![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_ddc31cb72a8aa21440e26147cfc64b1b.svg) | Lfm-a13 | IC50 | 61000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_ac9222422aa3967de001af41e8ffd43b.svg) | Wortmannin | IC50 | 48.0 [1], 49.0 [2], 220.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_6603a475932cb1632b1b43c2f664a423.svg) | 2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one | IC50 | 3000.0 [1], 88000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_44b484a9c1048f0607f62988f78cc00d.svg) | BI-2536 | IC50 | 20.78 [1], 90.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_6eb85432df5d02aab0b18480749b4c05.svg) | 5-(5,6-Dimethoxy-1-benzimidazolyl)-3-[[2-(trifluoromethyl)phenyl]methoxy]-2-thiophenecarboxamide | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_693b4dc5e5c2d34bce7645a52c5c3915.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-(8-phenyloctyl)imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 280.0 [1], 1200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_af4ffbf4dbfd01d2f1479cc420b05ad5.svg) | 3-[(E)-[3-[(E)-2-Pyridin-4-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_f1366eff0c7fe9a3f64ff9c8af68c3bc.svg) | 1-Methyl-8-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 1439.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_f622aa4e29ed2191958d7259f200be05.svg) | 8-[5-Amino-2-(trifluoromethoxy)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 154.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_593760634b5e73daf93d1b0d76afa02a.svg) | 1-Methyl-8-[5-[2-(1-methylpyrrolidin-2-yl)ethylamino]-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 485.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_2cd9f08f5dea65516c41f9c3534be4cf.svg) | Thymoquinone | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_e1bd3c1d60717a09fae0532edc016b5c.svg) | Axitinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_84fae1800055ebf670b925911d10e379.svg) | CFI-400945 (free base) | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_9ac8c17a1cd78f944fc3ce79f16d4238.svg) | Nms-P937 (nms1286937) | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_b800922b5c769ca9c52161d0b5a33c4a.svg) | 8-[2-Methoxy-5-(4-methylpiperazin-1-yl)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_93fd355a308bbc6a4f2d55c507cc6f63.svg) | 3-[(2-Chlorophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_380f5093e8c48de5971e557cdec1d4dc.svg) | CID 11328632 | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_ff17b6f8c0d6e75a664fb18c2f79a1b9.svg) | 5-[6-(1-Methylpiperidin-4-yl)oxybenzimidazol-1-yl]-3-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]thiophene-2-carboxamide | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_4d98885183dedb60fb4e060206ecfc34.svg) | 3-(1,3-Benzodioxol-5-yl)-N-[(1S)-1-phenylethyl]-[1,2]oxazolo[5,4-c]pyridin-5-amine | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_ae3cb292e66be9578004d2faaf9b275f.svg) | 8-Anilino-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_371bf7e5b9caef5f042b6633dc19c345.svg) | Benz[b]indeno[1,2-e]pyran-6,11-dione | IC50 | 8970.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_b684ab957065832f0929f6b907dcb29f.svg) | 3-[(E)-[3-[(E)-2-[4-[(Dimethylamino)methyl]phenyl]ethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_127674c15dddfb61d8f9a13c7daa5925.svg) | GSK 461364 analogue I | IC50 | 630.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 1085.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a5c5bae0fd3ddf532506780bb4f7f125.svg) | Khk-IN-1 | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_345a18e52d71f6ef064960bce460999a.svg) | 2-Pyrrolidin-1-yl-N-[3-(3-sulfamoylphenyl)-1H-indazol-5-yl]-2-thiophen-3-ylacetamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_0731e513dda8b4631f904dc8f0082e8c.svg) | 7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrile | Ki | 820.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_1fe60e6d13674f8cf1dfc82fac3410b2.svg) | 7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrile | Ki | 560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_029f5b4cad89a2c59efa869fd9853874.svg) | N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_c2aa7e0fb640ea7529d7330460976868.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamide | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_98598461b658b3f77425e67c797f8e2d.svg) | N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a3bd9a5a28d4f4d2890ccf5cdf08d883.svg) | N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_cde4e83180955e4849d8daba0837480d.svg) | N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamide | Ki | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_fc2bed3411d27892c4eee6ba2912d663.svg) | 5-[5,6-Bis(Methyloxy)-1h-Benzimidazol-1-Yl]-3-{[1-(2-Chlorophenyl)ethyl]oxy}-2-Thiophenecarboxamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_0f91699454b38a2b6da01a1d4e67d200.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-(2-fluoro-6-phenoxyphenyl)octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 1450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_5ac6d45a2decd47b9da10a8a7645b06e.svg) | 5-Methoxy-3-[(E)-[3-[(E)-2-[6-(4-methylpiperazin-1-yl)pyridin-3-yl]ethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a7dbdd6952b28399f700d51a83f5e290.svg) | 1-Methyl-8-(2-methylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_262c5527ba96216e81ae5e081ba9279f.svg) | 3-Methyl-N-[6-methylsulfanyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine | IC50 | 785.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_b80728998e0b173ed97842a79c1db051.svg) | 5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_77eb8e9cdf9ebb4dafaaacd9407e9c0b.svg) | 3-[(1R)-1-[(2S,6R)-2,6-Dimethylmorpholin-4-yl]ethyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_d177c352a8a90316beccdf76166341e8.svg) | N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_3d1aadff81b1eaa89d51e0ddb6f70b40.svg) | 8-(2-Methoxyanilino)-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_241ed90fbf6182a4fbaa5becdb0166c4.svg) | 1-Methyl-8-(2-(trifluoromethoxy)phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_c0567c6a189a92c4afaa9b25013eacd2.svg) | (2'S,3R)-2'-[3-[(E)-2-[4-[(Dimethylamino)methyl]phenyl]ethenyl]-1H-indazol-6-yl]spiro[1H-indole-3,1'-cyclopropane]-2-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_77724ee49e47eee53829f305dbaa4d17.svg) | 3-[(1R)-1-[4-[(Tert-butylamino)methyl]-2-(difluoromethoxy)phenyl]ethoxy]-5-imidazo[1,2-a]pyridin-3-ylthiophene-2-carboxamide | IC50 | 178.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_da63de9d92c2d79ff40b1d8ee8ae24af.svg) | 3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-N-(2-hydroxyethyl)-4-methylbenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a60212f39beebdf18c71eb0e0e1f5d97.svg) | 5-Methyl-5,11-dihydro-6H-indeno[2,1-b]quinoline-6,11-dione | IC50 | 200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_c9bdb8daaee16f4ae67bee958a08b36a.svg) | 3-[(E)-Benzotriazol-5-ylidenemethyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_c6bfd7ef500997029a4f4a83dcda424b.svg) | 3-[(E)-[3-[(E)-2-[4-[(Dimethylamino)methyl]phenyl]ethenyl]indazol-6-ylidene]methyl]-5-methoxy-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_26443a912f6919cd6b3ccaf7be5c82f6.svg) | (E)-3-((1H-Indazol-6-yl)methylene)indolin-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_bcde0b22d99ef699f2a357964c268cd8.svg) | 3-[(E)-[3-[(E)-2-Pyridin-3-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_72ca37613b1b8b338656d9af36efcf6c.svg) | 5-Methyl-3-[(E)-[3-[(E)-2-pyridin-4-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a4228653718e615f73d83355c1b50750.svg) | 5-Chloro-3-[(E)-indazol-6-ylidenemethyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_d9c1a80cf77465f57c5f3c8dd8216c0d.svg) | 3-[(E)-[3-[(E)-2-[6-(4-Methylpiperazin-1-yl)pyridin-3-yl]ethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_ba60118f3087f2f761dc154ba216f9de.svg) | 4-[(E)-2-[(6E)-6-[(2-Hydroxy-1H-indol-3-yl)methylidene]indazol-3-yl]ethenyl]benzoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_6ea52c61ef801f7365ee86d368781346.svg) | 3-[(E)-[3-[(E)-2-Pyridin-4-ylethenyl]indazol-6-ylidene]methyl]-1H-indole-2,5-diol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_cabd2e6fab372b9aa566eb0762c04990.svg) | 5-Methoxy-3-[(E)-[3-[(E)-2-pyridin-4-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_db21c925503b45a584fcf299a55fa9cf.svg) | 6-Chloro-3-[(E)-indazol-6-ylidenemethyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_1f13695cbfacb1264480451d1e4b5328.svg) | 3-[(E)-[3-[(E)-2-Pyridin-2-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_2b01fb11161878303fd35002d1a23b0f.svg) | 5-Chloro-3-[(E)-[3-[(E)-2-pyridin-4-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_5ab0095e232a80a23d7ad618654dcd30.svg) | 5-Methoxy-3-[(E)-[3-[(E)-2-pyridin-3-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_beaf9a24caa8dd47b0e72eeaf90ad09a.svg) | N-[2-Hydroxy-3-[(E)-indazol-6-ylidenemethyl]-1H-indol-6-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_2b4941de617b5ec75cb1be94b8902102.svg) | 3-[(E)-[3-[(E)-2-Phenylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_3881735a95965672a06ef2422397651c.svg) | 3-[(E)-Indazol-6-ylidenemethyl]-5-methoxy-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_f22c62ebccbf9cee5a0bfda184a6b639.svg) | 3-[(Z)-Indazol-5-ylidenemethyl]-1H-indol-2-ol | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_51ef8e4efb58dcc659a558eb6b9fe463.svg) | 5-Fluoro-3-[(Z)-indazol-6-ylidenemethyl]-1H-indol-2-ol | IC50 | 24000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_108893c23dc069f2bcfa2f301e8eefe1.svg) | N-[2-Hydroxy-3-[(E)-indazol-6-ylidenemethyl]-1H-indol-5-yl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_cd5aa2d2056f262fbc6243aa522193f1.svg) | 5-Ethyl-3-[(E)-[3-[(E)-2-pyridin-3-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_183eb5019a067b9f2e5855771d0b4450.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[4-(2-phenylmethoxyethyl)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_f4c8c14c2cecc1ac7506f9a3813e3b5f.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[2-fluoro-6-(3-hydroxyphenoxy)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_07fffdab16bf0b1c794aca31a2a18716.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[2-fluoro-6-(3-phenylmethoxyphenoxy)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 29500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_7f69691ef511378e1ee395481a0e78b0.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[4-(2-hydroxyethyl)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 960.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_5a6b146d753b9b31e92e18fa3daeb6f5.svg) | 4-[[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-(3-hydroxypropyl)benzenesulfonamide | IC50 | 165.3 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_759210e1410c76ade15fdbb39976692a.svg) | 4-[[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-methylbenzenesulfonamide | IC50 | 38.52 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_d7709963f640ef34e0031750dcff77bb.svg) | N-Cyclopentyl-4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]benzenesulfonamide | IC50 | 742.8 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_db6f62e6b87ffbe2467e45606cc0190d.svg) | N-Butyl-4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]benzenesulfonamide | IC50 | 245.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_be56a12187aa1116027c47e09fd6a323.svg) | 4-[[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-phenylbenzenesulfonamide | IC50 | 2403.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_73549a364dbc499fa734245c874f864e.svg) | 4-[[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]amino]-N-(2-hydroxyethyl)benzenesulfonamide | IC50 | 482.8 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_8947f23dd35aea4e08ba77c29086bf2b.svg) | 1-[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]-N-propan-2-ylindole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_a1959661e8b90a4d8199016c57af2739.svg) | 1-[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]indole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_dccfbcdd95191a834308abe84abd3e84.svg) | 1-[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]-N-(2-methylpropyl)indole-5-carboxamide | IC50 | 2789.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_73bcfccfde16fb90103034edbc08ea3c.svg) | 1-[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]-N-(2-methylpropyl)indole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_3897483b548b77284f9b51a28bccaea4.svg) | 1-[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]-N-ethylindole-5-carboxamide | IC50 | 4442.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_02d5af84dd7ae560bbebbafce149c1d5.svg) | 1-[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]-N-propan-2-ylindole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_60dd05ff4b13495a011dcb9e7c666348.svg) | 4-[[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]amino]-N-methylbenzenesulfonamide | IC50 | 1263.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_9385be292eaf7965e5dd629e7a38e326.svg) | (7R)-8-Cyclopentyl-7-ethyl-2-(5-fluoroindol-1-yl)-5-methyl-7H-pteridin-6-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_374edae18d57097f9bf30cddf554d578.svg) | N-Ethyl-1-[7-ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]indole-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_1bec560b50b56a5b5f0b1a0c951c3320.svg) | 7-Ethyl-2-(5-fluoroindol-1-yl)-5-methyl-8-(1-methylpyrazol-3-yl)-7H-pteridin-6-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_85eb96806551d135bf70a36289549bd4.svg) | 4-[[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]amino]-N-propylbenzenesulfonamide | IC50 | 1550.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_6682f6f2efe05b1916d61d178b1dc246.svg) | 4-[[7-Ethyl-5-methyl-8-(1-methylpyrazol-3-yl)-6-oxo-7H-pteridin-2-yl]amino]-N-(2-methylpropyl)benzenesulfonamide | IC50 | 1902.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk3_3c61c24e917d88dbb75257f38a040632.svg) | 4-[[(7R)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]benzenesulfonamide | IC50 | 80.72 [1] |