![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_006d0f3aa87eeac731a2bb8261074968.svg) | Fasudil | IC50 | 780.0 [1], 4000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_ec33dd540333b135ca60087b94fea344.svg) | Cyclohexanecarboxamide, 4-[(1R)-1-aminoethyl]-N-4-pyridinyl-, trans- | IC50 | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 2.2 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_07ed37209e0d1ed8b2069d600eb2723d.svg) | Y-27632 Dihydrochloride | IC50 | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_c77eb69f87d46b4d00314a6bfb851cf8.svg) | Crizotinib | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_fe739739798d5a426922dc4c74a41375.svg) | (4S,6Z,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_99d590530c99b53efc4907213bcd8b23.svg) | 7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrile | Ki | 8195.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_21aa752395444707db3d7c65ae53dc35.svg) | 1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acid | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_1565b2d807a215b6a10da52d9cb6c464.svg) | N'-(3-Pyridin-4-yl-2,6-naphthyridin-1-yl)ethane-1,2-diamine | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_b43f9b172387f2a84cebdafc2497da4c.svg) | cis-3-[4-Amino-7-(3-azetidin-1-ylmethyl-cyclobutyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]-phenol | IC50 | 2400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_dbc9774b4a10efc12e4d4309ee79f133.svg) | (13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dione | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_2b4938336d47e67252d45dde101abe28.svg) | N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(dimethylamino)-2-phenylacetamide | IC50 | 2300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_16ce37733bd768c6e666cdabec5d62d1.svg) | N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(cyclopropylamino)-2-phenylacetamide | IC50 | 8000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_da33bd60718fb74d356938fd32d1e232.svg) | N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(methylamino)-2-phenylacetamide | IC50 | 110.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_1156fb4b89335573c15a89baa29ae94b.svg) | 2-Methyl-N~1~-[3-(Pyridin-4-Yl)-2,6-Naphthyridin-1-Yl]propane-1,2-Diamine | IC50 | 17.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_947cf1c4060c0cf66f2ed2f8a80005fd.svg) | (3S,4R)-N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | IC50 | 14.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_6895eda4789a8360c158c764a4c5b856.svg) | 2-Amino-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamide | IC50 | 510.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_bd7ab61fd74e87578c2dfefbcc47d031.svg) | 7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_84ad2ce5fbf306770a6c850a5b17125a.svg) | 9-Cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_61551f1612b1d03b33f689e3fdae85ae.svg) | 2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Ki | 77.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_dc19af93aca15ed046c17748663ce5b7.svg) | 2-Methyl-1-N-(2-pyridin-4-ylpyrido[3,4-d]pyrimidin-4-yl)propane-1,2-diamine | IC50 | 58.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_371c3707e8831c9b0b53b88dc4f18976.svg) | 2-(1H-Indazol-5-yl)-4-piperazin-1-ylquinazoline | IC50 | 995.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_d74d4d16ec049016f870981de62b475f.svg) | 3-(1H-Indazol-5-yl)-1-piperazin-1-ylisoquinoline | IC50 | 920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_528cfaf5b96dd156938ca398d0e87e46.svg) | N'-[2-(1H-Indazol-5-yl)quinazolin-4-yl]ethane-1,2-diamine | IC50 | 951.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_1bd83937ae7bc58b4162f5b53407ff10.svg) | N'-[2-(1H-Indazol-5-yl)quinazolin-4-yl]propane-1,3-diamine | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_acb5d0f1f956d9a5855159b35889cb53.svg) | 2-(1H-Indazol-5-yl)-4-(4-methylpiperazin-1-yl)quinazoline | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_a0f8e89f029b8cd9d04f636375ccfa18.svg) | N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamide | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_984f1d19dd4f7aff4c8096322cf2c2cd.svg) | 4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_ba4191031ad1833485eab4917c42fd7c.svg) | N-[3-(4-Dimethylaminomethyl-phenylcarbamoyl)-benzyl]-3,4-dimethoxy-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_3d42f79fca7f259efedce4901f024390.svg) | 3-Chloro-N-[3-(4-dimethylaminomethyl-phenylcarbamoyl)-benzyl]-4-methoxy-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_0b6988c3cf36dab472a3ad574d320c7a.svg) | 3,4-Dimethoxy-N-[3-(3-piperidin-3-yl-propionylamino)-benzyl]-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_d2455f54fef1eacbfa124c42ccdfe21c.svg) | 3-[3-(4-Cyano-phenyl)-ureidomethyl]-N-(1,2,3,4-tetrahydro-isoquinolin-7-yl)-benzamide | IC50 | 1600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_292979b9b1bc0ecbad9a056b7c2ddb1a.svg) | 3-[3-(4-Cyano-phenyl)-ureidomethyl]-N-(2-piperidin-3-yl-ethyl)-benzamide | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_212e89804f13e737eec8680ba5410af1.svg) | 3-[3-(3-Cyano-phenyl)-ureidomethyl]-N-(2-piperidin-3-yl-ethyl)-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_ccc7ec8c9e66ce8127930267b47cd007.svg) | 3-[3-(4-Cyano-phenyl)-ureidomethyl]-N-(4-dimethylaminomethylphenyl)-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_88c6210996ec5f73c149549e4aef7dbc.svg) | 3,4-Dimethoxy-N-[3-(2-piperidin-3-yl-ethylcarbamoyl)-benzyl]-benzamide | IC50 | 4400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_f43a289da9112d38ebaad50830605e47.svg) | 3,4-Dimethoxy-N-[3-(1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_8c7c416cd2e77fda5ef21e47110b39ab.svg) | 3,4-Dimethoxy-N-[3-(2-piperidin-4-yl-ethylcarbamoyl)-benzyl]-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_47389838a9aec6294ab73cfa5f8df773.svg) | 3,4-Dimethoxy-N-[3-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamide | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_38eb3f174ec5b88705015915fd85d246.svg) | 3-[[(4-Carbamoylphenyl)carbamoylamino]methyl]-N-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamide | IC50 | 770.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_ef5580b860ce268bf20d4e34768a6fb7.svg) | 2-(Benzylamino)-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)acetamide | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_03e0d1a2e88126708ed3a73e7e36755b.svg) | N-[5-[6-(Methylamino)pyrazin-2-yl]-2-oxo-1H-pyridin-3-yl]-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]benzamide | Ki | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_657c8c4caed986ad8356aa0b751c2e39.svg) | (4S,6Z,10S)-10,18-Dihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_a840767d7ddb2c27c40164419a996160.svg) | Infigratinib phosphate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_700247dab7b9fdcc2d81fe4984afa76c.svg) | 2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_78dd939207cb0503fa3cbab2732a9f06.svg) | 7-[3-(Azetidin-1-ylmethyl)cyclobutyl]-5-[3-(7-oxabicyclo[2.2.1]heptan-1-ylmethoxy)phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_a7fde301c04af122ad328d1cb3f126ab.svg) | 1-[4-[3-[4-Amino-5-[2-fluoro-3-[[(2S)-oxolan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl]piperazin-1-yl]ethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_a71b8bbffb08d6de93d28151b96024da.svg) | N~1~-[2-(1h-Indazol-5-Yl)pyrido[3,4-D]pyrimidin-4-Yl]-2-Methylpropane-1,2-Diamine | IC50 | 742.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_ad946fa32618a037eb1c316583993f21.svg) | 9-[[8-Fluoro-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]sulfanyl]-4-methyl-[1,4]oxazino[3,2-c]quinolin-3-one | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n2_c1af48a2d7eaa6bdbe6dedeb932db20a.svg) | 2-(1H-Indazol-5-yl)-4-piperazin-1-ylpyrido[3,4-d]pyrimidine | IC50 | 974.0 [1] |