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Pyruvate kinase isozymes M1/M2 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
ShikoninIC508820.0 [1]
5-(2,5-Dimethyl-pyrrol-1-yl)-2-hydroxy-benzoic acidIC507000.0 [1], 12500.0 [2], 100000.0 [3]
ScutellareinIC5012500.0 [1], 100000.0 [2]
3-[2-(1H-Indol-3-yl)ethyl]-6-nitro-1H-indoleIC5054600.0 [1], 95900.0 [2]
[1,4-Dioxo-3-(piperidine-1-carbothioylsulfanylmethyl)naphthalen-2-yl]methyl piperidine-1-carbodithioateIC50880.0 [1], 5070.0 [2]
2-(1H-1,2,4-Triazol-3-yl)-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3-dioneIC5090000.0 [1]
2-Chloro-5-(2,5-dimethyl-pyrrol-1-yl)-benzoic acidIC50100000.0 [1]
PKM2 inhibitorIC5016710.0 [1]
5-Methylsulfanylthiophene-2-carboxylic acidIC5010000.0 [1]
(1,4-Dioxonaphthalen-2-yl)methyl N,N-diethylcarbamodithioateIC502580.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-(pyridin-4-ylmethyl)carbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl) N,N-dipropylcarbamodithioateIC509980.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-[2-(diethylamino)ethyl]carbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N,N-bis(prop-2-enyl)carbamodithioateIC5014110.0 [1]
(1,4-Dimethoxynaphthalen-2-yl)methyl N,N-dipropylcarbamodithioateIC5015660.0 [1]
(1,4-Dioxonaphthalen-2-yl)methyl 4-phenylpiperazine-1-carbodithioateIC506260.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N,N-diethylcarbamodithioateIC508780.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N,N-dipropylcarbamodithioateIC506790.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl 1,3-thiazolidine-3-carbodithioateIC505280.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-benzylcarbamodithioateIC502210.0 [1]
(1,4-Dioxonaphthalen-2-yl)methyl piperidine-1-carbodithioateIC501740.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-methylcarbamodithioateIC5020000.0 [1]
(1,4-Dioxonaphthalen-2-yl)methyl morpholine-4-carbodithioateIC504230.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl 2,6-dimethylmorpholine-4-carbodithioateIC5011700.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-(pyridin-2-ylmethyl)carbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl) morpholine-4-carbodithioateIC508500.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl thiomorpholine-4-carbodithioateIC505890.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-(pyridin-3-ylmethyl)carbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N,N-bis(2-hydroxyethyl)carbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N,N-dibutylcarbamodithioateIC504570.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl 4-propan-2-ylpiperazine-1-carbodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl) piperidine-1-carbodithioateIC504930.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl 4-methylpiperazine-1-carbodithioateIC5014240.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-(4-methylpiperazin-1-yl)carbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl 4-acetylpiperazine-1-carbodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-piperidin-1-ylcarbamodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl) 4-acetylpiperazine-1-carbodithioateIC5020000.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl N-(cyclohexylmethyl)carbamodithioateIC505080.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl pyrrolidine-1-carbodithioateIC5019730.0 [1]
(3-Methyl-1,4-dioxonaphthalen-2-yl)methyl morpholine-4-carbodithioateIC5015240.0 [1]
2-[(5Z)-5-[[4-(2-Iodobenzoyl)oxyphenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acidIC5020000.0 [1]
(2Z)-1-Butyl-2-[(E)-3-(1-butyl-5,6-dichloro-3-pentylbenzimidazol-3-ium-2-yl)prop-2-enylidene]-5,6-dichloro-3-pentylbenzimidazoleIC5010000.0 [1]
1-[4-(2,5-Dimethylpyrrol-1-yl)phenyl]sulfanylpropan-2-oneIC5090000.0 [1]
8-Methyl-2-[1-(propan-2-ylamino)ethenyl]thieno[3,2-c]chromen-4-oneIC5070000.0 [1]
Items per page: 1 - 10 of 44
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References

This online tool may be cited as follows

MLA

"Quest Database™ Pyruvate kinase isozymes M1/M2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/pyruvate-kinase-isozymes-m1-m2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Pyruvate kinase isozymes M1/M2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/pyruvate-kinase-isozymes-m1-m2-inhibitors-ic50-ki.
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