![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_fbdf65d01abe32bcfa6dbda4a0a90dcc.svg) | N2-(2-Chlorobenzyl)-N4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitropyrimidine-2,4-diamine | IC50 | 18.0 [1], 29.0 [2], 46.0 [3], 290.0 [4], 630.0 [5] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_6ce223fbd5241efea172edc836e9b6c1.svg) | Sotrastaurin | IC50 | 1.0 [1], 81.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_f06ae3a73167a2538deab22ad6195e18.svg) | Indolactam V | Ki | 8.7 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_5f951503cd8519971704b7d1444d5a7e.svg) | 5-(3,4-Dimethoxyphenyl)-4-(1H-indol-5-ylamino)nicotinonitrile | IC50 | 70.0 [1], 150.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_5f951503cd8519971704b7d1444d5a7e.svg) | 5-(3,4-Dimethoxyphenyl)-4-(1H-indol-5-ylamino)nicotinonitrile | Ki | 79.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_089400a91a1f447d0307ea048744acf0.svg) | 4-[(3-Bromophenyl)amino]-5-(3,4-dimethoxyphenyl)nicotinonitrile | IC50 | 150.0 [1], 4600.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_089400a91a1f447d0307ea048744acf0.svg) | 4-[(3-Bromophenyl)amino]-5-(3,4-dimethoxyphenyl)nicotinonitrile | Ki | 4900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_bf510744cb83a77fbc98859859fc334a.svg) | 2-[3-[(Dimethylamino)methyl]phenyl]-4-[(4-methyl-1H-indol-5-yl)amino]thieno[2,3-b]pyridine-5-carbonitrile | IC50 | 7.5 [1], 230.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_bf510744cb83a77fbc98859859fc334a.svg) | 2-[3-[(Dimethylamino)methyl]phenyl]-4-[(4-methyl-1H-indol-5-yl)amino]thieno[2,3-b]pyridine-5-carbonitrile | Ki | 9.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_672e7998b8a2d8ffbf57a9a8fcc11921.svg) | (2R)-2-[(2S)-4-[3-Chloro-5-fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | IC50 | 11.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_672e7998b8a2d8ffbf57a9a8fcc11921.svg) | (2R)-2-[(2S)-4-[3-Chloro-5-fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | Ki | 0.08 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_017dba2ebab49191d2376ab32875e32f.svg) | CID 76285722 | IC50 | 23.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_12522883f9a9aed57303234cc665f8b8.svg) | 8-Octyl-benzolactam-V9 | Ki | 290.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_4d09b7ab6f7f3cabdcfc17a7797a09aa.svg) | 4-(4-Methyl-1H-indol-5-ylamino)-5-(4-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)nicotinonitrile | IC50 | 7.4 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_08f3e7d3dec6f7ed4214557b200967be.svg) | (1S,3R,5R,9R,13R)-9-(Hydroxymethyl)-3-[4-(3-hydroxyphenyl)butyl]-16,16-dimethyl-2,6,10,17-tetraoxatricyclo[11.3.1.11,5]octadecane-7,11-dione | Ki | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_1565b2d807a215b6a10da52d9cb6c464.svg) | N'-(3-Pyridin-4-yl-2,6-naphthyridin-1-yl)ethane-1,2-diamine | IC50 | 77.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_7b6d64791d06a7e25ffce6c3c06aa871.svg) | 2,2-Dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-1-[(1R)-1-phenylethyl]-3H-quinazolin-4-one | IC50 | 0.25 [1], 11.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_2e4490abba951f4f3613d6878836b906.svg) | 8-Decyl-5-hydroxymethyl-2-isopropyl-1-methyl-1,2,5,6-tetrahydro-benzo[e][1,4]oxazocin-3-one | Ki | 1097.0 [1], 1100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_69ef1b0b7b21a72d0f8a8c6ad8b2fa0b.svg) | 5-(3,4-Dimethoxyphenyl)-4-(1H-indol-6-ylamino)pyridine-3-carbonitrile | IC50 | 2000.0 [1], 2300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_a919527161761a8a385e53b6176933f1.svg) | 5-(3,4-Dimethoxyphenyl)-4-(1H-indol-4-ylamino)pyridine-3-carbonitrile | IC50 | 13.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_27fcafcac574dd57e209554c040ba332.svg) | (2-Aminopyridine-3-yl)(6-(1,4-diazepan-1-yl)pyridine-2-yl)methanone | Ki | 164.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_1156fb4b89335573c15a89baa29ae94b.svg) | 2-Methyl-N~1~-[3-(Pyridin-4-Yl)-2,6-Naphthyridin-1-Yl]propane-1,2-Diamine | IC50 | 141.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_2d992db0f2ddb156295918bc8b096ec9.svg) | 3,5-Dihydro[1,2,4]triazino[3,4-C][1,4]benzoxazin-2(1h)-One | IC50 | 19000.0 [1], 453000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_692f505f66b5060fb479a0f5943dc69b.svg) | 3-(1H-Indol-3-yl)-4-[3-(4-methylpiperazin-1-yl)naphthalen-1-yl]pyrrole-2,5-dione | IC50 | 4.8 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_ab49707c1490889471a5730adcedee9d.svg) | 4-(1H-Indol-5-ylamino)-2-phenylthieno[2,3-b]pyridine-5-carbonitrile | IC50 | 52.0 [1], 460.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_83e87e5bdde1cffc75fd9476c6917bde.svg) | 4-(4-Methyl-1H-indol-5-ylamino)-5-(4-(2-(4-methylpiperazin-1-yl)ethoxy)styryl)nicotinonitrile | IC50 | 3.6 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_a7722e986ca7e025e7a2957059f71c54.svg) | (2-Aminopyridin-3-yl)-(6-piperazin-1-ylpyridin-2-yl)methanone | Ki | 32.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_02b601235c2eef4bc604ea317f51a9af.svg) | 3-(2-Chloro-6-dimethylaminomethyl-naphthalen-1-yl)-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione | IC50 | 19.0 [1], 185.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_5095f27b300a6371b7e5509e028c096a.svg) | 3-[2-Chloro-7-[(dimethylamino)methyl]naphthalen-1-yl]-4-(1H-indol-3-yl)pyrrole-2,5-dione | IC50 | 216.0 [1], 708.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_de8f28e51e9e9ab4d05b26fe0dfe32ba.svg) | 3-[2-Chloro-6-[(dimethylamino)methyl]naphthalen-1-yl]-4-(1H-indol-3-yl)pyrrole-2,5-dione | IC50 | 12.0 [1], 156.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_4fdd7b15b614d8927bd5a9cf0fe4cc0c.svg) | 1-Benzyl-2,2-dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-3H-quinazolin-4-one | IC50 | 0.46 [1], 16.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_e08d65c52500dfd17dd8259b9d4ef7c0.svg) | 1-(Cyclopropylmethyl)-2,2-dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-3H-quinazolin-4-one | IC50 | 170.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_4468db7bc251cef268e44d94e0d10b9f.svg) | 1-Ethyl-2,2-dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-3H-quinazolin-4-one | IC50 | 260.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_c9ac75a9df88809326649edd02cab760.svg) | 2,2-Dimethyl-1-(2-methylpropyl)-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-3H-quinazolin-4-one | IC50 | 45.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_d8e6836e631f2b47ba4f713386d8cd5d.svg) | 2,2-Dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-1-(2-phenylethyl)-3H-quinazolin-4-one | IC50 | 300.0 [1], 1000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_6f39b20811823139bfd5ed8b115443aa.svg) | 1-(Cyclopentylmethyl)-2,2-dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-3H-quinazolin-4-one | IC50 | 4.3 [1], 170.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_b5d03571a49075d84f795e482d555905.svg) | 5-Fluoro-2-[(3S)-3-[(2R)-2-hydroxy-3-methylbutan-2-yl]piperazin-1-yl]-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-3-ol | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_b5d03571a49075d84f795e482d555905.svg) | 5-Fluoro-2-[(3S)-3-[(2R)-2-hydroxy-3-methylbutan-2-yl]piperazin-1-yl]-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-3-ol | Ki | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_8a13c9aec7afef9a9d3145228777a307.svg) | 3-[2-Chloro-7-[[cyclopropyl(methyl)amino]methyl]naphthalen-1-yl]-4-(1-methylindol-3-yl)pyrrole-2,5-dione | IC50 | 316.0 [1], 3555.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_61bbc2a0191b8cbfcfe0a837c4cbf886.svg) | (2-Aminopyridin-3-yl)-[6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | IC50 | 165.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_61bbc2a0191b8cbfcfe0a837c4cbf886.svg) | (2-Aminopyridin-3-yl)-[6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | Ki | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_f4bd6c874d6513a81ee59f60c1e4a18d.svg) | (2-Aminopyridin-3-yl)-[3-cyclopropyl-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | IC50 | 2600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_f4bd6c874d6513a81ee59f60c1e4a18d.svg) | (2-Aminopyridin-3-yl)-[3-cyclopropyl-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | Ki | 28.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_07671e672ecb8716436948a27c13beed.svg) | (S)-(2-Aminopyridin-3-yl)(6-(3-isobutylpiperazin-1-yl)-3-(trifluoromethyl)pyridin-2-yl)methanone | IC50 | 52.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_07671e672ecb8716436948a27c13beed.svg) | (S)-(2-Aminopyridin-3-yl)(6-(3-isobutylpiperazin-1-yl)-3-(trifluoromethyl)pyridin-2-yl)methanone | Ki | 3.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_13c91843039eeb03797e384d139f3930.svg) | (2-Aminopyridin-3-yl)-[3-chloro-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | IC50 | 58.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_13c91843039eeb03797e384d139f3930.svg) | (2-Aminopyridin-3-yl)-[3-chloro-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | Ki | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_9be20be6caab186175a3a5ffe3b1283a.svg) | (2R)-2-[(2S)-4-[3,5-Difluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_9be20be6caab186175a3a5ffe3b1283a.svg) | (2R)-2-[(2S)-4-[3,5-Difluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | Ki | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_9cbba9236f9ba08f4eca7cc37b53ae52.svg) | 5-Fluoro-2-[(3S)-3-[(2R)-2-hydroxy-3-methylbutan-2-yl]piperazin-1-yl]-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridine-3-carbonitrile | IC50 | 120.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_9cbba9236f9ba08f4eca7cc37b53ae52.svg) | 5-Fluoro-2-[(3S)-3-[(2R)-2-hydroxy-3-methylbutan-2-yl]piperazin-1-yl]-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridine-3-carbonitrile | Ki | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_ca1babfe7a92a1c446a8c63e73be2dfe.svg) | (2R)-2-[(2S)-4-[5-Fluoro-3-(hydroxymethyl)-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | IC50 | 1.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_ca1babfe7a92a1c446a8c63e73be2dfe.svg) | (2R)-2-[(2S)-4-[5-Fluoro-3-(hydroxymethyl)-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | Ki | 0.1 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_82b1b719209b675377595001b058c03e.svg) | 3-(2-Chloro-7-dimethylaminomethyl-naphthalen-1-yl)-4-(1-methyl-1H-indol-3-yl)-pyrrole-2,5-dione | IC50 | 263.0 [1], 402.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_97b2c5c6469fdb343d3563869cf4f5b3.svg) | (2-Aminopyridin-3-yl)-[6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]-3-propylpyridin-2-yl]methanone | IC50 | 410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_97b2c5c6469fdb343d3563869cf4f5b3.svg) | (2-Aminopyridin-3-yl)-[6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]-3-propylpyridin-2-yl]methanone | Ki | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_134549be413feb40dec54ef3e063dcd7.svg) | (2-Aminopyridin-3-yl)-[3-(difluoromethoxy)-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | IC50 | 229.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_134549be413feb40dec54ef3e063dcd7.svg) | (2-Aminopyridin-3-yl)-[3-(difluoromethoxy)-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | Ki | 7.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_949c166b97b7630cd9052552b6352e67.svg) | (2-Aminopyridin-3-yl)-[6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]-3-phenylpyridin-2-yl]methanone | IC50 | 5.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_949c166b97b7630cd9052552b6352e67.svg) | (2-Aminopyridin-3-yl)-[6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]-3-phenylpyridin-2-yl]methanone | Ki | 0.6 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_0054bf14e96139589fa6ff8d49e23763.svg) | 4-[[(3R,5S)-4-Amino-1-adamantyl]methylamino]-2-[[2-(trifluoromethoxy)phenyl]methylamino]pyrimidine-5-carbonitrile | IC50 | 1.3 [1], 22.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_241b09a1a0949327cad8fdb81e94b3be.svg) | 4-[[(3R,5S)-4-Amino-1-adamantyl]methylamino]-2-(3-bromoanilino)pyrimidine-5-carbonitrile | IC50 | 3.9 [1], 100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_e614f8ab712fc2f3aa9201ab058b4fe7.svg) | 4-[[(3R,5S)-4-Amino-1-adamantyl]methylamino]-2-anilinopyrimidine-5-carbonitrile | IC50 | 28.0 [1], 660.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_37a3b2f3020a72e90775d189cd0d896a.svg) | 2-[[(1R,3S)-5-[[[5-Cyano-2-[[2-(trifluoromethoxy)phenyl]methylamino]pyrimidin-4-yl]amino]methyl]-2-adamantyl]amino]acetamide | IC50 | 1.9 [1], 41.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_5599fb249b65659a7bb9dac09668c6f2.svg) | 4-[[(3R,5S)-4-(2-Hydroxyethylamino)-1-adamantyl]methylamino]-2-[[2-(trifluoromethoxy)phenyl]methylamino]pyrimidine-5-carbonitrile | IC50 | 0.7 [1], 6.3 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_28aa37114a8a457f9c8b43134333f82d.svg) | 4-[[(3R,5S)-4-Amino-1-adamantyl]methylamino]-2-[(2-bromophenyl)methylamino]pyrimidine-5-carbonitrile | IC50 | 5.9 [1], 31.0 [2] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_93c21b71ad6e74f4964c81e68b18d8d5.svg) | (2-Aminopyridin-3-yl)-[4-methyl-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | IC50 | 410.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_93c21b71ad6e74f4964c81e68b18d8d5.svg) | (2-Aminopyridin-3-yl)-[4-methyl-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone | Ki | 24.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_ee4e586a9e26d338e60f7b4d788ed143.svg) | (2R)-2-[(2S)-4-[5-Fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | IC50 | 6.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_ee4e586a9e26d338e60f7b4d788ed143.svg) | (2R)-2-[(2S)-4-[5-Fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | Ki | 0.2 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_1c717d22d1378d2c01196c07d713b779.svg) | (2R)-2-[(2S)-4-[5-Chloro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | IC50 | 170.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_1c717d22d1378d2c01196c07d713b779.svg) | (2R)-2-[(2S)-4-[5-Chloro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-ol | Ki | 21.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_90491a5646ab353d88ec5ca044a2cd78.svg) | (2R)-3-Methyl-2-[(2S)-4-[6-(2H-pyrazolo[3,4-b]pyridin-3-yl)-5-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]butan-2-ol | IC50 | 420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_90491a5646ab353d88ec5ca044a2cd78.svg) | (2R)-3-Methyl-2-[(2S)-4-[6-(2H-pyrazolo[3,4-b]pyridin-3-yl)-5-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]butan-2-ol | Ki | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_8971c4c32e37132a094823a464bfcc9f.svg) | Phorbol 12,13-dibutyrate | Ki | 1.54 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_2ed4c94a2d5ffc8de608010761ebd89a.svg) | Bisindolylmaleimide i | IC50 | 6.7 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_5d9eab088a0c5589b89740e84fcbca6b.svg) | Xanthohumol | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_0a83b01cf93719a90ccaeda771089c43.svg) | Doramapimod | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_0f28c9659401d00170d1048c776a152f.svg) | Aplysiatoxin | Ki | 0.16 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_0ddf3e5dfb61c54e2addad647a866dcb.svg) | Isoxanthohumol | IC50 | 31600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_67f4e732a49bf39a183fb443d695bf12.svg) | Gsk-690693 | IC50 | 2.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_fe6203f147bd42417709582aca6cd0a9.svg) | Debromoaplysiatoxin | Ki | 0.11 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_c74a1b9d6feb1def6b7e3f6834b5761b.svg) | Tak-285 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_c71081a8619ec348ecd13cc61c9f2023.svg) | CID 46209401 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_836d58634120a742d63c1602f26addff.svg) | CID 59604787 | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_941408e43c25b505975eab00c707db56.svg) | 1-[2-Fluoro-4-(5-methylpyrrolo[3,2-d]pyrimidin-4-yl)oxyphenyl]-3-[3-(trifluoromethyl)phenyl]urea | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_9a65d2cfdcb6c2711e673a4cb101fbc0.svg) | 3-[5-[4-(2-Hydroxy-2-methylpropanoyl)piperazin-1-yl]-2-(trifluoromethyl)phenyl]-4-(1H-indol-3-yl)pyrrole-2,5-dione | IC50 | 68.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_aa78cc3183c29821fe7c015c8320a3ff.svg) | CID 44814409 | IC50 | 4100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_6c1930b58c3218f1026ffccbe15b146f.svg) | 17,20,23-Trioxa-4,12,14,26,28-pentazahexacyclo[24.6.1.17,14.02,6.08,13.027,32]tetratriaconta-1(33),2(6),7(34),8(13),9,11,27(32),28,30-nonaene-3,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_46bba2bc4a87a0013dc3991e2036a0ae.svg) | Indolylylmaleimide 1 | IC50 | 835.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_801c554a8abc4fae0624107ac463a91f.svg) | 4-[(4-Methyl-1H-indol-5-yl)amino]-2-phenylthieno[2,3-b]pyridine-5-carbonitrile | IC50 | 52.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_2005d21a1b798bf9f66b264bafeb149e.svg) | 8-Bromo-4-(3-chloro-4-fluoroanilino)-6-[(1-methylimidazol-4-yl)methylamino]quinoline-3-carbonitrile | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_a5c5bae0fd3ddf532506780bb4f7f125.svg) | Khk-IN-1 | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_b43f9b172387f2a84cebdafc2497da4c.svg) | cis-3-[4-Amino-7-(3-azetidin-1-ylmethyl-cyclobutyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]-phenol | IC50 | 230.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_7e5f0df77e5b12da5aed8824d56b0324.svg) | Indolylylmaleimide 2 | IC50 | 65.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_7aea6f53dbac020fb411fced9f88f70b.svg) | (2S,5S)-8-Decyl-5-(hydroxymethyl)-1-methyl-2-propan-2-yl-2,4,5,6-tetrahydro-1,4-benzodiazocin-3-one | Ki | 13.2 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_e5c7a1e990d1af735a4c6d894ba6d642.svg) | Methyl 6-bromo-2-[(4-methylsulfonylphenyl)methyl]-1-oxo-4-phenylisoquinoline-3-carboxylate | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_e02cc3fb3f4bb5b162cd68fe36b13b1e.svg) | 17,20,23,26-Tetraoxa-4,12,14,29,31-pentazahexacyclo[27.6.1.17,14.02,6.08,13.030,35]heptatriaconta-1(36),2(6),7(37),8(13),9,11,30(35),31,33-nonaene-3,5-dione | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_8ea7b06e4b92347c86bcac69316b8ba6.svg) | (2,6-Dimethylphenyl) N-[2-[3,5-dimethoxy-4-[3-(4-methylpiperazin-1-yl)propoxy]anilino]pyrimidin-4-yl]-N-(2,4-dimethoxyphenyl)carbamate | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/protein-kinase-c-theta_29efefc9afcac9feac082a17257c193b.svg) | 3-(1H-Indol-3-yl)-4-(2-piperazin-1-ylquinazolin-4-yl)pyrrole-2,5-dione | IC50 | 0.5 [1] |