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Ribosomal protein S6 kinase alpha 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Bisindolylmaleimide IXIC5010.0 [1]
1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)ureaIC501.0 [1]
CID 53246941IC501.1 [1]
CID 59604787IC5010000.0 [1]
(1S,2S,3R,4R)-3-[[5-Chloro-2-[[(7S)-4-methoxy-7-morpholin-4-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamideIC507.0 [1]
2-(4-Toluidinomethyl)-1H-isoindole-1,3(2H)-dioneIC504300.0 [1]
2-((4-Morpholinophenylamino)methyl)isoindoline-1,3-dioneIC50790.0 [1]
2-(((4-Methoxyphenyl)amino)methyl)isoindoline-1,3-dioneIC50470.0 [1]
N-(1-Methylbenzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC509.0 [1]
N-(3-Methyl-1,2-oxazol-5-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5019.0 [1]
N-(1-Methylpyrazol-4-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5011.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi940.0 [1]
2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
7-(2-Methoxyphenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC5020.0 [1]
29-(Dimethylamino)-4,14,24,30-tetrazaheptacyclo[26.2.2.14,11.117,24.05,10.012,16.018,23]tetratriaconta-1(30),5,7,9,11(34),12(16),17(33),18,20,22,28,31-dodecaene-13,15-dioneIC50850.0 [1]
N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-5-methyl-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC501.3 [1]
N-[2-(Cyclopentylcarbamoyl)-1-methylimidazol-4-yl]-4,4-dimethyl-1-oxo-2,3-dihydropyrazino[1,2-a]indole-7-carboxamideIC503.7 [1]
N-(1-Ethylbenzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC501.1 [1]
N-(6-Chloro-1-ethylbenzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5012.0 [1]
1-Oxo-N-[1-(pyridin-4-ylmethyl)pyrazol-4-yl]-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC501.9 [1]
(5S)-N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-5-methyl-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5014.0 [1]
N-(1H-Benzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC504.4 [1]
N-(4-Chlorophenyl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50190.0 [1]
4,4-Dimethyl-1-oxo-N-pyridin-3-yl-3,5-dihydro-2H-[1,4]diazepino[1,2-a]indole-8-carboxamideIC504600.0 [1]
1-Oxo-N-(1-propan-2-ylpyrazolo[3,4-b]pyridin-5-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5053.0 [1]
1-Oxo-N-(3-phenyl-1,2-oxazol-5-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5087.0 [1]
1-Oxo-N-phenyl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50290.0 [1]
N-(2-Methoxyphenyl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50400.0 [1]
N-(2-Carbamoylphenyl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5021.0 [1]
4,4-Difluoro-1-oxo-N-pyridin-3-yl-3,5-dihydro-2H-[1,4]diazepino[1,2-a]indole-8-carboxamideIC501700.0 [1]
1-Oxo-N-quinolin-2-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5070.0 [1]
N-[6-Chloro-1-[3-(dimethylamino)propyl]benzimidazol-2-yl]-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5020.0 [1]
N-(1H-Imidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5025.5 [1]
1-Oxo-N-pyridin-3-ylspiro[3,5-dihydro-2H-[1,4]diazepino[1,2-a]indole-4,1'-cyclopropane]-8-carboxamideIC50430.0 [1]
1-Oxo-N-pyridin-3-ylspiro[3,5-dihydro-2H-[1,4]diazepino[1,2-a]indole-4,1'-cyclobutane]-8-carboxamideIC503300.0 [1]
N-(1,3-Benzoxazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50370.0 [1]
N-[1-(Cyclohexylmethyl)pyrazol-4-yl]-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC507.4 [1]
1-Oxo-N-pyridin-4-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5039.0 [1]
N-(1-Methylimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC502200.0 [1]
1-Oxo-N-(1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5043.0 [1]
1-Oxo-N-quinolin-3-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5034.0 [1]
N-(3-Cyclopropyl-1,2-oxazol-5-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5018.0 [1]
N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-4,4-dimethyl-1-oxo-3,5-dihydro-2H-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5027.0 [1]
N-[3-(1H-Imidazol-5-yl)phenyl]-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5052.0 [1]
N-(1-Methylpyrazol-3-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50540.0 [1]
1-Oxo-N-(1-propan-2-ylbenzimidazol-2-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5020.0 [1]
1-Oxo-N-(1-phenylbenzimidazol-2-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5061.0 [1]
N-(3-Ethylimidazo[4,5-b]pyridin-2-yl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC504.4 [1]
1-Oxo-N-(3-propan-2-yl-1,2-oxazol-5-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5026.0 [1]
N-(3-Chlorophenyl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50270.0 [1]
5-Methyl-1-oxo-N-pyridin-3-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5041.0 [1]
(4R,5S)-4,5-Dimethyl-1-oxo-N-pyridin-3-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC501100.0 [1]
1-Oxo-N-(1H-pyrazol-5-yl)-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5093.0 [1]
N-(2-Chlorophenyl)-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC506000.0 [1]
1-Oxo-N-pyridin-2-yl-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC50220.0 [1]
N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-1-oxo-2,3,4,5-tetrahydro-[1,4]diazepino[1,2-a]indole-8-carboxamideIC5021.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
2-[(4-Ethoxyanilino)methyl]-5-nitroisoindole-1,3-dioneIC502830.0 [1]
7-(2-Fluoro-6-Methoxyphenyl)-N-(3,4,5-Trimethoxyphenyl)-1,3-Benzoxazol-2-AmineIC5020.0 [1]
7-(1h-Benzimidazol-7-Yl)-N-(3,4,5-Trimethoxyphenyl)-1,3-Benzoxazol-2-AmineIC504.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-N-[4-methoxy-3-[(3S)-pyrrolidin-3-yl]oxyphenyl]-1,3-benzoxazol-2-amineIC5010.0 [1]
7-(5-Fluoro-2-methoxyphenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC5040.0 [1]
7-(2-Methoxy-4-methylphenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC5040.0 [1]
7-(1H-Indazol-7-yl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC5050.0 [1]
N-(3,4-Dimethoxyphenyl)-7-(2-fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-amineIC5070.0 [1]
N-(3,5-Dimethoxyphenyl)-7-(2-fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-amineIC50210.0 [1]
1-N-[7-(2-Fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-yl]-4-methoxybenzene-1,3-diamineIC50220.0 [1]
7-(2-Fluorophenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC50220.0 [1]
3-[[7-(2-Fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-yl]amino]benzenesulfonamideIC50340.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-N-(3-methoxyphenyl)-1,3-benzoxazol-2-amineIC50410.0 [1]
7-(2-Ethoxy-6-fluorophenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC50490.0 [1]
7-(2,5-Dimethyl-1H-imidazol-4-yl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC50560.0 [1]
N-Cyclohexyl-7-(2-fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-amineIC50620.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-N-(6-methoxypyridin-2-yl)-1,3-benzoxazol-2-amineIC50620.0 [1]
N-(3-Ethoxyphenyl)-7-(2-fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-amineIC50730.0 [1]
7-(2-Fluoro-6-propan-2-yloxyphenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC50970.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-N-phenyl-1,3-benzoxazol-2-amineIC501000.0 [1]
7-(2-Methoxy-5-methylphenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC501100.0 [1]
7-(2,6-Dimethoxyphenyl)-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC501200.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-N-(4-methoxyphenyl)-1,3-benzoxazol-2-amineIC501400.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-1,3-benzoxazol-2-amineIC502800.0 [1]
7-(2-Fluoro-6-methoxyphenyl)-N-(oxan-4-yl)-1,3-benzoxazol-2-amineIC503200.0 [1]
7-[2-(Trifluoromethoxy)phenyl]-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC504000.0 [1]
7-[2-(1H-Pyrazol-4-yl)phenyl]-N-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineIC509300.0 [1]
1-[4-(Dimethylamino)-7-(3-hydroxypropyl)-5-(4-methylphenyl)pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoroethanoneIC5015.0 [1]
N-[2-[(4-Methoxyanilino)methyl]-1,3-dioxoisoindol-5-yl]benzamideIC502160.0 [1]
N-[2-[(4-Ethoxyanilino)methyl]-1,3-dioxoisoindol-4-yl]benzamideIC501340.0 [1]
N-[2-[(4-Ethoxyanilino)methyl]-1,3-dioxoisoindol-5-yl]benzamideIC504580.0 [1]
5-Amino-2-[(4-methoxyanilino)methyl]isoindole-1,3-dioneIC50590.0 [1]
N-[2-[(4-Morpholin-4-ylanilino)methyl]-1,3-dioxoisoindol-5-yl]benzamideIC501010.0 [1]
4-Amino-2-[(4-methoxyanilino)methyl]isoindole-1,3-dioneIC503530.0 [1]
2-[(4-Methoxy-N-methylanilino)methyl]isoindole-1,3-dioneIC503500.0 [1]
N-[2-[(4-Methoxyanilino)methyl]-1,3-dioxoisoindol-4-yl]benzamideIC50990.0 [1]
2-[[4-(Diethylamino)-2-methylanilino]methyl]isoindole-1,3-dioneIC50860.0 [1]
2-{[(4-Ethoxyphenyl)amino]methyl}-1H-isoindole-1,3(2H)-dioneIC50590.0 [1]
(3S,4R)-N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-3,4-dimethyl-1-oxo-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carboxamideIC5013.7 [1]
(4R)-N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-4-methyl-1-oxo-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carboxamideIC500.7 [1]
N-[1-[3-(Dimethylamino)propyl]benzimidazol-2-yl]-4-methyl-1-oxo-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carboxamideIC501.3 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Ribosomal protein S6 kinase alpha 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/ribosomal-protein-s6-kinase-alpha-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Ribosomal protein S6 kinase alpha 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/ribosomal-protein-s6-kinase-alpha-2-inhibitors-ic50-ki.
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