| 7-Bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide | IC50 | 25000.0 [1] |
| 3,4-Dihydro-1H-isoquinolin-2-yl-[2-(4-methoxyanilino)-1,3-thiazol-4-yl]methanone | IC50 | 1260.0 [1] |
| 4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide | IC50 | 39810.72 [1] |
| (4-Methylpiperidino)[2-(4-toluidino)-1,3-thiazol-4-yl]methanone | IC50 | 630.0 [1] |
| [2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-[(2S,3S)-2,3-dimethylpiperidin-1-yl]methanone | IC50 | 100.0 [1] |
| 4-[(3S,4R)-1-(2,4-Dichlorophenyl)sulfonyl-4-hydroxy-4-(hydroxymethyl)pyrrolidin-3-yl]oxy-2-fluorobenzonitrile | IC50 | 10000.0 [1] |
| {2-[(4-Methoxyphenyl)amino]-1,3-thiazol-4-yl}(4-methylpiperidin-1-yl)methanone | IC50 | 800.0 [1] |
| [2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone | IC50 | 500.0 [1] |
| [2-(4-Chloroanilino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone | IC50 | 800.0 [1] |
| [2-(2-Chloroanilino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone | IC50 | 6300.0 [1] |
| [2-(4-Chloro-2-fluoroanilino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone | IC50 | 1600.0 [1] |
| [2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(4-methylpiperidin-1-yl)methanone | IC50 | 400.0 [1] |
| [2-(4-Methylanilino)-1,3-thiazol-4-yl]-(2-methylpiperidin-1-yl)methanone | IC50 | 800.0 [1] |
| [2-(4-Methylanilino)-1,3-thiazol-4-yl]-(2-phenylpiperidin-1-yl)methanone | IC50 | 12600.0 [1] |
| [2-(4-Methylanilino)-1,3-thiazol-4-yl]-(3-phenylpiperidin-1-yl)methanone | IC50 | 25000.0 [1] |
| [2-(4-Methoxyanilino)-1,3-thiazol-4-yl]-(4-phenylpiperidin-1-yl)methanone | IC50 | 2500.0 [1] |
| (4-Cyclohexylpiperidin-1-yl)-[2-(4-methylanilino)-1,3-thiazol-4-yl]methanone | IC50 | 6300.0 [1] |
| (2,3-Dimethylpiperidin-1-yl)-[2-(4-methylanilino)-1,3-thiazol-4-yl]methanone | IC50 | 250.0 [1] |
| [2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(2,3-dimethylpiperidin-1-yl)methanone | IC50 | 80.0 [1] |
| (2,3-Dimethylpiperidin-1-yl)-[2-[(6-fluoro-1,3-benzodioxol-5-yl)amino]-5-methyl-1,3-thiazol-4-yl]methanone | IC50 | 160.0 [1] |
| [5-Chloro-2-[(6-fluoro-1,3-benzodioxol-5-yl)amino]-1,3-thiazol-4-yl]-(2,3-dimethylpiperidin-1-yl)methanone | IC50 | 32.0 [1] |
| [2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-(2,3-dimethylpiperidin-1-yl)methanone | IC50 | 250.0 [1] |
| [2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-[(2R,3R)-2,3-dimethylpiperidin-1-yl]methanone | IC50 | 1000.0 [1] |
| [2-(1,3-Benzodioxol-5-ylamino)-1,3-thiazol-4-yl]-(1-methyl-3,4-dihydro-1H-isoquinolin-2-yl)methanone | IC50 | 316.0 [1] |
| [2-(1,3-Benzodioxol-5-ylamino)-5-methyl-1,3-thiazol-4-yl]-(1-methyl-3,4-dihydro-1H-isoquinolin-2-yl)methanone | IC50 | 316.0 [1] |
| [2-(1,3-Benzodioxol-5-ylamino)-5-methyl-1,3-thiazol-4-yl]-(5-methyl-7,8-dihydro-5H-1,6-naphthyridin-6-yl)methanone | IC50 | 10000.0 [1] |
| [2-(4-Chloro-2-fluoroanilino)-5-methyl-1,3-thiazol-4-yl]-(7,8-dihydro-5H-1,6-naphthyridin-6-yl)methanone | IC50 | 20000.0 [1] |