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Proto-oncogene c-JUN Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
3-(4-Chloro-phenyl)-2-(4-methyl-2-methylamino-thiazol-5-yl)-3H-quinazolin-4-oneIC501200.0 [1], 3000.0 [2], 3300.0 [3]
2-[2-(4-Chloroanilino)-4-methyl-1,3-thiazol-5-yl]-3-(4-chlorophenyl)quinazolin-4-oneIC501200.0 [1], 3300.0 [2]
3-[5-(4-Cyclopentyloxy-2-hydroxybenzoyl)-2-[(3-oxo-1,2-benzoxazol-6-yl)methoxy]phenyl]propanoic acidIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-chloro-4-(trifluoromethyl)pyrimidine-5-carboxamideIC5050.0 [1]
CID 10407641IC5020.0 [1]
CID 10499355IC504000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2,4-bis(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-cyano-4-(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-6-chloro-4-(trifluoromethyl)pyridazine-3-carboxamideIC5010000.0 [1]
CID 10666814IC501700.0 [1]
N-(3,5-Bis-trifluoromethyl-phenyl)-4-chloro-2-trifluoromethyl-benzamideIC5030000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-fluoro-4-(trifluoromethyl)pyrimidine-5-carboxamideIC50100.0 [1]
CID 10741998IC50400.0 [1]
CID 10763720IC50200.0 [1]
2-(4-Methyl-2-phenylamino-thiazol-5-yl)-3-o-tolyl-3H-quinazolin-4-oneIC505500.0 [1]
3-(4-Acetylphenyl)-2-(5-morpholin-4-yl-4-pyridin-4-ylthiophen-2-yl)quinazolin-4-oneIC505000.0 [1]
Nagilactone FIC501500.0 [1]
2-(4-Methyl-2-methylamino-thiazol-5-yl)-3-o-tolyl-3H-quinazolin-4-oneIC505500.0 [1]
InumakilactoneIC504000.0 [1]
Rosmarinic acidIC5016200.0 [1]
(1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneIC5012800.0 [1]
(Z)-3-Amino-3-(4-aminophenylthio)-2-(2-(trifluoromethyl)phenyl)acrylonitrileIC502030.0 [1]
CyqualonIC507300.0 [1]
1-(5-Methoxy-2-(thiophen-2-yl)quinazolin-4-ylamino)-3-methyl-1H-pyrrole-2,5-dioneIC508.0 [1]
GlaucarubinoneIC5040.0 [1]
TylophorinidineIC5065.0 [1]
PergularinineIC50110.0 [1]
Unii-txf835U41KIC501067.0 [1]
Momordine IIC5030000.0 [1]
(1E,4E)-1,5-Di(pyridin-3-yl)penta-1,4-dien-3-oneIC504100.0 [1]
1,5-Bis(2-hydroxyphenyl)penta-1,4-dien-3-oneIC5011700.0 [1]
Tylophoridicine EIC503000.0 [1]
1-(6-Methoxy-2-thiophen-2-yl-quinazolin-4-ylamino)-3-methyl-pyrrole-2,5-dioneIC503.0 [1]
2-Anthracenecarboxylic acid, 9,10-dihydro-3,8-dihydroxy-9,10-dioxo-1-propyl-IC50100000.0 [1]
[4-[(1E,4E)-5-(4-Acetyloxy-3-methoxyphenyl)-3-oxopenta-1,4-dienyl]-2-methoxyphenyl] acetateIC508300.0 [1]
2-Phenyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC50100.0 [1]
Ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(trifluoromethyl)pyrimidine-5-carboxylateIC501000.0 [1]
TylophorinicineIC50300.0 [1]
[(1S,4S,5R,6R,7S,8R,11R,13S,17S,18S,19R)-4,5,17-Trihydroxy-6,14,18-trimethyl-9,16-dioxo-3,10-dioxapentacyclo[9.8.0.01,7.04,19.013,18]nonadec-14-en-8-yl] 2-methylbutanoateIC5032.0 [1]
2-(2-Thienyl)-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC5020.0 [1]
Ethyl 2-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-4-(5-methylthiophen-2-yl)pyrimidine-5-carboxylateIC5045.0 [1]
Ethyl 4-ethyl-2-[methyl-(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC5035.0 [1]
(1E,4E)-1,5-Bis(2,5-dimethoxyphenyl)penta-1,4-dien-3-oneIC501400.0 [1]
3-[2-Isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propionic acidIC505000.0 [1]
Ethyl 4-ethyl-2-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC50400.0 [1]
Ethyl 2-[methyl-(3-methyl-2,5-dioxopyrrol-1-yl)amino]-4-(trifluoromethyl)pyrimidine-5-carboxylateIC50300.0 [1]
1-[[5-Benzoyl-4-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methylpyrrole-2,5-dioneIC5098.0 [1]
Ethyl 2-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-4-(trifluoromethyl)pyrimidine-5-carboxylateIC502000.0 [1]
Tert-butyl 2-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-4-(trifluoromethyl)pyrimidine-5-carboxylateIC50210.0 [1]
1-[[5-Acetyl-4-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methylpyrrole-2,5-dioneIC504400.0 [1]
7-(1-Methylpyrazol-4-yl)-N-[4-(3-morpholin-4-yl-1,2,4-triazol-1-yl)phenyl]quinazolin-2-amineIC50310.0 [1]
Grassypeptolide FIC505200.0 [1]
Grassypeptolide GIC506000.0 [1]
2-Chloro-8-(trifluoromethyl)-6H-pyrimido[4,5-b][1,5]benzothiazepin-5-oneIC50100.0 [1]
(Z)-3-[(1S,2S,4S,5S,6S,7S)-5-Hydroxy-10-methoxycarbonyl-7-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-3,8-dioxatricyclo[4.4.0.02,4]dec-9-ene-5-carbonyl]oxy-2-(4-hydroxy-3-methoxyphenyl)prop-2-enoic acidIC5029000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-4-chloro-2-(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-chloro-4-(1,1,2,2,2-pentafluoroethyl)pyrimidine-5-carboxamideIC50600.0 [1]
CID 10666813IC50300.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2,6-dichloropyrimidine-4-carboxamideIC5010000.0 [1]
CID 10716536IC5010000.0 [1]
CID 10716588IC50500.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-chloro-6-(trifluoromethyl)pyrimidine-4-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-methyl-4-(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-chloro-6-methylpyrimidine-4-carboxamideIC5010000.0 [1]
CID 10787015IC50300.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-4-methyl-2-(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-chloro-4-thiophen-2-ylpyrimidine-5-carboxamideIC508000.0 [1]
N-Ethyl-4-[[4-(1H-indol-3-yl)-5-methylpyrimidin-2-yl]amino]piperidine-1-carboxamideIC5010000.0 [1]
N-[2-[4-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]-2-oxoethyl]acetamideIC501938.0 [1]
2-Chloro-N-(3,5-dichlorophenyl)-4-methylpyrimidine-5-carboxamideIC50500.0 [1]
N-[2,4-Bis(trifluoromethyl)phenyl]-2-chloro-6-(trifluoromethyl)pyrimidine-4-carboxamideIC5010000.0 [1]
N-[2,4-Bis(trifluoromethyl)phenyl]-2-chloro-6-methylpyrimidine-4-carboxamideIC5010000.0 [1]
[2-Chloro-4-(trifluoromethyl)pyrimidin-5-yl]-[7-(trifluoromethyl)-2,4-dihydro-3,1-benzoxazin-1-yl]methanoneIC5010000.0 [1]
6-[3,5-Bis(trifluoromethyl)phenyl]-2-chloropyrrolo[3,4-d]pyrimidine-5,7-dioneIC509400.0 [1]
6-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-2-chloropyrrolo[3,4-d]pyrimidine-5,7-dioneIC509400.0 [1]
2-Chloro-8-(trifluoromethyl)-6H-pyrimido[5,4-c]quinolin-5-oneIC506100.0 [1]
2-Chloro-8-(trifluoromethyl)-6,11-dihydropyrimido[5,4-c][1]benzazepin-5-oneIC508500.0 [1]
2-Chloro-8-(trifluoromethyl)-6,11-dihydropyrimido[5,4-c][1,5]benzodiazepin-5-oneIC5010000.0 [1]
2-Chloro-8-(trifluoromethyl)-6H-pyrimido[4,5-b][1,5]benzoxazepin-5-oneIC501900.0 [1]
1-[[4-Ethyl-5-(2-methyl-1,3-oxazol-4-yl)pyrimidin-2-yl]amino]-3-methylpyrrole-2,5-dioneIC50830.0 [1]
3-Methyl-1-[[5-(2-methyl-1,3-oxazol-4-yl)-4-thiophen-2-ylpyrimidin-2-yl]amino]pyrrole-2,5-dioneIC50760.0 [1]
(Z)-3-[(1S,4As,7S,7aS)-7-hydroxy-4-methoxycarbonyl-5-methyl-1-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-4a,7a-dihydro-1H-cyclopenta[c]pyran-7-carbonyl]oxy-2-(4-hydroxy-3-methoxyphenyl)prop-2-enoic acidIC5069600.0 [1]
(1E,4E)-1,5-Di(pyridin-4-yl)penta-1,4-dien-3-oneIC508200.0 [1]
(1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)-4-methylhepta-1,4,6-trien-3-oneIC506000.0 [1]
4-{[5-Chloro-4-(1h-Indol-3-Yl)pyrimidin-2-Yl]amino}-N-Ethylpiperidine-1-CarboxamideIC50704.0 [1]
Ethyl N-[5-[3-(4-chlorophenyl)-4-oxoquinazolin-2-yl]-4-methyl-1,3-thiazol-2-yl]carbamateIC5010000.0 [1]
3-(2-Methoxyphenyl)-2-[2-(methylamino)-4-phenyl-1,3-thiazol-5-yl]quinazolin-4-oneIC50500.0 [1]
4-[[5-Cyano-4-(6-fluoro-1H-indol-3-yl)pyrimidin-2-yl]amino]-N-ethylpiperidine-1-carboxamideIC503700.0 [1]
4-(4-(1H-Indol-3-yl)pyrimidin-2-ylamino)-N-ethylpiperidine-1-carboxamideIC508091.0 [1]
4-[(5-Chloro-4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]-N-ethylpiperidine-1-carboxamideIC507723.0 [1]
4-[(5-Chloro-4-indol-1-ylpyrimidin-2-yl)amino]-N-ethylpiperidine-1-carboxamideIC5010000.0 [1]
N-Ethyl-4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidine-1-carboxamideIC5019331.0 [1]
4-(4-(1H-Indol-1-yl)pyrimidin-2-ylamino)-N-ethylpiperidine-1-carboxamideIC5029891.0 [1]
3-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]-N-ethylpyrrolidine-1-carboxamideIC506268.0 [1]
3-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]-N-ethylazetidine-1-carboxamideIC504272.0 [1]
(3S)-3-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]-N-ethylpiperidine-1-carboxamideIC506995.0 [1]
2-[(3S)-3-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]-N-methylacetamideIC5014667.0 [1]
(3R)-3-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]-N-ethylpiperidine-1-carboxamideIC503883.0 [1]
2-[(3R)-3-[[5-Chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]-N-methylacetamideIC502807.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Proto-oncogene c-JUN Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/proto-oncogene-c-jun-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Proto-oncogene c-JUN Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/proto-oncogene-c-jun-inhibitors-ic50-ki.
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