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Serine/threonine-protein kinase TAO3 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-(Pyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-oneIC5010000.0 [1]
(7S)-2-(2-Aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-oneIC50126.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideIC5030000.0 [1]
4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideIC5030000.0 [1]
(6-Fluoro-1H-indol-2-yl)-[(3R)-1'-[(6R)-6-methylpiperidin-3-yl]spiro[2H-indole-3,3'-pyrrolidine]-1-yl]methanoneIC5030000.0 [1]
2-[[2-(4-Bromophenoxy)acetyl]amino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC5050.0 [1]
4-Heptoxy-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
N-[1-Oxo-1-(1,2,3,4-tetrahydronaphthalen-2-ylamino)propan-2-yl]-4-phenylmethoxybenzamideIC5050.0 [1]
2-[[2-(4-Phenylmethoxyphenoxy)acetyl]amino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC5050.0 [1]
4-Heptyl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-Hexoxy-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-Hexyl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-Butoxy-N-[1-oxo-1-(1,2,3,4-tetrahydronaphthalen-2-ylamino)propan-2-yl]benzamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-pentylbenzamideIC5050.0 [1]
2-Cyclopentyl-N-[2-oxo-1-pyridin-3-yl-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-2-phenylacetamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-pentoxybenzamideIC5050.0 [1]
N-[1-Oxo-1-(1,2,3,4-tetrahydronaphthalen-2-ylamino)propan-2-yl]-4-pentoxybenzamideIC5050.0 [1]
N-[2-(3-Chlorophenyl)ethyl]-5-[(E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxamideIC5050.0 [1]
3,5-Dimethyl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-phenylmethoxybenzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[1-oxo-1-(1,2,3,4-tetrahydronaphthalen-2-ylamino)propan-2-yl]benzamideIC5050.0 [1]
(2S)-N-Benzhydryl-2-[[(E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]amino]-3-phenylmethoxypropanamideIC5050.0 [1]
2-[[2-(4-Tert-butylphenoxy)acetyl]amino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC50500.0 [1]
N-[(2S)-4-Methyl-1-oxo-1-(1,2,3,4-tetrahydronaphthalen-1-ylamino)pentan-2-yl]-4-pentoxybenzamideIC5050.0 [1]
(2S)-2-[(4-Butoxyphenyl)carbamoylamino]-N-(2-phenylethyl)-3-phenylmethoxypropanamideIC5050.0 [1]
N-[(2S)-3-(1H-Indol-3-yl)-1-oxo-1-(1,2,3,4-tetrahydronaphthalen-1-ylamino)propan-2-yl]-5,6-dimethoxy-2,3-dihydro-1H-indole-2-carboxamideIC5050.0 [1]
N-[(3,4-Dichlorophenyl)methyl]-2-[4-(5-pyridin-2-ylpyrimidin-2-yl)phenoxy]acetamideIC5050.0 [1]
N-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-6-oxo-5,11-dihydrobenzo[b][1,4]benzodiazepine-3-carboxamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-phenylbenzamideIC5050.0 [1]
N-[3-Oxo-3-[[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]amino]-1-phenylpropyl]benzamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-phenoxybenzamideIC5050.0 [1]
2-[(6-Methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl 3-(benzoylamino)-3-phenylpropanoateIC5050.0 [1]
N-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-3-(3-ethoxypropyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]naphthalene-2-carboxamideIC50500.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-(trifluoromethoxy)benzamideIC5050.0 [1]
2-[(4-Phenylphenyl)methylamino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC505000.0 [1]
(2S)-2-Amino-1-N-(4-butylphenyl)-2-N-[(3,4-dichlorophenyl)methyl]pyrrolidine-1,2-dicarboxamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-4-ylamino)ethyl]benzamideIC50500.0 [1]
2-[[2-(3-Methoxyphenoxy)acetyl]amino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC5050.0 [1]
2-[[2-(4-Chlorophenoxy)acetyl]amino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC50500.0 [1]
N-[4-Methyl-1-oxo-1-(1,2,3,4-tetrahydronaphthalen-1-ylamino)pentan-2-yl]-4-phenylbenzamideIC50500.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl]benzamideIC5050.0 [1]
(2S)-2-Amino-2-N-[(3,4-dichlorophenyl)methyl]-1-N-(4-propan-2-ylphenyl)pyrrolidine-1,2-dicarboxamideIC5050.0 [1]
N-[3-[[2-[(6-Hydroxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]amino]-3-oxo-1-phenylpropyl]benzamideIC5050.0 [1]
N-[2-(Cyclohexylamino)-2-oxoethyl]-4-(4-ethylphenyl)benzamideIC505000.0 [1]
4-Butyl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC50500.0 [1]
2-[(4-Phenylphenyl)carbamoylamino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-phenylpiperazine-1-carboxamideIC505000.0 [1]
2-[4-(2-Naphthalen-1-ylethylsulfonyl)piperazin-1-yl]-N-pyridin-2-ylacetamideIC5050.0 [1]
N-[2-Oxo-2-(5,6,7,8-tetrahydronaphthalen-1-ylamino)ethyl]quinoline-3-carboxamideIC505000.0 [1]
N-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-4-(4-ethylphenyl)benzamideIC505000.0 [1]
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-2-[[2-[4-(trifluoromethoxy)phenoxy]acetyl]amino]acetamideIC50500.0 [1]
4-Hexoxy-N-[1-oxo-1-(1,2,3,4-tetrahydronaphthalen-2-ylamino)propan-2-yl]benzamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-5,6,7,8-tetrahydronaphthalene-2-carboxamideIC50500.0 [1]
N-[3-[(6-Hydroxy-1,3-benzothiazol-2-yl)amino]-3-oxo-1-phenylpropyl]benzamideIC505000.0 [1]
N-[2-(Benzylamino)-2-oxoethyl]-4-(4-ethylphenyl)benzamideIC505000.0 [1]
N-[2-Oxo-1-pyridin-3-yl-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-(1,2,4-triazol-1-yl)benzamideIC5050.0 [1]
N-[2-[(3,4-Dichlorophenyl)methylamino]-2-oxoethyl]-4-(4-ethylphenyl)benzamideIC505000.0 [1]
N-[2-Oxo-2-(5,6,7,8-tetrahydronaphthalen-1-ylamino)ethyl]quinoline-6-carboxamideIC505000.0 [1]
2-[[3,5-Bis(trifluoromethyl)phenyl]carbamoylamino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC505000.0 [1]
N-[2-(2,3-Dihydro-1,4-benzodioxin-3-ylmethylamino)-2-oxoethyl]-4-(4-ethylphenyl)benzamideIC505000.0 [1]
N-[3-[[2-[(6-Methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]amino]-3-oxo-1-phenylpropyl]benzamideIC5050.0 [1]
4-Cyclohexyl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-(naphthalen-1-ylamino)-2-oxoethyl]benzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]benzamideIC505000.0 [1]
2-Cyclopentyl-N-[2-oxo-2-[[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]amino]-1-pyridin-3-ylethyl]-2-phenylacetamideIC505000.0 [1]
2-[[2-(4-Bromophenoxy)acetyl]amino]-N-[(3,4-dichlorophenyl)methyl]acetamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]quinoline-3-carboxamideIC505000.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]benzamideIC505000.0 [1]
4-(4-Ethylphenyl)-N-methyl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC505000.0 [1]
4-Butoxy-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-(1-phenylethylamino)ethyl]benzamideIC5050.0 [1]
4-Imidazol-1-yl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-[[2-(trifluoromethyl)phenyl]methylamino]ethyl]benzamideIC5050.0 [1]
N-[3-[[2-[(4-Methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]amino]-3-oxo-1-phenylpropyl]benzamideIC505000.0 [1]
Tert-butyl 4-[[2-[[4-(4-ethylphenyl)benzoyl]amino]acetyl]amino]-3,4-dihydro-1H-isoquinoline-2-carboxylateIC50500.0 [1]
4-(1,3-Oxazol-5-yl)-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-piperidin-1-ylbenzamideIC5050.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-(2-phenylethylamino)ethyl]benzamideIC505000.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-(1-phenylpropylamino)ethyl]benzamideIC5050.0 [1]
2-Amino-4-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1-N-(3-ethoxypropyl)benzene-1,4-dicarboxamideIC505000.0 [1]
N-[2-Oxo-1-pyridin-3-yl-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-phenyldiazenylbenzamideIC5050.0 [1]
4-Morpholin-4-yl-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC50500.0 [1]
N-[3-[[2-(1,3-Benzothiazol-2-ylamino)-2-oxoethyl]amino]-3-oxo-1-phenylpropyl]benzamideIC5050.0 [1]
5,6-Dimethoxy-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-1H-indole-2-carboxamideIC5050.0 [1]
2-[2-(4-Phenylphenyl)ethylcarbamoylamino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC505000.0 [1]
N-[3-[[2-[(6-Methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]amino]-3-oxopropyl]benzamideIC505000.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-3-piperidin-1-ylpropanamideIC505000.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]-4-phenylmethoxybenzamideIC5050.0 [1]
3-Acetamido-N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-3-phenylpropanamideIC505000.0 [1]
4-(4-Ethylphenyl)-N-[2-[(2-methylphenyl)methylamino]-2-oxoethyl]benzamideIC5050.0 [1]
N-[2-Oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]quinoline-6-carboxamideIC5050.0 [1]
N-(6-Methoxy-1,3-benzothiazol-2-yl)-4-[[2-(4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-3-yl)acetyl]amino]butanamideIC5050.0 [1]
2-[(3-Ethylphenyl)carbamoylamino]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideIC505000.0 [1]
4-(4-Ethylphenyl)-N-[2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl]benzamideIC505000.0 [1]
N-[2-Oxo-2-(5,6,7,8-tetrahydronaphthalen-1-ylamino)ethyl]-4-piperidin-1-ylbenzamideIC505000.0 [1]
4-Hydroxy-N-[2-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]benzamideIC5050.0 [1]
2-[[2-(5,6-Dimethyl-4-oxothieno[2,3-d]pyrimidin-3-yl)acetyl]amino]-N-(6-methoxy-1,3-benzothiazol-2-yl)acetamideIC5050.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase TAO3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-tao3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Serine/threonine-protein kinase TAO3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-tao3-inhibitors-ic50-ki.
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