Scavenger receptor class B member 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	CID 62705299	IC50	1.5 [1]
	Rimcazole	IC50	1200.0 [1]
	Methyl 9-[3-(4,6-dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazole-3-carboxylate	IC50	1.5 [1]
	ITX-5061 free base	IC50	100.0 [1]
	3-(6-Cyano-1,2,3,4-tetrahydrocarbazol-9-yl)-N,N-dimethylpropane-1-sulfonamide	IC50	50.0 [1]
	9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-6-methylsulfonyl-1,2,3,4-tetrahydrocarbazole	IC50	50.0 [1]
	9-[3-[(4,6-Dimethoxypyrimidin-2-yl)amino]propyl]-5,6,7,8-tetrahydrocarbazole-3-carbonitrile	IC50	15.0 [1]
	Propan-2-yl 9-[3-[(3S,5R)-3,5-dimethylpiperazin-1-yl]propyl]carbazole-3-carboxylate	IC50	630.0 [1]
	Methyl 9-[3-[(3R,5S)-3,5-dimethylpiperazin-1-yl]propyl]carbazole-3-carboxylate	IC50	230.0 [1]
	Ethyl 9-[3-[(3S,5R)-3,5-dimethylpiperazin-1-yl]propyl]carbazole-3-carboxylate	IC50	600.0 [1]
	2-[9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-4,5-dihydro-1,3-oxazole	IC50	50.0 [1]
	2-[9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-1,3-oxazole	IC50	1.5 [1]
	CID 62705136	IC50	50.0 [1]
	CID 62705137	IC50	15.0 [1]
	CID 62705138	IC50	1.5 [1]
	CID 62705139	IC50	1.5 [1]
	CID 62705298	IC50	1.5 [1]
	CID 62705302	IC50	1.5 [1]
	CID 62705303	IC50	5.0 [1]
	CID 62705467	IC50	15.0 [1]
	5-[9-[3-(6-Fluoro-1H-benzimidazol-2-yl)propyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-3-methyl-1,2,4-oxadiazole	IC50	1.5 [1]
	5-[9-[3-(3,5-Difluorophenoxy)-2-fluoropropyl]-5,6,7,8-tetrahydrocarbazol-3-yl]-3-methyl-1,2,4-oxadiazole	IC50	1.5 [1]
	CID 62705642	IC50	5.0 [1]
	CID 62705643	IC50	1.5 [1]
	CID 62705646	IC50	15.0 [1]
	CID 62705816	IC50	15.0 [1]
	CID 62707244	IC50	10.0 [1]
	9-[3-(4,6-Diethylpyrimidin-2-yl)oxypropyl]-6-methylsulfonyl-1,2,3,4-tetrahydrocarbazole	IC50	30.0 [1]
	CID 62707406	IC50	500.0 [1]
	9-[3-(4,6-Dimethylpyrimidin-2-yl)oxypropyl]-5,6,7,8-tetrahydrocarbazole-3-carbonitrile	IC50	15.0 [1]
	CID 62707566	IC50	5.0 [1]
	CID 62707567	IC50	15.0 [1]
	CID 62707568	IC50	1.5 [1]
	CID 62707569	IC50	1.5 [1]
	CID 62707570	IC50	1.5 [1]
	CID 62707571	IC50	1.5 [1]
	N-[3-[3-[Bis(2-hydroxyethyl)amino]propylsulfonylamino]-5-tert-butyl-2-methoxyphenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide	IC50	39.81 [1]
	2-[3-[[5-Tert-butyl-2-methoxy-3-[[2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetyl]amino]phenyl]sulfamoyl]propyl-(carboxymethyl)amino]acetic acid	IC50	5011.87 [1]
	N-[5-Tert-butyl-3-[3-[[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]amino]propylsulfonylamino]-2-methoxyphenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide	IC50	50.12 [1]
	3-[[5-Tert-butyl-2-methoxy-3-[[2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetyl]amino]phenyl]sulfamoyl]propyl-triethylazanium;2,2,2-trifluoroacetate	IC50	158.49 [1]
	N-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-[4-[2-(4-methylmorpholin-4-ium-4-yl)ethoxy]naphthalen-1-yl]-2-oxoacetamide;2,2,2-trifluoroacetate	IC50	1000.0 [1]
	N-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-[4-(4-morpholin-4-ylbutoxy)naphthalen-1-yl]-2-oxoacetamide	IC50	50.12 [1]
	2-[4-[2-[(2-Aminoacetyl)amino]ethoxy]naphthalen-1-yl]-N-[5-tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-oxoacetamide	IC50	50.12 [1]
	3-[2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethylamino]-3-oxopropanoic acid	IC50	1000.0 [1]
	2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethyl-trimethylazanium;2,2,2-trifluoroacetate	IC50	501.19 [1]
	2-[[5-Tert-butyl-2-methoxy-3-[[2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetyl]amino]phenyl]sulfamoyl]acetic acid	IC50	199.53 [1]
	N-[3-(4-Aza-1-azoniabicyclo[2.2.2]octan-1-ylmethylsulfonylamino)-5-tert-butyl-2-methoxyphenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide;chloride	IC50	158.49 [1]
	2-[2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethyl-(carboxymethyl)amino]acetic acid	IC50	31622.78 [1]
	1-[2-[4-[2-[5-Tert-butyl-3-(methanesulfonamido)-2-methoxyanilino]-2-oxoacetyl]naphthalen-1-yl]oxyethyl]piperidine-4-carboxylic acid	IC50	1000.0 [1]
	2-[4-[2-[Bis(2-hydroxyethyl)amino]ethoxy]naphthalen-1-yl]-N-[5-tert-butyl-3-(methanesulfonamido)-2-methoxyphenyl]-2-oxoacetamide	IC50	79.43 [1]
	9-[3-(1H-Benzimidazol-2-yl)propyl]-6-methylsulfonyl-1,2,3,4-tetrahydrocarbazole	IC50	50.0 [1]
	9-[3-(1H-Benzimidazol-2-yl)propyl]-5,6,7,8-tetrahydrocarbazole-3-carbonitrile	IC50	50.0 [1]
	N-[5-Tert-butyl-2-methoxy-3-(propylsulfonylamino)phenyl]-2-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]-2-oxoacetamide	IC50	50.12 [1]
	9-[3-(4,6-Diethylpyrimidin-2-yl)oxypropyl]-6-nitro-1,2,3,4-tetrahydrocarbazole	IC50	1.5 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 54 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Scavenger receptor class B member 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/scavenger-receptor-class-b-member-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 20). Quest Database™ Scavenger receptor class B member 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/scavenger-receptor-class-b-member-1-inhibitors-ic50-ki.
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