![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_ab73d05fabc36590340ebf4c65ff52ff.svg) | 6-(4-Chlorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 15.7 [1], 168.0 [2] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_9931c7204127fed84870673d24299dc2.svg) | 5-[(4-Chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methyl-6-[3-(trifluoromethoxy)phenoxy]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 584.0 [2] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_858675c3f2704e10c03bd85d14b1e861.svg) | 5-[(4-Chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methyl-6-[3-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 1.91 [2] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_5883d849cdb1606e059476acc3cfdc35.svg) | 6-(3-Chlorophenoxy)-5-[(4-chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 117.0 [2] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_6741a7609f0d57af7c81e14c4a2de778.svg) | 6-(4-Chlorophenyl)-5-[(4-chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1.84 [1], 242.0 [2] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_177f2292db61c06d7c61cff315ee527e.svg) | 6-(3-Chlorophenyl)-5-[(4-chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methylfuro[2,3-d]pyrimidine-2,4-dione | IC50 | 1.0 [1], 134.0 [2] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_5022f7729dde6785cadadbeb2b57e139.svg) | 4-[(3S,4R)-1-(2,4-Dichlorophenyl)sulfonyl-4-hydroxy-4-(hydroxymethyl)pyrrolidin-3-yl]oxy-2-fluorobenzonitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_88a20d744c2c6c2a6eb62ab659c5d230.svg) | 3-(3-Hydroxypropyl)-1,5-dimethyl-6-naphthalen-2-ylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 34.9 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_413423556320dd91ae77fab4b4806bf5.svg) | 3-(3-Hydroxypropyl)-1,5-dimethyl-6-[2-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_cb1a8c9f9b55a9a7a8e9b092ac9b95da.svg) | 6-(3,4-Dichlorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_52f23b933f4c50720cff94112c9b26d4.svg) | 5-(1-Hydroxy-3-methylbutyl)-3-(3-hydroxypropyl)-1-methyl-6-[3-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 369.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_3d5a06b1c55616403e3edad32b84cd7d.svg) | 5-[(4-Chlorophenyl)-hydroxymethyl]-3-(3-hydroxypropyl)-1-methyl-6-[3-(trifluoromethoxy)phenoxy]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 194.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_77fd0c43e66dee2a80b7fa8107af1ced.svg) | 6-(3,4-Difluorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 112.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_e820ec1e7637a91c33a4bd53c765a079.svg) | 6-(3-Fluorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_a94f508d927362f4e90bd46702325a1f.svg) | 6-(3-Chlorophenyl)-5-[(4-chlorophenyl)methyl]-1,3-bis(3-hydroxypropyl)furo[2,3-d]pyrimidine-2,4-dione | IC50 | 4330.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_3d01f9dce626223d39fe196af7a99a2b.svg) | 6-(5-Chloropyridin-3-yl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_0829cfc6bcd7216f673efe2774940eb4.svg) | 6-(3-Chlorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 226.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_1a9f8e987929bd2fd6228fbd57e96054.svg) | 3-(3-Hydroxypropyl)-1-methyl-5-(3-methylbutyl)-6-[3-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_79e7c1aab4b79a79d515816be1e9a6db.svg) | 6-(2-Chlorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_bf4ce7b9346dae9a7f4e42bdd5c7b460.svg) | 6-(2,3-Dichlorophenyl)-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 31.6 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_ab08084c6eb7d1923018803c1bfb178c.svg) | 6-(3-Chlorophenyl)-5-[(4-chlorophenyl)-hydroxymethyl]-3-(3-hydroxypropyl)-1-methylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 55.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_3d452f33912b3bc4fb9bac05e862f753.svg) | 6-(3-Chlorophenyl)-5-[(4-chlorophenyl)methyl]-3-(3-hydroxypropyl)-1-methylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_c40153b261209ce61b8894e0260701df.svg) | 3-(3-Hydroxypropyl)-1,5-dimethyl-6-[3-(trifluoromethoxy)phenyl]thieno[2,3-d]pyrimidine-2,4-dione | IC50 | 82.2 [1] |
![](https://images.aatbio.com/dataset/ic50/short-transient-receptor-potential-channel-5_9e16adfb9a89259f53df24e84bfdd83e.svg) | 6-[4-Fluoro-3-(trifluoromethyl)phenyl]-3-(3-hydroxypropyl)-1,5-dimethylthieno[2,3-d]pyrimidine-2,4-dione | IC50 | 27.0 [1] |