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Serine/threonine-protein kinase D2 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
DoramapimodIC5030000.0 [1]
7-Hydroxy-2,3,4,5-tetrahydro-1H-benzofuro[2,3-c]azepin-1-oneIC50280.0 [1]
JNK Inhibitor VIIIKi5300.0 [1]
CID 53246941IC50139.0 [1]
CID 59604787IC5010000.0 [1]
BpkdiIC509.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi2500.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideKi5200.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi8980.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamideKi10000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi9000.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi9000.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi950.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi9000.0 [1]
(13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dioneIC501000.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amineIC50950.0 [1]
N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamideIC501000.0 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi1000.0 [1]
6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamideIC5010000.0 [1]
4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-iumIC5010000.0 [1]
N-Cyclohexyl-4-[6-piperazin-1-yl-4-(1H-pyrazol-5-yl)pyridin-2-yl]pyridin-2-amineIC5062.0 [1]
4-[6-Piperazin-1-yl-4-(1H-pyrazol-4-yl)pyridin-2-yl]-N-propan-2-ylpyridin-2-amineIC502.0 [1]
N-(Oxan-4-yl)-4-[6-piperazin-1-yl-4-(1H-pyrazol-4-yl)pyridin-2-yl]pyridin-2-amineIC502.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[[(3R)-pyrrolidin-3-yl]amino]pyridine-4-carboxamideIC5018.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[[(3S)-pyrrolidin-3-yl]amino]pyridine-4-carboxamideIC50540.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[(3R)-3-methylpiperazin-1-yl]pyridine-4-carboxamideIC5060.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[(3S)-3-methylpiperazin-1-yl]pyridine-4-carboxamideIC5086.0 [1]
2-(3-Aminopiperidin-1-yl)-6-[2-(cyclohexylamino)pyridin-4-yl]pyridine-4-carboxamideIC50168.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-(4-methylpiperazin-1-yl)pyridine-4-carboxamideIC50238.0 [1]
2-[4-(Aminomethyl)piperidin-1-yl]-6-[2-(cyclohexylamino)pyridin-4-yl]pyridine-4-carboxamideIC50212.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-(3,3-dimethylpiperazin-1-yl)pyridine-4-carboxamideIC50427.0 [1]
N-Cyclohexyl-4-[6-piperazin-1-yl-4-(trifluoromethyl)pyridin-2-yl]pyridin-2-amineIC50101.0 [1]
N-Cyclohexyl-4-[4-(difluoromethyl)-6-piperazin-1-ylpyridin-2-yl]pyridin-2-amineIC5076.0 [1]
2-(2-Anilinopyridin-4-yl)-6-piperazin-1-ylpyridine-4-carboxamideIC501.0 [1]
2-[2-(Oxan-4-ylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC509.0 [1]
2-Piperazin-1-yl-6-[2-(propan-2-ylamino)pyridin-4-yl]pyridine-4-carboxamideIC508.0 [1]
2-[2-[(1-Methylpyrazol-3-yl)amino]pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC507.0 [1]
2-[2-(2-Chloroanilino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC508.0 [1]
2-[2-(Cyclopentylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC5059.0 [1]
2-[2-(Ethylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC5031.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carbonitrileIC50130.0 [1]
2-(2-Anilinopyridin-4-yl)-6-piperazin-1-ylpyridine-4-carbonitrileIC5035.0 [1]
2-[2-[(1-Methylpyrazol-3-yl)amino]pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carbonitrileIC5068.0 [1]
N-Cyclohexyl-4-[6-piperazin-1-yl-4-(1H-pyrazol-4-yl)pyridin-2-yl]pyridin-2-amineIC501.0 [1]
N-[(1R)-1-Cyanoethyl]-3-[5-[4-[(oxan-4-ylamino)methyl]phenyl]-1,2-oxazol-3-yl]benzamideIC5048.0 [1]
4-Methoxy-8,14-dithia-3,5,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),2,4,6-tetraen-10-oneIC5050.0 [1]
4-[2-Amino-5-[4-[(dimethylamino)methyl]thiophen-2-yl]pyridin-3-yl]-2-[(Z,2R)-5,5,5-trifluoropent-3-en-2-yl]oxybenzamideIC50330.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC501000.0 [1]
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-PurineIC5046000.0 [1]
6-(2,9-Diazaspiro[5.5]undecan-9-Yl)-9h-PurineIC501300.0 [1]
3-(Tert-butylamino)-4-[[2-(4-pyridin-4-ylanilino)pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dioneKi175.0 [1]
Items per page: 1 - 10 of 58
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References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase D2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-d2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Serine/threonine-protein kinase D2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-d2-inhibitors-ic50-ki.
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