![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_08708cd7ba9d3e1d8e003535055a8693.svg) | Akt inhibitor VIII | IC50 | 58.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_37db551c0860118de4481a6c244df05d.svg) | (2S)-1-(1H-Indol-3-yl)-3-(5-isoquinolin-6-ylpyridin-3-yl)oxy-propan-2-amine | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_37db551c0860118de4481a6c244df05d.svg) | (2S)-1-(1H-Indol-3-yl)-3-(5-isoquinolin-6-ylpyridin-3-yl)oxy-propan-2-amine | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_67f4e732a49bf39a183fb443d695bf12.svg) | Gsk-690693 | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_67f4e732a49bf39a183fb443d695bf12.svg) | Gsk-690693 | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_6812a0dc7e759e339be173c8f272f1fd.svg) | 2-[4-[2-(2-Aminopyridin-3-yl)imidazo[4,5-b]pyridin-3-yl]phenyl]-N-phenylacetamide | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_56b551cfdb9317e13443c38423b1a446.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-6-cyclopentylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_8ef35a49211de1090d3d853bca1ba5f1.svg) | N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide | IC50 | 1800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_8ef35a49211de1090d3d853bca1ba5f1.svg) | N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide | Ki | 4500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_73575945a91f3d74ccca2eda2876f266.svg) | N-[[4-[5-(3-Acetamidophenyl)-2-(2-aminopyridin-3-yl)imidazo[4,5-b]pyridin-3-yl]phenyl]methyl]-3-fluorobenzamide | IC50 | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_a03b2bc5396480aff1ed022e73b139f2.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)imidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_1d843fa6553565b08ddc6e2696b75fe3.svg) | 2-[4-[5-(3-Acetamidophenyl)-2-(2-aminopyridin-3-yl)imidazo[4,5-b]pyridin-3-yl]phenyl]-N-phenylacetamide | IC50 | 49.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_d1328e0ad85c0aa0559c7383608d5b30.svg) | 2-[4-[2-(2-Aminopyridin-3-yl)-5-pyridin-3-ylimidazo[4,5-b]pyridin-3-yl]phenyl]-N-phenylacetamide | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_09969bd8aeaf50265ba6e1f7bb8fa890.svg) | N-[[4-[5-(3-Acetamidophenyl)-2-(2-aminopyridin-3-yl)imidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 140.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_e107b3835b19fcae47df4aed6fcd26c3.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-5-pyridin-3-ylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_a79dfc67e8c794dba6d33310d5f1f81c.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-6-pyridin-3-ylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 91.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_f24cb1f8b448a380aee42d3c31b0276f.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-6-bromoimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_cfbd925858204740376381e4aa1e2b0d.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-5-phenylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_bce0ce7b059a710af3b92d3d65e9b208.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-6-phenylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]benzamide | IC50 | 680.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_7d242a0f8ce50bcdc7b483c1d0e681f2.svg) | 2-[4-[5-(3-Acetamidophenyl)-2-(2-aminopyridin-3-yl)imidazo[4,5-b]pyridin-3-yl]phenyl]-N-(3-fluorophenyl)acetamide | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_2c45a906f8ed72199fea3852831c207b.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-5-pyridin-3-ylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]-3-fluorobenzamide | IC50 | 340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_ee88dd5df1db071a033c623dca81a680.svg) | N-[[4-[2-(2-Aminopyridin-3-yl)-6-pyridin-3-ylimidazo[4,5-b]pyridin-3-yl]phenyl]methyl]-3-fluorobenzamide | IC50 | 54.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_79ccba98dd462b1631c9db41481af774.svg) | (2S)-1-N-(5-Isoquinolin-6-yl-1,3,4-thiadiazol-2-yl)-3-[4-(trifluoromethyl)phenyl]propane-1,2-diamine | IC50 | 247.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_c8017cad0338655ba40f56b179d4c498.svg) | (2s)-1-(1h-Indol-3-Yl)-3-{[5-(3-Methyl-1h-Indazol-5-Yl)pyridin-3-Yl]oxy}propan-2-Amine | IC50 | 0.16 [1], 2.5 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_c8017cad0338655ba40f56b179d4c498.svg) | (2s)-1-(1h-Indol-3-Yl)-3-{[5-(3-Methyl-1h-Indazol-5-Yl)pyridin-3-Yl]oxy}propan-2-Amine | Ki | 0.16 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_87c771daffed6101d1b561019d6c2997.svg) | Medermycin | IC50 | 149.0 [1], 30400.0 [2], 38500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_7489af297ca5d99d886f106758e75d74.svg) | 2-[4-(3-Phenylquinoxalin-2-yl)phenyl]propan-2-amine | IC50 | 3400.0 [1], 250000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_9d38a171c31a3d0ddba7416e6ed4a947.svg) | (1S)-2-(1H-Indol-3-YL)-1-[({5-[(E)-2-pyridin-4-ylvinyl]pyridin-3-YL}oxy)methyl]ethylamine | IC50 | 14.0 [1], 360.0 [2], 3000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_534d0285debd563abec3aa43bce75378.svg) | A-674563 | IC50 | 14.0 [1], 125.0 [2], 100000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_534d0285debd563abec3aa43bce75378.svg) | A-674563 | Ki | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_6b7ed5d4bde8a2dd13f619c48594a177.svg) | Merck-22-6 | IC50 | 138.0 [1], 253.0 [2], 527.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_bc77633739634ca96b0eec21cde6deed.svg) | 3-[1-[[4-(5-Methyl-6-oxo-2-phenyl-1H-pyrazin-3-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_bc77633739634ca96b0eec21cde6deed.svg) | 3-[1-[[4-(5-Methyl-6-oxo-2-phenyl-1H-pyrazin-3-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | Ki | 760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_a818b5189c24e9661b349c41464a5f0e.svg) | 1-(1-{[4-(3-Phenylquinoxalin-2-yl)phenyl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one | IC50 | 290.0 [1], 295.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_e05034746040acbbed6c9ec341699487.svg) | 4-Amino-n-(1,3,4-thiadiazol-2-yl)benzenesulfonamide | IC50 | 20000.0 [1], 25000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_e05034746040acbbed6c9ec341699487.svg) | 4-Amino-n-(1,3,4-thiadiazol-2-yl)benzenesulfonamide | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_feb99200dbbf837d73959ae2cee6f935.svg) | 6-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]-2-chloropyridin-3-yl}isoquinoline | IC50 | 1.8 [1], 3000.0 [2], 5700.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_84d4445f65950334b0170a4ef5cacdef.svg) | 7-[4-[[4-(4-Aminopyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]methyl]phenyl]-6-phenylpyrido[2,3-d]pyrimidin-4-amine | IC50 | 14.0 [1], 295.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_984f82656ba80cc9ab3095abf59c5db4.svg) | N,N-Dimethyl-2-[4-[6-phenyl-7-[4-[[4-(3-pyridin-2-yl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl]phenyl]pyrido[2,3-d]pyrimidin-2-yl]piperazin-1-yl]ethanamine | IC50 | 4.0 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_444db87f8c2457450c5ba08be58c9a25.svg) | N-Methyl-6-phenyl-7-[4-[[4-(3-pyridin-2-yl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl]phenyl]pyrido[2,3-d]pyrimidin-2-amine | IC50 | 6.0 [1], 20.0 [2], 20.3 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_468e6ed5526669dd854c333ca0134c60.svg) | 7-[4-[[4-(6-Fluoro-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]phenyl]-6-phenylpyrido[2,3-d]pyrimidin-4-amine | IC50 | 18.0 [1], 277.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_152b6741b067e1e606c6d7ded30efa5e.svg) | 6-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}isoquinolin-3-amine | IC50 | 3.4 [1], 200.0 [2], 930.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_160a29879cd73d7dd09660bb28cdf816.svg) | Pictilisib | IC50 | 28.0 [1], 37.0 [2], 46.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_efa546891924580a73b05a0325d621e2.svg) | Frenolicin B | IC50 | 198.0 [1], 313.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_9fcfedb7cdf0eaede0e004d06409a22a.svg) | 4-Dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide | IC50 | 6300.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_9fcfedb7cdf0eaede0e004d06409a22a.svg) | 4-Dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide | Ki | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_302526c024c71396d28c3ce026dc5f5f.svg) | (S)-1-(4-(1H-Pyrazol-4-yl)phenyl)-2-amino-1-(4-chlorophenyl)ethanol | IC50 | 10.0 [1], 38.0 [2], 1100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_6fe0ae1f24c5b4eafe04bc46354e68fd.svg) | (11R,15R,17R)-17-Methyl-12,16-dioxatetracyclo[8.7.0.03,8.011,15]heptadeca-1(10),3,5,7-tetraene-2,9,13-trione | IC50 | 150.0 [1], 280.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_d2497ae1855cd4d782afa7fbefc515ee.svg) | 3-[4-[[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-2-phenylquinoxaline-6-carboxylic acid | IC50 | 166.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_924b685d38b27ec843b31a549e18baf2.svg) | 3-[(2S)-2-Amino-3-phenylpropoxy]-5-[(E)-2-(pyridin-4-yl)ethenyl]pyridine | IC50 | 690.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_25774502353a4c4c2828afb710c6fc93.svg) | 2-[4-[[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]phenyl]-3-phenylquinoxaline-6-carboxylic acid | IC50 | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_b2283fe1e6c3f6a8da3854a28b969289.svg) | (2s)-1-{[6-Furan-3-Yl-5-(3-Methyl-2h-Indazol-5-Yl)pyridin-3-Yl]oxy}-3-(1h-Indol-3-Yl)propan-2-Amine | IC50 | 1.0 [1], 500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_b011a91764627c80ffc0af9c6c144191.svg) | (2R)-2-Amino-3-(4-fluorophenyl)-1-[4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-one | IC50 | 3.0 [1], 160.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_29d1b4499723558170a904c2722059ae.svg) | 1-(2-Aminophenyl)-3-[[4-(2-methylsulfanyl-6-phenylpyrido[2,3-d]pyrimidin-7-yl)phenyl]methylamino]propan-1-one | IC50 | 15.0 [1], 78.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_069e9005245eb47a0f931083a057c4e1.svg) | 4-Spiro[2H-indole-3,4'-piperidine]-1-yl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | IC50 | 2.0 [1], 2.4 [2], 50.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_1434950707716d941f02c36e9f1dfe88.svg) | 9-Phenyl-8-[4-[[4-(3-pyridin-2-yl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl]phenyl]-[1,2,4]triazolo[3,4-f][1,6]naphthyridine | IC50 | 4.0 [1], 5.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_f86ae67818aea5f288640aff15868aa1.svg) | 6-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-3-fluoroisoquinoline | IC50 | 3.5 [1], 2300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_26b79855acfaf43486f6cc1e9ddde256.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[[(3R)-piperidin-3-yl]methoxy]imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 2.0 [1], 3.0 [2], 400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_eadb57fc4a7212f4b18b1eb5a4c39c2c.svg) | N-(4-(N-1,3,4-Thiadiazol-2-ylsulfamoyl)phenyl)decanamide | IC50 | 10000.0 [1], 15000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_eadb57fc4a7212f4b18b1eb5a4c39c2c.svg) | N-(4-(N-1,3,4-Thiadiazol-2-ylsulfamoyl)phenyl)decanamide | Ki | 21800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_2823a4294217c6f546ed47edeb7bb50a.svg) | N-(4-(N-1,3,4-Thiadiazol-2-ylsulfamoyl)phenyl)-2-(2-(2-methoxyethoxy)ethoxy)acetamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_2823a4294217c6f546ed47edeb7bb50a.svg) | N-(4-(N-1,3,4-Thiadiazol-2-ylsulfamoyl)phenyl)-2-(2-(2-methoxyethoxy)ethoxy)acetamide | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_03add6debfeca27fc25a13bf4d60e500.svg) | N-[5-Chloro-3-[4-(3-ethyl-2H-pyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]-2-methylphenyl]-N',N'-dimethylethane-1,2-diamine | IC50 | 371.0 [1], 9026.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_835873ee72f71781cc2e627e5a2365e7.svg) | N-[3-[4-(3-Bromo-2H-pyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]-5-chloro-2-methylphenyl]-N',N'-dimethylethane-1,2-diamine | IC50 | 53.0 [1], 4285.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_cf01f7adaf9e516ec2bed2f5c18024d8.svg) | N-(4-(N-1,3,4-Thiadiazol-2-ylsulfamoyl)phenyl)acetamide | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_cf01f7adaf9e516ec2bed2f5c18024d8.svg) | N-(4-(N-1,3,4-Thiadiazol-2-ylsulfamoyl)phenyl)acetamide | Ki | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_4bda03015536fc7046af2c82f82108e6.svg) | (2S)-1-N-[5-(3-Methyl-2H-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-[4-(trifluoromethyl)phenyl]propane-1,2-diamine | IC50 | 5.5 [1], 333.0 [2], 357.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_79901e7ea670d630405e5cef9aab7f8b.svg) | (2S)-1-N-[5-(1H-Indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-[4-(trifluoromethyl)phenyl]propane-1,2-diamine | IC50 | 6.0 [1], 154.0 [2], 444.0 [3] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_324a735f3dfd55339b078f5bfe295a89.svg) | MK-2206 | IC50 | 8.0 [1], 10.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_b3c4880e77322182637a22879b9e24d9.svg) | Capivasertib | IC50 | 3.0 [1], 34.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_4f3a477c8387451989e5d1602a9be1ec.svg) | Ipatasertib | IC50 | 5.0 [1], 157.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_fb5fc35767dd7c4ce20f234cb54827a4.svg) | 4-(4-Chlorobenzyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-amine | IC50 | 0.66 [1], 3.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_5f625f186b4b50ea97c3b1508240317a.svg) | Uprosertib | IC50 | 2.0 [1], 18.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_70587fa0659be3f28c8a2050d45e9fc9.svg) | N-[6-[6-Chloro-5-[[(4-fluorophenyl)sulfonyl]amino]-3-pyridinyl]-1,3-benzothiazol-2-yl]acetamide | IC50 | 6.3 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_1dabac911faf494befb86a22bfcb361a.svg) | (E)-3-(1H-Benzo[d]imidazol-2-yl)-1-(6-chloro-2-hydroxy-4-phenylquinolin-3-yl)prop-2-en-1-one | IC50 | 4500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_1dabac911faf494befb86a22bfcb361a.svg) | (E)-3-(1H-Benzo[d]imidazol-2-yl)-1-(6-chloro-2-hydroxy-4-phenylquinolin-3-yl)prop-2-en-1-one | Ki | 3900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_654c996963915ee5ba23b4e6bfb7b559.svg) | (S)-2-(2-(2-Methylindolin-1-yl)-2-oxoethyl)-6-morpholinopyrimidin-4(3H)-one | IC50 | 9.0 [1], 12.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_00776230c6ba5ad9b8574c1ff999bfb4.svg) | (Z)-3-((1H-Pyrrol-2-yl)methylene)indolin-2-one | IC50 | 2300.0 [1], 3000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_c14151f8a3f91d99bdd1903366b06e7d.svg) | (1S)-1-Methyl-2-[5-[2-(4-pyridyl)vinyl]-6-chloro-3-pyridyloxy]ethanamine | IC50 | 5290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_ee7a537c3497146dcd992de8a5f84845.svg) | [(2R)-2-Methoxy-3-octadecoxypropyl] [(1R,2S,3S,4R,6R)-2,3,4,6-tetrahydroxycyclohexyl] hydrogen phosphate | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_eb125c8f6ed93e5365c8ef9c8e72fb26.svg) | 5-[5-[(1,3-Dioxoindan-2-ylidene)methyl]-2-furyl]-2-hydroxy-benzoic acid | IC50 | 25100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_eb125c8f6ed93e5365c8ef9c8e72fb26.svg) | 5-[5-[(1,3-Dioxoindan-2-ylidene)methyl]-2-furyl]-2-hydroxy-benzoic acid | Ki | 20800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_7a4254b2b4cd2e9937dbe5863115462e.svg) | 3-(4'-Hydroxybiphenyl-4-Yl)-N-(4-Hydroxycyclohexyl)-1,4-Dihydroindeno[1,2-C]pyrazole-6-Carboxamide | IC50 | 4430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_f78ea3f034b7b643fcb19743ec512abb.svg) | AKT Kinase Inhibitor | IC50 | 2.0 [1], 1130.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_dbc94bb504996085040e4d04c5df6c07.svg) | Akt inhibitor | IC50 | 0.5 [1], 310.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_bd55926c7b3558be92fcb8361c526820.svg) | 3-(3-Iodobenzyl)-1-tert-butyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 28.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_d09cea2d1177b2565a86abbaa894d024.svg) | [(2R)-2-Methoxy-3-octadecoxypropyl] [(1R,2S,3S,4R,5S,6R)-2,3,4,6-tetrahydroxy-5-(hydroxymethyl)cyclohexyl] carbonate | IC50 | 5000.0 [1], 32000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_76250ddfa35d9c62332c9d413fe93396.svg) | 5-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}-1H-indazole | IC50 | 1.5 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_bd3a93680f902c529f9b1ba7108efe82.svg) | N-[4-[5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl]phenyl]acetamide | IC50 | 227.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_7ebd65d79417e4311f095890a7ac004e.svg) | 6-{5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]-6-chloropyridin-3-yl}isoquinoline | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_2480eb95bb869a86579a110bf3e85789.svg) | (E)-3-(4-Bromophenyl)-N-[2-[5-[(E)-2-pyridin-4-ylethenyl]pyridin-3-yl]oxyethyl]prop-2-en-1-amine | IC50 | 32250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_7d2f4f05b6737a782002cf9914762a02.svg) | 3-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]-6-(pyridin-4-yl)quinoline | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_f36517eb495346665a3f4ffc2fe37895.svg) | 3-[1-[[4-(6-Oxo-2-phenyl-1H-pyrazin-3-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 3029.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_e21e6973878706c2852ef43223046095.svg) | 3-[1-[[4-[5-(2-Methylpropyl)-6-oxo-3-phenyl-1H-pyrazin-2-yl]phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 20000.0 [1], 21200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_830a47cc46a5831b569bee4553d29dff.svg) | (2S)-2-Amino-3-(1H-indol-3-yl)-N-[5-[(E)-2-pyridin-4-ylethenyl]pyridin-3-yl]propanamide | IC50 | 278.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_5974605e294f40b3fcd0d2cb886080e6.svg) | 5-[(2S)-2-Amino-3-(1H-indol-3-yl)propoxy]-N-pyridin-4-ylpyridine-3-carboxamide | IC50 | 1659.0 [1], 2020.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_3ab784eb12726abfdb6630b2473a48dd.svg) | 3-N-[(2S)-2-Amino-3-(1H-indol-3-yl)propyl]-5-N-isoquinolin-5-ylpyridine-3,5-diamine | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_4461f456c4daa83fdcf137a7fd509ed8.svg) | (2S)-3-(1H-Indol-3-yl)-1-N-(5-isoquinolin-5-yloxypyridin-3-yl)propane-1,2-diamine | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-akt_0afde03be452af9a350e0d5b5b7da1cf.svg) | 3-[1-[[4-(6-Oxo-3-phenyl-1H-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one | IC50 | 1500.0 [1] |