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Sn1-specific diacylglycerol lipase alpha Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
OrlistatIC501.0 [1], 10.0 [2], 60.0 [3], 1000.0 [4]
(4-([1,1'-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)(2-benzylpiperidin-1-yl)methanoneIC506.31 [1], 125.89 [2], 2511.89 [3]
2-[(2,2-Dimethyl-3,4-dihydrochromen-6-yl)sulfonyl-[(4-phenoxyphenyl)methyl]amino]acetic acidIC5018.0 [1]
2-[(2,2-Dimethyl-3,4-dihydrochromen-6-yl)sulfonyl-[(4-phenoxyphenyl)methyl]amino]acetic acidKi700.0 [1]
[(2S)-2-Benzylpiperidin-1-yl]-[4-(4-phenylphenyl)triazol-1-yl]methanoneIC5039.81 [1], 794.33 [2]
[(2R)-2-Benzylpiperidin-1-yl]-[4-(4-phenylphenyl)triazol-1-yl]methanoneIC500.79 [1], 25.12 [2]
1,6-Bis(cyclohexyloximinocarbonyl)hexaneIC5060.0 [1], 65000.0 [2]
2-[[(1R)-1-[4-(2,4-Dichlorophenyl)phenyl]ethyl]-[4-(difluoromethoxy)phenyl]sulfonylamino]acetic acidIC5019.0 [1], 100.0 [2]
2-[3-(2,3-Dichlorophenyl)-N-[4-(difluoromethoxy)phenyl]sulfonylanilino]acetic acidIC502.4 [1], 14.3 [2]
2-[[3-(2,3-Dichlorophenyl)phenyl]methyl-[4-(difluoromethoxy)phenyl]sulfonylamino]acetic acidIC503.0 [1], 14.0 [2]
2-[[4-(Difluoromethoxy)phenyl]sulfonyl-[[3-[2-(trifluoromethoxy)phenyl]phenyl]methyl]amino]acetic acidIC5017.0 [1], 60.0 [2]
2-[[1-[3-(3,5-Dichlorophenyl)phenyl]cyclobutyl]-[(2,2-dimethyl-3,4-dihydrochromen-6-yl)sulfonyl]amino]acetic acidIC500.6 [1], 37.0 [2]
2-[[1-[4-(2,4-Dichlorophenyl)phenyl]cyclobutyl]-[4-(difluoromethoxy)phenyl]sulfonylamino]acetic acidIC506.0 [1], 88.0 [2]
2-[[4-(Difluoromethoxy)phenyl]sulfonyl-[1-[4-[2-(trifluoromethoxy)phenyl]phenyl]cyclobutyl]amino]acetic acidIC508.0 [1], 82.0 [2]
N,N-Dimethyl-5-[(4-phenylphenyl)methyl]-1-tetrazolecarboxamideIC5010000.0 [1]
1-Oxazolo[4,5-b]pyridin-2-yl-6-phenyl-hexan-1-oneIC5037.15 [1]
1-([1,3]Oxazolo[4,5-b]pyridin-2-yl)-7-phenylheptan-1-oneIC50524.81 [1]
1-(Oxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
Oleoyl oxazolopyridineIC5026.3 [1]
7-Phenyl-1-(5-phenyloxazol-2-yl)heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-[5-(Pyridin-2-Yl)-1,3,4-Oxadiazol-2-Yl]heptan-1-OneIC5010000.0 [1]
2-(7-Phenylheptanoyl)oxazole-5-carbonitrileIC5010000.0 [1]
5-([1,1'-Biphenyl]-4-ylmethyl)-N,N-dimethyl-2H-tetrazole-2-carboxamideIC50510.0 [1]
1-Oxazolo[4,5-B]pyridin-2-YL-1-dodecanoneIC5030.9 [1]
7-Phenyl-1-(5-(trifluoromethyl)oxazol-2-yl)heptan-1-oneIC5010000.0 [1]
Orlistat derivative, 17cIC502800.0 [1]
1-(Oxazolo[4,5-b]pyridin-2-yl)-8-phenyloctan-1-oneIC5046.77 [1]
1-(Oxazolo[4,5-b]pyridin-2-yl)-9-phenylnonan-1-oneIC503.63 [1]
7-Phenyl-1-(5-phenyl-1,3,4-oxadiazol-2-yl)heptan-1-oneIC5010000.0 [1]
Methyl 2-(7-phenylheptanoyl)oxazole-5-carboxylateIC5010000.0 [1]
1-(5-Methyl-2-oxazolyl)-7-phenyl-1-heptanoneIC5010000.0 [1]
1-([1,3]Oxazolo[4,5-b]pyridin-2-yl)octan-1-oneIC50630.96 [1]
1-Benzooxazol-2-yl-6-phenyl-hexan-1-oneIC503630.78 [1]
1-[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]-7-phenylheptan-1-oneIC5010000.0 [1]
1-(Oxazolo[4,5-b]pyridin-2-yl)-4-phenylbutan-1-oneIC502238.72 [1]
1-(Oxazolo[4,5-b]pyridin-2-yl)-5-phenylpentan-1-oneIC50204.17 [1]
CID 11991811IC5010000.0 [1]
7-Phenyl-1-(5-(2,2,2-trifluoroacetyl)oxazol-2-yl)heptan-1-oneIC501819.7 [1]
CID 11991890IC5010000.0 [1]
N,N-Dimethyl-2-(7-phenylheptanoyl)-1,3-oxazole-5-carboxamideIC5010000.0 [1]
2-(7-Phenylheptanoyl)oxazole-5-carbaldehydeIC5010000.0 [1]
1-(5-Bromooxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(5-Methylsulfanyl-1,3-oxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
[(2R,5R)-2-Benzyl-5-prop-2-ynoxypiperidin-1-yl]-[4-[bis(4-fluorophenyl)-hydroxymethyl]triazol-2-yl]methanoneIC501.26 [1]
1-(5-(2-Fluorophenyl)oxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(5-(3-Fluorophenyl)oxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(5-(4-Fluorophenyl)oxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(5-(4-Methoxyphenyl)oxazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-([1,3]Oxazolo[4,5-b]pyridin-2-yl)decan-1-oneIC5074.13 [1]
1-(Oxazolo[4,5-b]pyridin-2-yl)-1-oxo-pentaneIC5010000.0 [1]
7-Phenyl-1-(5-(pyridin-2-yl)-4H-1,2,4-triazol-3-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(2-(pyridin-2-yl)-2H-tetrazol-5-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(4H-1,2,4-triazol-3-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(2H-tetrazol-5-yl)-heptan-1-oneIC5010000.0 [1]
(5Z,8Z,11Z,14Z)-1-(Oxazolo[4,5-b]pyridin-2-yl)icosa-5,8,11,14-tetraen-1-oneIC502398.83 [1]
5-[[(4-Azido-3-iodobenzoyl)amino]methyl]-N,N-dimethyltetrazole-1-carboxamideIC50130.0 [1]
(2-Ethylpiperidin-1-yl)-[4-[hydroxy(diphenyl)methyl]triazol-2-yl]methanoneIC5063.1 [1]
7-Phenyl-1-(5-pyridin-4-yl-[1,3,4]oxadiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(5-pyridin-3-yl-[1,3,4]oxadiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
Leucine orlistat, (-)-IC505000.0 [1]
7-Phenyl-1-(5-(4-(2,2,2-trifluoroacetyl)phenyl)oxazol-2-yl)heptan-1-oneIC5010000.0 [1]
CID 16110650IC5010000.0 [1]
CID 16110720IC5010000.0 [1]
1-([1,3]Oxazolo[4,5-b]pyridin-2-yl)tetradecan-1-oneIC5074.13 [1]
1-([1,3]Oxazolo[4,5-b]pyridin-2-yl)hexadecan-1-oneIC5064.57 [1]
1-([1,3]Oxazolo[4,5-b]pyridin-2-yl)ethanoneIC5010000.0 [1]
1-(Oxazolo[4,5-b]pyridin-2-yl)-1-oxo-hexaneIC5010000.0 [1]
1-(5-(Furan-2-yl)-4H-1,2,4-triazol-3-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(2-(thiophen-2-yl)-2H-tetrazol-5-yl)-heptan-1-oneIC5010000.0 [1]
1-(1-Methyltetrazol-5-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
Methyl 3-(7-Phenylheptanoyl)-1,2,4-oxadiazole-5-carboxylateIC5010000.0 [1]
Methyl 5-(7-Phenylheptanoyl)-4H-1,2,4-triazole-3-carboxylateIC5010000.0 [1]
1-(3-(6-Chloropyridin-2-yl)-1,2,4-oxadiazol-5-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(3-(6-Bromopyridin-2-yl)-1,2,4-oxadiazol-5-yl)-7-phenylheptan-1-oneIC502041.74 [1]
1-(3-(6-Iodopyridin-2-yl)-1,2,4-oxadiazol-5-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
6-[5-(7-Phenylheptanoyl)-1,2,4-oxadiazol-3-yl]pyridine-2-carbonitrileIC501047.13 [1]
7-Phenyl-1-(5-(pyridin-2-yl)-thiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(5-(thiophen-2-yl)-thiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
1-(5-(Furan-2-yl)-1,3,4-thiadiazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
Methyl 5-(7-Phenylheptanoyl)-1,3,4-thiadiazole-2-carboxylateIC5010000.0 [1]
1-(6-(Furan-2-yl)-pyridazin-3-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(5-(thiophen-2-yl)-4H-1,2,4-triazol-3-yl)-heptan-1-oneIC5010000.0 [1]
1-(2-(Furan-2-yl)-2H-tetrazol-5-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(2-Methyl-2H-tetrazol-5-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
1-(1,3,4-Oxadiazol-2-yl)-7-phenylheptan-1-oneIC502691.53 [1]
1-(1,2,4-Oxadiazol-5-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)heptan-1-oneIC502754.23 [1]
1-(3-(Furan-2-yl)-1,2,4-oxadiazol-5-yl)-7-phenylheptan-1-oneIC50933.25 [1]
7-Phenyl-1-(3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl)-heptan-1-oneIC501949.84 [1]
Methyl 6-(5-(7-Phenylheptanoyl)-1,2,4-oxadiazol-3-yl)-picolinateIC5010000.0 [1]
6-(5-(7-Phenylheptanoyl)-1,2,4-oxadiazol-3-yl)-picolinic AcidIC5010000.0 [1]
7-Phenyl-1-(5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl)-heptan-1-oneIC5010000.0 [1]
1-(5-(Furan-2-yl)-1,2,4-oxadiazol-3-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl)-heptan-1-oneIC5010000.0 [1]
1-(5-(Furan-2-yl)-thiazol-2-yl)-7-phenylheptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(1,3,4-thiadiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(5-(pyridin-2-yl)-1,3,4-thiadiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(pyridazin-3-yl)-heptan-1-oneIC5010000.0 [1]
7-Phenyl-1-(6-(pyridin-2-yl)-pyridazin-3-yl)-heptan-1-oneIC5010000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Sn1-specific diacylglycerol lipase alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/sn1-specific-diacylglycerol-lipase-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Sn1-specific diacylglycerol lipase alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/sn1-specific-diacylglycerol-lipase-alpha-inhibitors-ic50-ki.
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