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Small conductance calcium-activated potassium channel protein 3 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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3-[(1R,4S,7S,13S,16S,19S,22S,25S,28R,31S,34S,37S,40R,47S,50R)-50-Amino-40-[[(2S)-5-amino-1-[[(2S)-5-amino-1-[[(2S)-1-amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-1,5-dioxopentan-2-yl]carbamoyl]-4-(4-aminobutyl)-47-(2-amino-2-oxoethyl)-34,37-bis(3-carbamimidamidopropyl)-19-[(1R)-1-hydroxyethyl]-7,22,31-trimethyl-25-(2-methylpropyl)-2,5,8,14,17,20,23,26,29,32,35,38,46,49-tetradecaoxo-42,43,52,53-tetrathia-3,6,9,15,18,21,24,27,30,33,36,39,45,48-tetradecazatricyclo[26.16.10.09,13]tetrapentacontan-16-yl]propanoic acidIC500.06 [1], 0.17 [2]
Pyridin-2-yl-(4-pyridin-2-yl-thiazol-2-yl)-amineIC5025.0 [1], 290.0 [2], 543.0 [3]
N-(4-Methylpyridin-2-yl)-4-(pyridin-2-yl)thiazol-2-amineIC504.0 [1], 56.0 [2], 59.0 [3]
Dequalinium chlorideIC501300.0 [1], 2000.0 [2]
5-Chloro-N-(thiophen-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineIC50350.0 [1], 580.0 [2]
N-Benzyl-5-chloropyrazolo[1,5-a]pyrimidin-7-amineIC501100.0 [1], 1600.0 [2]
2-Methyl-1-[[3-[(2-methyl-8-propan-2-ylisoquinolin-2-ium-1-yl)methyl]phenyl]methyl]-8-propan-2-ylisoquinolin-2-iumIC502970.0 [1]
2-Methyl-1-[[3-[(2-methyl-8-propan-2-ylisoquinolin-2-ium-1-yl)methyl]phenyl]methyl]-8-propan-2-ylisoquinolin-2-iumKi46.0 [1]
N-Phenyl-4-(pyridin-2-yl)thiazol-2-amineIC5030000.0 [1]
N-(4-(Pyridin-3-yl)thiazol-2-yl)pyridin-2-amineIC5030000.0 [1]
N-Pyridin-2-yl-4-pyridin-4-yl-1,3-thiazol-2-amineIC5030000.0 [1]
5-Chloro-N-(2-chlorobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5019100.0 [1]
5-Chloro-N-(4-(trifluoromethyl)benzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
N,4-Diphenyl-1,3-thiazol-2-amineIC5030000.0 [1]
2,4-Bis(2-pyridyl)thiazoleIC5030000.0 [1]
2,9-Diaza-17,23-diazoniahexacyclo[21.6.2.24,7.210,17.011,16.024,29]pentatriaconta-1(30),4,6,10(33),11,13,15,17(32),23(31),24,26,28,34-tridecaeneIC5060.0 [1]
(1S)-1-[3-[(1S)-6,7-Dimethoxy-2-methyl-3,4-dihydro-1H-isoquinolin-1-yl]propyl]-6,7-dimethoxy-2-methyl-3,4-dihydro-1H-isoquinoline;dihydrochlorideIC503000.0 [1]
N-(4-(Pyridin-2-yl)thiazol-2-yl)pyrimidin-2-amineIC5030000.0 [1]
N-[3-Chloro-5-(trifluoromethyl)pyridin-2-yl]-4-pyridin-2-yl-1,3-thiazol-2-amineIC5030000.0 [1]
5-Iodo-N-(4-(pyridin-2-yl)thiazol-2-yl)pyridin-2-amineIC5030000.0 [1]
N-(4-(Pyridin-2-yl)thiazol-2-yl)pyridin-4-amineIC5030000.0 [1]
2-(2-(Pyridin-2-ylmethyl)thiazol-4-yl)pyridineIC5030000.0 [1]
5-Chloro-N-(2-methylbenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5014600.0 [1]
5-Chloro-N-(2-(trifluoromethyl)benzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
5-Chloro-N-(2-methoxybenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5015900.0 [1]
5-Chloro-N-(2-(trifluoromethoxy)benzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5010000.0 [1]
5-Chloro-N-(3-chlorobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC505200.0 [1]
5-Chloro-N-(3-methylbenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5010700.0 [1]
5-Chloro-N-(3-(trifluoromethyl)benzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5014600.0 [1]
5-Chloro-N-(3-(trifluoromethoxy)benzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5011000.0 [1]
5-Chloro-N-(3-nitrobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC507900.0 [1]
5-Chloro-N-(4-chlorobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
5-Chloro-N-(4-methylbenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
5-Chloro-N-(4-(trifluoromethoxy)benzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5015400.0 [1]
5-Chloro-N-(4-nitrobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
5-Chloro-N-(4-phenoxybenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
5-Chloro-N-(3,4-dichlorobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
5-Chloro-N-(3,5-dichlorobenzyl)pyrazolo[1,5-a]pyrimidin-7-amineIC5030000.0 [1]
(R)-5-Chloro-N-(1-phenylethyl)pyrazolo[1,5-a]pyrimidin-7-amineIC501000.0 [1]
5-Chloro-N-(1,2-diphenylethyl)pyrazolo[1,5-a]pyrimidin-7-amineIC507500.0 [1]
2,10-Diaza-18,24-diazoniahexacyclo[22.6.2.211,18.14,8.012,17.025,30]pentatriaconta-1(31),4(35),5,7,11(34),12,14,16,18(33),24(32),25,27,29-tridecaeneIC5031.0 [1]
2-Methyl-1-[[4-[(2-methyl-8-propan-2-ylisoquinolin-2-ium-1-yl)methyl]phenyl]methyl]-8-propan-2-ylisoquinolin-2-iumKi1268.0 [1]
2-Methyl-1-[3-(2-methyl-8-propan-2-ylisoquinolin-2-ium-1-yl)propyl]-8-propan-2-ylisoquinolin-2-iumKi837.0 [1]
2-Methyl-1-[5-(2-methyl-8-propan-2-ylisoquinolin-2-ium-1-yl)pentyl]-8-propan-2-ylisoquinolin-2-iumKi575.0 [1]
2-Methyl-1-[4-(2-methyl-8-propan-2-ylisoquinolin-2-ium-1-yl)butyl]-8-propan-2-ylisoquinolin-2-iumKi214.0 [1]
Items per page: 1 - 10 of 45
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References

This online tool may be cited as follows

MLA

"Quest Database™ Small conductance calcium-activated potassium channel protein 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/small-conductance-calcium-activated-potassium-channel-protein-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Small conductance calcium-activated potassium channel protein 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/small-conductance-calcium-activated-potassium-channel-protein-3-inhibitors-ic50-ki.
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