![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_291fdc26c251ab1eb139e1406ed05831.svg) | Canertinib | IC50 | 10.0 [1], 14.0 [2], 27.0 [3], 31.0 [4] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_01384179eb1c1c1ef001bfbf31bfa500.svg) | Ibrutinib | IC50 | 0.1 [1], 1.8 [2] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 28.3 [1], 282.0 [2] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_e5e549ece7aea0a406367a90c52ffced.svg) | Dacomitinib | IC50 | 74.0 [1], 83.67 [2] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_9dd6da7cb57ea869429d2bb32c1c121c.svg) | 2-PropenaMide, N-[cis-4-[4-aMino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyriMidin-1-yl]cyclohexyl]- | IC50 | 3.2 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_3bd5dcd12d2ef57fd5cbefabf7849aa3.svg) | Gefitinib | IC50 | 476.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_e2f99194617c96946324b426e112d809.svg) | Erlotinib | IC50 | 1130.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_755000a88f2651809d912de0f446bcfe.svg) | Lapatinib | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_5a6f7b0bc67aeb9c222e12402dcf8759.svg) | Dacomitinib monohydrate | IC50 | 74.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a257c791d1de1df5d4a1fa04612f9c76.svg) | Nvp-aew541 | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_997fe095318226e799cbe61db5e4d8fd.svg) | 4-[(3-Bromophenyl)amino]-6-acrylamidoquinazoline | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_eb1729f98bdd8714dc7d292bc1ad0548.svg) | Cfms Receptor Tyrosine Kinase Inhibitor | IC50 | 24000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_302100520865fe19cc7f043083882d93.svg) | N-(4-((3-Bromophenyl)amino)quinazolin-6-yl)but-2-ynamide | IC50 | 12.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_20beeda5bb0152c29cef63a6468d977e.svg) | N6,N6-Dimethyl-N4-[1-(phenylmethyl)-5-indazolyl]pyrido[3,4-d]pyrimidine-4,6-diamine | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_c74a1b9d6feb1def6b7e3f6834b5761b.svg) | Tak-285 | IC50 | 260.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_24babf0b715d6efc28c3720939ee7d34.svg) | Bms-599626 | IC50 | 190.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_f02c1e14dc540300fe73303dae37c549.svg) | N-(2,6-Difluorophenyl)-5-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]-2-methoxybenzamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_c836f354b1a8144ea297d57d99d66267.svg) | PD-153035 hydrochloride | IC50 | 49.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_07d2d0af7904836ad3cf5ea2273c6a53.svg) | 1-((2S,5R)-5-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-yl)prop-2-en-1-one | IC50 | 25200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_9041d8083a937939ecc814af0ee443d4.svg) | Evobrutinib | IC50 | 37.9 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_f86db8122447b42c0e9cd9b49b1fcfd3.svg) | EGFR Inhibitor | IC50 | 7640.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_5652cbb626eaea3175445f98e056e324.svg) | EGFR/ErbB-2/ErbB-4 Inhibitor | IC50 | 0.5 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_e07c8cd6f81fa23b777a36d7d9709688.svg) | 4-Tert-Butyl-N-[6-(1h-Imidazol-1-Yl)imidazo[1,2-A]pyridin-2-Yl]benzamide | IC50 | 19952.62 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_7cd07c14c9a6699a18c59379f39dd9e2.svg) | N~3~-Cyclopropyl-N~4~'-(Cyclopropylmethyl)-6-Methylbiphenyl-3,4'-Dicarboxamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_601e453d7a089204e0a249b45693b4d5.svg) | 2-(4-Fluorophenyl)-3-(4-pyridinyl)pyrazolo[1,5-a]pyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_c33074e1aa4339917412ec783090268d.svg) | 2-Methyl-N-[2-[3-[[2-(prop-2-enoylamino)acetyl]amino]anilino]pyrimidin-5-yl]-5-[[3-(trifluoromethyl)benzoyl]amino]benzamide | IC50 | 3.3 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_628e796c331326ac7d59e9f8e229eaa5.svg) | 6,6-Dimethyl-8-[1-(oxan-4-ylmethyl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile | IC50 | 213.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_07a9a7dadcb6403aa1be2fdac16a78df.svg) | JAK3 covalent inhibitor-1 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a8db7d1164098dbe83e74bfac894881a.svg) | 4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide | Ki | 3800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 3750.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_db1cea5586701bc53652f3f79d33c46d.svg) | 2-Methyl-N-[2-[3-(prop-2-enoylamino)anilino]pyrimidin-5-yl]-5-[[3-(trifluoromethyl)benzoyl]amino]benzamide | IC50 | 5.5 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_0731e513dda8b4631f904dc8f0082e8c.svg) | 7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_1fe60e6d13674f8cf1dfc82fac3410b2.svg) | 7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrile | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_029f5b4cad89a2c59efa869fd9853874.svg) | N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamide | Ki | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_482caccce5577424472b4f30ef45663d.svg) | [6-Chloro-4-methyl-3-[[3-(methylsulfamoylamino)phenyl]methyl]-2-oxochromen-7-yl] N,N-dimethylcarbamate | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_b80728998e0b173ed97842a79c1db051.svg) | 5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_d177c352a8a90316beccdf76166341e8.svg) | N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamide | IC50 | 18.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_4f696c52d1e67bdfa2fa3a5dad0f0d31.svg) | CID 46927672 | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_335af318a60a5aef7318895fe8f1ffa2.svg) | N-[[2-[4-Amino-6-[3-chloro-4-(pyridin-2-ylmethoxy)anilino]pyrimidin-5-yl]-1,3-oxazol-4-yl]methyl]prop-2-enamide | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_f83aeef223e4cffa787f7bf871c66dc3.svg) | 1-(4-Fluorophenyl)-N-[3-fluoro-4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)oxyphenyl]-2-oxopyridine-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_400786f64062ecb5f10a9d3b11455207.svg) | 1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_84ad2ce5fbf306770a6c850a5b17125a.svg) | 9-Cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_cfc75c4c6279f580d70c524b8b3dff09.svg) | (E)-4-(Dimethylamino)-N-[7-fluoro-4-(2-methylanilino)imidazo[1,5-a]quinoxalin-8-yl]-N-methylbut-2-enamide | IC50 | 43.7 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_77f4b74dc836b9bdb4b558af6f5da27f.svg) | 6-(6-Fluoroindol-1-yl)-2-[2-[7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyethyl]pyridazin-3-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a39c97bae3f00a1b6b8da340592659ae.svg) | N-Cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a67b4a9432e9d562090f947d3c04935f.svg) | N-[4-Methyl-3-[2-methyl-4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl]-2-pyrrolidin-1-ylpyridine-4-carboxamide | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_0ce0167481b175c14fe1e1be1b692040.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-[di(propan-2-yl)amino]but-2-ynamide | IC50 | 538.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_870e7a8e13b27676c665793a0e944ab9.svg) | N-[4-(3-Chloro-4-fluoroanilino)quinazolin-6-yl]-4-morpholin-4-ylbut-2-ynamide | IC50 | 229.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_17eca8e9a13fdb5b6814b055548007cc.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-5-(4-methylpiperazin-1-yl)pent-2-ynamide | IC50 | 1.2 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a38029b1a4e785b051ad338e5c1d265a.svg) | N-[4-(3-Chloro-4-fluoroanilino)quinazolin-6-yl]-4-(dibutylamino)but-2-ynamide | IC50 | 624.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_e741bda6866d0137e01d8265edf78555.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]hept-2-ynamide | IC50 | 7.1 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a47f66b27465c169918987821c0d6fb6.svg) | N-[4-(3-Chloro-4-fluoroanilino)quinazolin-6-yl]-5-(diethylamino)pent-2-ynamide | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_fd856eadb598e69541c3332794f5bcd2.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-morpholin-4-ylbut-2-ynamide | IC50 | 6.2 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_74a8d1b1cda6db01284b7283b7473d56.svg) | N-[4-(3-Chloro-4-fluoroanilino)quinazolin-6-yl]-4-(diethylamino)but-2-ynamide | IC50 | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_4c9ec54ae04f7d7158fd20bcb5558a77.svg) | N-[4-[(3-Chloro-4-fluorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-5-(4-morpholinyl)-2-pentynamide | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_469d7b07597ef44d9809e6a1ffe62bb6.svg) | N-[4-[(3-Chloro-4-fluorophenyl)amino]-6-quinazolinyl]-5-(4-morpholinyl)-2-pentynamide | IC50 | 4.3 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_1d1e5de38328b8ebfd158425ca0d07ff.svg) | N-[4-(3-Chloro-4-fluoroanilino)quinazolin-6-yl]-4-hydroxybut-2-ynamide | IC50 | 7.3 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_f03132d47be7afe97651934dcab4d9e9.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-5-piperidin-1-ylpent-2-ynamide | IC50 | 1.8 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_028cc7e0b0772a62ab8acb6278b8146f.svg) | N-[4-(3-Bromo-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-5-(4-methylpiperazin-1-yl)pent-2-ynamide | IC50 | 0.8 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_b3a49261903ffca4c012d99dc469c899.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]hex-2-ynamide | IC50 | 2.4 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a4d77d6db5d2d76dd6f431905abd1061.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-(dibutylamino)but-2-ynamide | IC50 | 73.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_599ac957c297e940d4bcc72a0213f21e.svg) | 6,7-Diethoxy-N-(3-iodophenyl)quinazolin-4-amine;hydrochloride | IC50 | 59.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_0524a17543b3a059c97dc525160d0a55.svg) | 6,7-Diethoxy-N-[(4-fluorophenyl)methyl]quinazolin-4-amine | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_3661c98ac05b1b0da3a8a2c366e6cd56.svg) | N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-(diethylamino)but-2-ynamide | IC50 | 644.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_5f3a6add295ca6e973340645e7f663a8.svg) | N-[4-(3-Bromo-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-5-morpholin-4-ylpent-2-ynamide | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a1ed7c6cea78520168096b5b9d9f015a.svg) | N-[4-(3-Chloro-4-fluoroanilino)quinazolin-6-yl]-4-[di(propan-2-yl)amino]but-2-ynamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_9c16bdd1e37ef747e5b1a806c82a0b05.svg) | 2,3-Dimethyl-4-[2-methyl-3-(prop-2-enoylamino)phenyl]-1H-indole-7-carboxamide | IC50 | 240.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_73a64410e42f17bda47f701b7ae2ee93.svg) | 4-[3-(Ethenylsulfonylamino)-2-methylphenyl]-2,3-dimethyl-1H-indole-7-carboxamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_dc5ff7b87d06ec962585df9a614f5950.svg) | 6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_b50b2ac1c1cf1b547ee16b1027344c58.svg) | N-(3-Chloro-4-fluorophenyl)-6-(1-methylpyrazol-4-yl)quinazolin-4-amine | IC50 | 801.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_9629b092a7d5bcd59bbcdc59e87ec69e.svg) | 6-(1-Piperidin-4-ylpyrazol-4-yl)-N-quinolin-6-ylquinazolin-4-amine | IC50 | 1100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_b1ee86e2760c7f787b732ba0b40eb7a2.svg) | 6-(1-Methylpyrazol-4-yl)-N-quinolin-6-ylquinazolin-4-amine | IC50 | 930.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_81998d8b6de92df686e61cecd49b8ac9.svg) | N-(3-Ethynylphenyl)-6-(1-methylpyrazol-4-yl)quinazolin-4-amine | IC50 | 782.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_5bf61c46f69c300d824991cc6bab1557.svg) | N-(3-Chloro-4-fluorophenyl)-6-(1-piperidin-4-ylpyrazol-4-yl)quinazolin-4-amine | IC50 | 1603.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_6976739bd35c9001420ae84623837f06.svg) | Chmfl-egfr-202 | IC50 | 3.2 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_cf61d41cb0341078e0096c6957f8977e.svg) | 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(prop-2-enoylamino)phenyl]-6,7,8,9-tetrahydro-5H-carbazole-1-carboxamide | IC50 | 150.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a092c705c43630bc83f938c779c0b253.svg) | (E)-N-[4-[(1-Benzylindazol-5-yl)amino]-7-(2-methoxyethoxy)quinazolin-6-yl]-4-pyrrolidin-1-ylbut-2-enamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_3498c2639b4c7c7e9fc066a2830d44f5.svg) | (E)-N-[4-[(1-Benzylindazol-5-yl)amino]-7-ethoxyquinazolin-6-yl]-4-morpholin-4-ylbut-2-enamide | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_b133f61e369e9050fab2cb953f75cc71.svg) | (E)-N-[4-(4-Phenoxyanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-pyrrolidin-1-ylbut-2-enamide | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_41ea20ee93769a348b73d9ccf077f397.svg) | (E)-N-[4-[[1-(Benzenesulfonyl)indol-5-yl]amino]-7-ethoxyquinazolin-6-yl]-4-(dimethylamino)but-2-enamide | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_20f4fa13da8062625f5db74f52efe0af.svg) | (E)-N-[4-[3-Chloro-4-[(3-fluorophenyl)methoxy]anilino]pyrido[3,4-d]pyrimidin-6-yl]-4-pyrrolidin-1-ylbut-2-enamide | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_40d3959b0b1f8d426abd60b23a127d39.svg) | N-[4-[(1-Benzyl-2,3-dihydroindol-5-yl)amino]-7-methoxyquinazolin-6-yl]propanamide | IC50 | 82.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_07f5324df9d2dbe53069d0f824eb4145.svg) | (E)-N-[4-[[1-(Benzenesulfonyl)indol-5-yl]amino]-7-ethoxyquinazolin-6-yl]-4-pyrrolidin-1-ylbut-2-enamide | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_d33aaeaf7474072406ec189bab3c0471.svg) | (E)-N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-piperidin-1-ylbut-2-enamide | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_1f2620adb966ec041fe6e2f5f7694f69.svg) | N-[7-Methoxy-4-(4-phenylmethoxyanilino)quinazolin-6-yl]propanamide | IC50 | 460.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_98e391d6d0f6e1aea9a9fb229350034c.svg) | (E)-N-[7-Methoxy-4-[4-(pyridin-2-ylmethyl)anilino]quinazolin-6-yl]-4-pyrrolidin-1-ylbut-2-enamide | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_9c2a196aef3d3849897d56fb5fe7e8ba.svg) | (E)-N-[4-[(1-Benzylindazol-5-yl)amino]-7-ethoxyquinazolin-6-yl]-4-(dimethylamino)but-2-enamide | IC50 | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_7c027d3f703e9849dfcb5f94d565357b.svg) | (E)-N-[4-[[1-(Benzenesulfonyl)indol-5-yl]amino]-7-ethoxyquinazolin-6-yl]-4-morpholin-4-ylbut-2-enamide | IC50 | 27.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_89d49bf93cf28957c3cbe205f28bc264.svg) | N-[4-(3-Chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]propanamide | IC50 | 376.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_a215e47fbc47515ff0acab379db26e1a.svg) | N-[7-Methoxy-4-[[1-(pyridin-2-ylmethyl)indazol-5-yl]amino]quinazolin-6-yl]propanamide | IC50 | 15.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_b39f5c429b77ff897be38a8f2db69c6f.svg) | (E)-4-(4-Methylpiperazin-1-yl)-N-[4-[4-(pyridin-2-ylmethyl)anilino]pyrido[3,4-d]pyrimidin-6-yl]but-2-enamide | IC50 | 94.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_e9041270f0428e340744b7d91a5e873f.svg) | (E)-N-[7-Ethoxy-4-[4-(pyridin-2-ylmethoxy)anilino]quinazolin-6-yl]-4-(4-methylpiperazin-1-yl)but-2-enamide | IC50 | 94.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_4d71e8cdb9ed60c0a4e32417683ac49a.svg) | (E)-N-[4-[(1-Benzylindazol-5-yl)amino]-7-ethoxyquinazolin-6-yl]-4-(4-methylpiperazin-1-yl)but-2-enamide | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_ee10c01c9630797da106fa0d6f466b55.svg) | (E)-N-[4-(3-Chloro-4-fluoroanilino)pyrido[3,4-d]pyrimidin-6-yl]-4-(4-methylpiperazin-1-yl)but-2-enamide | IC50 | 302.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_ab726fd2372ae9c88ae9ed9e7811468b.svg) | (E)-N-[4-[(1-Benzylindazol-5-yl)amino]-7-ethoxyquinazolin-6-yl]-4-pyrrolidin-1-ylbut-2-enamide | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-protein-tyrosine-kinase-erbb-4_42bc2229e4304b106ebda57c28317a0f.svg) | N-[7-Methoxy-4-[[1-(pyridin-4-ylmethyl)indol-5-yl]amino]quinazolin-6-yl]propanamide | IC50 | 213.0 [1] |