![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_806b136a185c8f00c9c74936ccf7683c.svg) | N-[5-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl]cyclohexanecarboxamide | IC50 | 1330.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_83c9c8729ff2ddfdd825a53ccf71f553.svg) | Sulfuretin | IC50 | 5850.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_fa37ae125bcd4e6df1af4be57fbea491.svg) | 1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)urea | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_1475ac4f13187836f3e8e4e00ac9ba17.svg) | Tomivosertib | IC50 | 131.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_8b8fdaae6a146a7f296d159fd2da00a6.svg) | Chembl4126445 | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_e24fa70c5b8c357e90ebd4f344e9be85.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2,2-dimethylpropanamide | IC50 | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_622b018ed1691625cf365dac7954cc5e.svg) | (5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-one | IC50 | 12.8 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_18f755a79542e417268d9ff837b61c52.svg) | N-[2-(3,4-Dimethoxyphenyl)thieno[2,3-b]pyrazin-7-yl]cyclohexanecarboxamide | IC50 | 4940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_1e4bbde9f21e3138fb96719273dd8845.svg) | Drak2-IN-1 | IC50 | 51.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_a682b1bfa1a535556efb28ed6218469f.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-nitrobenzamide | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_db37cdf30fc9eda80ad073a81f50c378.svg) | 4-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide | IC50 | 780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_a52b1163d65a7f07443744f687135f41.svg) | 2-Fluoro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide | IC50 | 250.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_2bd57943226af678d59278df9c32bb2f.svg) | 4-Chloro-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_f0ab47a0ac7fcad965b239119ce673cc.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]benzamide | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_650de2349e85579dfefe2156fa254a7a.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclohexanecarboxamide | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_3e2a1b10ed3c1fcd2a4906212726fdcd.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclopropanecarboxamide | IC50 | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_2dc93255a79bbfa3194f8141aa6e8839.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-methylbut-2-enamide | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_b0b1c360177119ea2ded621b471ec9d2.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,3-dimethylbutanamide | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_f761aa5e4adec79c527f4bb51b7e0f18.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]butanamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_7d9dd20cedc747de13fdc65d444a00b6.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]naphthalene-1-carboxamide | IC50 | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_089f35321f0ded370e56a3e1cd303533.svg) | (E)-N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-phenylprop-2-enamide | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_2b96a10905096a33b05d36c3e8974eb0.svg) | 2-(3-Chlorophenoxy)-N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]acetamide | IC50 | 460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_570e6d5e29b8d2705e9b1168526b15e6.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2-(trifluoromethyl)benzamide | IC50 | 320.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_1ab2fd45e8e02c6fa777c7d360c7f8ca.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methoxybenzamide | IC50 | 360.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_ac00cd339a5b32e0d249945df4fe46a5.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-4-methylbenzamide | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_72b59a73bdb10afecdc799f83bad6710.svg) | N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,5-dinitrobenzamide | IC50 | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_5d3ca99ca14e64765fe9213bf17e538f.svg) | (2Z)-2-[(3,4-Dihydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-one | IC50 | 5810.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_8115d93fd3560bcae3c78bccf6272ac6.svg) | (2Z)-2-[(3-Ethoxy-4-hydroxyphenyl)methylidene]-5-methoxy-1-benzofuran-3-one | IC50 | 1410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_8db6cb051225bbef11f4324ad1c0eaf6.svg) | N-[5-(6-Aminopyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]-4,4,4-trifluoro-2,2-dimethylbutanamide | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-threonine-protein-kinase-17a_7001927caad7c36762b0d4d34597955f.svg) | (2R)-N-[5-(6-Aminopyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]-4,4,4-trifluoro-2-methylbutanamide | IC50 | 2900.0 [1] |