 | Pentamidine | IC50 | 53600.0 [1] |
 | PRL-3 Inhibitor | IC50 | 900.0 [1] |
 | 2-{5-[(E)-(4-Oxo-2-thioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acid | IC50 | 13300.0 [1], 53000.0 [2] |
 | 4-(2-((2,5-Dioxoimidazolidin-4-ylidene)methyl)-1H-pyrrol-1-yl)benzoic acid | IC50 | 28100.0 [1], 100000.0 [2] |
 | 7-Amino-2-phenyl-5H-thieno[3,2-c]pyridin-4-one | IC50 | 128.0 [1], 240.0 [2] |
 | 1-(3,4-Dihydroxyphenyl)-2-{[1-(4-methoxyphenyl)-1H-tetrazol-5-yl]thio}ethanone | IC50 | 44700.0 [1] |
 | 2-[[5-(3-Chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanone | IC50 | 43800.0 [1] |
 | 3-(2-{(E)-[1-(3-Chlorophenyl)-2,5-dioxoimidazolidin-4-ylidene]methyl}-1H-pyrrol-1-yl)benzoic acid | IC50 | 15400.0 [1] |
 | 5-Amino-6-[(Z)-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-(4-hydroxyphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one | IC50 | 33200.0 [1] |
 | (2Z)-2-(3,4-Dihydroxybenzylidene)[1,3]thiazolo[3,2-a]benzimidazol-3(2H)-one | IC50 | 11000.0 [1] |
 | N-(4-Butylphenyl)-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide | IC50 | 50000.0 [1] |
 | 5-(4-Benzyloxy-biphenyl-3-ylmethylene)-2-thioxo-thiazolidin-4-one | IC50 | 1700.0 [1] |
 | 2-[(E)-2-[5-(4-Chlorophenyl)furan-2-yl]ethenyl]-6-oxo-3-phenyl-4-sulfanyl-1,2-dihydropyrimidine-5-carbonitrile | IC50 | 18300.0 [1] |
 | (5Z)-5-[2-(Benzyloxy)-5-bromobenzylidene]-2-thioxo-1,3-thiazolidin-4-one | IC50 | 3000.0 [1] |
 | 5-(5-Bromo-2-hydroxy-benzylidene)-2-thioxo-thiazolidin-4-one | IC50 | 9500.0 [1] |
 | 5-(4-Hydroxy-3-methoxybenzylidene)-2-(o-toluidino)thiazol-4(5H)-one | IC50 | 41500.0 [1] |
 | 3-[[(5Z)-5-[(3-Chloro-5-ethoxy-4-hydroxyphenyl)methylidene]-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoic acid | IC50 | 40300.0 [1] |
 | (6Z)-6-(3,4-Dihydroxybenzylidene)-7-imino-2-methyl-6,7-dihydro-5H-isoxazolo[2,3-a]pyrimidin-5-one | IC50 | 100000.0 [1] |
 | 2-[6-(Pyrazin-2-yl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-3-yl]quinoline | IC50 | 100000.0 [1] |
 | 3-[5-[(Z)-(5-Imino-7-oxo-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-6-ylidene)methyl]furan-2-yl]benzoic acid | IC50 | 41700.0 [1] |
 | (5Z)-5-[[3-[3-[(2-Chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | IC50 | 27600.0 [1] |
 | N'-[1-[4-(4-Fluorophenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]-N-(pyridin-3-ylmethyl)oxamide | IC50 | 50000.0 [1] |
 | N-(Furan-2-ylmethyl)-N'-[1-[4-(4-methoxyphenyl)piperazin-1-yl]-1-thiophen-2-ylpropan-2-yl]oxamide | IC50 | 50000.0 [1] |
 | 5-(2-(2-Chlorobenzyloxy)-5-bromobenzylidene)-2-thioxothiazolidin-4-one | IC50 | 2400.0 [1] |
 | Prop-2-enyl (E)-3-(3-bromo-4-hydroxy-5-methoxyphenyl)-2-cyanoprop-2-enoate | IC50 | 31400.0 [1] |
 | 2-{[5,6-Di(furan-2-yl)-1,2,4-triazin-3-yl]sulfanyl}-N-(2-nitrophenyl)acetamide | IC50 | 57000.0 [1] |
 | 5-(5-(Benzo[b]thiophen-3-yl)-2-(benzyloxy)benzylidene)-2-thioxothiazolidin-4-one | IC50 | 900.0 [1] |
 | 5-((3-(Benzyloxy)naphthalen-2-yl)methylene)-2-thioxothiazolidin-4-one | IC50 | 2000.0 [1] |
 | 5-((3-(3,5-Dimethoxybenzyloxy)naphthalen-2-yl)methylene)-2-thioxothiazolidin-4-one | IC50 | 3100.0 [1] |
 | 5-[1-[3-(Biphenyl-4-ylmethoxy)-naphthalen-2-yl]-methylidene]-2-thioxo-thiazolidin-4-one | IC50 | 1900.0 [1] |
 | 5-((3-(2-Chloro-6-fluorobenzyloxy)naphthalen-2-yl)methylene)-2-thioxothiazolidin-4-one | IC50 | 1700.0 [1] |
 | 5-[(5-Bromo-2-phenylmethoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one | IC50 | 4000.0 [1] |
 | (5Z)-5-[[5-[4-(Dimethylamino)phenyl]-2-phenylmethoxyphenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | IC50 | 3700.0 [1] |
 | 5-(5-(Benzofuran-3-yl)-2-(benzyloxy)benzylidene)-2-thioxothiazolidin-4-one | IC50 | 1200.0 [1] |
 | Propan-2-yl (Z)-3-(3-bromo-4-hydroxyphenyl)-2-cyanoprop-2-enoate | IC50 | 167100.0 [1] |
 | Ethyl (2E)-2-cyano-3-(3,5-dibromo-4-hydroxyphenyl)prop-2-enoate | IC50 | 109200.0 [1] |
 | (Z)-5-((2-Methyl-2H-chromen-3-yl)methylene)-2-((E)-styryl)thiazolo[3,2-b][1,2,4]triazol-6(5H)-one | IC50 | 48700.0 [1] |
 | 5-(2-(4-Bromobenzyloxy)benzylidene)-2-thioxothiazolidin-4-one | IC50 | 1600.0 [1] |
 | 5-Amino-3-benzylsulfanyl-6-[(Z)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-[1,2,4]thiadiazolo[4,5-a]pyrimidin-7-one | IC50 | 27700.0 [1] |
 | Propan-2-yl (E)-3-(3-bromo-4-hydroxy-5-methoxyphenyl)-2-cyanoprop-2-enoate | IC50 | 69400.0 [1] |
 | 2-(1,3-Benzothiazol-2-ylamino)-6-phenylpyrimidine-4-carboxylic acid | IC50 | 37800.0 [1] |
 | Prop-2-enyl (E)-3-(3-bromo-4-hydroxyphenyl)-2-cyanoprop-2-enoate | IC50 | 47800.0 [1] |
 | 3-Hydroxy-2-phenyl-[1,3]thiazolo[3,2-a]pyridin-4-ium-8-carboxylic acid | IC50 | 102000.0 [1] |
 | [6-(2-Fluorophenyl)-5,8-dihydro-[1,3]dioxolo[4,5-g]quinolin-8-yl] dihydrogen phosphate | IC50 | 4930.0 [1] |