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Protein kinase C mu Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Cyclohexyl-[4-(1-piperazin-1-yl[2,6]naphthyridin-3-yl)pyridin-2-yl]amineIC500.6 [1], 32.0 [2]
Go-6976IC5027.0 [1], 62.0 [2]
7-Hydroxy-2,3,4,5-tetrahydro-1H-benzofuro[2,3-c]azepin-1-oneIC50182.0 [1], 11800.0 [2]
3,4-Dihydro-9-hydroxy-[1]benzothieno[2,3-f]-1,4-thiazepin-5(2H)-oneIC5028.3 [1], 2200.0 [2]
(1)Benzothieno(2,3-f)-1,4-thiazepin-5(2H)-one, 3,4-dihydro-9-methoxy-IC5082.5 [1], 3100.0 [2]
N'-(3-Pyridin-4-yl-2,6-naphthyridin-1-yl)ethane-1,2-diamineIC50321.0 [1], 5420.0 [2]
1-Piperazin-1-yl-3-pyridin-4-yl[2,6]naphthyridineIC5059.0 [1], 2096.0 [2]
3-[[3-[2-(Methylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]amino]propan-1-olIC50764.0 [1], 10000.0 [2]
2-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyridin-1-ylamino]ethanolIC50382.0 [1], 1000.0 [2]
Cyclohexyl-{4-[1-(4-methylpiperazin-1-yl)[2,6]naphthyridin-3-yl]pyridin-2-yl}amineIC502.0 [1], 206.0 [2]
3-(3-Pyridin-4-yl[2,6]naphthyridin-1-ylamino)propan-1-olIC5010000.0 [1], 40000.0 [2]
3-(2-Chloropyridin-4-yl)-1-piperazin-1-yl[2,6]naphthyridineIC5050.0 [1], 1000.0 [2]
Cyclohexyl-{4-[1-(4-isobutylpiperazin-1-yl)[2,6]naphthyridin-3-yl]pyridin-2-yl}amineIC506.0 [1], 299.0 [2]
N-(Oxan-4-yl)-4-(1-piperazin-1-yl-2,6-naphthyridin-3-yl)pyridin-2-amineIC500.4 [1], 10.0 [2]
{4-[1-(4-Isobutylpiperazin-1-yl)[2,6]naphthyridin-3-yl]pyridin-2-yl}(tetrahydropyran-4-yl)amineIC501.0 [1], 78.0 [2]
N-Cyclohexyl-4-[1-[(3S,5R)-3,5-dimethylpiperazin-1-yl]-2,6-naphthyridin-3-yl]pyridin-2-amineIC503.0 [1], 30.0 [2]
1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyridin-1-yl]piperidin-4-olIC5015.0 [1], 474.0 [2]
Cyclohexyl-{4-[1-(4-cyclopropylmethylpiperazin-1-yl)[2,6]naphthyridin-3-yl]pyridin-2-yl}amineIC502.0 [1], 221.0 [2]
Cyclohexyl-{4-[1-(4-cyclopropylpiperazin-1-yl)[2,6]naphthyridin-3-yl]pyridin-2-yl}amineIC5013.0 [1], 454.0 [2]
4-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyridin-1-yl]piperazin-2-oneIC501000.0 [1], 4931.0 [2]
4-[1-[4-(Aminomethyl)piperidin-1-yl]-2,6-naphthyridin-3-yl]-N-cyclohexylpyridin-2-amineIC501.0 [1], 49.0 [2]
2-Amino-1-[4-[3-[2-(oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperazin-1-yl]ethanoneIC505.0 [1], 749.0 [2]
1-[3-(2-Cyclohexylaminopyridin-4-yl)[2,6]naphthyridin-1-yl]-piperidine-4-carboxylic Acid AmideIC5083.0 [1], 204.0 [2]
1-[3-[2-(Oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperidine-4-carboxamideIC502.0 [1], 20.0 [2]
1-[3-[2-(Cyclohexylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]-N-methylpiperidine-4-carboxamideIC503.0 [1], 94.0 [2]
1-[3-[2-(Cyclohexylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]-N-(2-pyrrolidin-1-ylethyl)piperidine-4-carboxamideIC501.0 [1], 35.0 [2]
[1-[3-[2-(Cyclohexylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperidin-4-yl]-(4-hydroxypiperidin-1-yl)methanoneIC504.0 [1], 294.0 [2]
N-Ethyl-1-[3-[2-(oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperidine-4-carboxamideIC503.0 [1], 83.0 [2]
N-(2-Methylpropyl)-1-[3-[2-(oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperidine-4-carboxamideIC502.0 [1], 228.0 [2]
1-(1-Piperazinyl)-3-(2-cyclohexylaminopyrid-4-yl)isoquinolineIC5012.0 [1], 356.0 [2]
Cyclohexyl-[4-(8-piperazin-1-yl[1,7]naphthyridin-6-yl)pyridin-2-yl]amineIC50695.0 [1], 10000.0 [2]
Cyclohexyl-[4-(1-piperazin-1-yl[2,7]naphthyridin-3-yl)pyridin-2-yl]amineIC50191.0 [1], 1558.0 [2]
Cyclohexyl-[4-(5-piperazin-1-yl[1,6]naphthyridin-7-yl)pyridin-2-yl]amineIC5015.0 [1], 262.0 [2]
Cyclohexyl-[4-(4-piperazin-1-ylquinazolin-2-yl)pyridin-2-yl]-amineIC5043.0 [1], 1521.0 [2]
1-[3-[2-(Oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]-N-(2-pyrrolidin-1-ylethyl)piperidine-4-carboxamideIC501.0 [1], 96.0 [2]
N-(2-Hydroxyethyl)-1-[3-[2-(oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperidine-4-carboxamideIC502.0 [1], 60.0 [2]
1-[3-[2-(Cyclohexylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]-N-piperidin-4-ylpiperidine-4-carboxamideIC501.0 [1], 44.0 [2]
1-[4-[3-[2-(Cyclohexylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]piperazin-2-yl]ethanoneIC5019.0 [1], 1000.0 [2]
10-Hydroxy-2,3,4,5-tetrahydro-[1]benzothiolo[3,2-b][1,5]thiazocin-6-oneIC50111.0 [1], 2600.0 [2]
4-Methoxy-8,14-dithia-3,5,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),2,4,6-tetraen-10-oneIC50124.0 [1], 6800.0 [2]
9-Azido-3,4-dihydro-2H-[1]benzothiolo[2,3-f][1,4]thiazepin-5-oneIC5074.9 [1], 2200.0 [2]
10-Methoxy-2,3,4,5-tetrahydro-[1]benzothiolo[3,2-b][1,5]thiazocin-6-oneIC50193.0 [1], 18600.0 [2]
3,4,5,10-Tetrahydro-7-hydroxy-azepino[3,4-b]indol-1(2H)-oneIC50130.0 [1], 50000.0 [2]
CrizotinibIC5010000.0 [1]
DoramapimodIC5030000.0 [1]
1-Cyclopropyl-3-(3-(5-(morpholinomethyl)-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-4-yl)ureaIC5010.0 [1]
CK1 InhibitorIC509100.0 [1]
1-Tert-butyl-3-(naphthalen-1-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC50250.0 [1]
4-(7-Butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl)phenolIC50100000.0 [1]
1-(Tert-Butyl)-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineIC50900.0 [1]
CID 53246941IC5035.0 [1]
CID 59604787IC5010000.0 [1]
3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-imidazol-2-yl)methyl)benzamideIC50650.0 [1]
BpkdiIC501.0 [1]
(2R)-2-[(2S)-4-[3-Chloro-5-fluoro-6-(2H-pyrazolo[3,4-b]pyridin-3-yl)pyridin-2-yl]piperazin-2-yl]-3-methylbutan-2-olKi2420.0 [1]
Benzonitrile, 3-(((5-(6-methyl-2-pyridinyl)-4-(6-quinoxalinyl)-1H-imidazol-2-yl)methyl)amino)-IC501000.0 [1]
(13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dioneIC501000.0 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamideIC5010000.0 [1]
(S)-6-(Piperidin-3-yloxy)-2H-isoquinolin-1-oneIC50501.19 [1]
N-Cyclohexyl-4-[6-piperazin-1-yl-4-(1H-pyrazol-5-yl)pyridin-2-yl]pyridin-2-amineIC504.0 [1]
4-[6-Piperazin-1-yl-4-(1H-pyrazol-4-yl)pyridin-2-yl]-N-propan-2-ylpyridin-2-amineIC501.0 [1]
N-(Oxan-4-yl)-4-[6-piperazin-1-yl-4-(1H-pyrazol-4-yl)pyridin-2-yl]pyridin-2-amineIC501.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[[(3R)-pyrrolidin-3-yl]amino]pyridine-4-carboxamideIC502.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[[(3S)-pyrrolidin-3-yl]amino]pyridine-4-carboxamideIC5068.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[(3R)-3-methylpiperazin-1-yl]pyridine-4-carboxamideIC506.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-[(3S)-3-methylpiperazin-1-yl]pyridine-4-carboxamideIC508.0 [1]
2-(3-Aminopiperidin-1-yl)-6-[2-(cyclohexylamino)pyridin-4-yl]pyridine-4-carboxamideIC5014.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-(4-methylpiperazin-1-yl)pyridine-4-carboxamideIC5025.0 [1]
2-[4-(Aminomethyl)piperidin-1-yl]-6-[2-(cyclohexylamino)pyridin-4-yl]pyridine-4-carboxamideIC5046.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-(3,3-dimethylpiperazin-1-yl)pyridine-4-carboxamideIC5055.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-morpholin-4-ylpyridine-4-carboxamideIC501000.0 [1]
N-Cyclohexyl-4-[6-piperazin-1-yl-4-(trifluoromethyl)pyridin-2-yl]pyridin-2-amineIC5020.0 [1]
N-Cyclohexyl-4-[4-(difluoromethyl)-6-piperazin-1-ylpyridin-2-yl]pyridin-2-amineIC5017.0 [1]
1-[3-[2-(Oxan-4-ylamino)pyridin-4-yl]-2,6-naphthyridin-1-yl]-N-propan-2-ylpiperidine-4-carboxamideIC50391.0 [1]
6-(2-Cyclohexylaminopyridin-4-yl)-4-piperazin-1-yl-2,3-dihydropyrrolo[3,4-c]pyridin-1-oneIC5035.0 [1]
4-(2-Cyclohexylaminopyridin-4-yl)-6-(piperazin-1-yl)-2,3-dihydropyrrolo[3,4-c]pyridin-1-oneIC501.0 [1]
2-(2-Anilinopyridin-4-yl)-6-piperazin-1-ylpyridine-4-carboxamideIC501.0 [1]
2-[2-(Oxan-4-ylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC501.0 [1]
2-Piperazin-1-yl-6-[2-(propan-2-ylamino)pyridin-4-yl]pyridine-4-carboxamideIC501.0 [1]
2-[2-[(1-Methylpyrazol-3-yl)amino]pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC501.0 [1]
2-[2-(2-Chloroanilino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC501.0 [1]
2-[2-(Cyclopentylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC506.0 [1]
2-[2-(Ethylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carboxamideIC504.0 [1]
2-[2-(Cyclohexylamino)pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carbonitrileIC5018.0 [1]
2-(2-Anilinopyridin-4-yl)-6-piperazin-1-ylpyridine-4-carbonitrileIC505.0 [1]
2-[2-[(1-Methylpyrazol-3-yl)amino]pyridin-4-yl]-6-piperazin-1-ylpyridine-4-carbonitrileIC508.0 [1]
N-Cyclohexyl-4-[6-piperazin-1-yl-4-(1H-pyrazol-4-yl)pyridin-2-yl]pyridin-2-amineIC501.0 [1]
N-[(1R)-1-Cyanoethyl]-3-[5-[4-[(oxan-4-ylamino)methyl]phenyl]-1,2-oxazol-3-yl]benzamideIC505.5 [1]
5-(1,4-Diazepan-1-ylsulfonyl)isoquinolin-1-amineIC5010000.0 [1]
N-[(1R)-1-Cyanoethyl]-3-[5-[4-[(propan-2-ylamino)methyl]phenyl]-1H-pyrazol-3-yl]benzamideIC503.7 [1]
N-[(1R)-1-Cyanoethyl]-3-[5-[4-[(propan-2-ylamino)methyl]phenyl]-1,2-oxazol-3-yl]benzamideIC509.0 [1]
3-[5-[4-(4-Methylpiperazin-1-yl)phenyl]-1H-pyrazol-3-yl]-N-propan-2-ylbenzamideIC501000.0 [1]
N-[(1R)-1-Cyanoethyl]-3-[5-[4-(4-methylpiperazin-1-yl)phenyl]-1,2-oxazol-3-yl]benzamideIC5060.0 [1]
N-[(1S)-1-Cyanoethyl]-3-[5-[4-(4-methylpiperazin-1-yl)phenyl]-1,2-oxazol-3-yl]benzamideIC50430.0 [1]
N-[3-[5-[4-(4-Methylpiperazin-1-yl)phenyl]-1H-pyrazol-3-yl]phenyl]acetamideIC502300.0 [1]
3-[5-[3-Bromo-4-(4-methylpiperazin-1-yl)phenyl]-1H-pyrazol-3-yl]-N-propan-2-ylbenzamideIC50280.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Protein kinase C mu Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/protein-kinase-c-mu-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Protein kinase C mu Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-kinase-c-mu-inhibitors-ic50-ki.
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