 | 4-(4-Fluorobenzyl)-2-p-tolyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 30.0 [1], 30.1 [2] |
 | Unii-9egb3J3KI5 | IC50 | 100000.0 [1] |
 | 1-Benzyl-3-p-tolyl-1H-pyrrole-2,5-dione | IC50 | 93000.0 [1], 93300.0 [2] |
 | 4-Butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 14.4 [1] |
 | RGS4 inhibitor 13 | IC50 | 54.3 [1] |
 | 4-Benzyl-2-phenyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 23.5 [1] |
 | 4-Benzyl-2-(4-methoxyphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 23.9 [1] |
 | 4-Benzyl-2-(4-methyl-benzyl)-[1,2,4]thiadiazolidine-3,5-dione | IC50 | 7.2 [1] |
 | 2-Ethyl-4-methyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 22.3 [1] |
 | 2-Butyl-4-methyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 23.5 [1] |
 | 2,4-Dibutyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 29.8 [1] |
 | 4-[(4-Methoxyphenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 176.0 [1] |
 | 4-[(4-Fluorophenyl)methyl]-2-(3-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 121.0 [1] |
 | 2-(3-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 52.3 [1] |
 | 2-(4-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 13.5 [1] |
 | 2-Butyl-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 15.6 [1] |
 | 4-Benzyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 14.4 [1] |
 | 4-Benzyl-2-(4-chlorophenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 28.7 [1] |
 | 4-Benzyl-2-[3-(trifluoromethyl)phenyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 57.4 [1] |
 | 4-[(4-Chlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 5.4 [1] |
 | 4-[(3-Chlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 17.4 [1] |
 | 4-[(3,4-Dichlorophenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 34.2 [1] |
 | 4-Butyl-2-tert-butyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 53.6 [1] |
 | 2-Ethyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 26.3 [1] |
 | 2-Tert-butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 29.1 [1] |
 | 4-[(4-Fluorophenyl)methyl]-2-[(4-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 12.9 [1] |
 | 2-(4-Methylphenyl)-4-[(3-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 14.5 [1] |
 | 2-(4-Methylphenyl)-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 14.0 [1] |
 | 2-Butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 38.6 [1] |
 | 2-(3,4-Dichlorophenyl)-4-[(4-fluorophenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 35.7 [1] |
 | 4-Benzyl-2-(3-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 38.2 [1] |
 | 2-(4-Methylphenyl)-4-[(4-methylphenyl)methyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 8.6 [1] |
 | 4-[(4-Fluorophenyl)methyl]-2-(4-methoxyphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 10.9 [1] |
 | 2-Tert-butyl-4-methyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 27.8 [1] |
 | 4-[(4-Fluorophenyl)methyl]-2-[3-(trifluoromethyl)phenyl]-1,2,4-thiadiazolidine-3,5-dione | IC50 | 79.3 [1] |
 | 4-Benzyl-2-(3,4-dichlorophenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 88.9 [1] |
 | 4-Methyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 18.9 [1] |
 | 4-[(4-Fluorophenyl)methyl]-2-phenyl-1,2,4-thiadiazolidine-3,5-dione | IC50 | 16.3 [1] |
 | 4-Butyl-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 19.7 [1] |
 | 4-Benzyl-2-(3-chlorophenyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 32.5 [1] |
 | 2-Ethyl-4-(4-fluorobenzyl)-1,2,4-thiadiazolidine-3,5-dione | IC50 | 22.3 [1] |
 | 1-Benzyl-3-bromo-1H-pyrrole-2,5-dione | IC50 | 32000.0 [1] |