![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_2060f6287083a28c9ead968a2460ede5.svg) | Tozasertib | IC50 | 4.6 [1], 70.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_2060f6287083a28c9ead968a2460ede5.svg) | Tozasertib | Ki | 4.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_aea8e5cd5eedd851a20871e2fe5ff0da.svg) | Danusertib | IC50 | 61.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_aea8e5cd5eedd851a20871e2fe5ff0da.svg) | Danusertib | Ki | 61.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_899e7233470c1e6b0c695ac9e914d9bb.svg) | 3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea | IC50 | 6.5 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_899e7233470c1e6b0c695ac9e914d9bb.svg) | 3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea | Ki | 1.5 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_bf4bbfed2d9a84ce58724a3f96582d1c.svg) | N-(2,6-Diethylphenyl)-3-[[4-(4-methylpiperazin-1-yl)benzoyl]amino]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazole-5-carboxamide | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_90018542cb653c64f1d13e3042c3f13c.svg) | Ethyl (9S)-9-[3-(1H-benzimidazol-2-yloxy)phenyl]-8-oxo-2,4,5,6,7,9-hexahydropyrrolo[3,4-b]quinoline-3-carboxylate | IC50 | 3.0 [1], 91.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_cf650059ebadf876573929d505122599.svg) | 6-Bromoindirubin-3'-oxime | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_8aa951d1935df336d561e6b48c9639a1.svg) | Su6656 | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_5428ac790b8af307435e4cd8a8ff47bb.svg) | Indirubin-3'-monoxime | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_818e20960290ff06e97b77b6f2196c9f.svg) | Barasertib | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_37acee0cd10541aa0b3bd57948b54806.svg) | Orantinib | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_bd1c4c226d09bccaf8e1c9ed8e2ba78a.svg) | Azd-1152hqpa | Ki | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_b7658ddcd7d263fa59a78a027c0aecaa.svg) | N-(4-(3-(2-Aminopyrimidin-4-yl)pyridin-2-yloxy)phenyl)-4-(4-methylthiophen-2-yl)phthalazin-1-amine | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_102ec7c5ee0c4ac821e03c1f1a4333ee.svg) | MK-5108 | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_a2d32a1f7c79660a88d646bbda5ee232.svg) | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_4e8b5202a71aafe003ab207cc4576058.svg) | 3-(1H-Indol-5-yl)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrrolo[2,3-b]pyridine | IC50 | 290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_57b1a53e0843c3a5378b2a53d12b0246.svg) | 7-Bromo-3-[3-(hydroxyamino)-1H-indol-2-yl]indol-2-one | IC50 | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_056c9191a034ade62826fb324b220197.svg) | Cct-129202 | IC50 | 227.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_ebfe6297f32e2686e7c18db06b48c78f.svg) | 7-Bromoindirubin | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_588f2be4587722618ef7ac0ea5aa517b.svg) | 7-Fluoro-3-[3-(hydroxyamino)-1H-indol-2-yl]indol-2-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_459921ea52a3c083de5a04274a53ee71.svg) | 7-Chloro-3-[3-(hydroxyamino)-1H-indol-2-yl]indol-2-one | IC50 | 900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_8899da5b11f5a8577f6f65dc6a954bb6.svg) | 7-Chloroindirubin | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_0edf9f76354790e3c34cb7887cac0f1d.svg) | 7-Fluoroindirubin | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_63c811b726c5cb3bca95e2c0f3f889dd.svg) | 2-(2-Hydroxy-7-iodo-1H-indol-3-yl)indol-3-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_86184bd783d1d52b3257ec6b20c242fa.svg) | 7-Iodo-3-(3-nitroso-1H-indol-2-yl)-1H-indol-2-ol | IC50 | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_12adea5a0beab1cb5238674f1853b18c.svg) | N-(4-(4-(3-Methyl-1H-pyrazol-5-ylamino)quinazolin-2-ylthio)phenyl)acetamide | Ki | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_94e490915983085a98fddac87c39e7c3.svg) | 3-[(4-Morpholin-4-ylbenzoyl)amino]-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-thieno[3,2-c]pyrazole-5-carboxamide | IC50 | 62.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_aedad5e135aaf41fff76ab90c98f1d40.svg) | 4-(Prop-2-enoylamino)-N-[4-[(5,8,11-trimethyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamide | IC50 | 63.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_1745880f16ec42a4020815071cddd64c.svg) | Indirubin-3-methoxime | IC50 | 400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_25a83cc2323f61f5ea86dc91fc467353.svg) | Indirubin-3-acetoxime | IC50 | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_5200127bbb6461e37cb44e51a63a0d1d.svg) | 3-Chloro-N-(4-morpholin-4-ylphenyl)-6-pyridin-3-ylimidazo[1,2-a]pyrazin-8-amine | IC50 | 1950.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_ef431bf27ff7842bbb4caafd947b43c7.svg) | Tilfrinib | IC50 | 259.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_5b63ea15265b993819abd00ed6f2eee3.svg) | 2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_60a800a4e4f140f7ee106adafde00fce.svg) | 5-[(Z)-[6-[[3-(4-Methoxyanilino)-3-oxopropanoyl]amino]-2-oxo-1H-indol-3-ylidene]methyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid | IC50 | 153.5 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_d2281e2e3ba1777d2f6c5b1c058c9add.svg) | 4-(Propanoylamino)-N-[4-[(5,8,11-trimethyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamide | IC50 | 53.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_c35190032016ee50a0bbc56656308927.svg) | [(Z)-[2-(7-Chloro-2-hydroxy-1H-indol-3-yl)indol-3-ylidene]amino] acetate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_9d033f7532c295d7bd3c1e14385b76e4.svg) | 7-Chloro-3-[(3Z)-3-methoxyiminoindol-2-yl]-1H-indol-2-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_1448a37f7aedcca58f6d61c2c8df9a97.svg) | [(Z)-[2-(2-Hydroxy-7-iodo-1H-indol-3-yl)indol-3-ylidene]amino] acetate | IC50 | 28000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_b1bde89e81e014f412a79681fb866910.svg) | [(Z)-[2-(7-Bromo-2-hydroxy-1H-indol-3-yl)indol-3-ylidene]amino] acetate | IC50 | 4500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_8be5dcaa0ddcf25fb96528177369c695.svg) | [(Z)-[2-(7-Fluoro-2-hydroxy-1H-indol-3-yl)indol-3-ylidene]amino] acetate | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_cb7e8c08c693b10a5dba2af9939ef46d.svg) | 7-Fluoro-3-[(3Z)-3-methoxyiminoindol-2-yl]-1H-indol-2-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_ce17364e96dda25fd1db6aa2db160df9.svg) | 7-Bromo-3-[(3Z)-3-methoxyiminoindol-2-yl]-1H-indol-2-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_9b11445945e3bb5b6fec39885146bc4b.svg) | 7-Iodo-3-[(3Z)-3-methoxyiminoindol-2-yl]-1H-indol-2-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_86110ecbf86795d1fddd255ab21816c5.svg) | 3-[(3S)-3-Aminopyrrolidine-1-carbonyl]-5,10-dihydroxy-2-methylnaphtho[2,3-f][1]benzofuran-4,11-dione;methanesulfonic acid | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_8f5820710583b3c9cbd130f10c5d2153.svg) | 1-(3-Chlorophenyl)-3-[5-[2-(thieno[2,3-d]pyrimidin-4-ylamino)ethyl]-2,3-dihydro-1,3-thiazol-2-yl]urea | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_830c2170dfee7f045c3d8420a1443b51.svg) | (2E)-2-[(3,4-Dihydroxyphenyl)methylidene]-1-benzofuran-3-one | IC50 | 4750.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_89623b6920052a05e72d61dcb466f878.svg) | 3-[[4-[6-Bromo-2-(4-methylpiperazin-1-yl)-1H-imidazo[4,5-b]pyridin-7-yl]piperazin-1-yl]methyl]-5-methyl-1,2-oxazole | IC50 | 19.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_04588a23ef4514c75cdc02ecc45743ea.svg) | N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amine | Ki | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_42984ff3447d9d0a9a53124388f0cbfc.svg) | 4-[[(3S,4R)-1-(5-Cyanopyridin-2-yl)-3-fluoropiperidin-4-yl]amino]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_6c34bcbf82f1b210364bfc6af4eddca3.svg) | 2-{3-[3-(Piperidin-4-Yl)propoxy]phenyl}-N-[4-(Pyridin-4-Yl)-1,3-Thiazol-2-Yl]acetamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-c_651380adee49db89525ac807adc94982.svg) | N-(4-Fluorophenyl)-N'-[(3Z)-2-oxo-3-(1H-pyrrol-2-ylmethylidene)-1H-indol-6-yl]propanediamide | IC50 | 67.2 [1] |