| CID 62705299 | IC50 | 1.5 [1] |
| Rimcazole | IC50 | 1200.0 [1] |
| Methyl 9-[3-(4,6-dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazole-3-carboxylate | IC50 | 1.5 [1] |
| ITX-5061 free base | IC50 | 100.0 [1] |
| 3-(6-Cyano-1,2,3,4-tetrahydrocarbazol-9-yl)-N,N-dimethylpropane-1-sulfonamide | IC50 | 50.0 [1] |
| 9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-6-methylsulfonyl-1,2,3,4-tetrahydrocarbazole | IC50 | 50.0 [1] |
| 9-[3-[(4,6-Dimethoxypyrimidin-2-yl)amino]propyl]-5,6,7,8-tetrahydrocarbazole-3-carbonitrile | IC50 | 15.0 [1] |
| Propan-2-yl 9-[3-[(3S,5R)-3,5-dimethylpiperazin-1-yl]propyl]carbazole-3-carboxylate | IC50 | 630.0 [1] |
| Methyl 9-[3-[(3R,5S)-3,5-dimethylpiperazin-1-yl]propyl]carbazole-3-carboxylate | IC50 | 230.0 [1] |
| Ethyl 9-[3-[(3S,5R)-3,5-dimethylpiperazin-1-yl]propyl]carbazole-3-carboxylate | IC50 | 600.0 [1] |
| 2-[9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-4,5-dihydro-1,3-oxazole | IC50 | 50.0 [1] |
| 2-[9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-1,3-oxazole | IC50 | 1.5 [1] |
| CID 62705136 | IC50 | 50.0 [1] |
| CID 62705137 | IC50 | 15.0 [1] |
| CID 62705138 | IC50 | 1.5 [1] |
| CID 62705139 | IC50 | 1.5 [1] |
| CID 62705298 | IC50 | 1.5 [1] |
| CID 62705302 | IC50 | 1.5 [1] |
| CID 62705303 | IC50 | 5.0 [1] |
| CID 62705467 | IC50 | 15.0 [1] |
| 5-[9-[3-(6-Fluoro-1H-benzimidazol-2-yl)propyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-3-methyl-1,2,4-oxadiazole | IC50 | 1.5 [1] |
| 5-[9-[3-(3,5-Difluorophenoxy)-2-fluoropropyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-3-methyl-1,2,4-oxadiazole | IC50 | 1.5 [1] |
| CID 62705642 | IC50 | 5.0 [1] |
| CID 62705643 | IC50 | 1.5 [1] |
| CID 62705646 | IC50 | 15.0 [1] |
| CID 62705816 | IC50 | 15.0 [1] |
| CID 62707244 | IC50 | 10.0 [1] |
| 9-[3-(4,6-Diethylpyrimidin-2-yl)oxypropyl]-6-methylsulfonyl-1,2,3,4-tetrahydrocarbazole | IC50 | 30.0 [1] |
| CID 62707406 | IC50 | 500.0 [1] |
| 9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazole-3-carbonitrile | IC50 | 15.0 [1] |
| CID 62707566 | IC50 | 5.0 [1] |
| CID 62707567 | IC50 | 15.0 [1] |
| CID 62707568 | IC50 | 1.5 [1] |
| CID 62707569 | IC50 | 1.5 [1] |
| CID 62707570 | IC50 | 1.5 [1] |
| CID 62707571 | IC50 | 1.5 [1] |
| N-[3-[3-[Bis(2-hydroxyethyl)amino]propylsulfonylamino]-5-tert-butyl-2-methoxyphenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide | IC50 | 39.81 [1] |
| 2-[3-[[5-Tert-butyl-2-methoxy-3-[[2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetyl]amino]phenyl]sulfamoyl]propyl-(carboxymethyl)amino]acetic acid | IC50 | 5011.87 [1] |
| N-[5-Tert-butyl-3-[3-[[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]amino]propylsulfonylamino]-2-methoxyphenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide | IC50 | 50.12 [1] |
| 3-[[5-Tert-butyl-2-methoxy-3-[[2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetyl]amino]phenyl]sulfamoyl]propyl-triethylazanium;2,2,2-trifluoroacetate | IC50 | 158.49 [1] |
| N-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-[4-[2-(4-methylmorpholin-4-ium-4-yl)ethoxy]naphthalen-1-yl]-2-oxoacetamide;2,2,2-trifluoroacetate | IC50 | 1000.0 [1] |
| N-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-[4-(4-morpholin-4-ylbutoxy)naphthalen-1-yl]-2-oxoacetamide | IC50 | 50.12 [1] |
| 2-[4-[2-[(2-Aminoacetyl)amino]ethoxy]naphthalen-1-yl]-N-[5-tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-oxoacetamide | IC50 | 50.12 [1] |
| 3-[2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethylamino]-3-oxopropanoic acid | IC50 | 1000.0 [1] |
| 2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethyl-trimethylazanium;2,2,2-trifluoroacetate | IC50 | 501.19 [1] |
| 2-[[5-Tert-butyl-2-methoxy-3-[[2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetyl]amino]phenyl]sulfamoyl]acetic acid | IC50 | 199.53 [1] |
| N-[3-(4-Aza-1-azoniabicyclo[2.2.2]octan-1-ylmethylsulfonylamino)-5-tert-butyl-2-methoxyphenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide;chloride | IC50 | 158.49 [1] |
| 2-[2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethyl-(carboxymethyl)amino]acetic acid | IC50 | 31622.78 [1] |
| 1-[2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethyl]piperidine-4-carboxylic acid | IC50 | 1000.0 [1] |
| 2-[4-[2-[Bis(2-hydroxyethyl)amino]ethoxy]naphthalen-1-yl]-N-[5-tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-oxoacetamide | IC50 | 79.43 [1] |
| 9-[3-(1H-Benzimidazol-2-yl)propyl]-6-methylsulfonyl-1,2,3,4-tetrahydrocarbazole | IC50 | 50.0 [1] |
| 9-[3-(1H-Benzimidazol-2-yl)propyl]-5,6,7,8-tetrahydrocarbazole-3-carbonitrile | IC50 | 50.0 [1] |
| N-[5-Tert-butyl-2-methoxy-3-(propylsulfonylamino)phenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide | IC50 | 50.12 [1] |
| 9-[3-(4,6-Diethylpyrimidin-2-yl)oxypropyl]-6-nitro-1,2,3,4-tetrahydrocarbazole | IC50 | 1.5 [1] |