![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_6447577ef3aac74ffd5250fc02a69745.svg) | 4-[5-(1-Methylpiperidin-4-yl)oxybenzimidazol-1-yl]-2-[1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 230.0 [1], 570.0 [2], 910.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e505f05d4ff05f9e4a3028c686fa03a4.svg) | CID 49837564 | IC50 | 200.0 [1], 230.0 [2], 300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_9140e9101b9da500b4a936aa6720a331.svg) | 4-[3-Amino-6-(3,4,5-Trimethoxyphenyl)pyrazin-2-Yl]-2-Methoxybenzoic Acid | IC50 | 1300.0 [1], 2400.0 [2], 2500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_69b1407966a0b318a5a64756c567c0dc.svg) | 4-[3-Amino-6-(3,4,5-Trimethoxyphenyl)pyrazin-2-Yl]-2-Methylbenzoic Acid | IC50 | 1200.0 [1], 2300.0 [2], 2600.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_6a0a67080c3a5b1176390eee954b50b2.svg) | 4-[3-Amino-6-(3,4,5-Trimethoxyphenyl)pyrazin-2-Yl]benzoic Acid | IC50 | 710.0 [1], 1600.0 [2], 2300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_58b7cf1945ecdf9d6b0a8b49081ca1ba.svg) | 1-[3-Amino-6-(3,4,5-Trimethoxyphenyl)pyrazin-2-Yl]piperidine-4-Carboxylic Acid | IC50 | 410.0 [1], 870.0 [2], 940.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_7d457696cdd5d7df0bc22dcf3f33ba07.svg) | 1-[3-Amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]piperidine-4-carboxylic acid | IC50 | 720.0 [1], 1900.0 [2], 2100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_dda5b9608f3befcd50c2ed6a42585f02.svg) | 5-[6-(1-Methylpiperidin-4-yl)oxybenzimidazol-1-yl]-3-[1-[2-(trifluoromethyl)phenyl]ethoxy]thiophene-2-carboxamide | IC50 | 50.0 [1], 160.0 [2], 200.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_ff17b6f8c0d6e75a664fb18c2f79a1b9.svg) | 5-[6-(1-Methylpiperidin-4-yl)oxybenzimidazol-1-yl]-3-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]thiophene-2-carboxamide | IC50 | 25.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e5d5b888a75654a370c358b20f01e1e0.svg) | N-[(3Z)-3-[(2-Ethyl-5-methyl-1H-imidazol-4-yl)methylidene]-2-oxo-1H-indol-5-yl]prop-2-ynamide | IC50 | 770.0 [1], 1300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_0e1affdc51b1b7e26b10be1d860fb0d0.svg) | CID 16662746 | IC50 | 6.0 [1], 14000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_21eb54a8f38a4391a67c59038a9939e0.svg) | N-[(3Z)-2-Oxo-3-(1H-pyrrol-2-ylmethylidene)-1H-indol-5-yl]prop-2-ynamide | IC50 | 920.0 [1], 20000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_2016e1fb48c552930d228a3e7f6e1433.svg) | Quercetin | IC50 | 5730.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 4790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_4242da2ee2a3321b0efd00f1d63fdcf7.svg) | Neratinib | IC50 | 274.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_cf6bd891f5d6eaff35c3d4ff27fd3db0.svg) | Pelitinib | IC50 | 661.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_34d56ed9b81c1d4adb6e33de1f3909ba.svg) | 5-[(Z)-(5-Chloro-2-oxo-1H-indol-3-ylidene)methyl]-N-[2-(diethylamino)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e0e66b7329f74ac9e778459370265f14.svg) | Norlichexanthone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_ac9e30b723e2c9bf1debc2a45966acbb.svg) | 3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)pyrrole-2,5-dione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5a8e321781069aee089dcc439066b321.svg) | 2,3,6,8-Tetrahydroxy-1-methylxanthone | IC50 | 83900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5803643fba2a49f1581ea6790292d883.svg) | Epicoccolide B | IC50 | 3780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_d72e6a5f6bda112109d526c400d3a392.svg) | Astrogorgiadiol B | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e24a6ef90b6dda81406d577957bafbf2.svg) | (1S,9R)-5,6,12,13,14-Pentahydroxy-4,11-dimethyl-16-oxo-8,17-dioxatetracyclo[7.7.1.02,7.010,15]heptadeca-2(7),3,5,10,12,14-hexaene-3-carbaldehyde | IC50 | 1830.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_8547ec1c061a6923170866cf54d1c0d4.svg) | (1R,3As,4S,5R,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(2R)-6-methyl-5-methylideneheptan-2-yl]-1,2,3,3a,4,5,6,7-octahydroinden-5-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_9f0649c0af7300504c89d15a04caf360.svg) | Calicoferol B | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_127674c15dddfb61d8f9a13c7daa5925.svg) | GSK 461364 analogue I | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 9242.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_89f93b41ac7e8a2307bd8fc1d9fad8a4.svg) | Calicoferol E | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_a5c5bae0fd3ddf532506780bb4f7f125.svg) | Khk-IN-1 | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_0731e513dda8b4631f904dc8f0082e8c.svg) | 7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_1fe60e6d13674f8cf1dfc82fac3410b2.svg) | 7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_029f5b4cad89a2c59efa869fd9853874.svg) | N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_c2aa7e0fb640ea7529d7330460976868.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_98598461b658b3f77425e67c797f8e2d.svg) | N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_a3bd9a5a28d4f4d2890ccf5cdf08d883.svg) | N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_cde4e83180955e4849d8daba0837480d.svg) | N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamide | Ki | 9200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_7f4f13e5a533e76aa2b0be165fbe10d5.svg) | 3-(6-Methoxy-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyridine | IC50 | 3220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 268.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_b076cdaba7bb8b7d9a4e8120c86a34a8.svg) | N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_b80728998e0b173ed97842a79c1db051.svg) | 5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_d177c352a8a90316beccdf76166341e8.svg) | N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamide | IC50 | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 1830.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_eda1570f6e608eea37da447234534ac5.svg) | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_ac2ac44cc6c324cb845a2c77f9c11dd1.svg) | CID 71553154 | IC50 | 2510.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_ef431bf27ff7842bbb4caafd947b43c7.svg) | Tilfrinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_70b0d2cbc054446af80b12d3d42fd894.svg) | (8S,16S)-3,16-Dihydroxy-9,10-seco-1,3,5(10)-cholestatrien-9-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_c67b754da3023ab057380dedf2f5a397.svg) | Calicoferol A | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_3ba3cfff437203d3cd5cef3fe6f6283a.svg) | (1R,3As,4S,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(2R)-6-methyl-5-methylideneheptan-2-yl]-2,3,3a,4,6,7-hexahydro-1H-inden-5-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_0b37fcadf8f90dc3bf2f29ca0be2a519.svg) | Methyl 3-[[(1R,2S,4aR,8aS)-1,2,4a,5-tetramethyl-2,3,4,7,8,8a-hexahydronaphthalen-1-yl]methyl]-4,5-dihydroxybenzoate | IC50 | 14700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5b63ea15265b993819abd00ed6f2eee3.svg) | 2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5f823a33091057f5669d4eae1712e421.svg) | 4-[4-[3-[4-[(Propan-2-ylamino)methyl]anilino]-1H-pyrazol-5-yl]phenyl]benzene-1,3-diol | IC50 | 1040.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_0b43927816ebbc9be13e6e44e4f9f2e1.svg) | 5,5-Dimethyl-8-[[4-(2,2,2-trifluoroethylamino)furo[3,2-d]pyrimidin-2-yl]amino]-1H-4,1-benzoxazepin-2-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_eff8c0d79e17da61a4fc7f0961e63b5a.svg) | 4-[7-(1-Methylpiperidin-4-yl)oxyimidazo[1,2-a]pyridin-3-yl]-2-phenylmethoxybenzamide | IC50 | 808.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_472aca21221bca1c9b7c6b79f7fcf834.svg) | 4-[7-(4-Methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 2170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_da4002a4fb834455f7d91a06490ab4ce.svg) | 4-[7-(1-Methylpiperidin-4-yl)oxyimidazo[1,2-a]pyridin-3-yl]-2-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 591.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e93ac71a84d3e96fd4ecd266167cc03c.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[(3-fluorophenyl)methoxy]benzamide | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_6c1041b67565ff1f5edfcede95eded80.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-phenylmethoxybenzamide | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_22f01ab442021d510cadc152aa7d6b88.svg) | 4-[7-(4-Methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-phenylmethoxybenzamide | IC50 | 3210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_f56d3ff4c6290e3b16e428ee05b7050f.svg) | N-Methyl-4-[7-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 197000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_16d6d8c70abf4e85b65d94d78459518d.svg) | N-Hydroxy-4-[7-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e936ed8070d64824e3ee820df0783687.svg) | Tert-butyl 4-[3-[4-carbamoyl-3-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]phenyl]imidazo[1,2-a]pyridin-7-yl]oxypiperidine-1-carboxylate | IC50 | 11190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_8e4dd364b05ba69379527f40dba302a9.svg) | 4-(7-Piperidin-4-yloxyimidazo[1,2-a]pyridin-3-yl)-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide;2,2,2-trifluoroacetic acid | IC50 | 10030.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_875ff0c43a663b8d0169c73dee9bfcc8.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[(2-fluorophenyl)methoxy]benzamide | IC50 | 87.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_711f5c48271ce2de73e0bfcf5bf32c8b.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[[3-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_30d2c46029ed77347ee4d60e1187c4ca.svg) | 4-[7-(4-Methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[[2-(trifluoromethyl)phenyl]methoxy]benzoic acid | IC50 | 10030.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_76fe14c972df58a415d828d8d299bda6.svg) | 4-[7-(1-Methylpiperidin-4-yl)oxyimidazo[1,2-a]pyridin-3-yl]-2-[1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_192fba6004f87b3b2f87516fecf1e451.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 927.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_4c29a0250283c52b9e7da512a30cae18.svg) | 4-[7-(4-Methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 1190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_15a0160db92c0549ed84e0c7ad02290a.svg) | 4-[7-(4-Methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_548ab02de1cdc31675788f9790e521dc.svg) | Tert-butyl 4-[3-[4-carbamoyl-3-[[2-(trifluoromethyl)phenyl]methoxy]phenyl]imidazo[1,2-a]pyridin-7-yl]oxypiperidine-1-carboxylate | IC50 | 1037.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_c009120ca19478ba69924ce16dc2791c.svg) | 5-(1,3-Benzodioxol-5-yl)-7-[[(2R)-1-ethenylsulfonylpyrrolidin-2-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e894b608b0d86710a2be55c2b086fd6e.svg) | Methyl 4-[7-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[1-[2-(trifluoromethyl)phenyl]ethoxy]benzoate | IC50 | 42600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_1838d7c83f25e26557f8ddb2096d727f.svg) | 4-[7-(1-Methylpiperidin-4-yl)oxyimidazo[1,2-a]pyridin-3-yl]-2-[(1S)-1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5db0b0e91319e7417f0ed1e271a4a041.svg) | 4-(7-Chloroimidazo[1,2-a]pyridin-3-yl)-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_f820b9e8df702b49c8cae4e33d393e22.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[[4-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 386.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_52d7bbf132fb906db057cf1aa2e33757.svg) | N-(2-Aminoethyl)-4-[7-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_e909b8ea54b08177d2aa10445b919789.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 478.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_82ac1c613d5d19fec993db14d9973be7.svg) | 4-[7-(1-Methylpiperidin-4-yl)oxyimidazo[1,2-a]pyridin-3-yl]-2-[[2-(trifluoromethyl)phenyl]methoxy]benzamide | IC50 | 838.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_4602c8c7b43a2a15f69235c600a7e988.svg) | 2-Methoxy-4-[7-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyridin-3-yl]benzamide | IC50 | 19280.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_be3215402906f80de76893d9c9f28399.svg) | 2-[Ethyl-[[5-[[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino]-1,2-thiazol-3-yl]methyl]amino]ethanol | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_984f1d19dd4f7aff4c8096322cf2c2cd.svg) | 4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_09c777664a74d957394c48618430a40f.svg) | 2-(5-Methoxy-3-oxo-1H-isoindol-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide | IC50 | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_2db2a2d148038bcb7681f06d72b80a8e.svg) | N-[6-Methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-3-(pyridin-2-ylmethyl)-1,2-thiazol-5-amine | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_2b875aca7518d1f789a36583c912a0dd.svg) | 4-[3-Amino-6-(3,4,5-Trimethoxyphenyl)pyrazin-2-Yl]-2-Ethoxybenzoic Acid | IC50 | 16900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_5a7d5cf759b396d4e294ad392b59b37b.svg) | 1-[3-Amino-6-(3-Methoxyphenyl)pyrazin-2-Yl]piperidine-4-Carboxylic Acid | IC50 | 4200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_9d981d8ccb5ff890f413fec4659b3d7b.svg) | 1-(3-Amino-6-(3,4-dimethoxyphenyl)pyrazin-2-yl)piperidine-4-carboxylic acid | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_048278bf7021ea034affc0c7ab54d9cf.svg) | 1-(3-Amino-6-(3,5-dimethoxyphenyl)pyrazin-2-yl)piperidine-4-carboxylic acid | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_896d6d5039dde38cd5187b699e626dde.svg) | 1-(3-Amino-6-(4-methoxyphenyl)pyrazin-2-yl)piperidine-4-carboxylic acid | IC50 | 19800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_3dca04b6d083df85b1e46d1de3fb5e59.svg) | 1-(3-Amino-6-phenylpyrazin-2-yl)piperidine-4-carboxylic acid | IC50 | 7800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_26ce8919ccb44028427692a63abf9afe.svg) | 1-(3-Aminopyrazin-2-yl)piperidine-4-carboxylic acid | IC50 | 48500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-nek2_1f187d85418abf63f0784babde6382e9.svg) | 3-(Piperidin-1-yl)-5-(3,4,5-trimethoxyphenyl)pyrazin-2-amine | IC50 | 50000.0 [1] |