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Serine/threonine-protein kinase EEF2K Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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7-Amino-1-cyclopropyl-3-ethyl-2,4-dioxo-1,2,3,4-tetrahydropyrido[2,3-d]pyrimidine-6-carboxamideIC50280.0 [1], 420.0 [2], 510.0 [3]
2-((3,5-Dimethyl-4-hydroxyphenyl)-methylene)-4-cyclopentene-1,3-dioneIC50440.0 [1]
EntrectinibIC5010000.0 [1]
Nms-P937 (nms1286937)IC5010000.0 [1]
5-[2,4-Dihydroxy-6-(4-Nitrophenoxy)phenyl]-N-(1-Methylpiperidin-4-Yl)-1,2-Oxazole-3-CarboxamideIC5010.0 [1]
2-((3,5-Di-tert-Butyl-4-hydroxyphenyl)-methylene)-4-cyclopentene-1,3-dioneIC503200.0 [1]
3-Amino-5,6,7,8,9,10-hexahydrocycloocta[b]thieno[3,2-e]pyridine-2-carboxamideIC502500.0 [1]
5-(2-Aminopyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-carboxamideIC5010000.0 [1]
2-[1-(4,4-Difluorocyclohexyl)-piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamideIC5010000.0 [1]
6-Amino-8-(furan-2-yl)-4-thia-2-azatricyclo[7.7.0.03,7]hexadeca-1(9),2,5,7-tetraene-5-carboxamideIC50170.0 [1]
3-[[5-(1,3-Benzodioxol-5-yl)-[1,2,4]triazolo[1,5-c]quinazolin-8-yl]amino]propan-1-olIC5010000.0 [1]
7-Amino-1,3-diethyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamideIC501000.0 [1]
6-Amino-1-cyclopropyl-3-ethylpyrimidine-2,4-dioneIC5025000.0 [1]
6-Amino-1-cyclopropyl-3-ethyl-2,4-dioxopyrimidine-5-carbaldehydeIC5025000.0 [1]
7-Amino-1-cyclopropyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamideIC506600.0 [1]
7-Amino-1-cyclopropyl-3-methyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamideIC506100.0 [1]
7-Amino-1-cyclopropyl-2,4-dioxo-3-propylpyrido[2,3-d]pyrimidine-6-carboxamideIC50930.0 [1]
7-Amino-1-cyclopropyl-3-[(4-nitrophenyl)methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamideIC5025000.0 [1]
7-Amino-3-[(4-aminophenyl)methyl]-1-cyclopropyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamideIC5025000.0 [1]
7-Amino-1-cyclopropyl-3-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carbothioamideIC5025000.0 [1]
7-Amino-1,3-dimethyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamideIC5025000.0 [1]
5-[2-[4-(Dimethylamino)phenoxy]-4,6-dihydroxyphenyl]-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamideIC5010.0 [1]
5-[2,4-Dihydroxy-6-[4-(propan-2-ylamino)phenoxy]phenyl]-N-(1-methylpiperidin-4-yl)-1,2-oxazole-3-carboxamideIC5010.0 [1]
5-[2-[4-(Dimethylamino)phenoxy]-4,6-dihydroxyphenyl]-N-[1-(1,4-dioxaspiro[4.5]decan-8-yl)piperidin-4-yl]-1,2-oxazole-3-carboxamideIC5010.0 [1]
1-Benzyl-3-hexadecyl-2-methyl-4,5-dihydroimidazol-1-ium;iodideIC5060.0 [1]
3-(2,4-Dichlorophenyl)-3-[(4-fluorobenzoyl)amino]propanoic acidIC5017100.0 [1]
3-[(3-Bromobenzoyl)amino]-3-(2,4-dichlorophenyl)propanoic acidIC5028400.0 [1]
3-(2,4-Dichlorophenyl)-3-[(3,5-difluorophenyl)sulfonylamino]propanoic acidIC5012500.0 [1]
3-(2-Fluorophenyl)-3-[[4-(trifluoromethyl)phenyl]sulfonylamino]propanoic acidIC5011600.0 [1]
3-[(3-Bromobenzoyl)amino]-3-(2-fluorophenyl)propanoic acidIC5050000.0 [1]
3-[(2,4-Dichlorobenzoyl)amino]-3-(2-fluorophenyl)propanoic acidIC5033700.0 [1]
3-(4-Tert-butylphenyl)-3-[(4-fluorophenyl)sulfonylamino]propanoic acidIC5038500.0 [1]
3-[(4-Cyanophenyl)sulfonylamino]-3-(2-fluorophenyl)propanoic acidIC5027500.0 [1]
3-(2,4-Dichlorophenyl)-3-[(2-methoxybenzoyl)amino]propanoic acidIC5050000.0 [1]
3-(Benzenesulfonamido)-3-(2-fluorophenyl)propanoic acidIC5050000.0 [1]
3-(Benzenesulfonamido)-3-(2,4-dichlorophenyl)propanoic acidIC5033400.0 [1]
3-(4-Tert-butylphenyl)-3-[[4-(trifluoromethoxy)phenyl]sulfonylamino]propanoic acidIC5050000.0 [1]
3-[(2,6-Dichlorobenzoyl)amino]-3-phenylpropanoic acidIC5050000.0 [1]
3-(2-Fluorophenyl)-3-[[4-(trifluoromethyl)benzoyl]amino]propanoic acidIC5044500.0 [1]
3-[(2,4-Dichlorobenzoyl)amino]-3-(2,4-dichlorophenyl)propanoic acidIC5019900.0 [1]
3-[(2-Bromophenyl)sulfonylamino]-3-(2,4-dichlorophenyl)propanoic acidIC5050000.0 [1]
3-(4-Tert-butylphenyl)-3-[[4-(trifluoromethyl)benzoyl]amino]propanoic acidIC5022600.0 [1]
3-[(4-Fluorobenzoyl)amino]-3-(2-fluorophenyl)propanoic acidIC5036700.0 [1]
3-(4-Tert-butylphenyl)-3-[(2-methoxybenzoyl)amino]propanoic acidIC5050000.0 [1]
3-(4-Tert-butylphenyl)-3-[(2,6-dichlorobenzoyl)amino]propanoic acidIC5050000.0 [1]
3-[(4-Cyanophenyl)sulfonylamino]-3-(2,4-dichlorophenyl)propanoic acidIC505500.0 [1]
3-(2,4-Dichlorophenyl)-3-[(4-methoxybenzoyl)amino]propanoic acidIC5044400.0 [1]
3-(2,4-Dichlorophenyl)-3-[[4-(trifluoromethyl)benzoyl]amino]propanoic acidIC5011700.0 [1]
3-[(2,6-Dichlorobenzoyl)amino]-3-(2,4-dichlorophenyl)propanoic acidIC5050000.0 [1]
3-(Benzenesulfonamido)-3-(4-tert-butylphenyl)propanoic acidIC5050000.0 [1]
3-[(3,5-Difluorophenyl)sulfonylamino]-3-(2-fluorophenyl)propanoic acidIC5019400.0 [1]
3-(2,4-Dichlorophenyl)-3-[(3-nitrophenyl)sulfonylamino]propanoic acidIC5044500.0 [1]
3-(4-Tert-butylphenyl)-3-[[4-(trifluoromethyl)phenyl]sulfonylamino]propanoic acidIC5018400.0 [1]
3-(4-Tert-butylphenyl)-3-[(2-methoxyphenyl)sulfonylamino]propanoic acidIC5050000.0 [1]
3-(2,4-Dichlorophenyl)-3-[[4-(trifluoromethyl)phenyl]sulfonylamino]propanoic acidIC509500.0 [1]
1-(3-Chlorophenyl)-3-[4-[2-(ethylamino)pyridin-4-yl]-3-(trifluoromethyl)phenyl]ureaIC50762.0 [1]
7-Amino-1-cyclopropyl-3-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carbonitrileIC5025000.0 [1]
Ethyl 7-amino-1-cyclopropyl-3-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxylateIC5025000.0 [1]
3-[(2-Methoxybenzoyl)amino]-3-phenylpropanoic acidIC5050000.0 [1]
3-[(4-Fluorobenzoyl)amino]-3-phenylpropanoic acidIC5035100.0 [1]
3-[(2,4-Dichlorobenzoyl)amino]-3-phenylpropanoic acidIC5029300.0 [1]
3-[(3-Bromophenyl)formamido]-3-phenylpropanoic acidIC5050000.0 [1]
3-{[(3-Nitrophenyl)sulfonyl]amino}-3-phenylpropanoic acidIC5050000.0 [1]
3-{[(4-Fluorophenyl)sulfonyl]amino}-3-phenylpropanoic acidIC5031200.0 [1]
3-Phenyl-3-[(phenylsulfonyl)amino]propanoic acidIC5050000.0 [1]
Chembl4169894IC5031600.0 [1]
8-[(1-Acetylpiperidin-4-yl)amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5010000.0 [1]
8-[(1-Benzoylpiperidin-4-yl)amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5010000.0 [1]
3-[(3,5-Difluorophenyl)sulfonylamino]-3-phenylpropanoic acidIC5037800.0 [1]
3-[(2-Bromophenyl)sulfonylamino]-3-phenylpropanoic acidIC5050000.0 [1]
3-[(4-Cyanophenyl)sulfonylamino]-3-phenylpropanoic acidIC5018700.0 [1]
3-Phenyl-3-[[4-(trifluoromethoxy)phenyl]sulfonylamino]propanoic acidIC5050000.0 [1]
3-Phenyl-3-[[4-(trifluoromethyl)phenyl]sulfonylamino]propanoic acidIC5019600.0 [1]
3-{[(4-Tert-butylphenyl)sulfonyl]amino}-3-phenylpropanoic acidIC5050000.0 [1]
N,1-Dimethyl-8-[[1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-4-yl]amino]-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5010000.0 [1]
6-Amino-8-[(E)-2-(furan-2-yl)ethenyl]-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50320.0 [1]
6-Amino-8-methyl-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1,3(7),5,8-tetraene-5-carboxamideIC501100.0 [1]
6-Amino-8-(2-methylpropyl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50860.0 [1]
6-Amino-8-cyclopropyl-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC502000.0 [1]
6-Amino-8-(6-methylhept-5-en-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC5010000.0 [1]
6-Amino-8-(3,4-dichlorophenyl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50990.0 [1]
6-Amino-8-(4-chlorophenyl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC501100.0 [1]
6-Amino-8-phenyl-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC5020000.0 [1]
4-(6-Amino-5-carbamoyl-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraen-8-yl)benzoic acidIC50860.0 [1]
6-Amino-8-(2-fluoro-5-methoxyphenyl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC501300.0 [1]
6-Amino-8-(3-methylphenyl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC501200.0 [1]
6-Amino-8-(furan-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50640.0 [1]
6-Amino-8-(3-methylthiophen-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50460.0 [1]
6-Amino-8-pyridin-3-yl-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50940.0 [1]
6-Amino-8-(1-methylpyrrol-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50990.0 [1]
6-Amino-8-(furan-3-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC501100.0 [1]
6-Amino-8-(1,3-thiazol-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC501400.0 [1]
6-Amino-8-(3-methylpyridin-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC5020000.0 [1]
6-Amino-8-(2-phenylethyl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC5020000.0 [1]
6-Amino-8-(5-chlorofuran-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50280.0 [1]
6-Amino-8-[5-(trifluoromethyl)furan-2-yl]-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50300.0 [1]
6-Amino-8-(1-benzofuran-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50330.0 [1]
6-Amino-8-(5-ethylfuran-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50660.0 [1]
6-Amino-8-[5-(hydroxymethyl)furan-2-yl]-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC50800.0 [1]
6-Amino-8-(4,5-dimethylfuran-2-yl)-4-thia-2-azatricyclo[7.6.0.03,7]pentadeca-1(9),2,5,7-tetraene-5-carboxamideIC501100.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase EEF2K Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-eef2k-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Serine/threonine-protein kinase EEF2K Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-eef2k-inhibitors-ic50-ki.
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