![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 1.0 [1], 1.2 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_2016e1fb48c552930d228a3e7f6e1433.svg) | Quercetin | IC50 | 5800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_006d0f3aa87eeac731a2bb8261074968.svg) | Fasudil | IC50 | 1700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_e0e66b7329f74ac9e778459370265f14.svg) | Norlichexanthone | IC50 | 54900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_fe739739798d5a426922dc4c74a41375.svg) | (4S,6Z,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 4900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_5a8e321781069aee089dcc439066b321.svg) | 2,3,6,8-Tetrahydroxy-1-methylxanthone | IC50 | 45300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_5803643fba2a49f1581ea6790292d883.svg) | Epicoccolide B | IC50 | 9000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_d72e6a5f6bda112109d526c400d3a392.svg) | Astrogorgiadiol B | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_e24a6ef90b6dda81406d577957bafbf2.svg) | (1S,9R)-5,6,12,13,14-Pentahydroxy-4,11-dimethyl-16-oxo-8,17-dioxatetracyclo[7.7.1.02,7.010,15]heptadeca-2(7),3,5,10,12,14-hexaene-3-carbaldehyde | IC50 | 4480.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_8547ec1c061a6923170866cf54d1c0d4.svg) | (1R,3As,4S,5R,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(2R)-6-methyl-5-methylideneheptan-2-yl]-1,2,3,3a,4,5,6,7-octahydroinden-5-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_9f0649c0af7300504c89d15a04caf360.svg) | Calicoferol B | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_1565b2d807a215b6a10da52d9cb6c464.svg) | N'-(3-Pyridin-4-yl-2,6-naphthyridin-1-yl)ethane-1,2-diamine | IC50 | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_89f93b41ac7e8a2307bd8fc1d9fad8a4.svg) | Calicoferol E | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_b43f9b172387f2a84cebdafc2497da4c.svg) | cis-3-[4-Amino-7-(3-azetidin-1-ylmethyl-cyclobutyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]-phenol | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_1156fb4b89335573c15a89baa29ae94b.svg) | 2-Methyl-N~1~-[3-(Pyridin-4-Yl)-2,6-Naphthyridin-1-Yl]propane-1,2-Diamine | IC50 | 35.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_a7ee75d4a7ce2e8d7ffa73cb444c324f.svg) | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_bd7ab61fd74e87578c2dfefbcc47d031.svg) | 7,8-Dichloro-9-methyl-1-oxospiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | IC50 | 310.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_84ad2ce5fbf306770a6c850a5b17125a.svg) | 9-Cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine | IC50 | 6100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_51153882d3ab9f3566d96aeaf5c3eeab.svg) | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_eda1570f6e608eea37da447234534ac5.svg) | 2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_70b0d2cbc054446af80b12d3d42fd894.svg) | (8S,16S)-3,16-Dihydroxy-9,10-seco-1,3,5(10)-cholestatrien-9-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_c67b754da3023ab057380dedf2f5a397.svg) | Calicoferol A | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_3ba3cfff437203d3cd5cef3fe6f6283a.svg) | (1R,3As,4S,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(2R)-6-methyl-5-methylideneheptan-2-yl]-2,3,3a,4,6,7-hexahydro-1H-inden-5-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_0b37fcadf8f90dc3bf2f29ca0be2a519.svg) | Methyl 3-[[(1R,2S,4aR,8aS)-1,2,4a,5-tetramethyl-2,3,4,7,8,8a-hexahydronaphthalen-1-yl]methyl]-4,5-dihydroxybenzoate | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_dc19af93aca15ed046c17748663ce5b7.svg) | 2-Methyl-1-N-(2-pyridin-4-ylpyrido[3,4-d]pyrimidin-4-yl)propane-1,2-diamine | IC50 | 99.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_371c3707e8831c9b0b53b88dc4f18976.svg) | 2-(1H-Indazol-5-yl)-4-piperazin-1-ylquinazoline | IC50 | 990.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_d74d4d16ec049016f870981de62b475f.svg) | 3-(1H-Indazol-5-yl)-1-piperazin-1-ylisoquinoline | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_528cfaf5b96dd156938ca398d0e87e46.svg) | N'-[2-(1H-Indazol-5-yl)quinazolin-4-yl]ethane-1,2-diamine | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_1bd83937ae7bc58b4162f5b53407ff10.svg) | N'-[2-(1H-Indazol-5-yl)quinazolin-4-yl]propane-1,3-diamine | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_acb5d0f1f956d9a5855159b35889cb53.svg) | 2-(1H-Indazol-5-yl)-4-(4-methylpiperazin-1-yl)quinazoline | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_657c8c4caed986ad8356aa0b751c2e39.svg) | (4S,6Z,10S)-10,18-Dihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),6,15,17-tetraene-2,8-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_97782ec01f992a8c58c39479f3daac33.svg) | (1R,3As,4S,5S,7aR)-4-[2-(5-hydroxy-2-methylphenyl)ethyl]-7a-methyl-1-[(E,2R)-6-methylhept-3-en-2-yl]-1,2,3,3a,4,5,6,7-octahydroinden-5-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_a840767d7ddb2c27c40164419a996160.svg) | Infigratinib phosphate | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_78dd939207cb0503fa3cbab2732a9f06.svg) | 7-[3-(Azetidin-1-ylmethyl)cyclobutyl]-5-[3-(7-oxabicyclo[2.2.1]heptan-1-ylmethoxy)phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | IC50 | 9700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_4c1c8e479c2e24660577929dfcea7599.svg) | 1-[4-[3-[4-Amino-5-[2-fluoro-5-[[(2S)-oxolan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl]piperazin-1-yl]ethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_a7fde301c04af122ad328d1cb3f126ab.svg) | 1-[4-[3-[4-Amino-5-[2-fluoro-3-[[(2S)-oxolan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl]piperazin-1-yl]ethanone | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_9b03225f89ed1195cf6b61682b2da5be.svg) | 1-[(3-Hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea;methanesulfonic acid | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_2701abbecbbf9efa0380ee28c8506637.svg) | 5,6,7-Trihydroxy-3-methoxy-4-methyl-3H-2-benzofuran-1-one | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_612cf2f12be0491ec6322bc2fc5e0648.svg) | 3-[[(1R,2S,4Ar,8aS)-1,2,4a,5-tetramethyl-2,3,4,7,8,8a-hexahydronaphthalen-1-yl]methyl]-4-hydroxy-5-(3-methylbutylamino)cyclohexa-3,5-diene-1,2-dione | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_1b21d28ce8b966a8686d0a33c7f6b5b3.svg) | CID 76324771 | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_814f4d20d9ed3f1c6f4967b9222f070e.svg) | 4-Methyl-5,6,7-trihydroxy-1,3-dihydroisobenzofuran-1-one | IC50 | 18600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_003730b1b76f77cca5ee4ec12a87c84b.svg) | 7-[[(1R,2S,4Ar,8aS)-1,2,4a,5-tetramethyl-2,3,4,7,8,8a-hexahydronaphthalen-1-yl]methyl]-5-methoxy-2-methyl-1,3-benzoxazol-6-ol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_a71b8bbffb08d6de93d28151b96024da.svg) | N~1~-[2-(1h-Indazol-5-Yl)pyrido[3,4-D]pyrimidin-4-Yl]-2-Methylpropane-1,2-Diamine | IC50 | 547.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_ad946fa32618a037eb1c316583993f21.svg) | 9-[[8-Fluoro-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]sulfanyl]-4-methyl-[1,4]oxazino[3,2-c]quinolin-3-one | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-n1_c1af48a2d7eaa6bdbe6dedeb932db20a.svg) | 2-(1H-Indazol-5-yl)-4-piperazin-1-ylpyrido[3,4-d]pyrimidine | IC50 | 1000.0 [1] |