![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_2adbc4a307d22bed17e0f710542542e9.svg) | Entrectinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_9ac8c17a1cd78f944fc3ce79f16d4238.svg) | Nms-P937 (nms1286937) | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_ccd2c2ad74c22d5f6bde002b0c36d90e.svg) | 3-[4-(Morpholin-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 178.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_c33668b892afbb36d843e9dd0815b38f.svg) | 5-[2,4-Dihydroxy-6-(4-Nitrophenoxy)phenyl]-N-(1-Methylpiperidin-4-Yl)-1,2-Oxazole-3-Carboxamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_e7b7aadcdbe86ffb6055de4dc7c032a9.svg) | 5-(2-Aminopyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_ddd0fed9eb76e60e618c88402814404d.svg) | 2-[1-(4,4-Difluorocyclohexyl)-piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_2e8153acbaf4777559825f69210e1632.svg) | (7S)-2-(2-Aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_a5c5bae0fd3ddf532506780bb4f7f125.svg) | Khk-IN-1 | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_1e3ff778dd8b5ed89f456cd8d80834b6.svg) | 8-[(5-Amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_94e490915983085a98fddac87c39e7c3.svg) | 3-[(4-Morpholin-4-ylbenzoyl)amino]-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-thieno[3,2-c]pyrazole-5-carboxamide | IC50 | 412.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_eda1570f6e608eea37da447234534ac5.svg) | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 2220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_ac2ac44cc6c324cb845a2c77f9c11dd1.svg) | CID 71553154 | IC50 | 3840.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_ef431bf27ff7842bbb4caafd947b43c7.svg) | Tilfrinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_c89106c4a521532cda4c2bf5f9e882d3.svg) | 3-[[5-(1,3-Benzodioxol-5-yl)-[1,2,4]triazolo[1,5-c]quinazolin-8-yl]amino]propan-1-ol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_6751581577889e826fac050483c91970.svg) | 3-[4-[(2S)-2-(5-Methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 12095.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_26075b443bb235883f0fdbdcdc04cf50.svg) | 3-[4-(2,3,3a,4,6,6a-Hexahydrofuro[2,3-c]pyrrol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 10218.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_5f823a33091057f5669d4eae1712e421.svg) | 4-[4-[3-[4-[(Propan-2-ylamino)methyl]anilino]-1H-pyrazol-5-yl]phenyl]benzene-1,3-diol | IC50 | 1850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_1a299af4bf962c94a0e6439304c79b11.svg) | 5-[2-[4-(Dimethylamino)phenoxy]-4,6-dihydroxyphenyl]-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_a346f0c47c7f17cb53ca8e14347d4afa.svg) | 5-[2,4-Dihydroxy-6-[4-(propan-2-ylamino)phenoxy]phenyl]-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_6b43be1bed4bce2576e9e27a49ba5b81.svg) | 5-[2-[4-(Dimethylamino)phenoxy]-4,6-dihydroxyphenyl]-N-[1-(1,4-dioxaspiro[4.5]decan-8-yl)piperidin-4-yl]-1,2-oxazole-3-carboxamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_f43a289da9112d38ebaad50830605e47.svg) | 3,4-Dimethoxy-N-[3-(1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_8b6143ca04eb73cae880f8fa5f030280.svg) | 1-Methyl-2-[2-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]pyrimidin-4-yl]-6,7-dihydro-5H-pyrrolo[3,2-c]pyridin-4-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_3364ae456a84baff14078fdd57a6c673.svg) | 8-[(1-Acetylpiperidin-4-yl)amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_1253d90949f713eb03ad4d975a1fe238.svg) | 8-[(1-Benzoylpiperidin-4-yl)amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_8fd11039df3af8d857812e088012b95c.svg) | N,1-Dimethyl-8-[[1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-4-yl]amino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_6958152d8bd43f8d3de6beb98828a696.svg) | 2-{[2-Amino-5-(1,3-Benzodioxol-5-Ylmethyl)[1,2,4]triazolo[1,5-C]quinazolin-8-Yl]amino}ethanol | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_e0d5e7d8eee71e3a48cf4604210ca68e.svg) | 5-(1,3-Benzodioxol-5-ylmethyl)-[1,2,4]triazolo[1,5-c]quinazoline-2,8-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_50613ae2c7e7029d2dd4f7f991fae5e8.svg) | 5-(1,3-Benzodioxol-5-Ylmethyl)-10-Fluoro[1,2,4]triazolo[1,5-C]quinazolin-2-Amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_4fb25ecc940b9008100bb9548035dc2d.svg) | 5-(1,3-Benzodioxol-5-ylmethyl)-10-fluoro-8-(4-methylpiperazin-1-yl)-[1,2,4]triazolo[1,5-c]quinazolin-2-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_cb9251a0cfa16e102ce80133db5b82ef.svg) | 1-Methyl-5-[2-[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)anilino]pyrimidin-4-yl]pyrrole-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_264a7157e80f6120303d9f2e2d1c561f.svg) | 8-N-(Cyclopropylmethyl)-4-N-(2-methylsulfanylphenyl)-2-(4-piperidin-4-ylpiperazin-1-yl)pyrimido[5,4-d]pyrimidine-4,8-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_df2324f8c5c5af7d9efc7d738c460583.svg) | 2-[(4S)-7-(3-Chlorophenyl)-1-oxo-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-4-yl]-N-[(1S)-1-cyclohexyl-2-(4-methylpiperazin-1-yl)ethyl]acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_9775cdc9295a6f017c0e1ac0bcd40110.svg) | 2-(3,5-Dichloroanilino)-4-[[4-(dimethylamino)cyclohexyl]amino]-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_404ac985301936f567b8910c5b197396.svg) | 2-(3,5-Dichloroanilino)-4-[[(3R,4S)-4-hydroxyoxolan-3-yl]amino]-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_2b89b02ab43026c450cc4bc42e45268a.svg) | 3-{4-[(2S)-2-Methylmorpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | IC50 | 1099.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_2378e7beb901196da5e7ccf72b025a22.svg) | 3-[4-[2-(3-Methyl-1,2,4-oxadiazol-5-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 32000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_5513037833988b135e272a5562958f35.svg) | 4-[5-(3-Cyanophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine-2-carbonitrile | IC50 | 6208.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_b23dd9eac2da186da843d3ca4dd44790.svg) | N-(2,2-Dimethylpropyl)-2-(1-oxo-7-thiophen-3-yl-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-4-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst4_da42255b90b040406351a987cb379fdc.svg) | 3-[4-[(2R)-2-(5-Methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 9430.0 [1] |