Pyruvate dehydrogenase kinase isoform 3 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(3S)-3-Amino-4-[4-[[2-(2,4-dihydroxyphenyl)sulfonyl-1,3-dihydroisoindol-5-yl]amino]piperidin-1-yl]-4-oxobutanamide	IC50	1710.0 [1], 45800.0 [2]
	Dichloroacetic acid	IC50	5560000.0 [1]
	Radicicol	IC50	230000.0 [1]
	Dimorpholinethiuram disulfide	Ki	2851.0 [1]
	CID 86280454	IC50	40.0 [1]
	2-[(2,4-Dihydroxyphenyl)sulfonyl]-2,3-Dihydro-1h-Isoindole-4,6-Diol	IC50	21300.0 [1]
	(E)-3-[5-(5-Chloro-2,4-dihydroxyphenyl)-4-(4-hydroxyphenyl)-1,2-oxazol-3-yl]-1-[4-(2-methoxyphenyl)piperazin-1-yl]prop-2-en-1-one	IC50	5336.0 [1]
	[(3R)-3-(Methoxymethyl)morpholine-4-carbothioyl]sulfanyl (3R)-3-(methoxymethyl)morpholine-4-carbodithioate	Ki	2987.0 [1]
	1,4-Oxazepane-4-carbothioylsulfanyl 1,4-oxazepane-4-carbodithioate	Ki	7762.0 [1]
	2,4-Dihydroxy-N-(4-methoxyphenyl)-N-methylbenzamide	Ki	550.0 [1]

---

---

References

This online tool may be cited as follows

MLA	"Quest Database™ Pyruvate dehydrogenase kinase isoform 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/pyruvate-dehydrogenase-kinase-isoform-3-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, December 21). Quest Database™ Pyruvate dehydrogenase kinase isoform 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/pyruvate-dehydrogenase-kinase-isoform-3-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan