1b18c4c8894da448f66adf3cb6c54ec8.svg) | N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-4-bromo-1H-pyrrole-2-carboxamide | IC50 | 26000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_8889ba945b627a40a411d2b142f7e056.svg) | 4-[2-Methoxy-4-(trifluoromethyl)phenyl]-N-(1,3-thiazol-2-yl)quinazoline-7-sulfonamide | IC50 | 21000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_dcd280248d8c7b18cc8bf71bf481f140.svg) | N-[6-Amino-5-(2,3,5-trichlorophenyl)pyridin-2-yl]acetamide | IC50 | 3500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_ba3d0dbddcb0669e9014f069801a24f3.svg) | 3-Cyano-4-[2-[2-[(2-piperidin-4-ylethylamino)methyl]pyridin-4-yl]-4-[3-(trifluoromethyl)phenyl]phenoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 6438.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_66d69856f0ef8731cd6abe663649906d.svg) | 1-[1-(2-Fluorophenyl)indazol-4-yl]-3-[2-[(3S)-3-fluoropyrrolidin-1-yl]-2-oxoethyl]imidazolidin-2-one | IC50 | 7100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f867a3109129b1ce591f7eb629418ce7.svg) | 1-[5-Fluoro-2-methoxy-4-[3-(trifluoromethyl)phenyl]phenyl]-N-(1,2-oxazol-3-yl)isoquinoline-6-sulfonamide | IC50 | 6900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_786abf31dcee0e1f07502fa37feebdb1.svg) | (3Ar,6aS)-5-[1-(2-fluorophenyl)indazol-4-yl]-2-(3-hydroxy-3-methylbutanoyl)-3,3a,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-4-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f86d7f2921e68f79b7f280f1503786e2.svg) | 1-[2-[5-Fluoro-1-(2-fluorophenyl)indazol-3-yl]oxyethyl]imidazolidin-2-one | IC50 | 3400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_ebb64c3433c2250bec223cd53e16f554.svg) | 4-[(3S)-3-[(3R)-3-(3,5-Dichlorophenyl)pyrrolidin-1-yl]-2-oxopyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)benzenesulfonamide | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_ffa17f3d7692b3a5abc9d12d03c5daae.svg) | 6-Amino-N-methyl-5-(2,3,5-trichlorophenyl)pyridine-3-carboxamide | IC50 | 6900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_559063e2e8fd8aaf5795c40346020e09.svg) | N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-1-methylpyrrole-2-carboxamide | IC50 | 24000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_b3723f36b784a8338db080b677724938.svg) | N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-1H-pyrrole-2-carboxamide | IC50 | 28000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_a81c03ffc2f274731bc53b5d59b9f03f.svg) | N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]furan-2-carboxamide | IC50 | 27000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_2707061ddb43ed9590fdf090de29ef08.svg) | Tert-butyl (2S)-2-[[(6S)-2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]carbamoyl]pyrrolidine-1-carboxylate | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7b01705c1efd22e1983e6aa88081212b.svg) | (6S)-6-N-(1H-Pyrrol-2-ylmethyl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2,6-diamine | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7a6b4f7ad418e41de56a0e650f7edeb6.svg) | N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-1H-indole-2-carboxamide | IC50 | 16000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_0a9c89f01017d7dd735ce93ca3c00132.svg) | Tert-butyl (2S)-2-[(2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methylcarbamoyl]pyrrolidine-1-carboxylate | IC50 | 26000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_1e656542379786505b6e300e60ab7480.svg) | N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-1H-pyrrole-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f947367a55586daae82c2dbd51d184ce.svg) | N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]-4-bromo-1H-pyrrole-2-carboxamide | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_2370f036424df7df8422db7719f9b1f0.svg) | 2-Fluoro-N-(1,3-thiazol-2-yl)-4-[(3S)-3-[5-(trifluoromethyl)pyridin-2-yl]oxypyrrolidin-1-yl]sulfonylbenzenesulfonamide | IC50 | 851.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7ac9e46bfd36ff05be01f2d9e0a60b69.svg) | 2-Fluoro-N-(1,3-thiazol-2-yl)-4-[4-[6-(trifluoromethyl)pyridin-2-yl]piperidin-1-yl]sulfonylbenzenesulfonamide | IC50 | 1640.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_110fa2a5f67a35081953d2f2de4afb24.svg) | 2-Fluoro-4-(3-phenoxyazetidin-1-yl)sulfonyl-N-(1,3-thiazol-2-yl)benzenesulfonamide | IC50 | 959.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_2b1fa7b0e6a92be6f0b904ee8279cb3a.svg) | 2-Fluoro-N-(1,2,4-thiadiazol-5-yl)-4-[4-[2-(trifluoromethyl)pyrimidin-4-yl]piperidine-1-carbonyl]benzenesulfonamide | IC50 | 6675.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_cb1fa0e8a82eb69a0157fff62921b63e.svg) | 4-[[3-Chloro-4-(trifluoromethoxy)phenyl]methoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_2aca76c4ec167bcc12c8d2f176697d47.svg) | 4-[(3S)-3-(2,6-Dichlorophenoxy)pyrrolidin-1-yl]sulfonyl-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide | IC50 | 945.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_8846e54044f2acbebb0b9e49bcb8c2b2.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(1,2,4-thiadiazol-5-ylsulfamoyl)benzamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_76f70f1175f401aa0df38e5ed894d261.svg) | 4-N-(1,3-Thiazol-2-yl)-1-N-[[4-(trifluoromethyl)phenyl]methyl]benzene-1,4-disulfonamide | IC50 | 160.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_c5e4bd1ae0aaeeb1ec9cd1b68f5203e8.svg) | 4-[3-Chloro-4-(trifluoromethoxy)phenoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 296.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_96714352c4f9d40d14d7decd6e0925b6.svg) | 2-Fluoro-4-[2-(3-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]sulfonyl-N-(1,3-thiazol-2-yl)benzenesulfonamide | IC50 | 1830.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_d4b6162fc53a45f7bcbae5257f1c769c.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-[(5-fluoropyrimidin-2-yl)sulfamoyl]benzamide | IC50 | 993.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7c48d261e331d9610b6e822d1ba76b53.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(pyrimidin-5-ylsulfamoyl)benzamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_18ba39e01af04c2889878d91c28469c7.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(pyrimidin-2-ylsulfamoyl)benzamide | IC50 | 374.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_773e14259248ea9146f8c66633d8a5f7.svg) | 2-Fluoro-N-(1,2,4-thiadiazol-5-yl)-4-[4-[5-[2-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl]piperidine-1-carbonyl]benzenesulfonamide | IC50 | 1955.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_7ed8b6db2cdae9a7f06d38e575bc359f.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-N-methyl-4-(1,2,4-thiadiazol-5-ylsulfamoyl)benzamide | IC50 | 522.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f7c84b483e716750239a18d95af3c997.svg) | N-(1,3-Thiazol-2-yl)-4-[5-[[4-(trifluoromethyl)phenyl]methyl]-1H-1,2,4-triazol-3-yl]benzenesulfonamide | IC50 | 124.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_5766d489474bb06cbec1c83f4e0bb6fb.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(pyridazin-3-ylsulfamoyl)benzamide | IC50 | 1793.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_0621893c95997496abf785d461cf972c.svg) | 2-Fluoro-4-[(2R)-2-[(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)methyl]pyrrolidin-1-yl]sulfonyl-N-(1,3-thiazol-2-yl)benzenesulfonamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_8995e8cc1ba818c1abd8be63b1ec7200.svg) | 4-[[1-[3-Chloro-4-(trifluoromethoxy)benzoyl]azetidin-3-yl]oxymethyl]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide | IC50 | 237.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_bd01eb2189988ff925cf3999773efa04.svg) | 2-Phenyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]acetamide | IC50 | 3790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_9711f71077d3a7949cc5c0664de53681.svg) | 1-[2-(4-Fluorophenoxy)acetyl]-N-(1,3-thiazol-2-yl)-2,3-dihydroindole-5-sulfonamide | IC50 | 2506.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_42f974532d2b2082512a374b47fbbf6f.svg) | 4-[5-[(3,4-Dichlorophenyl)methyl]-1H-1,2,4-triazol-3-yl]-N-(1,3-thiazol-2-yl)benzenesulfonamide | IC50 | 45.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_3d71f5725985bf93de10325aa2e75bd7.svg) | N-(1,3-Thiazol-2-yl)-4-[2-[4-(trifluoromethyl)phenyl]ethylsulfonyl]benzenesulfonamide | IC50 | 155.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_dcca8af4971523e5cd5a6fdc5b1563b7.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-4-(1,3-thiazol-2-ylsulfamoyl)benzamide | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_f048aaa9685278fd01dc1f2f4b97d5dc.svg) | N-[[3-Chloro-4-(trifluoromethoxy)phenyl]methyl]-3-fluoro-4-(1,3-thiazol-2-ylsulfamoyl)benzamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_c9b602b49a9362ebccd3a82be1c0a292.svg) | 4-(1,3-Thiazol-2-ylsulfamoyl)-N-[[4-(trifluoromethyl)phenyl]methyl]benzamide | IC50 | 147.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_b29187ea7102832a457d5efb2ad3a7bf.svg) | 1-[2-(4-Fluorophenoxy)acetyl]-N-(1,2,4-thiadiazol-5-yl)-2,3-dihydroindole-5-sulfonamide | IC50 | 1273.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_e8a82b8c896b0c49c829c0bcc999b2fb.svg) | (2S)-N-[(2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl)methyl]pyrrolidine-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_1cc21e6f83bf2fb56551a0ac82346d18.svg) | (2S)-N-[(6S)-2-Amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]pyrrolidine-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_2f2f12b33ac4cdb9a381e604133afbd0.svg) | N-Benzyl-4-(1,3-thiazol-2-ylsulfamoyl)benzamide | IC50 | 4450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/sodium-channel-protein-type-iii-alpha-subunit_04fc175494b0c8b4ff541d4576158dca.svg) | 4-(1,3-Thiazol-2-ylsulfamoyl)-N-[[4-(trifluoromethoxy)phenyl]methyl]benzamide | IC50 | 197.0 [1] |