![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 0.41 [1], 4.72 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_8aa951d1935df336d561e6b48c9639a1.svg) | Su6656 | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_ccd2c2ad74c22d5f6bde002b0c36d90e.svg) | 3-[4-(Morpholin-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_15a4bcfb2ea319b026c020006e2b004c.svg) | Cep-11981 | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_d019ff4da979aeb51ea88bb93c1f1472.svg) | 5-(4-Chlorophenyl)-N-(4-piperazin-1-ylphenyl)furan-2-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_c2aa7e0fb640ea7529d7330460976868.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamide | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_98598461b658b3f77425e67c797f8e2d.svg) | N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_a3bd9a5a28d4f4d2890ccf5cdf08d883.svg) | N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_cde4e83180955e4849d8daba0837480d.svg) | N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamide | Ki | 8800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_f046ae8812a77e5cb35fd8b53bebf05d.svg) | Ripk1-IN-7 | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_262c5527ba96216e81ae5e081ba9279f.svg) | 3-Methyl-N-[6-methylsulfanyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_420c640ab3d9d5b9acd6e7f999ac08f0.svg) | CID 27666048 | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_b80728998e0b173ed97842a79c1db051.svg) | 5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine | IC50 | 570.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_d177c352a8a90316beccdf76166341e8.svg) | N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamide | IC50 | 650.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_ac2ac44cc6c324cb845a2c77f9c11dd1.svg) | CID 71553154 | IC50 | 470.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_da63de9d92c2d79ff40b1d8ee8ae24af.svg) | 3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-N-(2-hydroxyethyl)-4-methylbenzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_5b63ea15265b993819abd00ed6f2eee3.svg) | 2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_6751581577889e826fac050483c91970.svg) | 3-[4-[(2S)-2-(5-Methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 795.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_26075b443bb235883f0fdbdcdc04cf50.svg) | 3-[4-(2,3,3a,4,6,6a-Hexahydrofuro[2,3-c]pyrrol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 626.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_be3215402906f80de76893d9c9f28399.svg) | 2-[Ethyl-[[5-[[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino]-1,2-thiazol-3-yl]methyl]amino]ethanol | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_09c777664a74d957394c48618430a40f.svg) | 2-(5-Methoxy-3-oxo-1H-isoindol-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_2db2a2d148038bcb7681f06d72b80a8e.svg) | N-[6-Methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-3-(pyridin-2-ylmethyl)-1,2-thiazol-5-amine | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_afb5e7e5a90712192313a68bd86f002b.svg) | 3,4-Difluoro-2-(2-fluoro-4-iodoanilino)-5-[[(4-methylsulfonylphenyl)methylamino]methyl]benzoic acid | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_b0c469f17f10eac9e56951f48a0ce22f.svg) | 5-[[[(2S)-2,4-Diamino-4-oxobutanoyl]amino]methyl]-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzoic acid | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_af41b64ed99eadff0ae3aacb1130e3af.svg) | 3,4-Difluoro-2-(2-fluoro-4-iodoanilino)-5-[(E)-[[5-(hydroxymethyl)furan-2-carbonyl]hydrazinylidene]methyl]benzoic acid | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_3ceb0c09ea2a3dc24429b87ed6e06d57.svg) | 5-[(E)-[[2-(4-Chlorophenyl)sulfonylacetyl]hydrazinylidene]methyl]-3,4-difluoro-2-(2-fluoro-4-iodoanilino)benzoic acid | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_39cd3e38d141db7358e74e4495085145.svg) | Aurora inhibitor 1 | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_079d46552bd9bfffd84d80bdda6c59b9.svg) | 3-[Dideuterio-(3,3-difluoropyrrolidin-1-yl)methyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine;hydrochloride | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_03e0d1a2e88126708ed3a73e7e36755b.svg) | N-[5-[6-(Methylamino)pyrazin-2-yl]-2-oxo-1H-pyridin-3-yl]-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]benzamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_9296ce5228829a70797f4a55b8cdc874.svg) | 2-(4-Chlorophenyl)-8-piperazin-1-yl-5-[(2-pyridin-3-ylphenyl)methyl]-10H-furo[2,3-c][1]benzazepin-4-one | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_a24e3192a9ff50577fd7c3e72a2d7066.svg) | 3-[(3,3-Difluoropyrrolidin-1-yl)methyl]-N-[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]-1,2-thiazol-5-amine;hydrochloride | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_5efd76d03838ecc45636f311fa9c0a92.svg) | SCH-1473759 (hydrochloride) | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_2f905efdbe6d8f0fedfc64e5dcd53382.svg) | (3R)-1-[2-[4-(4-Acetylphenyl)piperazin-1-yl]-2-oxoethyl]-N-(3-chloro-4-hydroxyphenyl)pyrrolidine-3-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_afa8da84f1cb91bdbfe79048ab9b5517.svg) | 3-(Tert-butylamino)-4-[[2-(4-pyridin-4-ylanilino)pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dione | Ki | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_9775cdc9295a6f017c0e1ac0bcd40110.svg) | 2-(3,5-Dichloroanilino)-4-[[4-(dimethylamino)cyclohexyl]amino]-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_404ac985301936f567b8910c5b197396.svg) | 2-(3,5-Dichloroanilino)-4-[[(3R,4S)-4-hydroxyoxolan-3-yl]amino]-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_2b89b02ab43026c450cc4bc42e45268a.svg) | 3-{4-[(2S)-2-Methylmorpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | IC50 | 179.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_2378e7beb901196da5e7ccf72b025a22.svg) | 3-[4-[2-(3-Methyl-1,2,4-oxadiazol-5-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 2388.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_5513037833988b135e272a5562958f35.svg) | 4-[5-(3-Cyanophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine-2-carbonitrile | IC50 | 288.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_b7ca0698bccc77ef1082a2d7bc07bb14.svg) | 3-[4-[2-(1,2-Oxazol-5-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 1333.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_e634ce90d58ac4d15de46af6a54c8583.svg) | 3-[4-[2-(Cyanomethyl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 196.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_da42255b90b040406351a987cb379fdc.svg) | 3-[4-[(2R)-2-(5-Methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | IC50 | 3239.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-mst2_f28e47e67ea642604198866d9f11a2d4.svg) | 1-[4-[2-[5-(4-Chlorophenyl)furan-2-yl]imidazol-1-yl]phenyl]piperazine | IC50 | 30000.0 [1] |