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Serine/threonine-protein kinase haspin Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
HarmineIC50590.0 [1]
HarmolIC50770.0 [1]
N-[(1-Methylpiperidin-4-yl)methyl]-3-[3-(trifluoromethoxy)phenyl]imidazo[1,2-b]pyridazin-6-amineIC5034.0 [1]
CercosporamideIC5010000.0 [1]
Nms-P937 (nms1286937)IC5010000.0 [1]
CID 59604787IC5010000.0 [1]
5-[2,4-Dihydroxy-6-(4-Nitrophenoxy)phenyl]-N-(1-Methylpiperidin-4-Yl)-1,2-Oxazole-3-CarboxamideIC5010.0 [1]
2-[1-(4,4-Difluorocyclohexyl)-piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamideIC5010000.0 [1]
2-(4-Fluorophenyl)-N-[5-(4-pyridin-3-ylthiophen-2-yl)pyridin-3-yl]acetamideIC5036.0 [1]
(Arylindolyl)maleimide deriv. 27IC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
(5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC50259.0 [1]
3-[[5-(1,3-Benzodioxol-5-yl)-[1,2,4]triazolo[1,5-c]quinazolin-8-yl]amino]propan-1-olIC5010000.0 [1]
1-Methyl-4-[4-(4-{3-[(Piperidin-4-Yl)methoxy]pyridin-4-Yl}-1h-Pyrazol-1-Yl)phenyl]piperazineIC50190.0 [1]
(5Z)-5-(1,3-Benzothiazol-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC50255.0 [1]
6-(4-Methylpiperazin-1-yl)-2-naphthalen-1-yl-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(6-Methoxynaphthalen-1-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(6-Ethoxynaphthalen-1-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-5-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
[3-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]phenyl]-morpholin-4-ylmethanoneIC503900.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-3-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-phenylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-a]pyridineIC5010000.0 [1]
2-(2,3-Dihydro-1,4-benzodioxin-5-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-(4-phenylphenyl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-(3-phenylphenyl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-3-pyridin-4-yl-2-(3-thiophen-2-ylphenyl)imidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-3-pyridin-4-yl-2-(3-thiophen-3-ylphenyl)imidazo[1,2-b]pyridazineIC5010000.0 [1]
2-(2,3-Dihydro-1,4-benzodioxin-6-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
6-(4-Methylpiperazin-1-yl)-2-(5-phenylthiophen-2-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
[4-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]phenyl]-morpholin-4-ylmethanoneIC5010000.0 [1]
6-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]-1,3-benzothiazoleIC5010000.0 [1]
N-(4-Morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amineIC504.0 [1]
5-[2-[4-(Dimethylamino)phenoxy]-4,6-dihydroxyphenyl]-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamideIC5010.0 [1]
5-[2,4-Dihydroxy-6-[4-(propan-2-ylamino)phenoxy]phenyl]-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamideIC5010.0 [1]
5-[2-[4-(Dimethylamino)phenoxy]-4,6-dihydroxyphenyl]-N-[1-(1,4-dioxaspiro[4.5]decan-8-yl)piperidin-4-yl]-1,2-oxazole-3-carboxamideIC5010.0 [1]
3-Fluoro-4-(8,9,10,11-tetrahydro-3H-pyrazolo[4,3-a]phenanthridin-7-yl)phenolIC5012.0 [1]
Potassium;3-(3-aminoanilino)quinoxaline-2-carboxylateIC5010000.0 [1]
3-(3-Morpholin-4-ylanilino)quinoxaline-2-carboxylic acidIC5010000.0 [1]
3-(2-Hydroxyanilino)quinoxaline-2-carboxylic acidIC5010000.0 [1]
3-(4-Hydroxyanilino)quinoxaline-2-carboxylic acidIC5010000.0 [1]
4-Amino-7-hydroxy-9-oxo-1H-[1]benzofuro[3,2-d]pyrimidine-6-carboxamideIC5010000.0 [1]
4,7-Dihydroxy-2,9-dioxo-1,3-dihydro-[1]benzofuro[3,2-d]pyrimidine-6-carboxamideIC5010000.0 [1]
4,7-Dihydroxy-9-oxo-1H-[1]benzofuro[3,2-d]pyrimidine-6-carboxamideIC5010000.0 [1]
3-(3-Hydroxyanilino)quinoxaline-2-carboxylic acidIC5010000.0 [1]
6-[3-[1-Hydroxy-4-(1H-indol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanoic acidIC5010000.0 [1]
4-Hydroxy-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8,10,12,22,24,26-nonaene-3,5-dioneIC5010000.0 [1]
1-Hydroxy-3-(1H-indol-3-yl)-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
3-(1-Ethylindol-3-yl)-1-hydroxy-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
1-Hydroxy-3-(1H-indol-3-yl)-4-(1-methylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
1-Hydroxy-3-(1H-indol-3-yl)-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
6-[3-[4-[1-(5-Cyanopentyl)indol-3-yl]-1-hydroxy-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrileIC5010000.0 [1]
3-(1-Ethylindol-3-yl)-1-hydroxy-4-(1-methylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
1-Hydroxy-3,4-bis(1-methylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
6-[3-[4-[1-(5-Cyanopentyl)indol-3-yl]-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrileIC5010000.0 [1]
6-[3-[1-Hydroxy-4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrileIC5010000.0 [1]
1-Hydroxy-3-(1-methylindol-3-yl)-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dioneIC5010000.0 [1]
6-[3-[1-Hydroxy-4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanoic acidIC5010000.0 [1]
N-[5-(4-Pyridin-3-ylthiophen-2-yl)pyridin-3-yl]cyclopropanecarboxamideIC5076.3 [1]
2-(3-Methoxyphenyl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazineIC5010000.0 [1]
2-{[2-Amino-5-(1,3-Benzodioxol-5-Ylmethyl)[1,2,4]triazolo[1,5-C]quinazolin-8-Yl]amino}ethanolIC5010000.0 [1]
5-(1,3-Benzodioxol-5-ylmethyl)-[1,2,4]triazolo[1,5-c]quinazoline-2,8-diamineIC5010000.0 [1]
5-(1,3-Benzodioxol-5-Ylmethyl)-10-Fluoro[1,2,4]triazolo[1,5-C]quinazolin-2-AmineIC5010000.0 [1]
5-(1,3-Benzodioxol-5-ylmethyl)-10-fluoro-8-(4-methylpiperazin-1-yl)-[1,2,4]triazolo[1,5-c]quinazolin-2-amineIC5010000.0 [1]
3-(7-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)propan-1-amineIC50460.0 [1]
4-(7-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)butan-1-amineIC50170.0 [1]
4-(7-Methoxypyrido[3,4-b]indol-9-yl)butan-1-amineIC50300.0 [1]
4-(1-Ethyl-7-methoxypyrido[3,4-b]indol-9-yl)butan-1-amineIC50190.0 [1]
4-(7-Methoxy-1-propan-2-ylpyrido[3,4-b]indol-9-yl)butan-1-amineIC50460.0 [1]
9-(4-Aminobutyl)-1-methyl-2H-pyrido[3,4-b]indol-7-oneIC50160.0 [1]
4-(7-Fluoro-1-methylpyrido[3,4-b]indol-9-yl)butan-1-amineIC50580.0 [1]
4-(8-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)butan-1-amineIC50220.0 [1]
4-(6-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)butan-1-amineIC502400.0 [1]
4-(5-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)butan-1-amineIC502700.0 [1]
4-(8-Chloro-7-methoxy-1-methylpyrido[3,4-b]indol-9-yl)butan-1-amineIC50830.0 [1]
N-[9-(4-Aminobutyl)-1-methylpyrido[3,4-b]indol-7-yl]methanesulfonamideIC50690.0 [1]
4-(7-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)-N-methylbutan-1-amineIC50340.0 [1]
4-(7-Methoxy-1-methylpyrido[3,4-b]indol-9-yl)-N,N-dimethylbutan-1-amineIC50470.0 [1]
4-[1-Methyl-7-[(2-methylpropan-2-yl)oxy]pyrido[3,4-b]indol-9-yl]butan-1-amineIC504600.0 [1]
9-(4-Aminobutyl)-1-(trifluoromethyl)-2H-pyrido[3,4-b]indol-7-oneIC50220.0 [1]
4-(6-Methyl-12,14-dioxa-5,8-diazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2(7),3,5,9,11(15)-hexaen-8-yl)butan-1-amineIC50500.0 [1]
4-(7-Methoxy-1-(Trifluoromethyl)-9h-Pyrido[3,4-B]indol-9-Yl)butan-1-AmineIC50100.0 [1]
2-[(4S)-7-(3-Chlorophenyl)-1-oxo-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-4-yl]-N-[(1S)-1-cyclohexyl-2-(4-methylpiperazin-1-yl)ethyl]acetamideIC5010000.0 [1]
N-(2,2-Dimethylpropyl)-2-(1-oxo-7-thiophen-3-yl-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-4-yl)acetamideIC5010000.0 [1]
Items per page: 1 - 10 of 86
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase haspin Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-haspin-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Serine/threonine-protein kinase haspin Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-haspin-inhibitors-ic50-ki.
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