![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_44b484a9c1048f0607f62988f78cc00d.svg) | BI-2536 | IC50 | 0.83 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_44b484a9c1048f0607f62988f78cc00d.svg) | BI-2536 | Ki | 0.22 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_693b4dc5e5c2d34bce7645a52c5c3915.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-(8-phenyloctyl)imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 540.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_cb1e7ba59f998cc2b27041e168f413c4.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 300.0 [1], 16000.0 [2], 21500.0 [3], 300000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_ac9222422aa3967de001af41e8ffd43b.svg) | Wortmannin | IC50 | 5.8 [1], 24.0 [2], 1300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_925efe76edccc6dd4a09761b08a84cbb.svg) | Volasertib | IC50 | 0.87 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_2cdfd9e169f1049c63f9dafb36e00e41.svg) | Gsk-461364 | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_2cdfd9e169f1049c63f9dafb36e00e41.svg) | Gsk-461364 | Ki | 2.2 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_0f91699454b38a2b6da01a1d4e67d200.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-(2-fluoro-6-phenoxyphenyl)octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 6.6 [1], 66.0 [2], 127.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_f1366eff0c7fe9a3f64ff9c8af68c3bc.svg) | 1-Methyl-8-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 1.0 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_a7dbdd6952b28399f700d51a83f5e290.svg) | 1-Methyl-8-(2-methylanilino)-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 14.0 [1], 15.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_65b74ed48997f7677666c5a59a3766b5.svg) | 4-[2-(2-Hydroxyethoxy)-5-methyl-3-[4-(2H-tetrazol-5-yl)phenyl]phenyl]benzonitrile | IC50 | 139000.0 [1], 146000.0 [2], 151000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_2016e1fb48c552930d228a3e7f6e1433.svg) | Quercetin | IC50 | 5750.0 [1], 64000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_6603a475932cb1632b1b43c2f664a423.svg) | 2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one | IC50 | 2000.0 [1], 2100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e931253b26ac7f440c5f2cf0a5e84a1b.svg) | 4-[[(7S)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | IC50 | 32.5 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e931253b26ac7f440c5f2cf0a5e84a1b.svg) | 4-[[(7S)-8-Cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | Ki | 0.42 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_6eb85432df5d02aab0b18480749b4c05.svg) | 5-(5,6-Dimethoxy-1-benzimidazolyl)-3-[[2-(trifluoromethyl)phenyl]methoxy]-2-thiophenecarboxamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_6a827a1fd20a9764f3e9c5aa0ddebdfc.svg) | 5-Cyano-7-nitro-3-oxido-1,3-benzothiazol-3-ium-2-carboxamide | IC50 | 8000.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_9ac8c17a1cd78f944fc3ce79f16d4238.svg) | Nms-P937 (nms1286937) | IC50 | 2.0 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_b800922b5c769ca9c52161d0b5a33c4a.svg) | 8-[2-Methoxy-5-(4-methylpiperazin-1-yl)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 7.0 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_93fd355a308bbc6a4f2d55c507cc6f63.svg) | 3-[(2-Chlorophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_ae3cb292e66be9578004d2faaf9b275f.svg) | 8-Anilino-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 68.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_b60dbd9c454c8110a1338f2041b0efa3.svg) | 8-Anilino-N,1-dimethyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 4215.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_d0ac7695956546de9fc51c4ae190e5c8.svg) | 4-[4-(4-Methyl-2-methylamino-thiazol-5-YL)-pyrimidin-2-ylamino]-phenol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_ed62fcea38ea17aad2067edf2e0c925a.svg) | 4-[4-(2,4-Dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]phenol | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_4ad63faa434e4c83e8471e6a3dd1e232.svg) | 5-(1H-Benzimidazol-1-yl)-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamide | IC50 | 15.0 [1], 35.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_d0137bac43a6d197f7c91ff243b89163.svg) | 3-[[(2R)-3,3-Dimethylbutan-2-yl]amino]-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione | Ki | 2000.0 [1], 2200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e65399444f3639d55c4b15703501c828.svg) | 8-Anilino-1-methyl-N-phenyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_c087b1a38a24d81507e65bff41ef7823.svg) | Cyclapolin 9 | IC50 | 500.0 [1], 2400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_af4ffbf4dbfd01d2f1479cc420b05ad5.svg) | 3-[(E)-[3-[(E)-2-Pyridin-4-ylethenyl]indazol-6-ylidene]methyl]-1H-indol-2-ol | IC50 | 10000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_4423acfde4406ac0c29b030c2f0a51ff.svg) | 2-(3-Hydroxy-4-methoxyanilino)-5,7-dihydropyrimido[5,4-d][1]benzazepin-6-one | IC50 | 5700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_dffd7e10345b8ce4e536a28bb698106f.svg) | 3-Methyl-1-phenyl-N-[(1S)-1-phenylethyl]pyrazolo[4,3-c]pyridin-6-amine | IC50 | 1301.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_149de0ffa90c27f5589ee0ec12e15539.svg) | 1-(3-Chlorophenyl)-3-methyl-N-[(1S)-1-phenylethyl]pyrazolo[4,3-c]pyridin-6-amine | IC50 | 121.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_56c88a2236cbc6026fc3690ac7724f39.svg) | 5-(5,6-Dimethoxy-1H-benzimidazol-1-yl)-3-[[4-(methylsulfonyl)phenyl]methoxy]-2-thiophenecarboxamide | IC50 | 75.0 [1], 125.89 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_c11a11088c789cedc2c8db1dba421dc5.svg) | (2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-3-phosphonooxybutanoic acid | IC50 | 5270.0 [1], 32030.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_3d1aadff81b1eaa89d51e0ddb6f70b40.svg) | 8-(2-Methoxyanilino)-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_f622aa4e29ed2191958d7259f200be05.svg) | 8-[5-Amino-2-(trifluoromethoxy)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 60.0 [1], 87.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_593760634b5e73daf93d1b0d76afa02a.svg) | 1-Methyl-8-[5-[2-(1-methylpyrrolidin-2-yl)ethylamino]-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 123.0 [1], 149.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_241ed90fbf6182a4fbaa5becdb0166c4.svg) | 1-Methyl-8-(2-(trifluoromethoxy)phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 117.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_bd79e73489eebe20ef4206ce4afadd76.svg) | N-[(2,6-Dibromo-4-sulfamoylphenyl)carbamothioyl]benzamide | IC50 | 39800.0 [1], 95000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_3a9bf695c67492067b30acdbb19606bc.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[6-[(E)-benzylideneamino]oxyhexyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 558.0 [1], 5050.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_3524620b0e3d9e6e4db1baf3e5315ae3.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[6-[(Z)-(2-fluoro-6-phenoxyphenyl)methylideneamino]oxyhexyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 91.0 [1], 670.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_59ec338fc45c4d08f8c2e9f3f54b2289.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[5-[(E)-(2-fluoro-6-phenoxyphenyl)methylideneamino]oxypentyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 163.0 [1], 1550.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_64175f83bd86563ea5053f97a0522fe2.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[5-[(E)-benzylideneamino]oxypentyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 2380.0 [1], 9000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_183eb5019a067b9f2e5855771d0b4450.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[4-(2-phenylmethoxyethyl)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 9.7 [1], 152.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_f4c8c14c2cecc1ac7506f9a3813e3b5f.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[2-fluoro-6-(3-hydroxyphenoxy)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 5.5 [1], 188.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_07fffdab16bf0b1c794aca31a2a18716.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[2-fluoro-6-(3-phenylmethoxyphenoxy)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 11.2 [1], 862.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_7f69691ef511378e1ee395481a0e78b0.svg) | [(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-[3-[8-[4-(2-hydroxyethyl)phenyl]octyl]imidazol-4-yl]propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] dihydrogen phosphate | IC50 | 5.5 [1], 218.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_bf02fb83e982262374183313aa684e6e.svg) | [(1R)-1-[(9S,12S,15S)-15-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-12-(hydroxymethyl)-8,11,14-trioxo-18-(8-phenyloctyl)-7,10,13,18-tetraza-1-azoniabicyclo[15.2.1]icosa-1(19),17(20)-dien-9-yl]ethyl] dihydrogen phosphate | IC50 | 6.0 [1], 45.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_44c7f56b2b3308b90bc7cc28a2dc99e9.svg) | [(1R)-1-[(10S,13S,16S)-16-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-13-(hydroxymethyl)-9,12,15-trioxo-19-(8-phenyloctyl)-8,11,14,19-tetraza-1-azoniabicyclo[16.2.1]henicosa-1(20),18(21)-dien-10-yl]ethyl] dihydrogen phosphate | IC50 | 5.0 [1], 44.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_529a66f2e31278729b377d54299ae27a.svg) | [(1R)-1-[(8S,11S,14S)-14-[[(2S)-2-[[(2S)-1-Acetylpyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-11-(hydroxymethyl)-7,10,13-trioxo-17-(8-phenyloctyl)-6,9,12,17-tetraza-1-azoniabicyclo[14.2.1]nonadeca-1(18),16(19)-dien-8-yl]ethyl] dihydrogen phosphate | IC50 | 10.0 [1], 160.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_8be3ed872252bd010950ea0bc6bff5b8.svg) | [(1R)-1-[(9S,12S,15S)-15-Acetamido-12-(hydroxymethyl)-8,11,14-trioxo-18-(8-phenyloctyl)-7,10,13,18-tetraza-1-azoniabicyclo[15.2.1]icosa-1(19),17(20)-dien-9-yl]ethyl] dihydrogen phosphate | IC50 | 8.0 [1], 370.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_4d5733618730e70b232fa59cf550b6a0.svg) | 1-Methyl-8-[5-piperazin-1-yl-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_0ba65440b4be10bfa799b3c7b15bc9ee.svg) | 1-Methyl-8-[5-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 3.0 [1], 8.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_9b83e5b61ec3aa8796d919c574da220d.svg) | 1-Ethenyl-8-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 1.0 [1], 6.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_eda6ee59da92f3301e3017c93c279489.svg) | 1-(2-Fluoroethyl)-8-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 4.0 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_857ca3eb165bb184fe2ffdd3430b51e5.svg) | 1-(2-Chloroethyl)-8-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 7.0 [1], 13.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e2f99194617c96946324b426e112d809.svg) | Erlotinib | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_7b158b23bff97dd8343875cddc90f377.svg) | Sorafenib tosylate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_755000a88f2651809d912de0f446bcfe.svg) | Lapatinib | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_9b0846c6235f0aecda0470a6e161c35a.svg) | Ellagic acid | IC50 | 3340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_77af51390c508a620cda34b086ecd521.svg) | Morin | IC50 | 12600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_2cd9f08f5dea65516c41f9c3534be4cf.svg) | Thymoquinone | IC50 | 2180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e1bd3c1d60717a09fae0532edc016b5c.svg) | Axitinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_8edb893ba88c5700603edef201da4265.svg) | Nintedanib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_4fc4352b32d3da424f7de0a0fd6aa1e3.svg) | N-[4-[[6-Methoxy-7-[3-(4-morpholinyl)propoxy]-4-quinazolinyl]amino]phenyl]benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_68d239a89e61fef8a6572bb5c797ceaf.svg) | Reversine | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_f888f082cfdd181caa483bbe675439bc.svg) | Kenpaullone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_a257c791d1de1df5d4a1fa04612f9c76.svg) | Nvp-aew541 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_aea8e5cd5eedd851a20871e2fe5ff0da.svg) | Danusertib | IC50 | 3500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_cae93b345c0c1f11079edb76060ab346.svg) | Scytonemin | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_b345e1750a38bf95a72d038f7bf6d9ff.svg) | 5-Iodo-3-[(3,5-dibromo-4-hydroxyphenyl)methylene]-2-indolinone | IC50 | 4600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_ab85d24569e928a06874243ca8643053.svg) | Rigosertib | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_def2622457c2392ae7d83708b0039226.svg) | 4-[[9-Chloro-7-(2,6-difluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid | IC50 | 53000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_2adbc4a307d22bed17e0f710542542e9.svg) | Entrectinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_eb1729f98bdd8714dc7d292bc1ad0548.svg) | Cfms Receptor Tyrosine Kinase Inhibitor | IC50 | 24000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e7ecb06887875f4d78baf892d82c33a5.svg) | Bms-777607 | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_bd1c4c226d09bccaf8e1c9ed8e2ba78a.svg) | Azd-1152hqpa | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_8fc6ee09adb3fcc99c67a2a384c17924.svg) | 2-(Pyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one | IC50 | 980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_c74a1b9d6feb1def6b7e3f6834b5761b.svg) | Tak-285 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_495c00c0eebcec0612a883578e83da0a.svg) | Milciclib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_a2d32a1f7c79660a88d646bbda5ee232.svg) | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_3ac91c26cb3202821ba09ba5b9d46a48.svg) | Aminofurazanyl-azabenzimidazole 6n | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_c03f7d5f41fab476c99fd46f75d44073.svg) | Pha-793887 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_84fae1800055ebf670b925911d10e379.svg) | CFI-400945 (free base) | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_f2b267f547ea2e28f9989796b704ab4e.svg) | TCS JNK 5a | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_e0e66b7329f74ac9e778459370265f14.svg) | Norlichexanthone | IC50 | 75700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_96dd1c245db8fda5ee6b165b0c628ae0.svg) | CID 44556162 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_681512d30c057666e306c60d1de4f37b.svg) | N6-Cyclohexyl-N2-(2-methyl-4-morpholinophenyl)-9H-purine-2,6-diamine | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_70c3cfa7f2d0b69602d9a215cff33e29.svg) | CID 53357478 | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_dc59b8d69935f3897f9e4732572cf184.svg) | Poloxin | IC50 | 29400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 8900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_8234c79ad4f66a353350852beb5c645b.svg) | IKK-3 Inhibitor | IC50 | 794.33 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_d44bb541aaceb7d87194194110f1e1e1.svg) | CID 11634725 | Ki | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_81467d3dc0c7e26df63f1e5159d5ad46.svg) | CID 25015677 | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-plk1_ac9e30b723e2c9bf1debc2a45966acbb.svg) | 3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)pyrrole-2,5-dione | IC50 | 100000.0 [1] |