![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_504e59ee4045da4ae506be77aa698656.svg) | CID 67469084 | IC50 | 16.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_e43350a0ac7beff955f823aa958c8635.svg) | (Arylindolyl)maleimide deriv. 27 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_095208844347ed4785884243d31c5466.svg) | 6-(4-Methylpiperazin-1-yl)-2-naphthalen-1-yl-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 880.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_cc14546399c19786a8e34ea4abe17b74.svg) | 2-(6-Methoxynaphthalen-1-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_fbb7804d40a3ae1ebfb7d7cf37e7fdf7.svg) | 2-(6-Ethoxynaphthalen-1-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_9a057185021bbe902fcf631dd3406d34.svg) | 2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 2500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_8a457332a5089ca595e95f159187f6b6.svg) | 2-(1,3-Benzodioxol-5-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 7600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_9a2c1d6e75e6e5ab9fb20cb9a12434ed.svg) | [3-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]phenyl]-morpholin-4-ylmethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_9bb4ec9b3e247b9c396995a1b6b656ee.svg) | 2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-3-ylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_4179c8b8a594a5a8b1de8dea97dcfac2.svg) | 2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-phenylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_c2ccabfea2fc119543bf89ffbcd07768.svg) | 2-(1,3-Benzodioxol-4-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 5500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_06b68c999909561f030bd44c86d5fbe4.svg) | 2-(1,3-Benzodioxol-4-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-a]pyridine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_3980f86df9820029580b36fdaebb88e5.svg) | 2-(2,3-Dihydro-1,4-benzodioxin-5-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_f40bfbb88208fdd1726ca6fb1d4da9c6.svg) | 6-(4-Methylpiperazin-1-yl)-2-(4-phenylphenyl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_86096cfaa1f6e4566b6aa05210a0768c.svg) | 6-(4-Methylpiperazin-1-yl)-2-(3-phenylphenyl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 450.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_793d0f45e06bf796c171400e62b6ab3a.svg) | 6-(4-Methylpiperazin-1-yl)-3-pyridin-4-yl-2-(3-thiophen-2-ylphenyl)imidazo[1,2-b]pyridazine | IC50 | 270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_a3bae3acc04e170b2f03292430a67972.svg) | 6-(4-Methylpiperazin-1-yl)-3-pyridin-4-yl-2-(3-thiophen-3-ylphenyl)imidazo[1,2-b]pyridazine | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_114583446e436b91999a8f68bae6ac6b.svg) | 2-(2,3-Dihydro-1,4-benzodioxin-6-yl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_98879a9a4eb951de69a72cf1ae094fa6.svg) | 6-(4-Methylpiperazin-1-yl)-2-(5-phenylthiophen-2-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_104a9df79f0f09cb253a54329252ecfc.svg) | [4-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]phenyl]-morpholin-4-ylmethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_32c95bdfade523c5b499ad25f4ccdb3d.svg) | 6-[6-(4-Methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazin-2-yl]-1,3-benzothiazole | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_cde2b34342f2c82e5223761841788bea.svg) | 6-[3-[1-Hydroxy-4-(1H-indol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_d1915eab4f37b417115050297a065181.svg) | 4-Hydroxy-4,14,21-triazahexacyclo[19.6.1.17,14.02,6.08,13.022,27]nonacosa-1(28),2(6),7(29),8,10,12,22,24,26-nonaene-3,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_f873969fd5042c55a8277c91b514411e.svg) | 1-Hydroxy-3-(1H-indol-3-yl)-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_0d4dc5072f1b7f88ef2207cc09eadf13.svg) | 3-(1-Ethylindol-3-yl)-1-hydroxy-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_6591383b313289e743f4adb0d9dd6fa3.svg) | 1-Hydroxy-3-(1H-indol-3-yl)-4-(1-methylindol-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_128ce1c03082e1d9d76fb276fa7fa521.svg) | 1-Hydroxy-3-(1H-indol-3-yl)-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_9c9485c08e6915fd2f891ef59099ffe4.svg) | 6-[3-[4-[1-(5-Cyanopentyl)indol-3-yl]-1-hydroxy-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_5639401709f9c1e2aa7791dca7aa10fd.svg) | 3-(1-Ethylindol-3-yl)-1-hydroxy-4-(1-methylindol-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_a9489efdc3c6a620c8cf1cba16458928.svg) | 1-Hydroxy-3,4-bis(1-methylindol-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_d47123b6fcff0d1783bc89c9bce501de.svg) | 6-[3-[4-[1-(5-Cyanopentyl)indol-3-yl]-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_88c9b45a32473c6764e2e6ebabac122d.svg) | 6-[3-[1-Hydroxy-4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanenitrile | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_6ea4760351cb47c58bcdb6b72c5298e0.svg) | 1-Hydroxy-3-(1-methylindol-3-yl)-4-(1-propan-2-ylindol-3-yl)pyrrole-2,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_e09578c167e3e2b42a83526a023fdc1e.svg) | 6-[3-[1-Hydroxy-4-(1-methylindol-3-yl)-2,5-dioxopyrrol-3-yl]indol-1-yl]hexanoic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/receptor-interacting-serine-threonine-protein-kinase-3_ff4449330c1ba5385514c846cf0ac937.svg) | 2-(3-Methoxyphenyl)-6-(4-methylpiperazin-1-yl)-3-pyridin-4-ylimidazo[1,2-b]pyridazine | IC50 | 10000.0 [1] |