 | 4-Iodo-2,5-dimethoxyphenylisopropylamine | IC50 | 2.5 [1], 3.2 [2], 3.5 [3], 4.0 [4] |
| 4-Iodo-2,5-dimethoxyphenylisopropylamine | Ki | 1.6 [1], 2.0 [2], 42.7 [3] |
 | Serotonin | Ki | 12.0 [1], 13.0 [2], 13.49 [3] |
 | 1-(3-Chlorophenyl)piperazine | Ki | 10.0 [1], 24.0 [2], 32.0 [3] |
 | 6-Chloro-5-methyl-1-((2-(2-methylpyrid-3-yloxy)pyrid-5-yl)carbamoyl)indoline | Ki | 100.0 [1] |
 | 4-N-(3-Bromophenyl)-1,3,5-triazaspiro[5.5]undeca-1,4-diene-2,4-diamine | IC50 | 33.4 [1], 35.4 [2] |
| 4-N-(3-Bromophenyl)-1,3,5-triazaspiro[5.5]undeca-1,4-diene-2,4-diamine | Ki | 5.8 [1], 6.2 [2] |
 | Chlorpromazine | Ki | 39.81 [1], 52.0 [2], 80.0 [3] |
 | Aripiprazole | Ki | 0.36 [1], 1.26 [2], 1.4 [3] |
 | SB 243213 | Ki | 100.0 [1] |
 | 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b:4,5-b']difuran-4-yl)propan-2-amine | Ki | 1.15 [1], 1.6 [2] |
 | N-(Diaminomethylidene)-9-hydroxy-9-methylfluorene-2-carboxamide;hydrochloride | IC50 | 52.0 [1] |
| N-(Diaminomethylidene)-9-hydroxy-9-methylfluorene-2-carboxamide;hydrochloride | Ki | 4.3 [1] |
 | Pulicatin A | IC50 | 30000.0 [1] |
| Pulicatin A | Ki | 505.0 [1], 510.0 [2] |
 | N-[2-(1,3-Benzodioxol-5-yl)ethyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenylpropan-1-amine | IC50 | 794.33 [1] |
| N-[2-(1,3-Benzodioxol-5-yl)ethyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenylpropan-1-amine | Ki | 26.0 [1] |
 | N-[2-(1H-Indol-3-yl)ethyl]-1-(4-phenylbenzoyl)piperidine-4-carboxamide | IC50 | 14.1 [1], 18.7 [2] |
| N-[2-(1H-Indol-3-yl)ethyl]-1-(4-phenylbenzoyl)piperidine-4-carboxamide | Ki | 4.5 [1] |
 | Propranolol | IC50 | 5011.87 [1] |
| Propranolol | Ki | 218.0 [1] |
 | Clozapine | Ki | 3.16 [1], 7.18 [2] |
 | Risperidone | Ki | 15.0 [1], 19.95 [2] |
 | Olanzapine | Ki | 6.31 [1], 36.0 [2] |
 | Quetiapine | Ki | 135.9 [1], 251.19 [2] |
 | Raloxifene | Ki | 69.0 [1], 226.0 [2] |
 | Methysergide | Ki | 0.36 [1], 7.6 [2] |
 | Cisapride | Ki | 39.81 [1], 70.0 [2] |
 | Ketotifen | Ki | 29.0 [1], 31.62 [2] |
 | Methylergonovine | Ki | 0.8 [1], 0.96 [2] |
 | Lorcaserin | Ki | 1.3 [1], 189.0 [2] |
 | alpha-Methyl-5-HT | Ki | 13.0 [1] |
 | IB-Meca | Ki | 1080.0 [1] |
 | (R)-3-((2-(2-(4-Methylpiperidin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)phenol | Ki | 5.0 [1], 10000.0 [2] |
 | (S)-2-(6-Chloro-5-fluoro-indol-1-yl)-1-methyl-ethylamine | Ki | 5.1 [1] |
 | (R)-1-(4-Iodo-2,5-dimethoxyphenyl)propan-2-amine | Ki | 18.0 [1] |
 | S1RA | IC50 | 4700.0 [1] |
| S1RA | Ki | 328.0 [1] |
 | 4-(4-Fluoronaphthalen-1-yl)-6-isopropylpyrimidin-2-amine | IC50 | 0.7 [1], 19.0 [2] |
 | 5-Methoxy-alpha-methyltryptamine | Ki | 7.8 [1] |
 | 6-Chloro-5-methyl-N-quinolin-5-yl-2,3-dihydroindole-1-carboxamide | IC50 | 13.0 [1], 64.0 [2] |
 | N,N-Diallyl-5-methoxytryptamine | Ki | 31.62 [1], 58.88 [2] |
 | ATC-0175 free base | IC50 | 9.66 [1], 150.0 [2] |
 | 2-Phenethyl-5-hydroxychromone | IC50 | 8912.51 [1] |
| 2-Phenethyl-5-hydroxychromone | Ki | 2454.71 [1] |
 | SB 221284 | Ki | 12.59 [1] |
 | PRX-08066 free base | IC50 | 3.5 [1], 270.0 [2] |
 | Thalictruberine | Ki | 543.0 [1] |
 | N~2~-(3-Bromophenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-triazine-2,4-diamine | IC50 | 327.6 [1] |
| N~2~-(3-Bromophenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-triazine-2,4-diamine | Ki | 20.5 [1] |
 | 3-(Benzenesulfonyl)-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine | IC50 | 5130.0 [1] |
| 3-(Benzenesulfonyl)-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine | Ki | 1040.0 [1] |
 | 7-[4-[4-(2,3-Dichlorophenyl)-1,4-diazepan-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one | Ki | 0.6 [1] |
 | 5-Chloro-N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-3-methyl-1-benzothiophene-2-sulfonamide | Ki | 1000.0 [1] |
 | N~4~-(3-Methylphenyl)-1,3,5-triazaspiro[5.5]undeca-1,3-diene-2,4-diamine | IC50 | 459.4 [1] |
| N~4~-(3-Methylphenyl)-1,3,5-triazaspiro[5.5]undeca-1,3-diene-2,4-diamine | Ki | 19.8 [1] |
 | Watasemycin A | Ki | 3922.0 [1], 4700.0 [2] |
 | Watasemycin B | Ki | 3900.0 [1], 4695.0 [2] |
 | (4-(1H-Benzo[d]imidazol-2-yl)piperidin-1-yl)(phenyl)methanone | IC50 | 10000.0 [1] |
 | Ethyl 3-[(4-amino-1,3,5-triazaspiro[5.5]undeca-2,4-dien-2-yl)amino]benzoate | IC50 | 27.3 [1] |
| Ethyl 3-[(4-amino-1,3,5-triazaspiro[5.5]undeca-2,4-dien-2-yl)amino]benzoate | Ki | 7.2 [1] |
 | (4R,10As)-7-Chloro-4,6-dimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole | Ki | 19.0 [1], 40.0 [2] |
 | (4S,6R)-11-Bromo-9-methoxy-2-oxatricyclo[6.3.1.04,12]dodeca-1(11),8(12),9-trien-6-amine | Ki | 255.0 [1], 263.0 [2] |
 | 5-Methoxy-N-[6-(2-methylpyridin-3-yl)oxypyridin-3-yl]-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide | Ki | 50.12 [1] |
 | Pulicatin B | IC50 | 18000.0 [1] |
| Pulicatin B | Ki | 130.0 [1] |
 | Aerugine | Ki | 1360.0 [1], 1400.0 [2] |
 | Pulicatin G | Ki | 1260.0 [1], 1300.0 [2] |
 | Pulicatin F | Ki | 1000.0 [1], 1031.0 [2] |
 | (4R,10Ar)-7-Chloro-4,6-dimethyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole | Ki | 3.2 [1] |
 | N-Cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydrothiochromeno[4,3-c][1,2]oxazole-1-carboxamide | IC50 | 42.66 [1] |
| N-Cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydrothiochromeno[4,3-c][1,2]oxazole-1-carboxamide | Ki | 42.0 [1] |
 | (8S)-N-[2-(3-Fluorophenyl)ethyl]pentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 6983.0 [1] |
 | (8S)-N-[2-(3-Fluorophenyl)ethyl]-N-methylpentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 6086.0 [1] |
 | 5-Methyl-1,5-diazapentacyclo[10.8.1.02,7.08,21.013,18]henicosa-2(7),8(21),9,11,13,15,17-heptaene | Ki | 104.0 [1], 104.71 [2] |
 | N~2~-Phenyl-1,3,5-triazaspiro[5.5]undeca-1,3-diene-2,4-diamine | IC50 | 1641.3 [1] |
| N~2~-Phenyl-1,3,5-triazaspiro[5.5]undeca-1,3-diene-2,4-diamine | Ki | 151.3 [1] |
 | 5-Methyl-1-[2-(pyridin-2-ylmethyloxy)pyridin-5-ylcarbamoyl]-6-trifluoromethylindoline | Ki | 31.62 [1] |
 | 2-Chloro-N-[(3-chlorophenyl)methyl]-7H-purin-6-amine | IC50 | 890.0 [1] |
| 2-Chloro-N-[(3-chlorophenyl)methyl]-7H-purin-6-amine | Ki | 2160.0 [1] |
 | (2R)-1-(4-Bromo-2,3,6,7-tetrahydrofuro[2,3-f][1]benzofuran-8-yl)propan-2-amine | Ki | 1.15 [1], 1.6 [2] |
 | 2-(8-Methoxy-2,3,5,6-tetrahydrofuro[3,2-f][1]benzofuran-4-yl)ethanamine | Ki | 205.0 [1], 301.5 [2] |
 | 6,7-Dimethoxy-2,3-dihydrobenzofuran-4-ethanamine | Ki | 311.0 [1], 523.0 [2] |
 | (9R)-N-(Diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide | IC50 | 73.0 [1] |
| (9R)-N-(Diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide | Ki | 5.1 [1] |
 | (9S)-N-(Diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide | IC50 | 35.0 [1] |
| (9S)-N-(Diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide | Ki | 2.7 [1] |
 | 4-N-(3-Chlorophenyl)-1,3,5-triazaspiro[5.5]undeca-1,4-diene-2,4-diamine | IC50 | 46.9 [1] |
| 4-N-(3-Chlorophenyl)-1,3,5-triazaspiro[5.5]undeca-1,4-diene-2,4-diamine | Ki | 6.3 [1] |
 | Ethyl 3-[[4-(dimethylamino)-1,3,5-triazaspiro[5.5]undeca-1,4-dien-2-yl]amino]benzoate | IC50 | 284.5 [1] |
| Ethyl 3-[[4-(dimethylamino)-1,3,5-triazaspiro[5.5]undeca-1,4-dien-2-yl]amino]benzoate | Ki | 38.5 [1] |
 | 3-[(2-Amino-1,3,5-triazaspiro[5.5]undeca-1,4-dien-4-yl)amino]-N-ethylbenzamide | IC50 | 104.0 [1] |
| 3-[(2-Amino-1,3,5-triazaspiro[5.5]undeca-1,4-dien-4-yl)amino]-N-ethylbenzamide | Ki | 27.5 [1] |
 | 4-N-(3-Iodophenyl)-1,3,5-triazaspiro[5.5]undeca-1,4-diene-2,4-diamine | IC50 | 23.3 [1] |
| 4-N-(3-Iodophenyl)-1,3,5-triazaspiro[5.5]undeca-1,4-diene-2,4-diamine | Ki | 1.7 [1] |
 | N-(Diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide;hydrochloride | IC50 | 55.0 [1] |
| N-(Diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide;hydrochloride | Ki | 5.1 [1] |
 | (7S)-7-[(5-Fluoro-2-methylphenyl)methoxy]-2-[(2R)-2-methylpiperazin-1-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine | IC50 | 28.0 [1] |
| (7S)-7-[(5-Fluoro-2-methylphenyl)methoxy]-2-[(2R)-2-methylpiperazin-1-yl]-6,7-dihydro-5H-cyclopenta[b]pyridine | Ki | 7.7 [1] |
 | 5-(4-(2-Quinolylmethoxy)phenyl)-6-(4-fluorophenyl)pyridine-2(1H)-one | IC50 | 6.7 [1], 220.0 [2] |
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