 | CID 44464263 | IC50 | 2.9 [1], 170.0 [2] |
 | N~2~-(1h-Benzimidazol-6-Yl)-N~4~-(5-Cyclobutyl-1h-Pyrazol-3-Yl)quinazoline-2,4-Diamine | IC50 | 5.3 [1], 8.0 [2] |
 | 4-Amino-N-(3-amino-1H-indazol-5-yl)cyclohexane-1-carboxamide | IC50 | 1490.0 [1], 13960.0 [2] |
 | CID 10077147 | IC50 | 87.0 [1] |
 | CID 92044402 | IC50 | 108.0 [1] |
 | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
 | N-[3-[[4-[3-(Cyclopropanecarbonylamino)propylamino]-5-iodopyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamide | IC50 | 67.0 [1] |
 | Clk1-IN-1 | IC50 | 10000.0 [1] |
 | (1S,3R)-3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 3050.0 [1] |
 | (1S,3R)-3-Amino-N-(3-amino-1H-indazol-5-yl)cyclohexane-1-carboxamide | IC50 | 330.0 [1] |
 | N-(3-Amino-1H-indazol-5-yl)piperidine-4-carboxamide | IC50 | 560.0 [1] |
 | 3-(Dimethylamino)-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 4230.0 [1] |
 | N-[3-(Naphthalen-1-ylamino)-1H-indazol-5-yl]azetidine-3-carboxamide | IC50 | 4940.0 [1] |
 | 3-Amino-N-[3-(2-fluoroanilino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 840.0 [1] |
 | 3-Hydroxy-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 2220.0 [1] |
 | 3-Amino-N-(3-anilino-1H-indazol-5-yl)cyclohexane-1-carboxamide | IC50 | 2730.0 [1] |
 | 4-Amino-N-(3-amino-1H-indazol-5-yl)butanamide | IC50 | 33000.0 [1] |
 | 3-Amino-N-[3-(2-methoxyanilino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 110.0 [1] |
 | 3-Amino-N-(3-amino-1H-indazol-5-yl)benzamide | IC50 | 18100.0 [1] |
 | 3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 11.0 [1] |
 | Methyl 3-[[5-[(3-aminocyclohexanecarbonyl)amino]-1H-indazol-3-yl]amino]benzoate | IC50 | 183.0 [1] |
 | 3-Amino-N-[3-(quinolin-8-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 589.0 [1] |
 | N-(3-Amino-1H-indazol-5-yl)piperidine-3-carboxamide | IC50 | 670.0 [1] |
 | (1R,3S)-3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 45.0 [1] |
 | N-[3-(Naphthalen-1-ylamino)-1H-indazol-5-yl]oxane-4-carboxamide | IC50 | 1830.0 [1] |
 | 3-Amino-N-[3-(quinolin-4-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 239.0 [1] |
 | N-[3-(Naphthalen-1-ylamino)-1H-indazol-5-yl]piperidine-4-carboxamide | IC50 | 315.0 [1] |
 | (1R,3R)-3-Amino-N-[3-(naphthalen-1-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 24.0 [1] |
 | 3-Amino-N-[3-[(4-methoxyphenyl)methylamino]-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 477.0 [1] |
 | 3-Amino-N-[3-[3-(trifluoromethyl)anilino]-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 288.0 [1] |
 | N-[5-[(3-Aminocyclohexanecarbonyl)amino]-1H-indazol-3-yl]benzamide | IC50 | 242.0 [1] |
 | N'-[3-[[5-Cyclopropyl-2-[(2-methyl-3,4-dihydro-1H-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboximidamide | IC50 | 45.0 [1] |
 | N-(3-Amino-1H-indazol-5-yl)piperidine-2-carboxamide | IC50 | 840.0 [1] |
 | 3-Amino-N-[3-(4-bromoanilino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 416.0 [1] |
 | 3-Amino-N-(3-amino-1H-indazol-5-yl)cyclohexane-1-carboxamide | IC50 | 368.0 [1] |
 | 3-Amino-N-[3-(quinolin-5-ylamino)-1H-indazol-5-yl]cyclohexane-1-carboxamide | IC50 | 40.0 [1] |
 | 3-Amino-N-(1H-indazol-5-yl)cyclohexane-1-carboxamide | IC50 | 22400.0 [1] |
 | N-[3-({4-[(3-Aminopropyl)amino]-5-Iodopyrimidin-2-Yl}amino)phenyl]pyrrolidine-1-Carboxamide | IC50 | 120.0 [1] |