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Sialidase 3 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
2-Deoxy-2,3-dehydro-n-acetyl-neuraminic acidIC5048000.0 [1]
2-Deoxy-2,3-dehydro-n-acetyl-neuraminic acidKi1600.0 [1], 2200.0 [2]
ZanamivirIC504000.0 [1], 6800.0 [2], 7000.0 [3], 8170.0 [4]
ZanamivirKi620.0 [1]
OseltamivirIC50500000.0 [1], 10000000.0 [2]
(2R,3R,4S)-3-[(2-Azidoacetyl)amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC504400.0 [1], 4700.0 [2], 21000.0 [3]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-phenylphenyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50700.0 [1], 12000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-phenylphenyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidKi280.0 [1]
(2R,3R,4S)-3-Acetamido-4-(diaminomethylideneamino)-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-phenylphenyl)triazol-1-yl]propyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50580.0 [1], 3800.0 [2]
(2R,3R,4S)-3-Acetamido-4-(diaminomethylideneamino)-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-phenylphenyl)triazol-1-yl]propyl]-3,4-dihydro-2H-pyran-6-carboxylic acidKi320.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-azido-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5019700.0 [1], 70000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(2-hydroxyethyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5038000.0 [1], 400000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(2-hydroxypropan-2-yl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50180000.0 [1], 300000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-(4-phenyltriazol-1-yl)propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC504600.0 [1], 20000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-(4-ethoxytriazol-1-yl)-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5090000.0 [1], 300000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(3-hydroxypropyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5039000.0 [1], 500000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-benzamido-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5034000.0 [1], 320000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(hydroxymethyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5080000.0 [1], 300000.0 [2]
(2R,3R,4S)-4-Hydroxy-3-[[2-(4-phenyltriazol-1-yl)acetyl]amino]-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1], 1000000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(phenoxymethyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC505500.0 [1], 45000.0 [2]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-(pentanoylamino)propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50110000.0 [1]
4-Acetamido-2-fluoro-5-[(4-phenylbenzoyl)amino]benzoic acidIC505000000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1S,2S)-1,2-dihydroxy-3-(pentanoylamino)propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC501000000.0 [1]
(2S,3R,4S)-3-Acetamido-4-azido-2-[(phenylmethoxyamino)methyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC5024000.0 [1]
(2S,3R,4S)-3-Acetamido-4-azido-2-[(phenylmethoxyamino)methyl]-3,4-dihydro-2H-pyran-6-carboxylic acidKi8000.0 [1]
(2S,3R,4S)-3-Acetamido-4-azido-2-[(2-phenylhydrazinyl)methyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC5020000.0 [1]
(2S,3R,4S)-3-Acetamido-4-azido-2-[(2-phenylhydrazinyl)methyl]-3,4-dihydro-2H-pyran-6-carboxylic acidKi11000.0 [1]
N-Acetyl-Neuraminic AcidIC50500000.0 [1]
PeramivirIC50500000.0 [1]
CarzenideIC502500000.0 [1]
4-Amino-2-deoxy-2,3-dehydro-n-neuraminic acidIC50180000.0 [1]
Benzoic acid, 4-(acetylamino)-3-((aminoiminomethyl)amino)-IC502500.0 [1]
4-Acetamido-3-[(E)-hydroxyiminomethyl]benzoic acidIC505500000.0 [1]
3-Guanidino-4-(methanesulfonamido)benzoic acidIC50100000.0 [1]
3-Guanidino-4-(methylcarbamoyl)benzoic acidIC505000.0 [1]
3-Guanidino-4-sulfamoyl-benzoic acidIC509000.0 [1]
3,5-Diguanidinobenzoic acidIC501500000.0 [1]
4-(Benzoylamino)benzoic acidIC501500000.0 [1]
3,4-Bis(phenylmethoxy)furan-2,5-dicarboxylic acidIC50920000.0 [1]
(3s,4r,5r)-4-(Acetylamino)-3-Amino-5-(Pentan-3-Yloxy)cyclohex-1-Ene-1-Carboxylic AcidIC501000000.0 [1]
(3S,4R,5R)-4-Acetamido-3-[4-(3-hydroxypropyl)triazol-1-yl]-5-pentan-3-yloxycyclohexene-1-carboxylic acidIC501000000.0 [1]
(3S,4R,5R)-4-Acetamido-3-[4-(2-hydroxypropan-2-yl)triazol-1-yl]-5-pentan-3-yloxycyclohexene-1-carboxylic acidIC501000000.0 [1]
3-Guanidinobenzoic acidIC505000000.0 [1]
4-Acetamido-3-(2-nitroethyl)benzoic acidIC502500000.0 [1]
3-Guanidino-4-(methylsulfinylmethyl)benzoic acidIC50140000.0 [1]
Benzoic Acid deriv. 178IC50300000.0 [1]
3-(Diaminomethylideneamino)-5-[(E)-hydroxyiminomethyl]benzoic acidIC50500000.0 [1]
(3S,4R,5R)-4-Acetamido-3-[4-(1-hydroxypropyl)triazol-1-yl]-5-pentan-3-yloxycyclohexene-1-carboxylic acidIC501000000.0 [1]
(3S,4R,5R)-4-Acetamido-3-[4-(1-hydroxycyclohexyl)triazol-1-yl]-5-pentan-3-yloxycyclohexene-1-carboxylic acidIC501000000.0 [1]
(3S,4R,5R)-4-Acetamido-3-[4-(1-hydroxycyclopentyl)triazol-1-yl]-5-pentan-3-yloxycyclohexene-1-carboxylic acidIC501000000.0 [1]
3-(Cyanoamino)benzoic acidIC504000000.0 [1]
Benzoic Acid deriv. 149IC501000000.0 [1]
3-Amino-5-guanidinobenzoic acidIC502000000.0 [1]
(2R,3R,4S)-3-Acetamido-4-azido-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC5054000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-(cyclopropanecarbonylamino)-1,2-dihydroxypropyl]-4-(diaminomethylideneamino)-3,4-dihydro-2H-pyran-6-carboxylic acid;2,2,2-trifluoroacetic acidIC501000000.0 [1]
(2R,3R,4S)-3-Acetamido-4-(cyclopropanecarbonylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-4-(cyclobutanecarbonylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-methoxyphenyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC505900.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[4-(4-carboxyphenyl)triazol-1-yl]-1,2-dihydroxypropyl]-4-(diaminomethylideneamino)-3,4-dihydro-2H-pyran-6-carboxylic acidIC50610.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-phenoxyphenyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC501000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[4-(4-carboxyphenyl)triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC501100.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-[4-(trifluoromethyl)phenyl]triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC503300.0 [1]
(2R,3R,4S)-3-Acetamido-4-amino-2-[(1R,2R)-3-[4-(4-carboxyphenyl)triazol-1-yl]-1,2-dihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-[4-(4-methylphenyl)triazol-1-yl]propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC508200.0 [1]
(2R,3R,4S)-3-Acetamido-4-(propanoylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[4-(4-aminophenyl)triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC508700.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[4-[4-(dimethylamino)phenyl]triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC509300.0 [1]
(2R,3R,4S)-3-Acetamido-4-azido-2-[(1R,2R)-3-[4-(4-carboxyphenyl)triazol-1-yl]-1,2-dihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC5020000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[4-(4-acetamidophenyl)triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC505500.0 [1]
(2R,3R,4S)-3-Acetamido-4-(pentanoylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[4-(4-fluorophenyl)triazol-1-yl]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5017000.0 [1]
(2R,3R,4S)-3-Acetamido-4-(2-carboxyethylcarbamoylamino)-2-[(1R,2R)-3-[4-(4-carboxyphenyl)triazol-1-yl]-1,2-dihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-(Heptanoylamino)-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50210000.0 [1]
(2R,3R,4S)-4-Hydroxy-3-(4-methylpentanoylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50150000.0 [1]
(2R,3R,4S)-3-(Hexanoylamino)-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50210000.0 [1]
(2R,3R,4S)-4-Hydroxy-3-(pentanoylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50140000.0 [1]
(2R,3R,4S)-4-Hydroxy-3-[[2-[4-(4-methylphenyl)triazol-1-yl]acetyl]amino]-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-2-[(1R,2R)-3-Acetamido-1,2-dihydroxypropyl]-4-hydroxy-3-(pentanoylamino)-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[(4-acetamidobenzoyl)amino]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC507200.0 [1]
(2R,3R,4S)-2-[(1R,2R)-1,2-Dihydroxy-3-(propanoylamino)propyl]-3-(hexanoylamino)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-[[2-[4-(4-Aminophenyl)triazol-1-yl]acetyl]amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50430000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-(3-methylbutanoylamino)propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5072000.0 [1]
(2R,3R,4S)-3-[[2-[4-(4-Fluorophenyl)triazol-1-yl]acetyl]amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50240000.0 [1]
(2R,3R,4S)-3-(5-Aminopentanoylamino)-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-4-(Diaminomethylideneamino)-3-(4-methylpentanoylamino)-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50150000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[5-[(4-acetamidobenzoyl)amino]pentanoylamino]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5031000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[(3-acetamidobenzoyl)amino]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC507100.0 [1]
(2R,3R,4S)-2-[(1R,2R)-3-(Butanoylamino)-1,2-dihydroxypropyl]-3-(hexanoylamino)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-[[2-[4-[4-(Dimethylamino)phenyl]triazol-1-yl]acetyl]amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC5046000.0 [1]
(2R,3R,4S)-4-Hydroxy-3-[[2-[4-(4-methoxyphenyl)triazol-1-yl]acetyl]amino]-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[(3-aminobenzoyl)amino]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5035000.0 [1]
(2R,3R,4S)-3-[[2-[4-(4-Acetamidophenyl)triazol-1-yl]acetyl]amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-2-[(1R,2R)-3-Acetamido-1,2-dihydroxypropyl]-3-(hexanoylamino)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-(Hexanoylamino)-2-[(1R,2R)-3-(hexanoylamino)-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-[[2-[4-(4-Carboxyphenyl)triazol-1-yl]acetyl]amino]-4-hydroxy-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-2-[(1R,2R)-3-(Hexanoylamino)-1,2-dihydroxypropyl]-4-hydroxy-3-(propanoylamino)-3,4-dihydro-2H-pyran-6-carboxylic acidIC50260000.0 [1]
(2R,3R,4S)-2-[(1R,2R)-1,2-Dihydroxy-3-(pentanoylamino)propyl]-4-hydroxy-3-(pentanoylamino)-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-1,2-dihydroxy-3-(4-pentyltriazol-1-yl)propyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC506700.0 [1]
(2R,3R,4S)-3-Acetamido-2-[(1R,2R)-3-[(4-aminobenzoyl)amino]-1,2-dihydroxypropyl]-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylic acidIC5031000.0 [1]
(2R,3R,4S)-4-Hydroxy-3-[[2-[4-[4-(trifluoromethyl)phenyl]triazol-1-yl]acetyl]amino]-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acidIC50500000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Sialidase 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/sialidase-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Sialidase 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/sialidase-3-inhibitors-ic50-ki.
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