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Receptor tyrosine-protein kinase erbB-3 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
ErlotinibIC5010.0 [1]
OsimertinibIC502.1 [1]
RociletinibIC5046.0 [1]
SapitinibIC504.0 [1]
4-Fluoro-N-[6-(4-morpholinyl)-4-pyrimidinyl]benzamideIC5096.0 [1]
Unii-5IE92SK9EBIC5021.0 [1]
N-[(3R,4R)-4-Fluoro-1-[6-[(1-methylpyrazol-4-yl)amino]-9-propan-2-ylpurin-2-yl]pyrrolidin-3-yl]prop-2-enamideIC502.0 [1]
N-[(3R,4R)-1-[6-[(1,3-Dimethylpyrazol-4-yl)amino]-9-propan-2-ylpurin-2-yl]-4-fluoropyrrolidin-3-yl]prop-2-enamideIC509.0 [1]
N-[4-(3-Chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]prop-2-enamideIC501.0 [1]
MavelertinibIC504.0 [1]
4-N-(2,5-Dimethoxyphenyl)-6-N-(4-fluorophenyl)pyrimidine-4,6-diamineIC50230.0 [1]
4-N-(3-Chlorophenyl)-6-N-(3-methoxyphenyl)pyrimidine-4,6-diamineIC501573.0 [1]
6-N-(4-Chlorophenyl)-4-N-(3,4,5-trimethoxyphenyl)pyrimidine-4,6-diamineIC5010000.0 [1]
4-N-(2,5-Dimethoxyphenyl)-6-N-(3-methoxyphenyl)pyrimidine-4,6-diamineIC5018.0 [1]
Ethyl 4-[[6-(3-methoxyanilino)pyrimidin-4-yl]amino]benzoateIC501745.0 [1]
N-[(3R,4R)-4-Fluoro-1-[6-[(3-methoxy-1-methylpyrazol-4-yl)amino]-9-propan-2-ylpurin-2-yl]pyrrolidin-3-yl]prop-2-enamideIC502.0 [1]
N-[4-(4-Methylpiperazin-1-yl)phenyl]-9-(oxan-4-yl)-8-phenylsulfanylpurin-2-amineIC502.0 [1]
N-[4-[2-(Dimethylamino)ethoxy]phenyl]-9-(oxan-4-yl)-8-phenylsulfanylpurin-2-amineIC501.7 [1]
N-[4-[2-(Dimethylamino)ethoxy]phenyl]-8-(4-fluorophenyl)sulfanyl-9-(oxan-4-yl)purin-2-amineIC501.2 [1]
N-[4-[4-(Dimethylamino)piperidin-1-yl]phenyl]-9-(oxan-4-yl)-8-phenylsulfanylpurin-2-amineIC501.9 [1]
8-(Benzenesulfinyl)-N-[4-[2-(dimethylamino)ethoxy]phenyl]-9-(oxan-4-yl)purin-2-amineIC502.6 [1]
N-[4-[2-(Dimethylamino)ethoxy]phenyl]-8-(3-fluorophenyl)sulfanyl-9-(oxan-4-yl)purin-2-amineIC505.8 [1]
5-(4-Methylphenyl)-3-naphthalen-2-yl-2-phenyl-3,4-dihydropyrazoleIC5045300.0 [1]
8-(Benzenesulfinyl)-9-cyclopentyl-N-[4-(4-methylpiperazin-1-yl)phenyl]purin-2-amineIC504.2 [1]
4-[2-[4-(4-Methylpiperazin-1-yl)anilino]-8-phenylsulfanylpurin-9-yl]cyclohexan-1-olIC502.4 [1]
9-Cyclopentyl-N-[4-(4-methylpiperazin-1-yl)phenyl]-8-phenylsulfanylpurin-2-amineIC504.2 [1]
N-[2-[2-(Dimethylamino)ethyl-methylamino]-4-methoxy-5-[[2-(1-methylindol-3-yl)pyrimidin-4-yl]amino]phenyl]prop-2-enamideIC5036.0 [1]
4-N-(2,5-Dimethoxyphenyl)-6-N-(2-thiophen-2-ylethyl)pyrimidine-4,6-diamineIC50167.0 [1]
N-[6-(4-Chloroanilino)pyrimidin-4-yl]-4-fluorobenzamideIC501608.0 [1]
5-[[6-(3-Chloroanilino)pyrimidin-4-yl]amino]-5-oxopentanoic acidIC5021.0 [1]
Ethyl 5-[[6-(3-chloroanilino)pyrimidin-4-yl]amino]-5-oxopentanoateIC5010000.0 [1]
5-[(6-Anilinopyrimidin-4-yl)amino]-5-oxopentanoic acidIC50183.0 [1]
5-[[6-(2,5-Dimethoxyanilino)pyrimidin-4-yl]amino]-5-oxopentanoic acidIC5010000.0 [1]
4-[[6-(2,5-Dimethoxyanilino)pyrimidin-4-yl]amino]benzenesulfonamideIC50619.0 [1]
N-[6-(4-Ethoxyanilino)pyrimidin-4-yl]benzamideIC501209.0 [1]
5-[[6-(4-Chloroanilino)pyrimidin-4-yl]amino]-5-oxopentanoic acidIC501322.0 [1]
5-[[6-(4-Ethoxycarbonylanilino)pyrimidin-4-yl]amino]-5-oxopentanoic acidIC5069.0 [1]
4-N-(2,5-Dimethoxyphenyl)-6-N-[4-(4-methylpiperazin-1-yl)phenyl]pyrimidine-4,6-diamineIC50167.0 [1]
6-N-(4-Chlorophenyl)-4-N-(6-chloropyridin-2-yl)pyrimidine-4,6-diamineIC50236.0 [1]
N-[6-(4-Methoxyanilino)pyrimidin-4-yl]benzamideIC5060.0 [1]
4-[[6-(3-Methoxyanilino)pyrimidin-4-yl]amino]benzenesulfonamideIC501847.0 [1]
5-[[6-(3-Bromoanilino)pyrimidin-4-yl]amino]-5-oxopentanoic acidIC5010000.0 [1]
4-[[6-(4-Chloroanilino)pyrimidin-4-yl]amino]-4-oxobutanoic acidIC50825.0 [1]
5-[(6-Morpholin-4-ylpyrimidin-4-yl)amino]-5-oxopentanoic acidIC5027.0 [1]
Ethyl 4-[[6-(3-bromoanilino)pyrimidin-4-yl]amino]-4-oxobutanoateIC501345.0 [1]
5-[[6-(3-Methoxyanilino)pyrimidin-4-yl]amino]-5-oxopentanoic acidIC5031.0 [1]
4-N-(3-Chlorophenyl)-6-N-ethylpyrimidine-4,6-diamineIC5010000.0 [1]
3-(4-Methoxyphenyl)-5-(1-naphthyl)-2-pyrazoline-1-carbothioamideIC5055600.0 [1]
5-(4-Methoxyphenyl)-3-naphthalen-1-yl-2-phenyl-3,4-dihydropyrazoleIC5040200.0 [1]
5-(4-Methylphenyl)-3-naphthalen-2-yl-3,4-dihydropyrazole-2-carbothioamideIC5063200.0 [1]
5-(3,4-Dichlorophenyl)-3-naphthalen-2-yl-3,4-dihydropyrazole-2-carbothioamideIC5051700.0 [1]
1-Phenyl-3-(3,4-dichlorophenyl)-5-(2-naphthyl)-2-pyrazolineIC5035900.0 [1]
Items per page: 1 - 10 of 52
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References

This online tool may be cited as follows

MLA

"Quest Database™ Receptor tyrosine-protein kinase erbB-3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/receptor-tyrosine-protein-kinase-erbb-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Receptor tyrosine-protein kinase erbB-3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/receptor-tyrosine-protein-kinase-erbb-3-inhibitors-ic50-ki.
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