![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_c1fc56ca717493fcf185aef7cc38cc20.svg) | 2-Morpholino-6-(thianthren-1-yl)-4H-pyran-4-one | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_c1fc56ca717493fcf185aef7cc38cc20.svg) | 2-Morpholino-6-(thianthren-1-yl)-4H-pyran-4-one | Ki | 2.2 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_020b6857f8c252df41bc602b24cd6d1e.svg) | 2-(Morpholin-4-yl)-benzo[h]chromen-4-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_6603a475932cb1632b1b43c2f664a423.svg) | 2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one | IC50 | 10000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_bada19a1327cd523a6a347eb625a6ce2.svg) | CID 118502708 | IC50 | 0.04 [1], 0.57 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_375723c4a9d1079c63e87796be774461.svg) | 8-(4-Dibenzothienyl)-2-(4-morpholinyl)-4H-1-benzopyran-4-one | IC50 | 10000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_7c4643189efd94dd6459f3f9fd31dd92.svg) | 1-(6,7-Dimethoxyquinazolin-4-yl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-amine | IC50 | 20.0 [1], 400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_6e737d4108ad3bb1cffa3d9228e43f45.svg) | CID 46244454 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_7f2bb74101cfce19fa35628c8e2894af.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-3-methyl-1-(oxetan-3-yl)imidazo[4,5-c]quinolin-2-one | IC50 | 1.46 [1], 1.5 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_a1bce4efd367b97e0a479b10d0a375be.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-7-fluoro-3-methyl-1-(oxan-4-yl)imidazo[4,5-c]quinolin-2-one | IC50 | 0.78 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_748e14057b90f6bf99f5df94d9e79647.svg) | 1-(3-Methoxycyclobutyl)-3-methyl-8-[6-[3-(methylamino)propoxy]pyridin-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 0.25 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_3425f3ab476d36130ef22be2db575e67.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-3-methyl-1-[(3S)-oxan-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 0.33 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_eacec6ab64635ee014beadbb4f80e850.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-1-(3-methoxycyclobutyl)-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 0.25 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_f43240199a098e036fd675cc583e8ba3.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-1-(3-hydroxycyclobutyl)-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 0.24 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_fa207f8e5006a0f64b3062d54d6589dc.svg) | 1-(3-Methoxycyclobutyl)-3-methyl-8-[6-(3-pyrrolidin-1-ylpropoxy)pyridin-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 0.17 [1], 0.18 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_5f4ff6fcca0f0ddfa9ce15ab8e753316.svg) | 8-[6-[3-(Dimethylamino)propoxy]-2-fluoropyridin-3-yl]-1-(3-methoxycyclobutyl)-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 0.76 [1], 0.77 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_908543f51b37e595052a3a35e524d208.svg) | 8-[6-[3-(Dimethylamino)propoxy]-2-fluoropyridin-3-yl]-7-fluoro-1-(3-methoxycyclobutyl)-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 2.6 [1], 2.62 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_9d56ee2102343c5c6bc54325fa55d2cc.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-7-fluoro-1-(3-methoxycyclobutyl)-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 1.05 [1], 1.1 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_75aeef29c20e8eb552b756ba3050966b.svg) | 1-(3-Methoxycyclobutyl)-3-methyl-8-[6-(3-piperidin-1-ylpropoxy)pyridin-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 0.2 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_962fe80927980017a92d28a04633f6fe.svg) | 8-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-3-methyl-1-[(3R)-oxan-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 0.94 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_9fc327fc80c1bd270b0258d1113edfd2.svg) | 8-[6-[3-(Azetidin-1-yl)propoxy]pyridin-3-yl]-1-(3-methoxycyclobutyl)-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 0.29 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_14dac9d5896f074bcf45345c60981078.svg) | 7-Fluoro-3-methyl-1-[(3S)-oxan-3-yl]-8-[6-(3-piperidin-1-ylpropoxy)pyridin-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 0.8 [1], 1.1 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_a630bb15f2e8d7600f15f95886600af9.svg) | 7-Fluoro-3-methyl-1-(oxan-4-yl)-8-[6-(3-piperidin-1-ylpropoxy)pyridin-3-yl]imidazo[4,5-c]quinolin-2-one | IC50 | 1.1 [1], 1.2 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_b428cf9217fc5982a66db23284a81c8d.svg) | ATM Inhibitor-1 | IC50 | 0.7 [1], 2.8 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_7df46a3fe28fe326c6c4fce8db0fb27b.svg) | 6-[6-[3-(Dimethylamino)propoxy]pyridin-3-yl]-4-[[(1S)-1-(oxan-4-yl)ethyl]amino]cinnoline-3-carboxamide | IC50 | 0.29 [1], 1.9 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_0c7825c24504348a6d7541133c2c8b82.svg) | 7-Fluoro-1-(3-methoxycyclobutyl)-8-[6-(methoxymethyl)pyridin-3-yl]-3-methylimidazo[4,5-c]quinolin-2-one | IC50 | 100.0 [1], 160.0 [2] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_bec8eaadb51e755de26c3660866564ee.svg) | Caffeine | IC50 | 200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_0a25d9549eee718648f002f556162019.svg) | Thiourea | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_98871935c6dbd53bec1df41a5db7ba4b.svg) | Dactolisib | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_c8c9c64706e15ecb9a8ca87144ec4882.svg) | Schisandrin B | IC50 | 1740000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_a59db47f5f7aa063c6007dcf79b51cfe.svg) | PD173074 | IC50 | 17600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_d472d7090a10696dcf0b9f871e2dfba5.svg) | Alpelisib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_dd9878f1baa15961f1fb02150c92f8b5.svg) | 3-Amino-6-(4-(methylsulfonyl)phenyl)-N-phenylpyrazine-2-carboxamide | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_e79ac988804a5fa77d428b6b8fb01191.svg) | KU-60019 | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_338c5cd8892fdf32da2db54d84d39915.svg) | Imino-methyl-[1-[6-[(3R)-3-methylmorpholin-4-yl]-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrimidin-4-yl]cyclopropyl]-oxo-lambda6-sulfane | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_750b1a397f7e487203db00823ad4de11.svg) | CID 11964036 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_cee977367305601582d81c3f043802f5.svg) | Diphenyl acetamidotrichloroethyl fluoronitrophenyl thiourea | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_09527b215eb7dd103cade5a5e6c5aca4.svg) | 2-Methyl-2-[4-(2-oxo-9-quinolin-3-yl-4H-[1,3]oxazino[5,4-c]quinolin-1-yl)phenyl]propanenitrile | IC50 | 36.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_8bb67ece054465d2ce242d532d393a29.svg) | 2-Morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_bdc90869b5df3bb3a7b3dfc7f9e7065f.svg) | Cc-115 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_7f20db493f470456ad09c664f792426e.svg) | 2-(2-Methyl-morpholin-4-yl)-benzo[h]chromen-4-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_ed257503d8f1feb75721a05c23ee2799.svg) | 4-Hydroxy-3,5-dimethoxybenzaldehyde [4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]hydrazone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_3e3b93094c79027f91bdc18ac9a276c1.svg) | 3-Amino-n,6-diphenylpyrazine-2-carboxamide | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_a4f9524fc4012a16e5e07bc4b78069ff.svg) | 7-Fluoro-6-[6-(methoxymethyl)pyridin-3-yl]-4-[[(1S)-1-(1-methylpyrazol-3-yl)ethyl]amino]quinoline-3-carboxamide | IC50 | 33.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_b9a223d468c23cc73579020f8c72509c.svg) | CID 134694318 | IC50 | 46.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_ebffe9981e1dc0736f6dedfea14a6d71.svg) | 3-Amino-6-[4-[1-(dimethylamino)propan-2-ylsulfonyl]phenyl]-N-phenylpyrazine-2-carboxamide | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_cf9afc6bcb83d9eac22c9b1424c76bad.svg) | (3E)-3-(1H-Pyrrol-2-ylmethylidene)-1,3-dihydro-2H-indol-2-one | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_723b89fc06b04f1365e222de14d7f616.svg) | 3-(4-Methylpiperazin-1-yl)-N-[6-(6-morpholin-4-yl-4-oxopyran-2-yl)thianthren-2-yl]propanamide | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_f2022dfa8ed0c588327c68c084b15d42.svg) | (6R)-6-Methyl-3-(4-methylsulfonylphenyl)-5-(1H-pyrrolo[2,3-b]pyridin-4-yl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine | IC50 | 130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_09ddf72fb2d98e767ed479db83a03e50.svg) | (6R)-6-Methyl-3-(1-methylsulfonylpiperidin-4-yl)-5-(1H-pyrrolo[2,3-b]pyridin-4-yl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine | IC50 | 14000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_3232b055327db0b7131ee1d86ff0ce53.svg) | (6R)-5-(6-Chloro-1H-pyrrolo[2,3-b]pyridin-4-yl)-6-methyl-3-(1-methylsulfonylpiperidin-4-yl)-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine | IC50 | 4300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_3b057841c942a6c2d371657c19537146.svg) | (3R)-3-Methyl-4-[1-methyl-6-(1H-pyrrolo[2,3-d]pyridazin-4-yl)imidazo[4,5-c]pyridin-4-yl]morpholine | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_a4d8c0429243ad7d601586bd5fc2524e.svg) | 2-[4-[4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-6,7-dimethoxyquinazolin-2-yl]piperazin-1-yl]ethanol | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_d36c57c351c5ddf6e3f585a6e959110b.svg) | Ethyl 2-[[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-6,7-dimethoxyquinazolin-2-yl]amino]acetate | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_fb426c57aae75f8609470b7fd5413bf8.svg) | 2-[[4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-6,7-dimethoxyquinazolin-2-yl]amino]acetic acid | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_b107197ece21d99555496f256df7b832.svg) | 4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-N,N-diethyl-6,7-dimethoxyquinazolin-2-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_eb186a68a14c0d5a8b6af15e1ce51dd7.svg) | 2-(6,7-Dimethoxy-2-methylquinazolin-4-yl)-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 10100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_88f3bb350b67e1dcdff8ab03d8718b4c.svg) | 2-(6,7-Dimethoxy-2-phenylquinazolin-4-yl)-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_cea210d71b15d53ab25bb5ca9c11fa21.svg) | 2-[7-Methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_4924ac0179447b50dfc7882590d1fd1c.svg) | 2-[6-Methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_fe9f323a38676c08d2fb86ecef5e33bb.svg) | 2-[6-[3-(Dimethylamino)propoxy]-7-methoxyquinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 6600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_ab6451b089ff738d4ed9c75c5c84f2fa.svg) | 2-[6-[2-[Di(propan-2-yl)amino]ethoxy]-7-methoxyquinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 6100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_6f0ce903136ae57e1dc17b031968c116.svg) | 2-[7-Methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_981da4588b7f88d735cffbf7eadf9313.svg) | 2-[7-Methoxy-6-[2-(4-methylpiperidin-1-yl)ethoxy]quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_8dc4e3d4f66669ec26a396cea22b492e.svg) | 2-[6-[3-(2,6-Dimethylmorpholin-4-yl)propoxy]-7-methoxyquinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_32a5a76c8f4bb68e12d8a1f89c63ccad.svg) | 2-[4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxy-N,N-diethylacetamide | IC50 | 5300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_d7eab66a2ab736072375d9f389243605.svg) | N-[3-[4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetamide | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_15c0e702e52d82fe644b7b9afd830f13.svg) | Tert-butyl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_ea61cb7435a244bd24a56558aa159eb7.svg) | 4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-6,7-dimethoxyquinazolin-2-amine | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_432abe5b8bfb084227a9758f93d5cd92.svg) | 6,7-Dimethoxy-4-(3-pyridin-2-yl-1,2,4-triazol-1-yl)quinazoline | IC50 | 5300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_8ba29e8474bcc9d12c4cbdd5f09d5df9.svg) | 6,7-Dimethoxy-4-(4-pyridin-2-yltriazol-2-yl)quinazoline | IC50 | 13300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_f5168ffbc1738a71081cb11188247f05.svg) | 2-(6,7-Dimethoxyquinazolin-4-yl)-5-pyridin-2-ylpyrazol-3-amine | IC50 | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_9666e32cdbc945ca5c7c2e1c75f56175.svg) | 2-[7-Methoxy-6-(2-piperidin-1-ylethoxy)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 5600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_7289f1c8d96b449da2aa5bd71bb20920.svg) | Tert-butyl N-[4-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxybutyl]carbamate | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_4140c99188c911e3e0a6c14505891e88.svg) | 2,2,2-Trifluoroethyl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_9bc48e986e3fb14bcfe4560293e13275.svg) | 2-[(2R,6S)-2,6-Dimethylmorpholin-4-yl]-N-[6-(6-morpholin-4-yl-4-oxopyran-2-yl)thianthren-2-yl]acetamide | IC50 | 6.3 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_45afe9fad38d97ac33e94d74a266d9c3.svg) | Tert-butyl N-[2-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxyethyl]carbamate | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_8d3cf641bb36b8a003d60c650ee68e02.svg) | Ethyl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_859a1d4bd3ca10792ad95636952253b5.svg) | Propan-2-yl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_b0e5572245beb23a29aeb259012624b0.svg) | 2-(6-Methoxy-7-phenylmethoxyquinazolin-4-yl)-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_f63397bc4e28c72d90ded6701bc2a19a.svg) | Hexyl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 28600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_d62af30716b29357275d68d42601b39e.svg) | Phenyl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 23500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_748c95f7a6d480ec2ea256228c2f27ac.svg) | 2,2-Dimethylpropyl N-[3-[4-(5-amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]carbamate | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_5666acaa29604c670c2a489734e3a48f.svg) | N-[3-[4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-yl]oxypropyl]-2,2,2-trifluoroacetamide | IC50 | 2900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_e96067054cdfe821057221ec4c03376c.svg) | 2-[6,7-Bis(cyclopropylmethoxy)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_01a355c48c3816a9d51ceb0925e7b97e.svg) | 2-(6,7-Dimethoxy-2-morpholin-4-ylquinazolin-4-yl)-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_daacace21bfd9581896028e9f1fd4327.svg) | 2-[6,7-Dimethoxy-2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_d3d416fb8a3dd8042c67e14de9942893.svg) | 2-(6,7-Dimethoxyquinazolin-4-yl)-5-(4-methylphenyl)pyrazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_dfe8173fe2ec92e45966b000b2d8edd7.svg) | 5-(4-Chlorophenyl)-2-(6,7-dimethoxyquinazolin-4-yl)pyrazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_6d6cec60ae1eb9d2d361ed44ab9be146.svg) | 1-(6,7-Dimethoxyquinazolin-4-yl)-1,2,4-triazole-3,5-diamine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_8539c3e2717d3b79451e646be6c7e9af.svg) | 2-(7-Methoxy-6-phenylmethoxyquinazolin-4-yl)-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 8600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_c53587d398b816ad9a79071059c6f479.svg) | 2-(2-Chloro-6,7-dimethoxyquinazolin-4-yl)-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_ccafc38689791bb4f0505ac14f02380f.svg) | 6,7-Dimethoxy-N-(4-pyridin-2-ylphenyl)quinazolin-4-amine | IC50 | 12500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_6bd011053bef291d795fb89718e6300b.svg) | 2-[6,7-Bis(2-methoxyethoxy)quinazolin-4-yl]-5-pyridin-2-yl-1,2,4-triazol-3-amine | IC50 | 2300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_e32018f53f3da78be1a906f325d15b18.svg) | 5-Cyclohexyl-2-(6,7-dimethoxyquinazolin-4-yl)-1,2,4-triazol-3-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_4a2557bb87385b77c9c277763005a7c5.svg) | 6,7-Dimethoxy-N-pyridin-2-ylquinazolin-4-amine | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_4f4d59f3f69afb8f8647bc3fe0ffbe9d.svg) | 2-(6,7-Dimethoxyquinazolin-4-yl)-4-pyridin-2-ylpyrazol-3-amine | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_ef6eecc476d5166d1cac2d15dd4bc2c6.svg) | 4-(5-Amino-3-pyridin-2-yl-1,2,4-triazol-1-yl)-7-methoxyquinazolin-6-ol | IC50 | 12600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/serine-protein-kinase-atm_d24be83001ec7d43f9198328f867c85e.svg) | 2-(6,7-Dimethoxyquinazolin-4-yl)-5-phenyl-1,2,4-triazol-3-amine | IC50 | 2000.0 [1] |