![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_0b2d442cd2d2265f4a4038b1178e2c93.svg) | Sgk1-IN-1 | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_041542b729950f52dcfeabb7da303944.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2,3-dichlorobenzenesulfonamide | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_d94d247b8d94478d48a3fd855a726fd7.svg) | Sgk1-IN-2 | IC50 | 5.0 [1], 25.0 [2], 630.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_67aa92f0a6e60d097a170a03a339d586.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluorophenyl]-5-chloro-2-fluorobenzenesulfonamide | IC50 | 2.0 [1], 50.0 [2], 2100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_e62b641671c6988040eff4527b1b8e4b.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluorophenyl]-2,5-dichlorobenzenesulfonamide | IC50 | 2.0 [1], 13.0 [2], 2600.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_e8bd31b5e73fd5543e38a7040f8d09e5.svg) | 5-Chloro-2-fluoro-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 4.0 [1], 88.0 [2], 1500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_719f39e8e6a3cbc3c8fd0eb89d4f1c7e.svg) | 2-Cyano-5-methyl-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 3.0 [1], 580.0 [2], 2900.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_4d1202127105cb1daa2d64e2e46f4ee9.svg) | 2-Fluoro-5-methyl-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 2.0 [1], 29.0 [2], 2400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_1b180f4117b68f6bcd8ac8dac3547357.svg) | 2-Chloro-5-methoxy-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 2.0 [1], 34.0 [2], 1500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_71ca2f2933f11b8728f61d95bd17cf54.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-cyano-5-methoxybenzenesulfonamide | IC50 | 2.0 [1], 40.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_2768d169a3912e09f95a7fddbd8e5314.svg) | 2,5-Dichloro-N-[4-(1H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 439.0 [1], 4550.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ab1ff539d6b95e799ed77fccd8889d84.svg) | 2,5-Dichloro-N-[2-fluoro-4-(1H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 496.0 [1], 3330.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_747f5415641441921a6433c90d916309.svg) | 2,3-Dichloro-N-[2-fluoro-4-(1H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 419.0 [1], 5730.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_6df6079f69293475aa6b7ebcec1bb541.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-5-chloro-2-hydrazinylbenzenesulfonamide | IC50 | 196.0 [1], 639.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_6464fd06aba489bbb0577d82b65b2c8f.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)-2-fluorophenyl]-2,3-dichlorobenzenesulfonamide | IC50 | 3.0 [1], 182.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ae53dd1a37c66e841eebcdb099863705.svg) | 2,5-Dichloro-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 2.0 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_48e4b79466daca25e0d4150617611ecc.svg) | 2,3-Dichloro-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 13.0 [1], 605.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_5172170c3d60774669800a36dedd7f8d.svg) | 5-Chloro-2-cyano-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 3.0 [1], 150.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_8d7b405a8d44ff166aafe4bc2df8d7e5.svg) | 5-Chloro-2-fluoro-N-[4-[4-(4-hydroxycyclohexyl)oxy-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]benzenesulfonamide | IC50 | 1.2 [1], 1.5 [2], 120.0 [3], 670.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_5d5314ac5efd12bafc43f7cde6d4a0bc.svg) | 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | IC50 | 13.0 [1], 580.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_48ae6690fff47b99703a334519252771.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-chlorobenzenesulfonamide | IC50 | 14.0 [1], 910.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_df8788468b5f8539a3186617bf4e3f9e.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-chloro-3-fluorobenzenesulfonamide | IC50 | 21.0 [1], 1260.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_adfc00125a30e567a31d48f869458309.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-fluorobenzenesulfonamide | IC50 | 22.0 [1], 1490.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_820e1e1e5303b3cfa3d63f56e4f7503c.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2,5-difluorobenzenesulfonamide | IC50 | 15.0 [1], 730.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_c1ba0f18b824b5bde22b32a30ffa7e20.svg) | N3-(4-Fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,4-diamine | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_d936f3dbad41727bd0deb9f9d3361e5f.svg) | 4-(5-Phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | IC50 | 40.0 [1], 1300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_7a4254b2b4cd2e9937dbe5863115462e.svg) | 3-(4'-Hydroxybiphenyl-4-Yl)-N-(4-Hydroxycyclohexyl)-1,4-Dihydroindeno[1,2-C]pyrazole-6-Carboxamide | IC50 | 1320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ec7101480603cb0553f102e7ea0b87e1.svg) | [4-(5-Naphthalen-2-Yl-1h-Pyrrolo[2,3-B]pyridin-3-Yl)phenyl]acetic Acid | IC50 | 63.0 [1], 880.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_00bfc608b564b72293041f1d78ddc15b.svg) | 2-Isobutyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | IC50 | 5.0 [1], 580.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_c26d95ea90ccec3e055894eb75178ff3.svg) | 2-Ethyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | IC50 | 20.0 [1], 710.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_4cbddc50029db49457c28e2e7350a4cd.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2,3-dichlorobenzenesulfonamide | IC50 | 2.0 [1], 261.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1], 5000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_472070ed1ed8bcedd050cf5e24588670.svg) | 5-Chloro-2-cyano-N-[4-[4-(4-hydroxycyclohexyl)oxy-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]benzenesulfonamide | IC50 | 1.5 [1], 110.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_efb825d6621ce2fdcc0cf594d8277947.svg) | N-[4-[4-(3-Aminopropoxy)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]-2,5-dichlorobenzenesulfonamide | IC50 | 1.2 [1], 280.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_65cb8f9dc24434bca9f1261e8ca1fc2b.svg) | 2-Fluoro-N-[4-[4-(4-hydroxycyclohexyl)oxy-3-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]-5-methoxybenzenesulfonamide | IC50 | 1.5 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_664eeca9ac43667086a0c79a514a817f.svg) | 2-Fluoro-N-[4-(4-methoxy-1H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl]-5-methylbenzenesulfonamide | IC50 | 1.5 [1], 50.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_859e1e7ff5e29eea05d381c0dada0708.svg) | N-[4-(4-Cyclopropyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl]-2-fluoro-5-methylbenzenesulfonamide | IC50 | 6.5 [1], 150.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_415f89e2894d8bb4806d9a15d6b0348d.svg) | 2-Fluoro-5-methyl-N-[4-[4-(morpholin-2-ylmethoxy)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]benzenesulfonamide | IC50 | 6.2 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_7d261ca75cf628ad2d48e3d7448ae45d.svg) | N-[4-[3-Amino-4-(2-methylpropoxy)-2H-pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]-2,5-dichlorobenzenesulfonamide | IC50 | 130.0 [1], 220.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_03c1abb8300d1e100aedbf677c054fed.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl]-5-chloro-2-fluorobenzenesulfonamide | IC50 | 19.0 [1], 390.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_e8080c4c06060d646c51b5eb37e46806.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-1-(2,5-difluorophenyl)methanesulfonamide | IC50 | 28.0 [1], 9830.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_181b8f1a3cd0e2642bcee59206df68a1.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-5-bromothiophene-2-sulfonamide | IC50 | 3.0 [1], 718.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_8f061e4323f5ae29407d3cd99b48fb9b.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-1-methyl-3-(trifluoromethyl)pyrazole-4-sulfonamide | IC50 | 14.0 [1], 518.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_59cfd20f4c681ff4fe1e4d8aac0edc7c.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]furan-2-sulfonamide | IC50 | 19.0 [1], 6840.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ab8494cdf78c54ea570f0c2792bc096e.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2,5-dichlorothiophene-3-sulfonamide | IC50 | 1.0 [1], 63.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_71cd4594c674a08a8cd460a4062d09a9.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]benzenesulfonamide | IC50 | 124.0 [1], 9720.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_0ee5eb877ff33ff7871d744ecbefc8f2.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2-chlorobenzenesulfonamide | IC50 | 1.0 [1], 396.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_45c52de2c5ede1d6f3f8c94a546a62f8.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2,5-dichlorobenzenesulfonamide | IC50 | 1.0 [1], 14.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_372b51b4f1b8a8ea3269207e4557168e.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-3-chloro-2-cyanobenzenesulfonamide | IC50 | 6.0 [1], 199.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_1e2c7256df9324872b2d50e13b60d9b7.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-5-cyano-2-methylbenzenesulfonamide | IC50 | 46.0 [1], 1970.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_5aa75ae73e1884a806af91a812f5c354.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-5-chloro-2-cyanobenzenesulfonamide | IC50 | 2.0 [1], 17.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_a70679b79a6c9a97071dd8a8073cd811.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2-fluoro-5-(trifluoromethyl)benzenesulfonamide | IC50 | 1.0 [1], 129.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_4d48a055fa8363d8e595d6b3a317ca04.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2-fluorobenzenesulfonamide | IC50 | 1.0 [1], 1110.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_89756428f3920532d916ff5c635b51f1.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2,3-difluorobenzenesulfonamide | IC50 | 9.0 [1], 2580.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_0b745985aa8e0a7518750d8c6d6ab8d0.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2,5-difluorobenzenesulfonamide | IC50 | 1.0 [1], 186.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_52e484549752238eb845d353fe871b4d.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-2-chloro-5-methoxybenzenesulfonamide | IC50 | 1.0 [1], 51.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_66bbab2a504a7f840dcac75b564ac8b2.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-5-bromo-2-chlorobenzenesulfonamide | IC50 | 1.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_9b2d58a6f5e4f6c9408867797bfb3953.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-5-bromo-2-fluorobenzenesulfonamide | IC50 | 5.0 [1], 6.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ece2b29716bab2b6e60285623c252a40.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-3-chloro-2-fluorobenzenesulfonamide | IC50 | 5.0 [1], 169.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_2529216ec231416ea7e332f0d1bc18ae.svg) | N-[4-(3-Amino-1H-indazol-6-yl)phenyl]-5-chloro-2-fluorobenzenesulfonamide | IC50 | 1.0 [1], 7.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_3f4e4bad084da46334514b3b13bd7395.svg) | 2,5-Difluoro-N-[4-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]benzenesulfonamide | IC50 | 29.0 [1], 1340.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_05f576155567981ba046bac9ea504cb1.svg) | 2-Methyl-2-(4-(5-(naphthalen-2-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)propanoic acid | IC50 | 63.0 [1], 870.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_236a608fa7a5e7c483abf27fa575a0fb.svg) | 2-Methyl-2-(4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)propanoic acid | IC50 | 50.0 [1], 1460.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_8c1771d412e43677072bdbd6d419a5b6.svg) | 2-(4-(5-(3-Cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)phenyl)-2-methylpropanoic acid | IC50 | 40.0 [1], 2000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_c0dafbb26d443d750405f366dc607672.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-fluoro-5-methoxybenzenesulfonamide | IC50 | 2.0 [1], 4.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_97a59b0a2cff7570cbe7fe87a24ee0d0.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-cyano-5-methylbenzenesulfonamide | IC50 | 3.0 [1], 61.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_81d4d4c59b75780863024a276bb241a7.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-chloro-5-methoxybenzenesulfonamide | IC50 | 2.0 [1], 34.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_0d26d675a2631d6927d92d7216129431.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-fluoro-5-methylbenzenesulfonamide | IC50 | 2.0 [1], 39.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_3c47523c8a6a7a8c6d644aa9e59de0d4.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-5-chloro-2-cyanobenzenesulfonamide | IC50 | 10.0 [1], 293.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_777dc13203dcdd300cf50c41b4182fb3.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2,5-dichlorothiophene-3-sulfonamide | IC50 | 4.0 [1], 183.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ebda4ebfc5e6d74eb9240ed1cdc435ef.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]naphthalene-1-sulfonamide | IC50 | 16.0 [1], 760.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_46962734d082e25b02afd7b701eaa110.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-5-chloro-2,4-difluorobenzenesulfonamide | IC50 | 2.0 [1], 41.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_be942fb7ce53b9b16b6c240008607ee6.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-2-chloro-4-(trifluoromethyl)benzenesulfonamide | IC50 | 407.0 [1], 18900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ec4ce706d23eda6fc97c252269f35dbb.svg) | N-[4-(3-Amino-4-cyclopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl]-2-cyano-5-methoxybenzenesulfonamide | IC50 | 1.5 [1], 61.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_4a933442e65177279215ed668a9abfb3.svg) | 2,5-Dichloro-N-[4-(3-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl]benzenesulfonamide | IC50 | 1.2 [1], 830.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_0dcf017614298724cb9a70e000610083.svg) | N-[4-(3-Amino-2H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl]-5-cyano-2-fluorobenzenesulfonamide | IC50 | 47.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_baaf5d744d6a6cfce80c91a2d9f5d31e.svg) | 5-Chloro-N-[4-[3-[(5-chloro-2,4-difluorophenyl)sulfonylamino]-1H-pyrazolo[3,4-b]pyrazin-6-yl]phenyl]-2,4-difluorobenzenesulfonamide | IC50 | 413.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_af6c849cab29e175678bc52964f46c9c.svg) | Tofacitinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_1970071dd3288d1434749caa6fc51ef1.svg) | 4,5,6,7-Tetrabromo-N,N-dimethyl-1H-benzimidazol-2-amine | IC50 | 3570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_4e8b5202a71aafe003ab207cc4576058.svg) | 3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 201.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_ab2268bff60761ec9560ebfb5b03f869.svg) | CID 6918852 | Ki | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_f556b5bb65759c4a8d3410b88a5c8036.svg) | JNK Inhibitor V | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 9400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_d44bb541aaceb7d87194194110f1e1e1.svg) | CID 11634725 | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_7489af297ca5d99d886f106758e75d74.svg) | 2-[4-(3-Phenylquinoxalin-2-yl)phenyl]propan-2-amine | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_6b7ed5d4bde8a2dd13f619c48594a177.svg) | Merck-22-6 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_a6b96a46d036a13f6af94a3ab0ae6bb0.svg) | 4-(Pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_5a8c83043b67c6f0ac7a7140b45ffee9.svg) | (3Z)-6-(4-Hydroxy-3-methoxyphenyl)-3-(1H-pyrrol-2-ylmethylene)-1,3-dihydro-2H-indol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_7cd07c14c9a6699a18c59379f39dd9e2.svg) | N~3~-Cyclopropyl-N~4~'-(Cyclopropylmethyl)-6-Methylbiphenyl-3,4'-Dicarboxamide | IC50 | 33000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_1f3d98cabb62838272ebe2a447268da2.svg) | 10,11-Dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_d2497ae1855cd4d782afa7fbefc515ee.svg) | 3-[4-[[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-2-phenylquinoxaline-6-carboxylic acid | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_79ccba98dd462b1631c9db41481af774.svg) | (2S)-1-N-(5-Isoquinolin-6-yl-1,3,4-thiadiazol-2-yl)-3-[4-(trifluoromethyl)phenyl]propane-1,2-diamine | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 9400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 9400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_25774502353a4c4c2828afb710c6fc93.svg) | 2-[4-[[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-3-phenylquinoxaline-6-carboxylic acid | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-sgk1_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 8176.0 [1] |