![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 0.09 [1], 0.1 [2], 0.5 [3], 1.2 [4] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_c1fedebb567a4bbe6300695b40b3887d.svg) | 4-(4-Fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_7de5848be93196a6906eba944a298431.svg) | Sunitinib | IC50 | 131.3 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_986db0437f20070dfb14143a9f1b018d.svg) | Dasatinib | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_d2aaae557a3df420b61b69998679cc44.svg) | Dorsomorphin | IC50 | 210.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_1970071dd3288d1434749caa6fc51ef1.svg) | 4,5,6,7-Tetrabromo-N,N-dimethyl-1H-benzimidazol-2-amine | IC50 | 10280.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_67f4e732a49bf39a183fb443d695bf12.svg) | Gsk-690693 | IC50 | 1260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_3ac91c26cb3202821ba09ba5b9d46a48.svg) | Aminofurazanyl-azabenzimidazole 6n | IC50 | 132.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_27d3a5b4d06517b7e7f7d0e79a2b07e5.svg) | CID 44219749 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_2d4a41d2946c525e47a927da216ebe9a.svg) | CID 11373846 | IC50 | 780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_c3246aa6b96004698c3662ec45bb1de3.svg) | 1-(4-Methoxyphenyl)-3-[(2-oxo-3-indolyl)amino]thiourea | IC50 | 34900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_c9334335ebac282148ba5756199ea5fb.svg) | CID 11548023 | IC50 | 398.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_801b71b496c9e614d27c57f59ce0b9c5.svg) | (1S,2S,3R,4R)-3-[[5-Chloro-2-[[(7S)-4-methoxy-7-morpholin-4-yl-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | IC50 | 61.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_2c0a0e63fcc4b586a819f779a22a9560.svg) | 4-(3,4-Dichlorophenyl)-N-1H-indazol-5-yl-2-methyl-6-oxo-1,4,5,6-tetrahydropyridine-3-carboxamide | IC50 | 620.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_3f5d91104bea51924b42efba028274f1.svg) | N-(1H-Indazol-5-yl)-2-methyl-4-(naphthalen-2-yl)-6-oxo-1,4,5,6-tetrahydropyridine-3-carboxamide | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_f46848857eadb7aa4e51f68ae566468c.svg) | N-(7-Chloro-1H-indazol-5-yl)-6-methyl-2-oxo-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyridine-5-carboxamide | IC50 | 90.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_771a3e3be9214cf922dd59d632cab01b.svg) | 6-Methyl-N-(3-methyl-2H-indazol-5-yl)-2-oxo-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyridine-5-carboxamide | IC50 | 1950.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_4c2c70178609eb610c2ed8f1c8904f26.svg) | [2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethylimidazo[4,5-c]pyridin-7-yl]-[(3S)-3-aminopyrrolidin-1-yl]methanone | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_f78ea3f034b7b643fcb19743ec512abb.svg) | AKT Kinase Inhibitor | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_30ed6f9f9f64fdc67231237d542155b2.svg) | 4-[2-[4-(3-Pyridin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenoxy]ethyl]morpholine | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_2d6824ed4663109c98dca83443bd727c.svg) | 3-{[(1R)-1-Phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione | IC50 | 810.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_26b79855acfaf43486f6cc1e9ddde256.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[[(3R)-piperidin-3-yl]methoxy]imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 1580.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_37c7d87ae1e9271852ba4e05a57e8cac.svg) | CID 25207521 | IC50 | 290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_a393d807e71b1e743502e2b63e78a618.svg) | 3-[7-[4-[(1S,4S)-5-Methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]phenyl]-2-pyridin-4-ylpyrazolo[1,5-a]pyrimidin-3-yl]phenol | IC50 | 9710.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_9fca32ea610aad3b71b7d2f2c910911b.svg) | 5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4-difluorophenyl)-1,3-oxazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_7cdd83797fcf6ca18f71a608554760f2.svg) | 5-(3-Propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_b4dd7a10209bc305502c2cafde0001da.svg) | N-(1H-Indazol-5-yl)-6-methyl-2-oxo-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyridine-5-carboxamide | IC50 | 740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_ca56256dbfde6e99e0d7f49305cc3fb4.svg) | 4-[7-(3-Aminopropoxy)-1-ethyl-4-phenyl-1H-imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine | IC50 | 44.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_397a11e5d1e1ab8f6c5ab11957468e6c.svg) | 4-(4-Fluorophenyl)-N-1H-indazol-5-yl-2-methyl-6-oxo-1,4,5,6-tetrahydro-3-pyridinecarboxamide | IC50 | 1410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_5b5057f07ba36d969b42e83280bc9205.svg) | 2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_4fb3c780ee43b04b2acef5f8dad95f87.svg) | CID 11641672 | IC50 | 510.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 2000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_29a968cc679eba6bc716916267bc1ddb.svg) | 4-(4-Fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-phenyl-1,4-dihydropyrimidine-5-carboxamide | IC50 | 5300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_dc5ff7b87d06ec962585df9a614f5950.svg) | 6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_9d109cefe6f21cc70e74499a7c9999ec.svg) | 3-(5-Cyclopropyl-1,2-oxazol-3-yl)-1-propan-2-ylpyrazolo[3,4-d]pyrimidin-4-amine | IC50 | 311.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_f0a6d7d789748b78fa1d4f10c4672780.svg) | (5R)-4-[4-[4-[4-Fluoro-3-(trifluoromethyl)phenyl]-1-(2-pyrrolidin-1-ylethyl)imidazol-2-yl]piperidin-1-yl]-5-methyl-6,8-dihydro-5H-pyrido[2,3-d]pyrimidin-7-one | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_e93ac71a84d3e96fd4ecd266167cc03c.svg) | 4-[7-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-3-yl]-2-[(3-fluorophenyl)methoxy]benzamide | IC50 | 5.4 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_c009120ca19478ba69924ce16dc2791c.svg) | 5-(1,3-Benzodioxol-5-yl)-7-[[(2R)-1-ethenylsulfonylpyrrolidin-2-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_82bdac609f1a790e6d1a099d41b52a0a.svg) | N-(4-Fluoro-1H-indazol-5-yl)-6-methyl-2-oxo-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyridine-5-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_4c803290f0783d34222108e90172986d.svg) | 4-(2-Chloro-4-fluorophenyl)-5-(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-1,3-oxazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_56301d3a39833378c6b79294f2d7372e.svg) | N-Ethyl-6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-[1,2,4]triazolo[4,3-a]pyridin-3-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_fef81667a3c53467d05ea74c906edaac.svg) | 6-[5-(2,5-Difluorophenyl)-1H-pyrazol-4-yl]-3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_3f6d20bf74fd3158df4e50f5c54bf91b.svg) | 4-[(4-Methyl-1H-indol-5-yl)amino]-2-[(E)-3-oxo-3-pyrrolidin-1-ylprop-1-enyl]thieno[2,3-b]pyridine-5-carbonitrile | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_984f1d19dd4f7aff4c8096322cf2c2cd.svg) | 4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_cb053db390b2dde80b6fbaed2e18b924.svg) | 4-[7-(3-Aminopropoxy)-1-ethyl-4-(1H-pyrrol-2-yl)imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_67b1cbb25b30e03b9707e8442212bc24.svg) | 4-[7-(3-Aminopropoxy)-1-ethyl-4-(furan-3-yl)-1H-imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine | IC50 | 71.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_d33144cf34d45ce61c86d3279e8ce441.svg) | 4-[7-(3-Aminopropoxy)-4-(2-cyclopropylethynyl)-1-ethylimidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine | IC50 | 251.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_087850d81c02bfd5f3366989218cbe3f.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-7-(3-aminopropoxy)-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 1259.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_e7efc820b81f8550f5b246fa48c28182.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-7-(3-aminopropoxy)-1-ethylimidazo[4,5-c]pyridin-4-yl]but-3-yn-1-ol | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_f47fcae7b9325332760994745656cbfb.svg) | 4-[7-(4-Aminobutoxy)-2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 790.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_9d95da8be764a008fd84869f506a7eca.svg) | 4-[7-(2-Aminoethoxy)-2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_6b2df43f1c29435cc7e9821804998561.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-7-[(3S)-3-amino-4-phenylbutoxy]-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 1560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_b9f74dfbdf11995a7472448fffeec1e1.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-(pyrrolidin-3-ylmethoxy)imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 1990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_501d3543fd30778d492a661357182b3f.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[3-[2-(4-methoxyphenyl)ethylamino]propoxy]imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | IC50 | 2510.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_196a7a15c719c2eca6b5a2782fd41350.svg) | (2S)-3-[3-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-4-(3-hydroxy-3-methylbut-1-ynyl)imidazo[4,5-c]pyridin-7-yl]oxypropylamino]propane-1,2-diol | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_7a3912873517dd8f1c884dd46dd15a56.svg) | 2-{[3,4-Dioxo-2-(pyridin-4-ylamino)cyclobut-1-en-1-yl]amino}-2-phenylacetamide | IC50 | 780.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_fe36d92f25988fc0fb64ee4465475cb6.svg) | 5-[(E)-4-[(3R)-3-Aminopiperidin-1-yl]but-1-enyl]-4-[(4-methyl-1H-indol-5-yl)amino]pyridine-3-carbonitrile | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_84998d632a3b7b87a4bacd4e0d531dc0.svg) | 2-[9-(4-Amino-3-methoxyphenyl)-6-oxo-5,11-dihydrobenzo[b][1,4]benzodiazepin-3-yl]-2-methyl-N-(4-morpholin-4-ylphenyl)propanamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_68e0b5867fb9bf360f7aed3ad8804faf.svg) | N-(2-Hydroxyethyl)-4-[3-[(Z)-(4-hydroxy-3-oxo-1-benzofuran-2-ylidene)methyl]-1-methylpyrrolo[2,3-b]pyridin-4-yl]benzamide | IC50 | 45.9 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_87da122e718d4820b2d4f08b5fa3813e.svg) | 3-[[2-(2-Fluorophenyl)pyridin-4-yl]amino]-4-[[(1R)-1-phenylethyl]amino]cyclobut-3-ene-1,2-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_c6ccd24d8a2edf38937b57a99646617e.svg) | 3-[[2-(Furan-2-yl)pyridin-4-yl]amino]-4-[[(1R)-1-phenylethyl]amino]cyclobut-3-ene-1,2-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_f6fb842344d10989aa562e5395045b64.svg) | 3-[[(1R)-1-Phenylethyl]amino]-4-[(2-thiophen-3-ylpyridin-4-yl)amino]cyclobut-3-ene-1,2-dione | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_eb6227e6c3f665cde5788efe127c843a.svg) | Methyl 4-(6-(4-aminophenyl)-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carboxylate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_603383508252a1d5c473147ffda04752.svg) | Tert-butyl 4-[6-(4-aminophenyl)-4-morpholin-4-ylpyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carboxylate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_793d8427574718310b36bfc2f5b0ef6e.svg) | 4-(4-Methyl-1H-indol-5-ylamino)-5-(3-(4-methylpiperazin-1-ylsulfonyl)styryl)nicotinonitrile | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_e504da47f712ca636f26a8738cbed8f0.svg) | 6-Methyl-4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-methylpiperazin-1-ylsulfonyl)styryl)nicotinonitrile | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_856f48d6d8e8440f40e1ed1695d741b8.svg) | CID 46179972 | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_59c709e56f1adb4cd0a96f4865747914.svg) | 1-[4-[4-(3-Oxa-8-azabicyclo[3.2.1]octan-8-yl)-6-(oxan-4-yl)-1,3,5-triazin-2-yl]phenyl]-3-[4-(4-propan-2-ylpiperazine-1-carbonyl)phenyl]urea | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_d34c75fb9050e2e16397466a936a127d.svg) | 29-(Dimethylamino)-4,14,24,30-tetrazaheptacyclo[26.2.2.14,11.117,24.05,10.012,16.018,23]tetratriaconta-1(30),5,7,9,11(34),12(16),17(33),18,20,22,28,31-dodecaene-13,15-dione | IC50 | 1900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_19d87806bfcd06e051f3ad2c806548b2.svg) | 5-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-1H-pyridin-2-one | IC50 | 2100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_28b548e15ef703a72464d59e93c458d0.svg) | Akt-IN-2 | IC50 | 568.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_03e0d1a2e88126708ed3a73e7e36755b.svg) | N-[5-[6-(Methylamino)pyrazin-2-yl]-2-oxo-1H-pyridin-3-yl]-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]benzamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_b4f0fb1c5a1f23c97d46151f60f2159e.svg) | 4-(5-(3,4-Dihydroxyphenyl)oxazol-2-ylamino)benzenesulfonamide | IC50 | 3400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_2e820b24c0c89f65339aac9834e3d3d1.svg) | 4-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzene-1,2-diol | IC50 | 560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_83d53ff1245d9b17889c7c10e764e869.svg) | 4-[2-[4-[3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl]phenoxy]ethyl]morpholine | IC50 | 220.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_ced669c6e974600b4fc1c63722455698.svg) | 4-[6-[4-(2-Morpholin-4-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]pyridin-2-amine | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_03a1795ee46dd948346d1e0ae5e605bc.svg) | 4-(5-(6-Oxo-1,6-dihydropyridin-3-yl)oxazol-2-ylamino)benzenesulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_db3389b08cd7eeba89e218d8e3620d0a.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-(piperidin-4-ylmethoxy)imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol;2,2,2-trifluoroacetic acid | IC50 | 2510.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_ea81e59641f070d6bdb71c4cde14fed5.svg) | 4-[7-(3-Aminopropoxy)-4-(3-aminoprop-1-ynyl)-1-ethylimidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amine;2,2,2-trifluoroacetic acid | IC50 | 251.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_5bbe27113bc0daec23d38c87d11d8e85.svg) | 4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-piperidin-4-yloxyimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol;2,2,2-trifluoroacetic acid | IC50 | 3980.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_c6ea55529c818434f91884d3809a48a0.svg) | Chembl4126067 | IC50 | 699.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_963a77fd6dd698cea005ea3cf04aa4de.svg) | Chembl4129817 | IC50 | 272.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_0e0ca8b60f9e9baede875ef91e8a629c.svg) | 6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine | IC50 | 63000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_5925762966e15aa06de5e931b537fef1.svg) | 6-(2,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine | IC50 | 13000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_9b03225f89ed1195cf6b61682b2da5be.svg) | 1-[(3-Hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea;methanesulfonic acid | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_67a68f362dc2cbc72a35c44ed3ac2e77.svg) | 3-Isopropyl-6-(4-phenyl-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_bd46bf00317ff4d1e5227df76c07b701.svg) | 5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_87054ec7135bf0559e1278aece50ce7a.svg) | N-[2-(4-Chloro-3-fluorophenyl)ethyl]-7-(oxan-4-ylamino)-1,6-naphthyridine-2-carboxamide | IC50 | 476.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_b91719d8853b88df8a8feb22bde556f7.svg) | (3S,4S)-3-Methoxy-4-(methylamino)-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-16-one | IC50 | 0.19 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_ac3fd06308fe296febb2c43876a782a7.svg) | 2-[(Z)-[2-Bromo-6-(4-nitrophenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylideneamino]guanidine | IC50 | 1181.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_ddcbe403a159fe5f332550634fa54596.svg) | 6-(4-Fluorophenyl)sulfanyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 4253.0 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_610ea39af2773554c8f5fcb5e76f716d.svg) | N-[(1S)-1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl]-7-[(2-methylpyrazol-3-yl)amino]-1,6-naphthyridine-2-carboxamide | IC50 | 9.84 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_bff94d522ed8dbbb960f088c8819d644.svg) | N-[(S)-(3-Fluoro-4-methoxyphenyl)-(1-methylpyrazol-4-yl)methyl]-7-[[(2S)-1-hydroxypropan-2-yl]amino]-1,6-naphthyridine-2-carboxamide | IC50 | 37.8 [1] |
![](https://images.aatbio.com/dataset/ic50/ribosomal-protein-s6-kinase-alpha-1_670812feaa492318332d5980c167f4e3.svg) | N-[(1S)-1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl]-3-(oxan-4-ylamino)isoquinoline-6-carboxamide | IC50 | 14.8 [1] |