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Serine/threonine-protein kinase ILK-1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(4E)-4-[4-(1,3-Benzothiazol-2-yl)-1,2-dihydropyrazol-3-ylidene]-3-hydroxycyclohexa-2,5-dien-1-oneIC503300.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-methyl-1,3-benzothiazole-5-sulfonamideIC501900.0 [1]
4-(4-Benzothiazol-2-YL-1H-pyrazol-3-YL)phenolIC503400.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-(1H-imidazol-2-ylmethylideneamino)-1H-pyrazol-5-amineIC501000.0 [1]
2-[4-(1,3-Benzothiazol-2-yl)-1H-pyrazol-5-yl]phenolIC504600.0 [1]
4-(1,3-Benzothiazol-2-yl)-1H-pyrazole-3,5-diamineIC50700.0 [1]
4-Benzothiazol-2-YL-2H-pyrazol-3-ylamineIC50300.0 [1]
4-(1,3-Benzothiazol-2-yl)-5-ethyl-1H-pyrazol-3-amineIC50800.0 [1]
4-(1,3-Benzothiazol-2-yl)-5-phenyl-1H-pyrazol-3-amineIC50900.0 [1]
4-(1,3-Benzothiazol-2-yl)-5-cyclopropyl-1H-pyrazol-3-amineIC50600.0 [1]
4-Benzothiazol-2-YL-5-furan-2-YL-2H-pyrazol-3-ylamineIC50100.0 [1]
4-(1,3-Benzothiazol-2-yl)-5-thiophen-2-yl-1H-pyrazol-3-amineIC50900.0 [1]
3-Methyl-4-(benzothiazole-2-yl)-5-amino-1H-pyrazoleIC50300.0 [1]
3-(3-Aminopropyl)-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-5-amineIC5010.0 [1]
4-[5-(Trifluoromethyl)-1,3-benzothiazol-2-yl]-1H-pyrazol-5-amineIC501100.0 [1]
2-(5-Methyl-1H-pyrazol-4-yl)-1,3-benzothiazoleIC50900.0 [1]
2-(1H-Pyrazol-4-yl)benzo[d]thiazoleIC501600.0 [1]
5-Methyl-4-(6-pyrrolidin-1-ylmethyl-benzothiazol-2-YL)-2H-pyrazol-3-ylamineIC50900.0 [1]
5-Cyclopropyl-4-(5-fluoro-6-methoxy-benzothiazol-2-YL)-2H-pyrazol-3-ylamineIC501000.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-3-N-[2-(1H-imidazol-5-yl)ethyl]-1H-pyrazole-3,5-diamineIC50200.0 [1]
4-(6-Methoxy-1,3-benzothiazol-2-yl)-3-piperazin-1-yl-1H-pyrazol-5-amineIC50200.0 [1]
4-[[5-Amino-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]butanoic acidIC504300.0 [1]
3-[[5-Amino-4-(5-fluoro-6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]propan-1-olIC50500.0 [1]
4-(6-Methoxy-1,3-benzothiazol-2-yl)-5-methyl-1H-pyrazol-3-amineIC50340.0 [1]
4-[2-[[5-Amino-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]ethyl]phenolIC502900.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(2-methoxyethyl)-1,3-benzothiazole-6-sulfonamideIC50600.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-[2-(1H-imidazol-5-yl)ethyl]-1,3-benzothiazole-6-sulfonamideIC50200.0 [1]
N-[2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-1,3-benzothiazol-6-yl]acetamideIC50400.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(2-phenylethyl)-1,3-benzothiazole-6-sulfonamideIC50800.0 [1]
4-(6-Chloro-1,3-benzothiazol-2-yl)-5-methyl-1H-pyrazol-3-amineIC50300.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-benzyl-1,3-benzothiazole-6-sulfonamideIC50800.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(4-fluorophenyl)-1H-pyrazol-3-amineIC502400.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-[2-(dimethylamino)ethyl]-1,3-benzothiazole-6-sulfonamideIC50300.0 [1]
3-N-(2-Aminoethyl)-4-(1,3-benzothiazol-2-yl)-1H-pyrazole-3,5-diamineIC5020.0 [1]
4-(7-Chloro-4-methoxy-1,3-benzothiazol-2-yl)-5-methyl-1H-pyrazol-3-amineIC501000.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(2-fluorophenyl)-1H-pyrazol-3-amineIC504000.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-fluoro-N-(2-hydroxyethyl)-1,3-benzothiazole-4-sulfonamideIC50150.0 [1]
4-(4-Fluorobenzothiazol-2-yl)-5-methyl-2H-pyrazol-3-ylamineIC50400.0 [1]
4-(5-Fluorobenzothiazol-2-YL)-5-methyl-2H-pyrazol-3-ylamineIC5040.0 [1]
4-(6-Nitro-1,3-benzothiazol-2-yl)-1H-pyrazol-5-amineIC503400.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(3-nitrophenyl)-1H-pyrazol-3-amineIC50900.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-thiophen-2-yl-1H-pyrazol-3-amineIC50700.0 [1]
[2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-fluorobenzothiazol-6-yl]methanolIC50100.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-N-(3-imidazol-1-ylpropyl)-1H-pyrazole-3,5-diamineIC50500.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-YL)-benzothiazole-6-carboxylic acid methyl esterIC50300.0 [1]
4-(5-Methoxy-benzothiazol-2-yl)-5-methyl-2H-pyrazol-3-ylamineIC503700.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(cyclopropylmethyl)-1,3-benzothiazole-6-sulfonamideIC50700.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-N-(2-pyrrolidin-1-ylethyl)-1H-pyrazole-3,5-diamineIC501900.0 [1]
4-(6-Dimethylaminomethyl-5-fluorobenzothiazol-2-yl)-5-methyl-1H-pyrazol-3-ylamineIC50600.0 [1]
4-(5-Fluoro-6-methoxybenzothiazol-2-yl)-5-methyl-2H-pyrazol-3-ylamineIC5060.0 [1]
4-[[[5-Amino-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]methyl]benzenesulfonamideIC502900.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(pyridin-4-ylmethyl)-1,3-benzothiazole-6-sulfonamideIC5040.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(2-hydroxyethyl)-1,3-benzothiazole-6-sulfonamideIC50200.0 [1]
3-[[2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-1,3-benzothiazol-6-yl]methylamino]benzenesulfonamideIC50800.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-N-[2-(ethylamino)ethyl]-1H-pyrazole-3,5-diamineIC50150.0 [1]
5-Methyl-4-[5-(trifluoromethyl)-1,3-benzothiazol-2-yl]-1H-pyrazol-3-amineIC502800.0 [1]
4-Benzothiazol-2-YL-5-piperidin-4-YL-2H-pyrazol-3-ylamineIC5060.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-N-[2-(1H-indol-3-yl)ethyl]-1H-pyrazole-3,5-diamineIC503300.0 [1]
Methyl 2-(3-amino-5-methyl-1H-pyrazol-4-yl)-5-fluoro-1,3-benzothiazole-6-carboxylateIC5060.0 [1]
3-[[5-Amino-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]propan-1-olIC50400.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-fluoro-N-(2-hydroxyethyl)-1,3-benzothiazole-6-sulfonamideIC5050.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-benzothiazole-6-carboxylic acidIC501100.0 [1]
5-Methyl-4-[6-(4-methylpiperazin-1-ylmethyl)-benzothiazol-2-yl]-2H-pyrazol-3-ylamineIC505000.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-N-[3-(dimethylamino)propyl]-1H-pyrazole-3,5-diamineIC50300.0 [1]
N-[2-[[2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-1,3-benzothiazol-6-yl]sulfonylamino]ethyl]acetamideIC50700.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(2-thiophen-2-ylethyl)-1,3-benzothiazole-6-sulfonamideIC501700.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-pyrrolidin-1-yl-1H-pyrazol-5-amineIC503700.0 [1]
4-(1,3-Benzothiazol-2-yl)-N-[2-(1H-imidazol-5-yl)ethyl]-1H-pyrazol-5-amineIC50200.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-(2-morpholin-4-ylethyl)-1,3-benzothiazole-6-sulfonamideIC503000.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(5-nitrofuran-2-yl)-1H-pyrazol-3-amineIC50300.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-phenyl-1H-pyrazol-3-amineIC502300.0 [1]
4-(6-Fluoro-1,3-benzothiazol-2-yl)-5-methyl-1H-pyrazol-3-amineIC50400.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-3-piperazin-1-yl-1H-pyrazol-5-amineIC5070.0 [1]
2-(5-Amino-3-methyl-1H-pyrazol-4-yl)benzothiazole-6-sulfonic acid 4-chlorobenzylamideIC50900.0 [1]
2-(5-Amino-3-methyl-1H-pyrazol-4-yl)benzothiazole-6-sulfonic acid 4-methoxybenzylamideIC501000.0 [1]
N-[2-[[5-Amino-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]ethyl]acetamideIC501100.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-1,3-benzothiazole-6-sulfonamideIC5010.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-piperazin-1-yl-1H-pyrazol-5-amineIC50190.0 [1]
4-(6-Dimethylaminomethylbenzothiazol-2-yl)-5-methyl-2H-pyrazol-3-ylamineIC50200.0 [1]
N-[2-[[5-Amino-4-(5-fluoro-6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]ethyl]acetamideIC501800.0 [1]
4-Benzothiazol-2-YL-5-(4-nitrophenyl)-2H-pyrazol-3-ylamineIC504000.0 [1]
4-(5-Fluoro-6-methyl-1,3-benzothiazol-2-yl)-5-methyl-1H-pyrazol-3-amineIC50300.0 [1]
4-Benzothiazol-2-YL-5-(3-methylamino-propyl)-2H-pyrazol-3-ylamineIC5020.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(4-methoxyphenyl)-1H-pyrazol-3-amineIC502000.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(3-fluorophenyl)-1H-pyrazol-3-amineIC502300.0 [1]
4-[[5-Amino-4-(1,3-benzothiazol-2-yl)-1H-pyrazol-3-yl]amino]butan-1-olIC501700.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-N-[2-(4-aminophenyl)ethyl]-1,3-benzothiazole-6-sulfonamideIC50200.0 [1]
4-Benzothiazol-2-yl-5-(4-methylaminobutyl)-2H-pyrazol-3-ylamineIC50100.0 [1]
4-(7-Chloro-5-fluoro-6-methoxybenzothiazol-2-YL)-5-methyl-1H-pyrazol-3-ylamineIC50400.0 [1]
2-(5-Amino-3-methyl-1H-pyrazol-4-yl)benzothiazol-5-olIC50200.0 [1]
4-(5-Amino-4-benzothiazol-2-yl-1H-pyrazol-3-yl)butan-1-olIC501000.0 [1]
5-Methyl-4-[6-(4-methylpiperazine-1-sulfonyl)-benzothiazol-2-yl]-2H-pyrazol-3-ylamineIC504900.0 [1]
3-(5-Amino-4-benzothiazol-2-YL-2H-pyrazol-3-YL)-propan-1-OLIC50200.0 [1]
4-(5-Fluoro-6-methyl-1,3-benzothiazol-2-yl)-1H-pyrazol-5-amineIC5050.0 [1]
5-Methyl-4-(6-methylsulfonyl-1,3-benzothiazol-2-yl)-1H-pyrazol-3-amineIC50500.0 [1]
3-N-[3-(Dimethylamino)propyl]-4-(5-fluoro-6-methoxy-1,3-benzothiazol-2-yl)-1H-pyrazole-3,5-diamineIC50200.0 [1]
2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-5-fluoro-N-methyl-1,3-benzothiazole-6-sulfonamideIC5040.0 [1]
4-(5-Fluoro-6-methoxy-1,3-benzothiazol-2-yl)-5-(2-phenylcyclopropyl)-1H-pyrazol-3-amineIC502100.0 [1]
4-(1,3-Benzothiazol-2-yl)-3-N-(2-methoxyethyl)-1H-pyrazole-3,5-diamineIC50700.0 [1]
4-(6-Bromobenzothiazol-2-YL)-5-methyl-2H-pyrazol-3-ylamineIC50400.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase ILK-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-ilk-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Serine/threonine-protein kinase ILK-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-ilk-1-inhibitors-ic50-ki.
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