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Retinoic acid receptor beta Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
TretinoinIC500.9 [1], 0.94 [2], 13.0 [3], 3000.0 [4]
TretinoinKi0.4 [1], 0.5 [2], 4.1 [3], 7.0 [4], 17.4 [5]
BexaroteneKi1000.0 [1], 5353.0 [2]
AlitretinoinIC507.0 [1]
AlitretinoinKi0.5 [1], 0.7 [2], 10.9 [3]
TtnpbIC505.0 [1]
TtnpbKi0.5 [1], 5.0 [2]
AdapaleneKi34.0 [1]
6-(1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopropyl)nicotinic acidKi1000.0 [1], 9901.0 [2]
(2E,4E,6Z)-7-[3,5-Ditert-butyl-2-(2,2-difluoroethoxy)phenyl]-3-methylocta-2,4,6-trienoic acidKi4687.0 [1], 9513.0 [2]
6-(1,2,3,4-Tetrahydro-1,1,4,4-tetramethyl-6-naphthyl)-2-naphthalenecarboxylic acidKi13.0 [1]
6-(3-Tert-butyl-4-hydroxyphenyl)-2-naphthoic acidKi3000.0 [1], 3550.0 [2]
(2E,4E)-3-Methyl-5-[2-[(E)-2-(3,3,6,6-tetramethylcyclohexen-1-yl)ethenyl]cyclopropyl]penta-2,4-dienoic acidKi11.0 [1], 13.0 [2]
(2Z,4E)-3-Methyl-5-[2-[(E)-2-(3,3,6,6-tetramethylcyclohexen-1-yl)ethenyl]cyclopropyl]penta-2,4-dienoic acidKi1100.0 [1], 1200.0 [2]
TamibaroteneKi30.0 [1]
6-[3-(1-Adamantyl)-4-hydroxyphenyl]-2-naphthalenecarboxylic AcidKi2480.0 [1]
4-[2-[5,5-Dimethyl-8-(4-methylphenyl)-6H-naphthalen-2-yl]ethynyl]benzoic acidIC5020.0 [1]
4-(2,18,18,21,21-Pentamethyl-2,14-diazapentacyclo[13.8.0.03,12.04,9.017,22]tricosa-1(15),3(12),4,6,8,10,13,16,22-nonaen-13-yl)benzoic acidKi500.0 [1]
4-(5,7,7,10,10-Pentamethyl-8,9-dihydronaphtho[2,3-b][1,4]benzodiazepin-13-yl)benzoic acidKi220.0 [1]
(2E,4E,6Z)-3-Methyl-7-(5,5,8,8-tetramethyl-3-propoxy-6,7-dihydronaphthalen-2-yl)octa-2,4,6-trienoic acidKi2587.0 [1]
4-(5,6,7,8-Tetrahydro-5,5,8,8-tetramethyl-2-anthracenyl)benzoic acidKi3.0 [1]
4-(7,7,10,10-Tetramethyl-8,9-dihydronaphtho[2,3-b][1,5]benzothiazepin-12-yl)benzoic acidKi320.0 [1]
4-(5,7,7,10,10-Pentamethyl-8,9-dihydronaphtho[2,3-b][1,5]benzodiazepin-12-yl)benzoic acidKi680.0 [1]
6-(4-Methoxy-3-(1-methylcyclohexyl)phenyl)-2-naphthalenecarboxylic acidKi26.0 [1]
7-(3,5-Ditert-butylphenyl)-3-methylocta-2,4,6-trienoic acidKi0.7 [1]
Benzoic acid, 4-(4-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-quinoxalinyl)-2-thiazolyl)-IC5021.0 [1]
6-[[3-[(2S)-1-Methoxypropan-2-yl]oxy-5-[(2S)-1-phenylpropan-2-yl]oxybenzoyl]amino]pyridine-3-carboxylic acidIC5032000.0 [1]
4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydronaphthalene-2-carbonyl)benzoic acidKi10000.0 [1]
4-[5-(4-Phenyl-8-propan-2-ylquinolin-2-yl)-1H-pyrrol-2-yl]benzoic acidIC503000.0 [1]
4-(2-(5,6,7,8-Tetrahydro-3,5,5,8,8-pentamethyl-2-naphthalenyl)-1-propenyl) benzoic acidIC501169.0 [1]
(2E,4E,6E,8E)-3,7-Dimethyl-9-[2,6,6-trimethyl-3-(1,2,4-triazol-1-yl)cyclohexen-1-yl]nona-2,4,6,8-tetraenoic acidIC501000000.0 [1]
Benzoic acid, 4-(5-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-quinoxalinyl)-1H-pyrrol-2-yl)-IC50230.0 [1]
4-((+/-)-(1H-Imidazol-1-yl)-(E)-retinoic acidIC50175000.0 [1]
(2E,4E,6E,8E)-3,7-Dimethyl-9-[2,6,6-trimethyl-3-(1,2,4-triazol-4-yl)cyclohexen-1-yl]nona-2,4,6,8-tetraenoic acidIC50250000.0 [1]
4-[(5,5,8,8-Tetramethyl-6,7-dihydroquinoxaline-2-carbonyl)amino]benzoic acidIC50140.0 [1]
4-[(E)-2-(3-Tert-Butyl-4-methoxy-phenyl)-propenyl]-benzoic acidKi12.0 [1]
(S)-6-(3-(3,5-Difluorophenoxy)-5-(1-methoxypropan-2-yloxy)benzamido)nicotinic acidIC501.0 [1]
(2E,4E,6E)-7-[3,5-Ditert-butyl-2-(2,2-difluoroethoxy)phenyl]-6-fluoro-3-methylocta-2,4,6-trienoic acidKi5681.0 [1]
4-[1-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-vinyl]-benzoic acidKi909.0 [1]
(2E,4E,6Z)-7-[2-(2,2-Difluoroethoxy)-5-(2-fluorophenyl)-3-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi3927.0 [1]
4-[(E)-2-(3-Ethyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-propenyl]-benzoic acidIC5075.0 [1]
(2E,4E)-5-[2-[3,5-Di(propan-2-yl)-2-(2,2,2-trifluoroethoxy)phenyl]cyclopenten-1-yl]-3-methylpenta-2,4-dienoic acidKi4742.0 [1]
6-(3-Isobutoxy-5-isopropoxy-benzoylamino)-nicotinic acidIC50135.0 [1]
4-(7,7,10,10-Tetramethyl-8,9-dihydronaphtho[2,3-b][1,5]benzoxazepin-12-yl)benzoic acidKi320.0 [1]
4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-anthracen-2-yl)-benzoic acidIC5022.0 [1]
4-[5,5-Dimethyl-8-(5-methyl-2-thienyl)-5,6-dihydroanthracene-2-yl]benzoic acidIC5015.0 [1]
6-[3-Adamantan-1-yl-4-(1,2-dihydroxy-ethyl)-phenyl]-naphthalene-2-carboxylic acidKi288.0 [1]
6-[3-Adamantan-1-yl-4-(2,3-dihydroxy-propoxy)-phenyl]-naphthalene-2-carboxylic acidKi89.0 [1]
4-{(E)-4-[2-(4-Tert-Butyl-phenyl)-6,6-dimethyl-cyclohex-1-enyl]-but-3-en-1-ynyl}-benzoic acidIC5025.0 [1]
4-(8,8,11,11-Tetramethyl-10,13-dihydro-9H-naphtho[2,3-c][1]benzazepin-6-yl)benzoic acidKi810.0 [1]
4-[(E)-2-(3-Isopropyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-propenyl]-benzoic acidIC50150.0 [1]
4-[(E)-4-(3,3-Dimethyl-6-p-tolyl-cyclohexa-1,5-dienyl)-but-3-en-1-ynyl]-benzoic acidIC5053.0 [1]
4-[(E)-2-(3-Adamantan-1-yl-4-hydroxy-phenyl)-propenyl]-benzoic acidKi1245.0 [1]
6-[3-(1-Adamantyl)-4-(2,3-dihydroxypropyl)phenyl]-2-naphthoic acidKi158.0 [1]
4-(2,2-Dimethyl-4-p-tolyl-2H-1-thia-anthracen-6-yl)-benzoic acidIC502.0 [1]
4-[(E)-2-(3-Tert-butyl-4-hydroxyphenyl)propenyl]benzoic acidKi105.0 [1]
4-[(E)-2-[3-(1-Adamantyl)-4-hydroxyphenyl]ethenyl]benzoic acidKi70.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)thiophen-3-yl]benzoic acidIC504.5 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)furan-3-yl]benzoic acidIC502.5 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)thiophen-2-yl]benzoic acidIC5036.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)furan-2-yl]benzoic acidIC5039.0 [1]
(2E,4E,6Z)-7-(3-Ethoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-3-methylocta-2,4,6-trienoic acidKi3115.0 [1]
4-{(E)-2-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl]-propenyl}-benzoic acidKi90.0 [1]
4-[(E)-2-(3-(1-Methylcyclohexyl)-4-methoxyphenyl)propenyl]benzoic acidKi17.0 [1]
4-[5-(5,5,8,8-Tetramethyl-6,7-dihydroquinoxalin-2-yl)-1H-pyrazol-3-yl]benzoic acidIC50290.0 [1]
6-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl]-naphthalene-2-carboxylic acidKi660.0 [1]
4-[(E)-2-(3-Adamantan-1-yl-4-methoxy-phenyl)-propenyl]-benzoic acidKi105.0 [1]
6-(3-Adamantan-1-yl-4-carboxy-phenyl)-naphthalene-2-carboxylic acidKi10000.0 [1]
6-[3-(1-Adamantyl)-4-(3-hydroxypropyl)phenyl]-2-naphthoic acidKi21.0 [1]
(2E,4E)-5-[3-[3,5-Di(propan-2-yl)-2-(2,2,2-trifluoroethoxy)phenyl]pyridin-4-yl]-3-methylpenta-2,4-dienoic acidKi2056.0 [1]
(2E,4E)-5-[3-[2-(3-Fluoropropoxy)-3,5-di(propan-2-yl)phenyl]thiophen-2-yl]-3-methylpenta-2,4-dienoic acidKi10000.0 [1]
(2E,4E)-5-[3-[3,5-Di(propan-2-yl)-2-(2,2,2-trifluoroethoxy)phenyl]thiophen-2-yl]-3-methylpenta-2,4-dienoic acidKi10000.0 [1]
(2E,4E)-5-[3-[3,5-Ditert-butyl-2-(3,3-difluoropropoxy)phenyl]thiophen-2-yl]-3-methylpenta-2,4-dienoic acidKi10000.0 [1]
(2E,4E,6E,8E)-3,7-Dimethyl-1-(1,2,4-triazol-1-yl)-9-(2,6,6-trimethylcyclohexen-1-yl)nona-2,4,6,8-tetraen-1-oneIC5090000.0 [1]
(2Z,4E,6E,8E)-9-(3-Imidazol-1-yl-2,6,6-trimethylcyclohexen-1-yl)-3,7-dimethylnona-2,4,6,8-tetraenoic acidIC50175000.0 [1]
(2E,4E,6E,8E)-1-Imidazol-1-yl-3,7-dimethyl-9-(2,6,6-trimethylcyclohexen-1-yl)nona-2,4,6,8-tetraen-1-oneIC50500000.0 [1]
(2E,4E,6Z)-7-(3-Methoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)-3-methylocta-2,4,6-trienoic acidKi400.0 [1]
6-(3-Adamantan-1-yl-4-hexyloxy-phenyl)-naphthalene-2-carboxylic acidKi10000.0 [1]
4-[5-(1,1,4,4-Tetramethyltetralin-6-yl)-1H-pyrrole-2-yl]benzoic acidIC50100.0 [1]
(2E,4E,6Z)-7-[2-(2,2-Difluoroethoxy)-3-propan-2-yl-5-thiophen-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi2112.0 [1]
(2E,4E,6E)-7-[2-Butoxy-3,5-di(propan-2-yl)phenyl]-6-fluoro-3-methylocta-2,4,6-trienoic acidKi4623.0 [1]
(2E,4E,6Z)-7-[2-(2,2-Difluoroethoxy)-5-(3-fluorophenyl)-3-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi3597.0 [1]
(2E,4E,6Z)-7-[2-(2,2-Difluoroethoxy)-5-(3,5-difluorophenyl)-3-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi1956.0 [1]
(2E,4E,6Z)-3-Methyl-7-[3-(1,1,2,2,2-pentafluoroethyl)-5-propan-2-yl-2-propoxyphenyl]octa-2,4,6-trienoic acidKi10000.0 [1]
(2E,4E,6Z)-7-[2-(2,2-Difluoroethoxy)-3-phenyl-5-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi2612.0 [1]
(2E,4E,6Z)-3-Methyl-7-[5-(1,1,2,2,2-pentafluoroethyl)-3-propan-2-yl-2-propoxyphenyl]octa-2,4,6-trienoic acidKi1984.0 [1]
(2E,4E,6Z)-7-[2-Ethoxy-5-(1,1,2,2,2-pentafluoroethyl)-3-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi10000.0 [1]
6-(4,4-Dimethyl-chroman-6-yl)-naphthalene-2-carboxylic acidKi210.0 [1]
6-[3,5-Bis-(2-fluoro-benzyloxy)-benzoylamino]-nicotinic acidIC507.0 [1]
(2E,4E)-2,4-Dimethyl-5-(6,6,9,9-tetramethyl-4-oxo-7,8-dihydrobenzo[g]chromen-3-yl)penta-2,4-dienoic acidIC5040.0 [1]
6-(3-Tert-butyl-4-methoxyphenyl)naphthalene-2-carboxylic acidKi36.0 [1]
4-[(E)-4-(6,6-Dimethyl-2-p-tolyl-cyclohex-1-enyl)-but-3-en-1-ynyl]-benzoic acidIC5022.0 [1]
(2E,4E)-5-[3-[2-(2,2-Difluoroethoxy)-3,5-di(propan-2-yl)phenyl]thiophen-2-yl]-3-methylpenta-2,4-dienoic acidKi4064.0 [1]
(2E,4E)-5-[2-[3,5-Ditert-butyl-2-(3-fluoropropoxy)phenyl]phenyl]-3-methylpenta-2,4-dienoic acidKi10000.0 [1]
6-(3-Adamantan-1-yl-4-hydroxymethyl-phenyl)-naphthalene-2-carboxylic acidKi156.0 [1]
4-[2,2-Dimethyl-4-(5-methyl-thiophen-2-yl)-2H-benzo[g]chromen-7-yl]-benzoic acidIC506.5 [1]
(2E,4E,6Z)-7-[2-Butoxy-5-(1,1,2,2,2-pentafluoroethyl)-3-propan-2-ylphenyl]-3-methylocta-2,4,6-trienoic acidKi2270.0 [1]
4-[(Z)-(Hydroxyimino)(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphthalene-2-yl)methyl]benzoic acidKi10000.0 [1]
4-{(E)-4-[2-(4-Ethyl-phenyl)-6,6-dimethyl-cyclohex-1-enyl]-but-3-en-1-ynyl}-benzoic acidIC5040.0 [1]
(2E,4E)-5-[2-[2-(2,2-Difluoroethoxy)-3,5-di(propan-2-yl)phenyl]cyclopenten-1-yl]-3-methylpenta-2,4-dienoic acidKi10000.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Retinoic acid receptor beta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/retinoic-acid-receptor-beta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Retinoic acid receptor beta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/retinoic-acid-receptor-beta-inhibitors-ic50-ki.
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