![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_2060f6287083a28c9ead968a2460ede5.svg) | Tozasertib | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_2060f6287083a28c9ead968a2460ede5.svg) | Tozasertib | Ki | 0.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 3.67 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_862f3cfaa60202128fbfbc33e055b61e.svg) | Alisertib | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_def2622457c2392ae7d83708b0039226.svg) | 4-[[9-Chloro-7-(2,6-difluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_4fc4352b32d3da424f7de0a0fd6aa1e3.svg) | N-[4-[[6-Methoxy-7-[3-(4-morpholinyl)propoxy]-4-quinazolinyl]amino]phenyl]benzamide | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_84a2f5d5b278f1bed3a9d83403c2d697.svg) | 2-(1,3-Dimethyl-1H-pyrazole-4-yl)-6-chloro-7-[4-(phenylcarbamoyl)phenoxy]-3H-imidazo[4,5-b]pyridine | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_102ec7c5ee0c4ac821e03c1f1a4333ee.svg) | MK-5108 | IC50 | 0.06 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_0bee5512594d9568f74893cb44175367.svg) | 2-({2-[(4-Carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acid | IC50 | 6.1 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_f96a5edb05c83804d0da83e40786432f.svg) | 4-[[6-Chloro-2-(1,3-dimethylpyrazol-4-yl)-1H-imidazo[4,5-b]pyridin-7-yl]oxy]-N-cyclobutylbenzamide | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_83c234bb8d1f466b89c0cd84a644d9f8.svg) | (E)-N-(5-Methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-1-yl)-2-styrylpyrimidin-4-amine | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_9418e91bfb92ccb1c06068bf56f8b8e2.svg) | 2,4-Bisanilinopyrimidine, 10 | IC50 | 3.4 [1], 390.0 [2], 2000.0 [3], 2500.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_d9011c12d7c3d6bcc4e3d1cc48df3c6e.svg) | N~4~-(2-Chlorophenyl)-N~2~-[4-(1h-Tetrazol-5-Yl)phenyl]pyrimidine-2,4-Diamine | IC50 | 3.1 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_c8494007663098abb5d227cb27cc738b.svg) | Sorafenib | IC50 | 3800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_aea8e5cd5eedd851a20871e2fe5ff0da.svg) | Danusertib | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_aea8e5cd5eedd851a20871e2fe5ff0da.svg) | Danusertib | Ki | 2.5 [1], 13.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_bf4bbfed2d9a84ce58724a3f96582d1c.svg) | N-(2,6-Diethylphenyl)-3-[[4-(4-methylpiperazin-1-yl)benzoyl]amino]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazole-5-carboxamide | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_e9c3476c230de7c77add29dc12235adb.svg) | 4-[[2-[4-[2-(4-Acetylpiperazin-1-yl)-2-oxoethyl]anilino]-5-fluoropyrimidin-4-yl]amino]-N-(2-chlorophenyl)benzamide | IC50 | 4.3 [1], 1600.0 [2], 2500.0 [3], 2800.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_3db90beb4f1bfe22d142bb667aa03f48.svg) | 6-[[4-[(Z)-[2-(4-Ethylphenyl)imino-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene]methyl]pyridin-2-yl]amino]pyridine-3-carboxylic acid | IC50 | 1.7 [1], 2.0 [2], 760.0 [3], 1400.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_d29de6ebcabe40c57ebc93753789c45b.svg) | 5-[[4-(2-Chloroanilino)-5-fluoropyrimidin-2-yl]amino]-2-(2H-tetrazol-5-yl)phenol | IC50 | 17.3 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a2841d948c6ad9a30524728b0509b75d.svg) | 4-{[4-(Phenylamino)pyrimidin-2-Yl]amino}benzoic Acid | IC50 | 8.9 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_2af00ba7f2b061e301a1a72866d3a7fb.svg) | 4-({4-[(2-Chlorophenyl)amino]pyrimidin-2-Yl}amino)benzoic Acid | IC50 | 0.74 [1], 2.5 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_594674b17fb97eccb42d35b3e65f7f2b.svg) | 4-({4-[(2-Chlorophenyl)amino]-5-Fluoropyrimidin-2-Yl}amino)benzoic Acid | IC50 | 0.2 [1], 0.8 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_7cc96c149983e405a2f2d0348e089908.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]benzamide | IC50 | 1.0 [1], 30.2 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_f6a52f6f8c2daa1b32c556a67607fa56.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]-N-(2-morpholin-4-ylethyl)benzamide | IC50 | 28.1 [1], 216.0 [2], 1000.0 [3], 5500.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_7c37679fdbefeadb1e0a95ab83833db4.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]-N-[2-(dimethylamino)ethyl]benzamide | IC50 | 28.1 [1], 216.0 [2], 1000.0 [3], 5500.0 [4] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_b9a2f4f57430b9cd003516055c5ddcf3.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]-N-(2-methoxyethyl)benzamide | IC50 | 18.0 [1], 1000.0 [2], 5500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_65cacd8dbf18d21018d8373b0d18d645.svg) | 4-N-(2-Chlorophenyl)-2-N-(4-methylsulfonylphenyl)pyrimidine-2,4-diamine | IC50 | 44.9 [1], 1000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_11dfaaf69310ebf6beb4505e0dd9edb2.svg) | 5-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]-1,3-dihydrobenzimidazol-2-one | IC50 | 316.0 [1], 3000.0 [2], 5500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a95dcbe2f2dae028101844456676338c.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]-2-methoxybenzoic acid | IC50 | 116.5 [1], 3000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_db7cd66d2bb2e93bbc5246d729342daa.svg) | 4-N-(2-Chlorophenyl)-2-N-(4-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | IC50 | 1.0 [1], 27.0 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_6599a78ecb94da62e058f09eb31924e9.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]benzenesulfonamide | IC50 | 1.0 [1], 253.0 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_d050c3a3bc34262d218251cd90fc5a98.svg) | 4-N-(2-Chlorophenyl)-5-fluoro-2-N-(4-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | IC50 | 1.0 [1], 21.4 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a6aad1ecdc828860912a5ba3f2ee83a1.svg) | 4-N-(2-Chlorophenyl)-5-fluoro-2-N-[4-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamine | IC50 | 1.0 [1], 23.2 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_9a31128d659068c00609c2110750c8fa.svg) | 4-[[4-(2-Chloroanilino)pyrimidin-2-yl]amino]-N-(2-hydroxyethyl)benzamide | IC50 | 1.0 [1], 12.3 [2], 1000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_5971f27f0b39700aa4adb9202d4f344e.svg) | 4-[[4-(2-Chloroanilino)-5-fluoropyrimidin-2-yl]amino]benzamide | IC50 | 1.0 [1], 14.4 [2], 300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_096dcab51752a8bdd38cfc6d9d82ccc3.svg) | 4-[[4-(2-Chloroanilino)-5-fluoropyrimidin-2-yl]amino]benzenesulfonamide | IC50 | 21.2 [1], 1000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_0ef2949985eb1f420652843cc4735320.svg) | 4-N-(2-Chlorophenyl)-5-fluoro-2-N-[4-(2H-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamine | IC50 | 2.9 [1], 3000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_7708f9395995c3be752ce2a2478da343.svg) | 5-Chloro-4-N-(2-chlorophenyl)-2-N-[4-(2H-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamine | IC50 | 3.0 [1], 3000.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_4e38800d1c310079b3b3e65c5db78d0d.svg) | Linifanib | IC50 | 760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_899e7233470c1e6b0c695ac9e914d9bb.svg) | 3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea | IC50 | 1259.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_899e7233470c1e6b0c695ac9e914d9bb.svg) | 3-[4-[4-[2-[3-[(Dimethylamino)methyl]phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethylpyrazol-3-yl]phenyl]-1,1-dimethylurea | Ki | 490.0 [1], 492.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_056c9191a034ade62826fb324b220197.svg) | Cct-129202 | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_8e3a7b12efcabb8e696346a7543944c0.svg) | N-(5-Methyl-1H-pyrazol-3-yl)-2-phenylquinazolin-4-amine | IC50 | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_8e3a7b12efcabb8e696346a7543944c0.svg) | N-(5-Methyl-1H-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Ki | 58.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_25447d1e3d43e096411d83a6f2d5a804.svg) | Aurora Kinase Inhibitor III | IC50 | 42.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_5ae8149f1ff59936cf23699cfca9f10b.svg) | Aurora Kinase Inhibitor II | IC50 | 310.0 [1], 393.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_e7638f99a26af4af2719625e6b5039d6.svg) | CID 9916282 | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_ae3cb292e66be9578004d2faaf9b275f.svg) | 8-Anilino-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_b60dbd9c454c8110a1338f2041b0efa3.svg) | 8-Anilino-N,1-dimethyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 312.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_8cf847d7bdf94a72b8c35ca7d8e5c6f4.svg) | 4-(4-Methylpiperazin-1-yl)-N-[5-(2-phenylacetyl)-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-3-yl]benzamide | IC50 | 130.0 [1], 140.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_e65399444f3639d55c4b15703501c828.svg) | 8-Anilino-1-methyl-N-phenyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_ae8e8ef09ff81545fc80ae0fc208fb79.svg) | N-[5-[[6-Methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]amino]pyrimidin-2-yl]benzamide | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_03ec9c8cc776552156467ae00eaba53c.svg) | 1-{5-[2-(Thieno[3,2-D]pyrimidin-4-Ylamino)ethyl]-1,3-Thiazol-2-Yl}-3-[3-(Trifluoromethyl)phenyl]urea | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_45dd68e411be9ba0d2534c497f840315.svg) | 1-Phenyl-3-[5-(2-{thieno[3,2-d]pyrimidin-4-ylamino}ethyl)-1,3-thiazol-2-yl]urea | IC50 | 52.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_77437fd353bcc1f8cb6daf81b795ba65.svg) | 4-(6-Chloro-1H-imidazo[4,5-b]pyridin-2-yl)-N,N-dimethyl-aniline | IC50 | 570.0 [1], 4970.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_2da32a891f5c71bb743df161b283d30a.svg) | 6-Chloro-7-[4-[(4-chlorophenyl)methyl]piperazin-1-yl]-2-(1,3-dimethylpyrazol-4-yl)-1H-imidazo[4,5-b]pyridine | IC50 | 30.0 [1], 38.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_95b1b6a854f1ad22b69c67dae323c503.svg) | 4-(6,7-Dimethoxy-9H-pyrimido[4,5-b]indol-4-yl)-N-[4-(pyrimidin-2-ylsulfamoyl)phenyl]piperazine-1-carbothioamide | IC50 | 94.0 [1], 900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_3df995f8d535df6b573fa7c0acafe8fc.svg) | Unii-LM7NL857V1 | IC50 | 4.0 [1], 80.0 [2], 160.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_32e8b0bc3d6e2ad4f5cb769f6f564a12.svg) | N-(2-Chlorophenyl)-4-[[5-fluoro-2-(4-hydroxyanilino)pyrimidin-4-yl]amino]benzamide | IC50 | 10.0 [1], 1600.0 [2], 5000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_81737edee35af2ee5d9b4f240bd72f7a.svg) | 4-({4-[(2-Fluorophenyl)amino]pyrimidin-2-Yl}amino)benzoic Acid | IC50 | 3.7 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_300af1465c51e5afb7c8315bce7f83e6.svg) | 4-{[4-(Biphenyl-2-Ylamino)pyrimidin-2-Yl]amino}benzoic Acid | IC50 | 149.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_913dddb57182590b5a9c322c43f2341e.svg) | 4-[(4-{[2-(Trifluoromethyl)phenyl]amino}pyrimidin-2-Yl)amino]benzoic Acid | IC50 | 35.0 [1], 35.1 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_e9c176e5a070fe07c7e1c7e7c7c24556.svg) | 4-({4-[(2-Bromophenyl)amino]pyrimidin-2-Yl}amino)benzoic Acid | IC50 | 2.1 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a9557c7092aadbddb0143b2589e60b04.svg) | 4-({4-[(2-Cyanophenyl)amino]pyrimidin-2-Yl}amino)benzoic Acid | IC50 | 43.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_99c9973f1a1eb0e0a8264b8e43a031c3.svg) | (3S,6S,9R,14R,17S,20S,23S,26S)-9-Amino-N-(2-amino-2-oxoethyl)-3-[3-(diaminomethylideneamino)propyl]-6-[(1R)-1-hydroxyethyl]-20,23-bis(1H-indol-3-ylmethyl)-17-(2-methylpropyl)-2,5,8,16,19,22,25-heptaoxo-11,12-dithia-1,4,7,15,18,21,24-heptazabicyclo[24.3.0]nonacosane-14-carboxamide | IC50 | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_99c9973f1a1eb0e0a8264b8e43a031c3.svg) | (3S,6S,9R,14R,17S,20S,23S,26S)-9-Amino-N-(2-amino-2-oxoethyl)-3-[3-(diaminomethylideneamino)propyl]-6-[(1R)-1-hydroxyethyl]-20,23-bis(1H-indol-3-ylmethyl)-17-(2-methylpropyl)-2,5,8,16,19,22,25-heptaoxo-11,12-dithia-1,4,7,15,18,21,24-heptazabicyclo[24.3.0]nonacosane-14-carboxamide | Ki | 27200.0 [1], 31500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_15ac436087bff5fd4c0e6f2c7a3173eb.svg) | 2-[[2-(4-Carboxyanilino)-5-methylpyrimidin-4-yl]amino]benzoic acid | IC50 | 145.0 [1], 281.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_818e20960290ff06e97b77b6f2196c9f.svg) | Barasertib | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_818e20960290ff06e97b77b6f2196c9f.svg) | Barasertib | Ki | 1368.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_1575317431cf6bb218d1789cccd6e0ea.svg) | Quizartinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_2adbc4a307d22bed17e0f710542542e9.svg) | Entrectinib | IC50 | 215.0 [1], 338.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_fa37ae125bcd4e6df1af4be57fbea491.svg) | 1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)urea | IC50 | 3.0 [1], 3.3 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_bd1c4c226d09bccaf8e1c9ed8e2ba78a.svg) | Azd-1152hqpa | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_bd1c4c226d09bccaf8e1c9ed8e2ba78a.svg) | Azd-1152hqpa | Ki | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_ad2e213c6bc5eb972596bba5a265d460.svg) | 1-(3-Chlorophenyl)-3-{5-[2-(Thieno[3,2-D]pyrimidin-4-Ylamino)ethyl]-1,3-Thiazol-2-Yl}urea | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a2d32a1f7c79660a88d646bbda5ee232.svg) | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | IC50 | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a2d32a1f7c79660a88d646bbda5ee232.svg) | 4-Methyl-5-(2-((4-morpholinophenyl)amino)-pyrimidin-4-yl)thiazol-2-amine | Ki | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_4ba3d76a313e9fc701d70ea02c97c366.svg) | 2-N,4-N-Diphenylpyrimidine-2,4-diamine | IC50 | 423.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_96dd1c245db8fda5ee6b165b0c628ae0.svg) | CID 44556162 | IC50 | 10000.0 [1], 30000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_580efe2e66439369c377fd174fde96fb.svg) | Ilorasertib | IC50 | 12.0 [1], 4743.1 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_ac9e30b723e2c9bf1debc2a45966acbb.svg) | 3-(1H-Indol-3-yl)-4-(3,4,5-trimethoxyphenyl)pyrrole-2,5-dione | IC50 | 5400.0 [1], 9900.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_9c1d0d8977acecc130ed64ff3fc51acc.svg) | PF-03814735 | IC50 | 0.8 [1], 20.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_956156183a357df1d821ce052bc65dc0.svg) | 2-[4-(Dimethylamino)phenyl]-1H-imidazo[4,5-b]pyridine | IC50 | 4300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_e2209e7758c6438055a026dffd3ba884.svg) | Chembl272125 | IC50 | 560.0 [1], 15100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_76c6c2c22bae9bce4fe3eb463989d0c9.svg) | 2-[(5,6-Diphenylfuro[2,3-D]pyrimidin-4-YL)amino]ethanol | IC50 | 273.0 [1], 309.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_8adeb6b2698b431f81231231182e167f.svg) | 2-(4-Methoxyphenyl)-1H-imidazo[4,5-b]pyridine | IC50 | 6600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_c6a4dbbed41189365b44881da3e90691.svg) | N-[5-[(2S)-2-Methoxy-2-phenylacetyl]-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-3-yl]-4-(4-methylpiperazin-1-yl)benzamide | IC50 | 354.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_6ae0eaede4a2033a87c45ee2183b55cc.svg) | 2-(1H-Pyrazol-3-yl)-1H-benzimidazole | IC50 | 910.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a9ab9fc62402963601c82ac3738f0779.svg) | N-[4-[4-(4-Methylpiperazin-1-yl)-6-[(5-methyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]sulfanylphenyl]propanamide | IC50 | 1.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_a9ab9fc62402963601c82ac3738f0779.svg) | N-[4-[4-(4-Methylpiperazin-1-yl)-6-[(5-methyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]sulfanylphenyl]propanamide | Ki | 1.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_f4d7f253fba38490b7fb35e70010bf9b.svg) | 2-(2-Methoxyphenyl)-1H-imidazo[4,5-b]pyridine | IC50 | 29000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_7a4254b2b4cd2e9937dbe5863115462e.svg) | 3-(4'-Hydroxybiphenyl-4-Yl)-N-(4-Hydroxycyclohexyl)-1,4-Dihydroindeno[1,2-C]pyrazole-6-Carboxamide | IC50 | 8090.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_2e8153acbaf4777559825f69210e1632.svg) | (7S)-2-(2-Aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_b301e590b6fa2ee3f8bfd342e6c37901.svg) | 2-{[5-Fluoro-2-(phenylamino)pyrimidin-4-yl]amino}benzoic acid | IC50 | 11.3 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_995601d80f8b663e21c02593d674ff7b.svg) | 2-[[4-(3,4-Dimethoxyanilino)-6-(quinolin-6-ylamino)-1,3,5-triazin-2-yl]amino]-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)propanamide | IC50 | 0.27 [1], 270.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_66ee537084332a28fb4fd921d6adf367.svg) | CID 56673651 | IC50 | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_342b866f5828340558231cb6af2ee22a.svg) | N-(4-(4-(5-Methyl-1H-pyrazol-3-ylamino)-6-morpholinopyrimidin-2-ylthio)phenyl)propionamide | IC50 | 1.7 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_342b866f5828340558231cb6af2ee22a.svg) | N-(4-(4-(5-Methyl-1H-pyrazol-3-ylamino)-6-morpholinopyrimidin-2-ylthio)phenyl)propionamide | Ki | 1.7 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-aurora-a_ff35a372ba5e94efa622cf6bcdb424b0.svg) | 4-Tert-butyl-N-[5-(2-phenylacetyl)-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-3-yl]benzamide | IC50 | 130.0 [1] |