![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_3fd8675cbf0c411f7aee264529c5cf97.svg) | 7,18-Bis[3-(dimethylamino)propyl]-7,18-diazaheptacyclo[14.6.2.22,5.03,12.04,9.013,23.020,24]hexacosa-1(23),2,4,9,11,13,15,20(24),21,25-decaene-6,8,17,19-tetrone | IC50 | 4500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_185ccb0cf3b983095272dcb588dd6eff.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 31000.0 [1], 35000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_185ccb0cf3b983095272dcb588dd6eff.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 15000.0 [1], 15500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_80fea5a9c0b55644141c8d025df24518.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[(2S)-2-[[(2S)-5-amino-1-[[(2S,3S)-1-[[(2S)-1-amino-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1,5-dioxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_31f753ac82aa9f3f78966dff2729a404.svg) | CID 53388144 | IC50 | 6800.0 [1], 19700.0 [2], 25600.0 [3] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_31f753ac82aa9f3f78966dff2729a404.svg) | CID 53388144 | Ki | 12800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_c8868c5b2b3ebb0020b42eba86a5415a.svg) | 2-Hydroxy-4-(2-(tosyloxy)acetamido)benzoic acid | IC50 | 84000.0 [1], 86000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_c8868c5b2b3ebb0020b42eba86a5415a.svg) | 2-Hydroxy-4-(2-(tosyloxy)acetamido)benzoic acid | Ki | 80000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_ac539ec1473267b3ea601e275753ac34.svg) | (1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | IC50 | 19250.0 [1], 33900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1a984ff2199cd3c90025d2a20db04a81.svg) | [4-[(E)-3-[[(2S)-1-[(2S)-2-[[(2S)-5-Amino-1-(benzylamino)-1,5-dioxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-3-oxoprop-1-enyl]phenyl] dihydrogen phosphate | IC50 | 135.0 [1], 138.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2974b5c10bb99da4b725e487cf6e31f2.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[(2S)-2-[[(2S)-1,5-diamino-1,5-dioxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | IC50 | 856.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_6fc7e40d17e3ad6997edb14858ca4fbe.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[(4-methylphenyl)sulfonyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 15800.0 [1], 115000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_6fc7e40d17e3ad6997edb14858ca4fbe.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[(4-methylphenyl)sulfonyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 7900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_5f5e7b227a8e5501c2ebc247f0bc2bbe.svg) | Stattic | IC50 | 5100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_bf5a4354e8299b78af102d81e8b2d6bd.svg) | Azd-1480 | IC50 | 23.0 [1], 80.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2d23a40b2f578d0d13066a710e0d7a4b.svg) | 4-[({3-[(Carboxymethyl)thio]-4-hydroxy-1-naphthyl}amino)sulfonyl]benzoic acid | IC50 | 20000.0 [1], 73000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_271358a0b38f21e9a43d969b7a893a36.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[(2S)-2-[[(2S)-5-amino-1-(benzylamino)-1,5-dioxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | IC50 | 409.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_63bb1f621cbe984baeb03da0aa23d324.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl-(2,4,6-trimethylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_ee476b92cfc790b0955549a2a31482be.svg) | [(1R,2E,8S,10R,11S)-6-(Acetyloxymethyl)-11-hydroxy-1,10-dimethyl-5-oxo-4,14-dioxatricyclo[9.2.1.03,7]tetradeca-2,6-dien-8-yl] (E)-2-methylbut-2-enoate | IC50 | 2200.0 [1], 2300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_3a2ea3008aa7d22b6720034a66c50870.svg) | [(2S)-3-(Benzylamino)-2-[[(2S)-1-[(2S)-4-methyl-2-[[(E)-3-(4-phosphonooxyphenyl)prop-2-enoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-3-oxopropyl] carbamate | IC50 | 379.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_46ae016b267325ee8678151546641a6b.svg) | [(2R,3S)-4-(Benzylamino)-3-[[(2S)-1-[(2S)-4-methyl-2-[[(E)-3-(4-phosphonooxyphenyl)prop-2-enoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutan-2-yl] carbamate | IC50 | 850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_ead4b824359611814c4360cd418e43c7.svg) | 4-[[2-[(4-Chlorophenyl)sulfonyl-methylamino]acetyl]-[(4-cyclohexylphenyl)methyl]amino]-2-hydroxybenzoic acid | Ki | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_e8cf17287faf0cd218c3638784ff8624.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl-(4-phenylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 6200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_66132e429df54e59916d5c9db9cbd2ba.svg) | 4-[[4-[1-(4-Cyanophenyl)sulfonylpiperidin-4-yl]phenyl]methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 8400.0 [1], 21500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1d982edc275fe83a58b4eae367b8ebf8.svg) | 4-[[4-[4-(4-Carbamoylphenyl)phenyl]phenyl]methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 8400.0 [1], 16700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_71e1df0fd5ef507d20147f6abe79f132.svg) | Vernolide-B | IC50 | 3200.0 [1], 4100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f2983f2ec2d6bdf8dfe3f7f629f31301.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-(4-methylphenyl)sulfonyloxyacetyl]amino]-2-hydroxybenzoic acid | IC50 | 43000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f2983f2ec2d6bdf8dfe3f7f629f31301.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-(4-methylphenyl)sulfonyloxyacetyl]amino]-2-hydroxybenzoic acid | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1619845a566e17328cb3d1b4fc1a3e4f.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[[(2S)-6-amino-1-[[(2S,3R)-1-[[(2S)-6-amino-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1619845a566e17328cb3d1b4fc1a3e4f.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[[(2S)-6-amino-1-[[(2S,3R)-1-[[(2S)-6-amino-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | Ki | 25900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_261812e8df72712f5234a5867dae1db5.svg) | 5,8-Dioxo-6-(2-piperazin-1-ylanilino)naphthalene-1-sulfonamide | Ki | 440.0 [1], 2420.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_609116da8750024b0bc56e31740c9139.svg) | Methyl 4-({[3-(2-methoxy-2-oxoethyl)-4,8-dimethyl-2-oxo-2H-chromen-7-yl]oxy}methyl)benzoate | IC50 | 63000.0 [1], 137000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_ef30c366d28792262453e396f9c81edc.svg) | 3-[[2-Chloro-4-[(1,3-dioxoinden-2-ylidene)methyl]-6-ethoxyphenoxy]methyl]benzoic acid | IC50 | 144000.0 [1], 256000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f5d2cbadfe1eb7e83fb57da27121f677.svg) | 4-[5-[(Z)-(3-Ethyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl]benzoic acid | IC50 | 18000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_cc6b275fe72e98f96332e70d392ffb48.svg) | [4-[(2S)-2-Acetamido-3-[[(2S)-1-[(2S)-2-[[(2S)-5-amino-1-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]amino]-1,5-dioxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate | IC50 | 600.0 [1], 739.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_337b9097ddc3813ceafbd10a1511f329.svg) | 4-[3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-oxo-propenyl]-benzoic acid | IC50 | 91000.0 [1], 447000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1716559248d6e99dae51113b4029254e.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 50000.0 [1], 95000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_eadd24cfebcc8b849dd92bf5f8c8fc18.svg) | [(1R,2E,8S,10R,11S)-8,11-Dihydroxy-1,10-dimethyl-5-oxo-4,14-dioxatricyclo[9.2.1.03,7]tetradeca-2,6-dien-6-yl]methyl (E)-2-methylbut-2-enoate | IC50 | 2400.0 [1], 2600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_3c392cd036d16f9a3c65f13b41f7ea9d.svg) | 4-Chloro-3-[5-[(1,3-diethyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]furan-2-yl]benzoic acid | IC50 | 60000.0 [1], 114000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_a25c64a0a197d46c1e033ae7abf19b3d.svg) | Genistein | IC50 | 24800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_a837c9a65d4411ddec4c52c49375903b.svg) | Oleanolic acid | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_875d19b61a74837bbc42b69de0d2d765.svg) | Niclosamide | IC50 | 250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_8af2d67dbbaf9354c2c59ae7499e9a91.svg) | Cryptotanshinone | IC50 | 4600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_e0db1010c174f6516b9baee0e4519cc2.svg) | Levomenol | IC50 | 73000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_39a4bcc2a4e088d25e2adb9476bfda0c.svg) | Bardoxolone methyl | IC50 | 2380.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_7eda287f73dc74dc97b540866ce3eb03.svg) | Loganin | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_5b92c2dc0f8499dcb6b85c3a0f704774.svg) | Piperlongumine | IC50 | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f6e456094f2ce08634f2eac277f787ea.svg) | Tetrahydrocurcumin | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_a5f32b5de0797b96bdca4c50f9e7f34e.svg) | Sweroside | IC50 | 89500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_d1e906454e7c1cdda2898196748bdfac.svg) | Morroniside | IC50 | 6900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_7c6d3954f60351d56e23c47f7327ded4.svg) | Ar-Turmerone | IC50 | 14210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_fc12d901759ca3c33d8822ad75c7ac75.svg) | (1E,4E)-1,5-Bis(4-hydroxy-3-methoxyphenyl)penta-1,4-dien-3-one | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_af14baaa637846b747237c907bdfdc77.svg) | Hydrazinocurcumin | IC50 | 16200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1e2d353fc507148e6ffecadeafbfd820.svg) | Incensole | IC50 | 15840.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_4cf999ac8c5530b16bc656fa121d0a24.svg) | [(E,6R)-6-[(2S,8S,9R,10S,13R,14S,16R,17R)-2,16-Dihydroxy-4,4,9,13,14-pentamethyl-3,11-dioxo-2,7,8,10,12,15,16,17-octahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-hydroxy-2-methyl-5-oxohept-3-en-2-yl] acetate | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_bb295b22ea7409ed7ec09d10443d4b8d.svg) | Incensole acetate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_294cba05fb9a42f9e7ce5c970f030307.svg) | N-[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]-2-phenylquinoline-4-carboxamide | IC50 | 74000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_16604a68fa586e4ee5393012d280f055.svg) | (2S,3R,4S)-3,4-Dihydroxy-6-methoxy-3-methyl-7-methylidene-2-pentyl-2,4-dihydropyrano[2,3-c]pyrrol-5-one | IC50 | 610000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_12e4ce3db9d117af0148fcb9fe2e01d0.svg) | 5,15-Diphenyl-21H,23H-porphine | IC50 | 280.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_3d828f908be01273f753bb2da73b0871.svg) | 4,6,8-Trimethyl-N-(4,4,6-trimethyl-1,4-dihydropyrimidin-2-yl)quinazolin-2-amine | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_503f5f913a6a7a4f6a78e8e4ad6983ce.svg) | Methyl (4aS,6aR,6aS,6bR,8aR,12aR,14bS)-2,2,6a,6b,9,9,12a-heptamethyl-10-oxo-3,4,5,6,6a,7,8,8a,11,12,13,14b-dodecahydro-1H-picene-4a-carboxylate | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_84c15cedad7a842175f9454486ad5ee5.svg) | 6-(4-Chlorophenyl)-3-(3-phenyl-1H-pyrazol-5-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | IC50 | 9600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f9c6ee5352cf80950ff89f853f6795ca.svg) | 2-Phenyl-N-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)quinoline-4-carboxamide | IC50 | 75000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_996c8778114b0cfe326bf14e93f54dcb.svg) | CID 4378002 | IC50 | 15700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2d998e2489195d9ad2f498af492971f2.svg) | (7-Ethoxy-4-methylquinazolin-2-yl)(4,4,6-trimethyl-1,4-dihydropyrimidin-2-yl)amine | IC50 | 20700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_fc13892ca06da1da8f73d605c2f1adc7.svg) | 6-(4-Chlorophenyl)-3-(1,4,5,6-tetrahydrocyclopenta[c]pyrazol-3-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | IC50 | 26800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f11eb4fd512939bd81ae34b2402854df.svg) | 6-Phenyl-3-(3-phenyl-1H-pyrazol-5-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | IC50 | 27000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_fdddb6b9f925303e88588554c567fef0.svg) | 6-Methyl-3-(3-phenyl-1H-pyrazol-5-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_5461b107735ff0cec611b9f1afe168ca.svg) | 6-Phenyl-3-(1,4,5,6-tetrahydrocyclopenta[c]pyrazol-3-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | IC50 | 21200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_003f3f83adf9a422e5848ff8d1df404b.svg) | 6-Methyl-3-(1,4,5,6-tetrahydrocyclopenta[c]pyrazol-3-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_36a27034df59fed9f50a62a1242d70af.svg) | CID 665910 | IC50 | 6800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_1dd6cbb974f0d7a6d321075f46185d52.svg) | 6-(3-Pyridylamino)-5,8-dioxo-5,8-dihydronaphthalene-1-sulfonamide | Ki | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_777440f6eb1e211b108f56938e32ab31.svg) | 4-Bromo-2-[3-(2,4-dichlorophenyl)acryloyl]-7-(methylamino)-2,4,6-cycloheptatrien-1-one | Ki | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_4af9423c072ca946db6b52ebfece6fd8.svg) | 8-Epiloganin | IC50 | 22900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_d381e8313772af3863be81ad753c065e.svg) | CID 72188643 | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_7dec959069bf3496e02c90052ff4ee32.svg) | Methyl (1S,3R,4aS,8S,8aS)-3-methoxy-1-methyl-8-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,3,4,4a,8,8a-hexahydropyrano[3,4-c]pyran-5-carboxylate | IC50 | 24800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_906c5add44bd876f8c4d6c7592c9c8b9.svg) | (1S,3E,7E,11E)-4,8,12-Trimethyl-1-propan-2-ylcyclotetradeca-3,7,11-trien-1-ol | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_32f5315d3b2e2ea6ea8e9c39a8701167.svg) | 5-[(4-Cyclohexylphenyl)methyl-(4-phenoxybenzoyl)amino]-2-hydroxybenzoic acid | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_5853da7c8f6dc32da2a80a7d09b00dd7.svg) | 5,6-Dimethyl-2-[(4,6,8-trimethylquinazolin-2-yl)amino]pyrimidin-4(1H)-one | IC50 | 6400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_4558afdb91559eda9ac65c352b12da24.svg) | 5-Benzyl-2-[(6-ethoxy-4-methylquinazolin-2-yl)amino]-6-methylpyrimidin-4(1H)-one | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_a9fccecec264cd161e67508caa6de878.svg) | 2-[(6-Ethoxy-4-methylquinazolin-2-yl)amino]-5,6-dimethylpyrimidin-4(1H)-one | IC50 | 11700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_b3af5963bd2243b3ee68247e497dfd7e.svg) | 6-Methyl-2-[(4,6,8-trimethylquinazolin-2-yl)amino]pyrimidin-4(3H)-one | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_47af915c52fbea418a5531455346bb66.svg) | 2-[(7-Methoxy-4-methylquinazolin-2-yl)amino]-6-methylpyrimidin-4-ol | IC50 | 33900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_64b9a5111ed09462ca5976dc60128957.svg) | 4-[(E)-2-[3-(4-Hydroxy-3-methoxyphenyl)-1H-pyrazol-5-yl]ethenyl]-2-methoxyphenol | IC50 | 18200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_5b3f7540324dd96a2af8af21a1b21e66.svg) | Methyl (4aS,6aR,6aS,6bR,8aR,12aR,14bS)-2,2,6a,6b,9,9,12a-heptamethyl-10-oxo-3,4,5,6,6a,7,8,8a,13,14b-decahydro-1H-picene-4a-carboxylate | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_a52938d7d44b8133452804910299c5d9.svg) | (7alpha-Hydroxy)-Morroniside | IC50 | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2b64d0c908e74a05ab4a0c47aff391d7.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl(quinolin-8-ylsulfonyl)amino]acetyl]amino]-2-hydroxybenzoic acid | Ki | 41000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2d957d1f60a775a2202a5027cf89a63d.svg) | Methyl (1S,3S,4aS,8S,8aS)-3-methoxy-1-methyl-8-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1,3,4,4a,8,8a-hexahydropyrano[3,4-c]pyran-5-carboxylate | IC50 | 32500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_ac38c0453d287b5fe4fc8654765028b3.svg) | 1,7-Bis[4-hydroxy-3-methoxy-5-(3-methylbutyl)phenyl]heptane-3,5-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_4c1e069f6fae2552f7f76ab1b4bb30ed.svg) | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl-(2,3,4,5,6-pentafluorophenyl)sulfonylamino]acetyl]amino]-N-hydroxybenzamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_03d49def98e02464f7ba7c19f56cc563.svg) | (1E,6E)-1,7-Bis[4-hydroxy-3-methoxy-5-(3-methylbut-2-enyl)phenyl]hepta-1,6-diene-3,5-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2ff667e517b58402e262b45f7e4f62cf.svg) | (2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2R)-1-(2-Aminoacetyl)pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-N-[(2S,3S)-1-[[(2S)-1-amino-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]pentanediamide | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_f557029ac4615b77c3a9b8b2e489a60d.svg) | (1E,4E)-1,5-Bis[4-hydroxy-3-methoxy-5-(3-methylbut-2-enyl)phenyl]penta-1,4-dien-3-one | IC50 | 22400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_2fcbc460cb3e88fdd9f2927ba87c6b67.svg) | (2S)-2-[[(2S)-2-[(4-Cyanobenzoyl)amino]-3-(4-phosphonooxyphenyl)propanoyl]amino]-4-methylpentanoic acid | IC50 | 310000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_c748ff13d45e1956c7987ae2adf279d4.svg) | (6S)-2-Methyl-6-[(2R,3R,5R,8R,9R,10R,12R,13R,14R,17S)-2,3,12-trihydroxy-4,4,8,10,14-pentamethyl-2,3,5,6,7,9,11,12,13,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-2-yl]oxyhept-1-en-3-one | IC50 | 590.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_4f5ea2060fbc5a77a6346e3e50a87e7d.svg) | (2R,3R,4R,5R,6S)-2-[[(2R,3S,4S,5R,6S)-6-[(E,2S)-2-[(2R,3R,5R,8R,9R,10R,12R,13R,14R,17S)-2,12-Dihydroxy-4,4,8,10,14-pentamethyl-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-2,3,5,6,7,9,11,12,13,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]-6-hydroxy-6-methylhept-4-en-2-yl]oxy-3,4,5-trihydroxyoxan-2-yl]methoxy]-6-methyloxane-3,4,5-triol | IC50 | 17100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_c5f593cd67286e38273a6c682d470fc1.svg) | 4-[[2-[(4-Chlorophenyl)methyl-(2,3,4,5,6-pentafluorophenyl)sulfonylamino]acetyl]-[(3,5-ditert-butylphenyl)methyl]amino]-2-hydroxybenzoic acid | Ki | 143800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_33e468c8b03774b7a71e527fc5f13108.svg) | (4Ar,6aR,6bS,8aS,12aS,14aR,14bR)-8a-methoxycarbonyl-4,4,6a,6b,11,11,14b-heptamethyl-3-oxo-5,6,7,8,9,10,12,12a,14,14a-decahydro-4aH-picene-2-carboxylic acid | IC50 | 25740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_dc250610c42de7a535bc9fb1bc951958.svg) | Methyl (4aS,6aR,6aS,6bR,8aR,12aR,14bS)-11-cyano-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,12,13,14b-dodecahydropicene-4a-carboxylate | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/signal-transducer-and-activator-of-transcription-3_fa44beb9835ce279475ab26c2940ec13.svg) | Dimethyl (4aR,6aR,6bS,8aS,12aS,14aR,14bR)-4,4,6a,6b,11,11,14b-heptamethyl-3-oxo-5,6,7,8,9,10,12,12a,14,14a-decahydro-4aH-picene-2,8a-dicarboxylate | IC50 | 25000.0 [1] |