![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 0.64 [1], 5.0 [2], 10.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_08708cd7ba9d3e1d8e003535055a8693.svg) | Akt inhibitor VIII | IC50 | 2119.0 [1], 2200.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_67f4e732a49bf39a183fb443d695bf12.svg) | Gsk-690693 | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_67f4e732a49bf39a183fb443d695bf12.svg) | Gsk-690693 | Ki | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_7489af297ca5d99d886f106758e75d74.svg) | 2-[4-(3-Phenylquinoxalin-2-yl)phenyl]propan-2-amine | IC50 | 50000.0 [1], 250000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_6b7ed5d4bde8a2dd13f619c48594a177.svg) | Merck-22-6 | IC50 | 7200.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_37db551c0860118de4481a6c244df05d.svg) | (2S)-1-(1H-Indol-3-yl)-3-(5-isoquinolin-6-ylpyridin-3-yl)oxy-propan-2-amine | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_a818b5189c24e9661b349c41464a5f0e.svg) | 1-(1-{[4-(3-Phenylquinoxalin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one | IC50 | 27000.0 [1], 50000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_d2497ae1855cd4d782afa7fbefc515ee.svg) | 3-[4-[[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-2-phenylquinoxaline-6-carboxylic acid | IC50 | 3200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_25774502353a4c4c2828afb710c6fc93.svg) | 2-[4-[[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-3-phenylquinoxaline-6-carboxylic acid | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_207042f7b18553f1c569f31eac2549a5.svg) | (2S,3S,4R,5R)-N-[6-[[(2R)-6-Amino-1-[[6-[[(2R)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-6-oxohexyl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolane-2-carboxamide | IC50 | 774.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_9d38a171c31a3d0ddba7416e6ed4a947.svg) | (1S)-2-(1H-Indol-3-YL)-1-[({5-[(E)-2-pyridin-4-ylvinyl]pyridin-3-YL}oxy)methyl]ethylamine | IC50 | 354.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_89f61185eee292e1e6d2c25ed4035afc.svg) | 3-[1-[[4-[3-Phenyl-7-(2H-tetrazol-5-yl)quinoxalin-2-yl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 1613.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_034fc7c19a4d28443b7b19a9dd7db8e2.svg) | 3-[1-[[4-[3-Phenyl-6-(2H-tetrazol-5-yl)quinoxalin-2-yl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 1228.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_27557c2f98908fe2029875dee5f2c27d.svg) | 4-[1-Ethyl-7-(piperidin-4-yloxy)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine | IC50 | 398.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_59ef2d062dc026381e0e01653a1e9675.svg) | N-[2-(Diethylamino)ethyl]-2-[4-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-3-phenylquinoxaline-6-carboxamide | IC50 | 7400.0 [1], 8000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_3a709edc2c27733406eb7da0d246c509.svg) | N-[(2S)-1-Amino-3-(2,4-dichlorophenyl)propan-2-yl]-5-[2-(methylamino)pyrimidin-4-yl]thiophene-2-carboxamide | IC50 | 2.6 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_8ef35a49211de1090d3d853bca1ba5f1.svg) | N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_324a735f3dfd55339b078f5bfe295a89.svg) | MK-2206 | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_3013791590a95a7fa1113a8967c19298.svg) | Neflamapimod | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_b3c4880e77322182637a22879b9e24d9.svg) | Capivasertib | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_2049621c606555281145c6a04f93a189.svg) | 4-Amino-N-[1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_c8017cad0338655ba40f56b179d4c498.svg) | (2s)-1-(1h-Indol-3-Yl)-3-{[5-(3-Methyl-1h-Indazol-5-Yl)pyridin-3-Yl]oxy}propan-2-Amine | IC50 | 51.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_4f3a477c8387451989e5d1602a9be1ec.svg) | Ipatasertib | IC50 | 8.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_5547e46f002aaa1621f16458dc38d88f.svg) | Afuresertib | IC50 | 1.58 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_3ac91c26cb3202821ba09ba5b9d46a48.svg) | Aminofurazanyl-azabenzimidazole 6n | IC50 | 1510.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_9ed259c362899d08e63c398effcfd25b.svg) | 4-[1-Ethyl-7-[(piperidin-4-ylamino)methyl]imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine | IC50 | 646.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_478f8c74275fce83224a96edad0f0b1f.svg) | JNK Inhibitor VIII | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_302526c024c71396d28c3ce026dc5f5f.svg) | (S)-1-(4-(1H-Pyrazol-4-yl)phenyl)-2-amino-1-(4-chlorophenyl)ethanol | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_d44bb541aaceb7d87194194110f1e1e1.svg) | CID 11634725 | Ki | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_b8cdecfced6d89a62d42ca41bd225e1d.svg) | H-89 Dihydrochloride | IC50 | 662.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_229be97168f5a1e19a21ea31c162ddf6.svg) | 3-(4-{4-Aminofuro[2,3-d]pyrimidin-5-yl}phenyl)-1-[2-fluoro-5-(trifluoromethyl)phenyl]urea | IC50 | 17378.01 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_601e453d7a089204e0a249b45693b4d5.svg) | 2-(4-Fluorophenyl)-3-(4-pyridinyl)pyrazolo[1,5-a]pyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_bc77633739634ca96b0eec21cde6deed.svg) | 3-[1-[[4-(5-Methyl-6-oxo-2-phenyl-1H-pyrazin-3-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_22bd102537d7b56bbf2c70ad165bf06a.svg) | 3-(4-Amino-3-(3-chloro-4-fluorophenyl)thieno[3,2-c]pyridin-7-yl)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_c788cb71f5b83be51026b4415777f07f.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-6-(pyrrolidin-1-ylmethyl)imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 22.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_67f0ff5bd04e3d7a478d5957f7a69b75.svg) | 2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-N-[2-(methylamino)ethyl]imidazo[4,5-c]pyridine-7-carboxamide | IC50 | 1410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_d4e3e73d15905aa05522ff356e411d48.svg) | 4-[1-Ethyl-7-(piperazin-1-ylcarbonyl)-1H-imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine | IC50 | 1549.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_c4efceda17e53de30b363a8b6106fac2.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamide | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_4c2c70178609eb610c2ed8f1c8904f26.svg) | [2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethylimidazo[4,5-c]pyridin-7-yl]-[(3S)-3-aminopyrrolidin-1-yl]methanone | IC50 | 1290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_dbc94bb504996085040e4d04c5df6c07.svg) | Akt inhibitor | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_bd55926c7b3558be92fcb8361c526820.svg) | 3-(3-Iodobenzyl)-1-tert-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 7157.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_b2283fe1e6c3f6a8da3854a28b969289.svg) | (2s)-1-{[6-Furan-3-Yl-5-(3-Methyl-2h-Indazol-5-Yl)pyridin-3-Yl]oxy}-3-(1h-Indol-3-Yl)propan-2-Amine | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_bdae19e34d614a34fa53af1ff2fb0dc4.svg) | N-[(2S)-1-Amino-3-(3,4-difluorophenyl)propan-2-yl]-5-chloro-4-(4-chloro-2-methylpyrazol-3-yl)thiophene-2-carboxamide | IC50 | 7.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_f36517eb495346665a3f4ffc2fe37895.svg) | 3-[1-[[4-(6-Oxo-2-phenyl-1H-pyrazin-3-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_e21e6973878706c2852ef43223046095.svg) | 3-[1-[[4-[5-(2-Methylpropyl)-6-oxo-3-phenyl-1H-pyrazin-2-yl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 21870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_0afde03be452af9a350e0d5b5b7da1cf.svg) | 3-[1-[[4-(6-Oxo-3-phenyl-1H-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_feb99200dbbf837d73959ae2cee6f935.svg) | 6-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]-2-chloropyridin-3-yl}isoquinoline | IC50 | 73.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_98723df6e7ca4ea1a41dc0b50c67865b.svg) | 3-[1-[[4-(5-Methyl-6-oxo-3-phenyl-1H-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 33100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_e107dc426fee102f1e388322c53e206c.svg) | 3-[1-[[4-[5-(2-Methylpropyl)-6-oxo-2-phenyl-1H-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_62bcbf995bfc1d6be18aa9eeb3cf42b9.svg) | 3-[1-[[4-(7-Phenyl-1H-pyrazolo[3,4-g]quinoxalin-6-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_0731e513dda8b4631f904dc8f0082e8c.svg) | 7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrile | Ki | 4890.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_1fe60e6d13674f8cf1dfc82fac3410b2.svg) | 7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_029f5b4cad89a2c59efa869fd9853874.svg) | N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_c2aa7e0fb640ea7529d7330460976868.svg) | N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamide | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_98598461b658b3f77425e67c797f8e2d.svg) | N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_a3bd9a5a28d4f4d2890ccf5cdf08d883.svg) | N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamide | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_cde4e83180955e4849d8daba0837480d.svg) | N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamide | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_444db87f8c2457450c5ba08be58c9a25.svg) | N-Methyl-6-phenyl-7-[4-[[4-(3-pyridin-2-yl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl]phenyl]pyrido[2,3-d]pyrimidin-2-amine | IC50 | 2474.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_fa8a748abfe5f3e63aba0da3b4b9b9ee.svg) | 4-Amino-N-(4-chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | IC50 | 57.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_152b6741b067e1e606c6d7ded30efa5e.svg) | 6-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}isoquinolin-3-amine | IC50 | 76.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_aeca0c938bd9ec574de75fc664797a90.svg) | 3-[1-[[4-[5-[(4-Hydroxyphenyl)methyl]-6-oxo-2-phenyl-1H-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_26b79855acfaf43486f6cc1e9ddde256.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[[(3R)-piperidin-3-yl]methoxy]imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_4b806c10a2e22c1d6dbf620f3d7721c4.svg) | (2S,3S,4R,5R)-N-[6-[[(2R)-6-Amino-1-[[6-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-6-oxohexyl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolane-2-carboxamide | IC50 | 14.6 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_66548acb2d44e83d2ca79fa99ad169ca.svg) | (S)-1-(5-(3-Methyl-7-propyl-1H-indazol-5-yl)pyridin-3-yloxy)-3-(1H-indol-3-yl)propan-2-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_2861b3ce0b87adf7f4bbd001d31f6700.svg) | (2S)-1-[6-(Furan-3-yl)-5-(3-methyl-2H-pyrazolo[3,4-b]pyrazin-5-yl)pyridin-3-yl]oxy-3-(1H-indol-3-yl)propan-2-amine | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_b80728998e0b173ed97842a79c1db051.svg) | 5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_a4dbb1e5595d742f8f809304f788246f.svg) | N-[6-[[(2R)-6-Amino-1-[[6-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-6-oxohexyl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]-5-(2-aminopyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_d177c352a8a90316beccdf76166341e8.svg) | N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_eda1570f6e608eea37da447234534ac5.svg) | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_ef431bf27ff7842bbb4caafd947b43c7.svg) | Tilfrinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_5b7a4e9c52ae12a8e6cf55da8661f320.svg) | 3-[1-[[4-(5-Butan-2-yl-6-oxo-2-phenyl-1H-pyrazin-3-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_cffe6067e6b3631ffc9ef0a866dbf46b.svg) | 3-[1-[[4-(5-Butan-2-yl-6-oxo-3-phenyl-1H-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_6c792bb84322ebc0685ceb9aac9f9d21.svg) | (R)-2-Amino-3-(4-chlorophenyl)-1-(4-(quinazolin-4-yl)piperazin-1-yl)propan-1-one | IC50 | 179.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_0920e6c896cd6c50407213a99d87f364.svg) | 4-[1-Ethyl-7-(piperidin-4-ylmethoxy)-1H-imidazo[4,5-c]pyridin-2-yl]-furazan-3-ylamine | IC50 | 380.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_20887592341bbe8a142e214d31f207ea.svg) | N-(4-Fluorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_fd22bf7632b85ee69bb7214183437e9a.svg) | N-(2,4-Dichlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_65873f674fd6cfcf9e4db049dac35282.svg) | N-(2,4-Dichlorophenethyl)-5-(2-(ethylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_6a6aa43ed6c7f59fde44a1b1688317bd.svg) | 5-[2-(Methylamino)pyrimidin-4-yl]-N-[2-(4-sulfamoylphenyl)ethyl]thiophene-2-carboxamide | IC50 | 19000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_6d5b40f7023a875b90a37f38a380a760.svg) | N-(4-Fluorobenzyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 4700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_8406ea63473c57dc0e66b721abc2235b.svg) | N-(3-Chlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 5400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_7b4cf1a6b44949dbdc94a54842388703.svg) | 5-(2-(Methylamino)pyrimidin-4-yl)-N-phenethylthiophene-2-carboxamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_a25c54038759864d0e01aee35def46d5.svg) | N-(2-Chlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_065f5b794815e1be2c40409f7bd82ec6.svg) | N-(2,4-Dichlorophenethyl)-5-(2-aminopyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 610.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_c5e657867262d8c524cb6085509d17f6.svg) | N-[(2S)-1-(2,4-Dichlorophenyl)-3-hydroxypropan-2-yl]-5-[2-(methylamino)pyrimidin-4-yl]thiophene-2-carboxamide | IC50 | 280.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_79be4e785f7f3cd85cd1e01131c4adbf.svg) | N-(4-Chlorophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_48949b4f1b828cb75b5835ab1e843ca5.svg) | N-(3-(4-Fluorophenyl)propyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 18000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_629b3ccaa97dd2a2e1b232faf4ff8293.svg) | N-(4-Bromophenethyl)-5-(2-(methylamino)pyrimidin-4-yl)thiophene-2-carboxamide | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_e7c828047235bb3390e5e95ba5a3070b.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-6-[(2R)-2-amino-3-phenylpropoxy]-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt3_655599d0ad37639cd9b6c6bd2931936c.svg) | 4-[6-(Aminomethyl)-2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 70.0 [1] |