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Serine/threonine-protein kinase 17B Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
N-[5-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl]cyclohexanecarboxamideIC50720.0 [1]
Drak2-IN-1IC503.0 [1]
Drak2-IN-1Ki0.26 [1]
StaurosporineIC5025.8 [1]
IndirubinIC5010000.0 [1]
Indirubin-3'-monoximeIC50710.0 [1]
AuroneIC5024640.0 [1]
SulfuretinIC501020.0 [1]
3-(1,3-Dihydro-3-oxo-2H-indol-2-ylidene)-1,3-dihydro-5-iodo-2H-indol-2-oneIC506200.0 [1]
5'-FluoroindirubinoximeIC50620.0 [1]
(3Z)-5-Methyl-3-(3-oxoindolin-2-ylidene)indolin-2-oneIC5010000.0 [1]
(3Z)-5-Fluoro-3-(3-oxoindolin-2-ylidene)indolin-2-oneIC5010000.0 [1]
(3Z)-5-Chloro-3-(3-oxoindolin-2-ylidene)indolin-2-oneIC5010000.0 [1]
(Z)-2-(3,4-Dimethoxybenzylidene)benzofuran-3(2H)-oneIC5021430.0 [1]
2-(4-Hydroxybenzylidene)-1-benzofuran-3(2H)-oneIC5053030.0 [1]
2-[(Z)-3,4-Dihydroxybenzylidene]-2,3-dihydrobenzofuran-3-oneIC503080.0 [1]
2-(3,4-Dihydroxybenzylidene)indan-1-oneIC5013290.0 [1]
2-(5-Amino-2-hydroxy-1H-indol-3-yl)indol-3-oneIC501400.0 [1]
5-Amino-3-(3-nitroso-1H-indol-2-yl)-1H-indol-2-olIC50250.0 [1]
2-(4-Fluorobenzylidene)benzofuran-3(2H)-oneIC5040550.0 [1]
2-[(Z)-3-Methoxy-4-hydroxybenzylidene]-2,3-dihydrobenzofuran-3-oneIC503110.0 [1]
(2Z)-2-[(3-Hydroxy-4-methoxyphenyl)methylidene]-1-benzofuran-3-oneIC5012100.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2,2-dimethylpropanamideIC5021.0 [1]
5-Chloro-7-methyl-3-(3-nitroso-1H-indol-2-yl)-1H-indol-2-olIC5010000.0 [1]
2-[(Z)-3-Ethoxy-4-hydroxybenzylidene]-2,3-dihydrobenzofuran-3-oneIC503240.0 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
(2Z)-2-(Pyridin-3-ylmethylidene)-1-benzofuran-3-oneIC5039390.0 [1]
SulferetolIC50990.0 [1]
N-[2-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyrazin-7-yl]cyclohexanecarboxamideIC501780.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-nitrobenzamideIC501300.0 [1]
4-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamideIC501200.0 [1]
2-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamideIC50290.0 [1]
4-Chloro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamideIC503200.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamideIC50200.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclohexanecarboxamideIC50120.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclopropanecarboxamideIC508.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-methylbut-2-enamideIC5014.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,3-dimethylbutanamideIC5014.0 [1]
4-Bromo-2-(2-hydroxy-5-nitro-1H-indol-3-yl)indol-3-oneIC5010000.0 [1]
2-(5-Chloro-2-hydroxy-7-methyl-1H-indol-3-yl)indol-3-oneIC5010000.0 [1]
2-(2-Hydroxy-5,7-dimethyl-1H-indol-3-yl)indol-3-oneIC5010000.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]butanamideIC5010.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]naphthalene-1-carboxamideIC501500.0 [1]
(E)-N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-phenylprop-2-enamideIC50700.0 [1]
2-(3-Chlorophenoxy)-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]acetamideIC50950.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2-(trifluoromethyl)benzamideIC50120.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methoxybenzamideIC50330.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methylbenzamideIC501300.0 [1]
N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,5-dinitrobenzamideIC5077.0 [1]
4-Bromo-2-(2-hydroxy-1H-indol-3-yl)indol-3-oneIC5010000.0 [1]
2-[(3,4-Dihydroxyphenyl)methyl]-1-benzofuran-3-oneIC5027810.0 [1]
5-(3-Amino-5-thiophen-3-ylthieno[2,3-b]pyridin-2-yl)-3H-1,3,4-oxadiazole-2-thioneIC5029.0 [1]
(2Z)-2-[[4-(Hydroxymethyl)phenyl]methylidene]-1-benzofuran-3-oneIC5011090.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-fluoro-1-benzofuran-3-oneIC501050.0 [1]
(2Z)-5-Butoxy-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC503660.0 [1]
(2Z)-2-[(3,4-Dihydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-oneIC50250.0 [1]
(2Z)-6-Chloro-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC5040540.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-iodo-1-benzofuran-3-oneIC5042520.0 [1]
(2Z)-2-[(4-Hydroxy-3-propan-2-yloxyphenyl)methylidene]-1-benzofuran-3-oneIC5017390.0 [1]
(2Z)-5-Ethoxy-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC50410.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-7-methoxy-1-benzofuran-3-oneIC501290.0 [1]
(2Z)-2-[(4-Hydroxy-3,5-dimethoxyphenyl)methylidene]-1-benzofuran-3-oneIC506650.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-4-methoxy-1-benzofuran-3-oneIC507260.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-oneIC50330.0 [1]
(2Z)-5-Amino-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC507160.0 [1]
1-Benzofuran-2-yl-(3,4-dihydroxyphenyl)methanoneIC5022910.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-6-fluoro-1-benzofuran-3-oneIC5060400.0 [1]
(2Z)-2-[(3-Butoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC5029100.0 [1]
[(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-3-oxo-1-benzofuran-5-yl] acetateIC50690.0 [1]
(2Z)-2-[(4-Hydroxy-3-propoxyphenyl)methylidene]-1-benzofuran-3-oneIC505370.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-6-methoxy-1-benzofuran-3-oneIC502440.0 [1]
(2Z)-5-Bromo-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC5028150.0 [1]
(2Z)-5-Chloro-2-[(3-ethoxy-4-hydroxyphenyl)methylidene]-1-benzofuran-3-oneIC5013710.0 [1]
(2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-methyl-1-benzofuran-3-oneIC50960.0 [1]
(2Z)-2-Furfurylidenebenzofuran-3(2H)-oneIC5063960.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Serine/threonine-protein kinase 17B Inhibitors (IC50, Ki)." AAT Bioquest, Inc.21 Dec2024https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-17b-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024December 21). Quest Database™ Serine/threonine-protein kinase 17B Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/serine-threonine-protein-kinase-17b-inhibitors-ic50-ki.
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