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Serine/threonine-protein kinase/endoribonuclease IRE1 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
3,5-DibromosalicylaldehydeIC50720.0 [1], 20000.0 [2]
CID 25160990IC505665.0 [1], 20000.0 [2]
2-Hydroxy-3-methoxybenzaldehydeIC505750.0 [1]
5-BromosalicylaldehydeIC501330.0 [1]
2,3-DihydroxybenzaldehydeIC5020250.0 [1]
5-ChlorosalicylaldehydeIC503120.0 [1]
2-Hydroxy-5-nitrobenzaldehydeIC501280.0 [1]
3,5-DichlorosalicylaldehydeIC501750.0 [1]
2-Hydroxy-5-methoxybenzaldehydeIC508850.0 [1]
3-Bromo-5-chloro-2-hydroxybenzaldehydeIC501300.0 [1]
3,5-DiiodosalicylaldehydeIC50440.0 [1]
5-Bromo-2-hydroxy-3-methoxybenzaldehydeIC50240.0 [1]
4,6-DimethoxysalicylaldehydeIC506830.0 [1]
5-Chloro-2-hydroxyisophthalaldehydeIC50400.0 [1]
2-Hydroxy-3-methoxy-5-nitrobenzaldehydeIC50170.0 [1]
2-Hydroxy-5-iodobenzaldehydeIC501400.0 [1]
6-Bromo-2-hydroxy-3-methoxybenzaldehydeIC5080.0 [1]
3-FluorosalicylaldehydeIC502850.0 [1]
3-NitrosalicylaldehydeIC505500.0 [1]
4-N-[4-[2-[4-(1H-Benzimidazol-2-ylamino)naphthalen-1-yl]oxypyridin-3-yl]pyrimidin-2-yl]cyclohexane-1,4-diamineIC5011.0 [1], 43.0 [2]
2-(2-Hydroxyethyliminomethyl)-4-bromo-6-methoxyphenolIC50154.0 [1]
CID 59599728IC505.0 [1]
3-Hydroxy-4-methoxynaphthalene-2-carbaldehydeIC502260.0 [1]
2-Hydroxy-5-(pyridin-3-yl)benzaldehydeIC50141.0 [1]
2-Hydroxy-5-(pyridin-4-yl)benzaldehydeIC50147.0 [1]
6-Hydroxyquinoline-5-carbaldehydeIC50170.0 [1]
7-Hydroxyquinoline-8-carbaldehydeIC501240.0 [1]
2-Methoxy-6-[(4-methoxyphenyl)methyliminomethyl]-4-thiophen-2-ylphenolIC5023.0 [1]
2-(2-Hydroxyethyliminomethyl)-6-methoxy-4-thiophen-2-ylphenolIC5015.0 [1]
2-(Cyclopropyliminomethyl)-6-methoxy-4-thiophen-2-ylphenolIC5034.0 [1]
2-Methoxy-6-[(E)-pyridin-2-yliminomethyl]-4-thiophen-2-ylphenolIC5020000.0 [1]
6-(5-Formyl-6-hydroxynaphthalen-2-yl)pyridine-2-carboxylic acidIC50125.0 [1]
6-(5-Formyl-6-hydroxynaphthalen-2-yl)-N-(2-morpholin-4-ylethyl)pyridine-2-carboxamideIC5048.0 [1]
2-Hydroxy-6-[6-(morpholine-4-carbonyl)pyridin-2-yl]naphthalene-1-carbaldehydeIC50645.0 [1]
2-Hydroxy-3-nitro-5-quinolin-5-ylbenzaldehydeIC50333.0 [1], 3333.0 [2]
2-Hydroxy-3-methoxy-5-pyridin-4-ylbenzaldehydeIC50104.0 [1]
4-Bromo-2-hydroxy-3-[(4-methoxyphenyl)methyliminomethyl]benzoic acidIC5020000.0 [1]
4-Bromo-3-(cyclopropyliminomethyl)-2-hydroxybenzoic acidIC509523.0 [1]
2-Hydroxy-3-methoxy-5-pyridin-2-ylbenzaldehydeIC50108.0 [1]
2-[2-[2-[(2-Hydroxy-3-methoxy-5-thiophen-2-ylphenyl)methylideneamino]ethyldisulfanyl]ethyliminomethyl]-6-methoxy-4-thiophen-2-ylphenolIC501348.0 [1]
2-Hydroxy-6-quinolin-5-ylnaphthalene-1-carbaldehydeIC506277.0 [1]
6-(5-Formyl-6-hydroxynaphthalen-2-yl)-N-propan-2-ylpyridine-2-carboxamideIC5047.0 [1]
6-Hydroxy-N-[(4-methoxyphenyl)methyl]-5-[(4-methoxyphenyl)methyliminomethyl]naphthalene-2-carboxamideIC5020000.0 [1]
3-Fluoro-2-hydroxy-5-quinolin-5-ylbenzaldehydeIC50305.0 [1]
4-Bromo-2-[2-[2-[(5-bromo-2-hydroxy-3-methoxyphenyl)methylideneamino]ethyldisulfanyl]ethyliminomethyl]-6-methoxyphenolIC502117.0 [1]
6-Hydroxy-N-[(4-methoxyphenyl)methyl]-5-[(4-methoxyphenyl)methyliminomethyl]naphthalene-1-carboxamideIC5020000.0 [1]
2-Hydroxy-3-methoxy-5-quinolin-5-ylbenzaldehydeIC50932.0 [1]
5-Isoquinolinecarboxaldehyde, 6-hydroxy-IC50427.0 [1]
4-Bromo-2-methoxy-6-[(4-methoxyphenyl)methyliminomethyl]phenolIC50221.0 [1]
2-Hydroxy-6-[6-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]naphthalene-1-carbaldehydeIC50389.0 [1]
4-Bromo-2-methoxy-6-[(E)-1,3-thiazol-2-yliminomethyl]phenolIC50641.0 [1]
4-Bromo-2-(cyclopropyliminomethyl)-6-methoxyphenolIC50110.0 [1]
2-Hydroxy-3-methoxy-5-thien-2-ylbenzaldehydeIC5022.0 [1]
3'-Formyl-4'-hydroxy[1,1'-biphenyl]-4-carboxylic acidIC50172.0 [1]
3'-Formyl-4'-hydroxy[1,1'-biphenyl]-3-carboxylic acidIC50371.0 [1]
Methyl 3'-formyl-4'-hydroxy[1,1'-biphenyl]-4-carboxylateIC50351.0 [1]
Methyl 3'-formyl-4'-hydroxy[1,1'-biphenyl]-3-carboxylateIC50421.0 [1]
2-Hydroxy-5-(3-thienyl)benzaldehydeIC50699.0 [1]
5-(Furan-2-yl)-2-hydroxybenzaldehydeIC50223.0 [1]
2-Hydroxy-5-(5-pyrimidinyl)benzaldehydeIC50170.0 [1]
3'-Formyl-4'-hydroxy-5'-methoxybiphenyl-3-carboxylic acidIC50102.0 [1]
N-Cyclohexyl-3-(3-formyl-4-hydroxy-5-methoxyphenyl)benzamideIC5019.0 [1]
6-Bromo-2-hydroxy-3-(morpholine-4-carbonyl)benzaldehydeIC50526.0 [1]
5-(1,3-Dimethyl-2,4-dioxopyrimidin-5-yl)-2-hydroxy-3-methoxybenzaldehydeIC501581.0 [1]
2-Hydroxy-6-pyridin-3-ylnaphthalene-1-carbaldehydeIC5023.0 [1]
2-Hydroxy-6-[3-(morpholine-4-carbonyl)phenyl]naphthalene-1-carbaldehydeIC5074.0 [1]
3-Hydroxy-2-methylquinoline-4-carbaldehydeIC5036370.0 [1]
Ethyl 2-(5-bromo-2-hydroxy-3-methoxyphenyl)-1,3-thiazolidine-5-carboxylateIC5017662.0 [1]
4-Bromo-2-methoxy-6-(1,3-thiazolidin-2-yl)phenolIC504146.0 [1]
4-Bromo-2-hydroxy-3-(1,3-thiazolidin-2-yl)benzoic acidIC5020000.0 [1]
2-Methoxy-6-(1,3-thiazolidin-2-yl)-4-thiophen-2-ylphenolIC5020000.0 [1]
3,5-Difluoro-2-hydroxybenzaldehydeIC503060.0 [1]
1-[(2-Mercaptoethyl)iminomethyl]-2-naphtholIC5020000.0 [1]
2-Hydroxy-3-methoxy-5-thiophen-3-ylbenzaldehydeIC50199.0 [1]
5-(2-Fluorophenyl)-2-hydroxy-3-methoxybenzaldehydeIC50400.0 [1]
2-Hydroxy-3-methoxy-5-(4-methoxyphenyl)benzaldehydeIC501380.0 [1]
2-Hydroxy-3-methoxy-5-(3-methoxyphenyl)benzaldehydeIC50400.0 [1]
2-Hydroxy-3-methoxy-5-(2-methoxyphenyl)benzaldehydeIC501590.0 [1]
5-(2-Chlorophenyl)-2-hydroxy-3-methoxybenzaldehydeIC501280.0 [1]
5-(4-Chlorophenyl)-2-hydroxy-3-methoxybenzaldehydeIC501830.0 [1]
5-(3,4-Dimethoxyphenyl)-2-hydroxy-3-methoxybenzaldehydeIC50380.0 [1]
5-(5-Chloro-2-methoxyphenyl)-2-hydroxy-3-methoxybenzaldehydeIC501640.0 [1]
2-Hydroxy-3-methoxy-5-(1H-pyrazol-4-yl)benzaldehydeIC50310.0 [1]
2-Hydroxy-3-methoxy-5-pyridin-3-ylbenzaldehydeIC50149.0 [1]
2-Hydroxy-3-methoxy-5-pyrimidin-5-ylbenzaldehydeIC5039.0 [1]
2-Hydroxy-3-methoxy-5-(1-methylpyrazol-4-yl)benzaldehydeIC50772.0 [1]
3-(3-Formyl-4-hydroxy-5-methoxyphenyl)benzamideIC50173.0 [1]
N-Benzyl-3-(3-formyl-4-hydroxyphenyl)benzamideIC50106.0 [1]
N-Benzyl-3-(3-formyl-4-hydroxy-5-methoxyphenyl)benzamideIC506.0 [1]
3-(3-Fluoro-5-formyl-4-hydroxyphenyl)benzamideIC5046.0 [1]
2,3-Dibromo-6-hydroxy-5-methoxybenzaldehydeIC5030.0 [1]
5-Chloro-2-hydroxy-3-methoxybenzaldehydeIC50280.0 [1]
5-(3,5-Dimethyl-1,2-oxazol-4-yl)-2-hydroxybenzaldehydeIC501011.0 [1]
3'-Formyl-4'-hydroxy[1,1'-biphenyl]-3-carboxamideIC50197.0 [1]
4-[Benzo(B)thiophen-2-YL]-2-formylphenolIC5020000.0 [1]
3'-Formyl-4'-hydroxy-N,N-dimethyl[1,1'-biphenyl]-3-carboxamideIC50147.0 [1]
4-[4-(N,N-Dimethylaminocarbonyl)phenyl]-2-formylphenolIC50420.0 [1]
4-(3-Formyl-4-hydroxy-5-nitrophenyl)benzoic acidIC50101.0 [1]
3-(3-Formyl-4-hydroxy-5-nitrophenyl)benzoic acidIC50132.0 [1]
Methyl 4-(3-formyl-4-hydroxy-5-nitrophenyl)benzoateIC5021.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase/endoribonuclease IRE1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-endoribonuclease-ire1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Serine/threonine-protein kinase/endoribonuclease IRE1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-endoribonuclease-ire1-inhibitors-ic50-ki.
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