| Clozapine | IC50 | 12.0 [1] |
| Clozapine | Ki | 6.3 [1], 9.1 [2] |
| Ketanserin | IC50 | 14.0 [1] |
| Aripiprazole | IC50 | 1100.0 [1], 2790.0 [2] |
| Olanzapine | IC50 | 9.0 [1], 100.0 [2] |
| Olanzapine | Ki | 2.3 [1] |
| Haloperidol | IC50 | 288.0 [1] |
| Haloperidol | Ki | 435.0 [1] |
| Risperidone | IC50 | 4.67 [1] |
| Risperidone | Ki | 0.81 [1] |
| Serotonin | Ki | 8.2 [1] |
| Mianserin | IC50 | 10.47 [1], 20.89 [2] |
| Mianserin | Ki | 4.3 [1], 8.1 [2] |
| Ziprasidone | IC50 | 0.42 [1] |
| Volinanserin | Ki | 0.1 [1] |
| Lysergide | Ki | 2.6 [1], 3.1 [2], 3.16 [3], 3.5 [4], 4.0 [5] |
| Spiperone | IC50 | 5.67 [1] |
| Spiperone | Ki | 1.1 [1], 1.58 [2], 2.24 [3], 2.9 [4] |
| Chlorpromazine | IC50 | 3.4 [1] |
| Chlorpromazine | Ki | 1.1 [1], 5.9 [2], 6.31 [3] |
| Sumatriptan | IC50 | 7943.28 [1], 10000.0 [2] |
| Sumatriptan | Ki | 376.0 [1], 1000.0 [2] |
| Cyproheptadine | Ki | 0.28 [1], 0.46 [2], 1.6 [3], 3.0 [4] |
| 6-Chloro-5-methyl-1-((2-(2-methylpyrid-3-yloxy)pyrid-5-yl)carbamoyl)indoline | Ki | 158.49 [1] |
| Cinanserin | Ki | 13.0 [1], 17.0 [2], 22.0 [3], 24.0 [4] |
| Benzo(1,2-b:4,5-b')dipyrrole-1(2H)-carboxamide, 3,5-dihydro-5-methyl-N-3-pyridinyl- | Ki | 1621.81 [1], 1995.26 [2] |
| (S)-2-(6-Chloro-5-fluoro-indol-1-yl)-1-methyl-ethylamine | Ki | 31.62 [1], 38.0 [2], 39.0 [3] |
| SB 243213 | IC50 | 32.4 [1] |
| SB 243213 | Ki | 158.49 [1] |
| 2,2-Diphenylethylamine | Ki | 4140.0 [1], 4610.0 [2] |
| 1-(2,4-Difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine | Ki | 0.42 [1] |
| (S)-1-(5,6-Difluoro-1H-indol-1-yl)propan-2-amine | Ki | 12.0 [1], 39.0 [2], 100.0 [3] |
| Imipramine | IC50 | 220.0 [1] |
| Imipramine | Ki | 94.0 [1], 160.0 [2] |
| Buspirone | Ki | 653.0 [1], 851.0 [2], 3240.0 [3] |
| N,N-Dimethyl-5-methoxytryptamine | Ki | 15.0 [1], 620.0 [2] |
| Zotepine | Ki | 0.5 [1], 0.91 [2], 2.7 [3] |
| Cariprazine | Ki | 22.0 [1], 23.0 [2] |
| Brolamfetamine | Ki | 0.6 [1], 41.0 [2] |
| 4-Bromo-2,5-dimethoxyphenethylamine | Ki | 0.66 [1], 1.0 [2], 34.0 [3] |
| Fananserin | Ki | 0.04 [1], 0.37 [2] |
| Nelotanserin | IC50 | 0.63 [1] |
| Nelotanserin | Ki | 0.51 [1], 0.63 [2] |
| 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b:4,5-b']difuran-4-yl)propan-2-amine | Ki | 0.48 [1], 10.73 [2] |
| 4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)butan-1-one | Ki | 30.9 [1] |
| 7-[4-[4-(2,3-Dichlorophenyl)-1,4-diazepan-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one | Ki | 0.6 [1], 2.0 [2], 16.0 [3] |
| N,N-Dimethyl-1-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)methanamine | IC50 | 22.91 [1], 1000.0 [2] |
| 1-(2,4-Difluorophenethyl)-4-fluoro-4-(4-fluorophenylsulfonyl)piperidine | Ki | 0.39 [1] |
| 9-(Methylaminomethyl)-9,10-dihydroanthracene | Ki | 52.0 [1] |
| 2-Phenyl-3-(2-piperidin-1-yl-ethyl)-1H-indole | Ki | 2.6 [1], 2.7 [2] |
| 6-Chloro-5-methyl-N-pyridin-3-yl-2,3-dihydroindole-1-carboxamide | Ki | 158.49 [1], 159.0 [2] |
| 5-[2-[4-(6-Fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-6,7-dihydro-5H-1-benzofuran-4-one | Ki | 0.56 [1], 0.72 [2] |
| N-[2-(1,3-Benzodioxol-5-yl)ethyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenylpropan-1-amine | IC50 | 5011.87 [1] |
| N-[2-(1,3-Benzodioxol-5-yl)ethyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenylpropan-1-amine | Ki | 165.0 [1] |
| N-[4-[2-[4-(1,2-Benzothiazol-3-yl)piperazin-1-yl]ethyl]cyclohexyl]furan-2-carboxamide | IC50 | 31.75 [1] |
| N-[4-[2-[4-(1,2-Benzothiazol-3-yl)piperazin-1-yl]ethyl]cyclohexyl]furan-2-carboxamide | Ki | 0.19 [1], 0.23 [2] |
| N-[4-[2-[4-(6-Chloro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]cyclohexyl]-2-(4-methoxy-4-methylcyclohexyl)acetamide | Ki | 14.0 [1], 16.0 [2], 19.0 [3] |
| Propranolol | IC50 | 5011.87 [1] |
| Propranolol | Ki | 419.0 [1] |
| Promethazine | IC50 | 23.0 [1] |
| Promethazine | Ki | 19.0 [1] |
| Methysergide | Ki | 3.83 [1], 10.0 [2] |
| Cisapride | Ki | 1.1 [1], 6.31 [2] |
| Ketotifen | Ki | 8.98 [1], 15.85 [2] |
| Phenethylamine | Ki | 16800.0 [1] |
| 5-Methoxytryptamine | Ki | 4.8 [1], 300.0 [2] |
| Sertindole | Ki | 0.6 [1], 0.85 [2] |
| Amoxapine | Ki | 0.44 [1], 1.77 [2] |
| Lorcaserin | Ki | 1.3 [1], 2782.0 [2] |
| GR-127935 | Ki | 15.85 [1], 42.7 [2] |
| (R)-3-((2-(2-(4-Methylpiperidin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)phenol | Ki | 5.0 [1], 10000.0 [2] |
| Altanserin | Ki | 0.13 [1], 0.3 [2] |
| 3-((4-(4-Chlorophenyl)piperazin-1-yl)methyl)-1H-pyrrolo[2,3-b]pyridine | Ki | 200.0 [1], 453.0 [2] |
| 5-Chloro-N-(4-methoxy-3-(piperazin-1-yl)phenyl)-3-methylbenzo[b]thiophene-2-sulfonamide | Ki | 1740.0 [1], 2511.89 [2] |
| Glemanserin | Ki | 2.5 [1] |
| 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide | IC50 | 2000.0 [1], 3000.0 [2] |
| 1-(1-Methylindol-5-yl)-3-(3-methyl-1,2-thiazol-5-yl)urea | Ki | 6309.57 [1] |
| 2,5-Dimethoxyamphetamine | Ki | 211.0 [1], 5200.0 [2] |
| SB 200646 hydrochloride | Ki | 6309.57 [1] |
| 3-[2-[4-(6-Fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-2lambda6-thia-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-triene 2,2-dioxide | Ki | 0.81 [1] |
| 2,4,5-Trimethoxyamphetamine | Ki | 57.9 [1], 1200.0 [2] |
| N,N-Diallyl-5-methoxytryptamine | Ki | 218.0 [1], 549.54 [2] |
| N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide | Ki | 330.0 [1], 430.0 [2] |
| CID 9820261 | IC50 | 150.0 [1] |
| CID 9820261 | Ki | 500.0 [1] |
| (S)-2-(7-Ethyl-1H-furo(2,3-g)indazol-1-yl)-1-methylethylamine | Ki | 13.0 [1] |
| SB 221284 | Ki | 398.11 [1] |
| 1,2,3,4-Tetrahydropyrazino[1,2-a]indole | Ki | 635.0 [1], 1040.0 [2] |
| 5-Methoxy-N-methyltryptamine | Ki | 4.1 [1], 450.0 [2] |
| Temanogrel | IC50 | 5.2 [1] |
| Temanogrel | Ki | 4.9 [1] |
| 3-[4-(4-Fluorobenzoyl)piperidinomethyl]tetralin-1-one | Ki | 1.62 [1], 23.44 [2] |
| 4-(3-(4-Chlorophenyl)-3-hydroxypyrrolidin-1-yl)-1-(4-fluorophenyl)butan-1-one | Ki | 75.8 [1], 241.5 [2] |