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Rap guanine nucleotide exchange factor 4 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
CID 6077765IC504400.0 [1], 7000.0 [2], 9000.0 [3]
Cyclic AMPIC5040000.0 [1], 48000.0 [2]
Mesityl P-tolyl sulfoneIC50400.0 [1], 500.0 [2]
(2R)-5,7-Dibromo-6-fluoro-2-methyl-3,4-dihydro-2H-quinoline-1-carbaldehydeIC5017000.0 [1], 22300.0 [2]
(E)-3-(3,4,5-Trihydroxy-6-oxoxanthen-9-yl)prop-2-enoic acidIC503800.0 [1]
2,4-Dimethyl-1-(2,4,6-trimethyl-benzenesulfonyl)-1H-pyrroleIC50300.0 [1]
1-(2,4,6-Trimethylphenyl)sulfonylindoleIC501200.0 [1]
Benzenesulfonic acid, 5-amino-2-[(4-aminophenyl)amino]-IC5018000.0 [1]
5-((2-Hydroxy-1-naphthyl)diazenyl)-2-naphthalenesulfonic acidIC501700.0 [1]
4-Cyclohexyl-2-[(2,5-dimethylphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrileIC508400.0 [1]
N-(5-Cyano-15,22-dioxo-13-oxa-3-thiapentacyclo[12.8.0.02,6.07,12.016,21]docosa-1(14),2(6),4,7,9,11,16,18,20-nonaen-4-yl)-2,2,2-trifluoroacetamideIC507900.0 [1]
N-(3,5-Dimethylphenyl)-2,4,6-trimethylanilineIC501700.0 [1]
3-N-(2,4,6-Trimethylphenyl)benzene-1,3-diamineIC5034000.0 [1]
2,4,6-Trimethyl-N-(4-methylphenyl)anilineIC503800.0 [1]
N-(4-Bromophenyl)-2,4,6-trimethylanilineIC501600.0 [1]
N-(2,4-Dimethylphenyl)-2,4,6-trimethylanilineIC502200.0 [1]
N-(3-Chloro-4-fluorophenyl)-2,4,6-trimethylanilineIC502900.0 [1]
N-[3-Chloro-5-(trifluoromethyl)phenyl]-2,4,6-trimethylanilineIC50500.0 [1]
N-(3,5-Difluorophenyl)-2,4,6-trimethylanilineIC505700.0 [1]
N-(3,4-Difluorophenyl)-2,4,6-trimethylanilineIC508700.0 [1]
N-(5-Chloro-2-methylphenyl)-2,4,6-trimethylanilineIC501400.0 [1]
N-(2,4-Dichloro-6-methylphenyl)-2,4,6-trimethylanilineIC50700.0 [1]
N-(3-Fluorophenyl)-2,4,6-trimethylanilineIC505800.0 [1]
N-(3-Bromophenyl)-2,4,6-trimethylanilineIC501500.0 [1]
2,4,6-Trimethyl-N-(3,4,5-trichlorophenyl)anilineIC501100.0 [1]
2,4,6-Trimethyl-N-(2,4,6-trifluorophenyl)anilineIC502700.0 [1]
N-(2,3-Dimethylphenyl)-2,4,6-trimethylanilineIC501000.0 [1]
N-(3-Chloro-5-fluorophenyl)-2,4,6-trimethylanilineIC502900.0 [1]
N-(3,4-Dichlorophenyl)-2,4,6-trimethylanilineIC501100.0 [1]
N-(4-Chloro-3-fluorophenyl)-2,4,6-trimethylanilineIC503300.0 [1]
N-(2,4,6-Trimethylphenyl)-2,3-dihydro-1H-inden-5-amineIC501800.0 [1]
N-(3-Ethylphenyl)-2,4,6-trimethylanilineIC501800.0 [1]
2,4,6-Trimethyl-N-[3-(trifluoromethyl)phenyl]anilineIC502000.0 [1]
2,4,6-Trimethyl-N-[3-[2-(2,4,6-trimethylphenyl)ethynyl]phenyl]anilineIC50300000.0 [1]
2,4,6-Trimethyl-N-(3,4,5-trifluorophenyl)anilineIC503000.0 [1]
3-(2,4,6-Trimethylanilino)phenolIC5046000.0 [1]
N-(3-Chloro-4-methylphenyl)-2,4,6-trimethylanilineIC501800.0 [1]
(1E)-2-(4-Tert-butylphenyl)-N-(3,5-dichloroanilino)-2-oxoethanimidoyl cyanideIC502500.0 [1]
(1E)-N-(3,5-Dichloroanilino)-2-naphthalen-2-yl-2-oxoethanimidoyl cyanideIC502500.0 [1]
(1E)-2-(4-Tert-butylphenyl)-N-(3-chloro-5-fluoroanilino)-2-oxoethanimidoyl cyanideIC503400.0 [1]
(1E)-2-(4-Tert-butylphenyl)-N-[4-chloro-3-(trifluoromethyl)anilino]-2-oxoethanimidoyl cyanideIC5012400.0 [1]
(1E)-2-(4-Tert-butylphenyl)-2-oxo-N-(3,4,5-trifluoroanilino)ethanimidoyl cyanideIC5015800.0 [1]
(1E)-2-(4-Tert-butylphenyl)-N-[3-chloro-5-(trifluoromethyl)anilino]-2-oxoethanimidoyl cyanideIC505400.0 [1]
(1E)-2-(4-Tert-butylphenyl)-2-oxo-N-(3,4,5-trichloroanilino)ethanimidoyl cyanideIC503000.0 [1]
2-Benzylsulfanyl-4-cyclohexyl-6-hydroxy-pyrimidine-5-carbonitrileIC5030500.0 [1]
2-[(5-Cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N-(4-methylphenyl)acetamideIC50300000.0 [1]
2-[(2,5-Dimethylphenyl)methylsulfanyl]-6-oxo-4-propan-2-yl-1H-pyrimidine-5-carbonitrileIC5012700.0 [1]
4-Cyclohexyl-2-[(2,4-dimethylphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrileIC5015700.0 [1]
2-[(5-Cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]acetic acidIC50300000.0 [1]
4-Cyclohexyl-6-oxo-2-[(2,4,6-trimethylphenyl)methylsulfanyl]-1H-pyrimidine-5-carbonitrileIC5011600.0 [1]
2-[(2,5-Dimethylphenyl)methylsulfanyl]-4-(1-methylpiperidin-4-yl)-6-oxo-1H-pyrimidine-5-carbonitrileIC50127000.0 [1]
2-Anilino-4-cyclohexyl-6-oxo-1H-pyrimidine-5-carbonitrileIC50300000.0 [1]
4-Cyclohexyl-2-[(3,5-dimethylphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrileIC507000.0 [1]
4-Cyclopropyl-2-[(2,5-dimethylphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrileIC504000.0 [1]
4-Cyclopentyl-2-[(2,5-dimethylphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrileIC505900.0 [1]
4-Cyclohexyl-2-[(4-methylphenyl)methylsulfanyl]-6-oxo-1H-pyrimidine-5-carbonitrileIC5038700.0 [1]
2-(4-Chloroanilino)-4-cyclohexyl-6-oxo-1H-pyrimidine-5-carbonitrileIC50300000.0 [1]
2-[(5-Cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N-(2,4,6-trimethylphenyl)acetamideIC50300000.0 [1]
2-[(2,5-Dimethylphenyl)methylsulfanyl]-6-oxo-4-piperidin-4-yl-1H-pyrimidine-5-carbonitrileIC50300000.0 [1]
2-[(5-Cyano-4-cyclohexyl-6-oxo-1H-pyrimidin-2-yl)sulfanyl]-N-phenylacetamideIC50300000.0 [1]
N-(3-Methoxyphenyl)-2,4,6-trimethylanilineIC5010700.0 [1]
5-Cyano-6-cyclohexyl-2-thiouracilIC50300000.0 [1]
2-(4-Methoxyphenyl)sulfonyl-1,3,5-trimethyl-benzeneIC501900.0 [1]
N-(2,5-Dimethylphenyl)-2,4,6-trimethylanilineIC501800.0 [1]
4-(2,4,6-Trimethylbenzenesulfonyl)PhenolIC5013500.0 [1]
2-Fluoro-5-[4-(2,4,6-trimethylphenyl)sulfonylphenyl]pyridineIC50300000.0 [1]
4,5-Dimethyl-N-(2,4,6-trimethylphenyl)-1,3-thiazol-2-amineIC50300000.0 [1]
1,3,5-Trimethyl-2-(2,4,5-trimethylphenyl)sulfonylbenzeneIC50700.0 [1]
1,3,5-Trimethyl-2-(4-pentylphenyl)sulfonylbenzeneIC50300000.0 [1]
2-(4-Cyclohexylphenyl)sulfonyl-1,3,5-trimethylbenzeneIC50300000.0 [1]
2-(4-Cyclohexyloxyphenyl)sulfonyl-1,3,5-trimethylbenzeneIC50300000.0 [1]
Tert-butyl 4-[4-(2,4,6-trimethylphenyl)sulfonylphenoxy]piperidine-1-carboxylateIC50300000.0 [1]
4-[4-(2,4,6-Trimethylphenyl)sulfonylphenoxy]piperidineIC50300000.0 [1]
2-[4-(2,4,6-Trimethylphenyl)sulfonylphenoxy]ethanamineIC50300000.0 [1]
N-(3,5-Dichlorophenyl)-2,4,6-trimethylanilineIC50900.0 [1]
(2,5-Dichlorophenyl)-(2,4,6-trimethylphenyl)-amineIC50400.0 [1]
2-Ethyl-1-(2,4,6-trimethylphenyl)sulfonylpyrroleIC50500.0 [1]
2-Ethyl-1-(4-methylphenyl)sulfonylpyrroleIC504000.0 [1]
2-Ethyl-1-(4-methoxyphenyl)sulfonylpyrroleIC508000.0 [1]
1-(4-Chloro-benzenesulfonyl)-2-ethyl-1H-pyrroleIC508000.0 [1]
2-Ethyl-1-[4-(trifluoromethyl)phenyl]sulfonylpyrroleIC50300000.0 [1]
2-Ethyl-1-(2-methylphenyl)sulfonylpyrroleIC505300.0 [1]
1-(3,5-Dimethylphenyl)sulfonyl-2-ethylpyrroleIC504700.0 [1]
1-(2,4-Dimethylphenyl)sulfonyl-2-ethylpyrroleIC501300.0 [1]
Methyl 1-(2,4,6-trimethylphenyl)sulfonylindole-5-carboxylateIC50300000.0 [1]
1-(2,4,6-Trimethylphenyl)sulfonylindole-5-carboxylic acidIC5010800.0 [1]
1-(2,4,6-Trimethylphenyl)sulfonylpyrrolo[3,2-b]pyridineIC503800.0 [1]
1-(2,4,6-Trimethylphenyl)sulfonylpyrrolo[3,2-c]pyridineIC508900.0 [1]
1-(2,4,6-Trimethylphenyl)sulfonylpyrrolo[2,3-c]pyridineIC5012600.0 [1]
1-(2,4,6-Trimethylphenyl)sulfonylpyrrolo[2,3-b]pyridineIC502400.0 [1]
2-(4-Iodophenyl)sulfonyl-1,3,5-trimethylbenzeneIC504000.0 [1]
(2S)-5,7-Dibromo-6-fluoro-2-methyl-3,4-dihydro-2H-quinoline-1-carbaldehydeIC5017100.0 [1]
2-(Mesitylamino)-3-(3-methoxypropyl)-4-methylthiazole-3-iumIC50600.0 [1]
Items per page: 1 - 10 of 93
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References

This online tool may be cited as follows

MLA

"Quest Database™ Rap guanine nucleotide exchange factor 4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/rap-guanine-nucleotide-exchange-factor-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Rap guanine nucleotide exchange factor 4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/rap-guanine-nucleotide-exchange-factor-4-inhibitors-ic50-ki.
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