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Protein-glutamine gamma-glutamyltransferase K Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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N-(4-Bromophenyl)acrylamideIC5010000.0 [1]
N-[(5S)-6-[4-(6-Methylpyridin-2-yl)piperazin-1-yl]-6-oxo-5-[(2-phenylacetyl)amino]hexyl]prop-2-enamideIC5015000.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-2-nitro-benzenesulfonamideIC508100.0 [1]
Benzyl N-[(2S)-1-[4-(2-chlorophenyl)piperazin-1-yl]-1-oxo-6-(prop-2-enoylamino)hexan-2-yl]carbamateIC5012900.0 [1]
1-Ethyl-3-(4-methoxyphenyl)-6-methylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dioneIC5018.0 [1]
{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitro-benzenesulfonylamino)-hexyl]-amino}-acetic acidIC5017000.0 [1]
2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitro-benzenesulfonylamino)-hexyl]-amino}-acetamideIC5032000.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-methyl-amino)-hexyl]-2-nitro-benzenesulfonamideIC506200.0 [1]
(5-Bromothiophen-2-yl)(4-methyl-1H-pyrazol-1-yl)methanoneIC5011000.0 [1]
(2S)-1-Acetyl-N-[(2S)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-6-diazo-1,5-dioxohexan-2-yl]pyrrolidine-2-carboxamideIC5045000.0 [1]
N-[4-(Pyrrolidine-1-sulfonyl)phenyl]prop-2-enamideIC5025000.0 [1]
N-[4-[4-(Adamantane-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC503400.0 [1]
(2,3-Difluorophenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC506700.0 [1]
Cyclopentyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC502500.0 [1]
N-[4-[4-(Piperidine-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC504100.0 [1]
N-[4-[4-(Pyrrolidine-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC505400.0 [1]
N-[4-[4-(3-Phenylpropyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC5015000.0 [1]
Benzyl 4-[6-(prop-2-enoylamino)pyridin-3-yl]sulfonylpiperazine-1-carboxylateIC506400.0 [1]
N-[4-[4-(4-Phenylbutyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC5022000.0 [1]
N-[4-[4-(Cyclopropanecarbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC506000.0 [1]
N-[4-[4-(Cyclopentanecarbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC505600.0 [1]
N-[4-[4-(4,4-Difluoropiperidine-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC505400.0 [1]
Tert-butyl 4-[6-(prop-2-enoylamino)pyridin-3-yl]sulfonylpiperazine-1-carboxylateIC503800.0 [1]
Benzyl 5-[4-(prop-2-enoylamino)phenyl]sulfonyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-2-carboxylateIC509500.0 [1]
(3-Phenoxyphenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5012000.0 [1]
Benzyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC503700.0 [1]
Benzyl 4-[3-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC504100.0 [1]
Benzyl 4-[4-(prop-2-enoylamino)phenyl]sulfonyl-1,4-diazepane-1-carboxylateIC504600.0 [1]
4-(4-Acryloylamino-benzenesulfonyl)-piperazine-1-carboxylic acid tert-butyl esterIC504900.0 [1]
4-(4-Acryloylamino-benzenesulfonylamino)-piperidine-1-carboxylic acid benzyl esterIC502700.0 [1]
[1-(4-Acryloylamino-benzenesulfonyl)-piperidin-4-yl]-carbamic acid benzyl esterIC504600.0 [1]
4-(4-Acryloylamino-benzenesulfonyl)-piperazine-1-carboxylic acid 2-chloro-benzyl esterIC506100.0 [1]
Benzyl (3R)-3-[[4-(prop-2-enoylamino)phenyl]sulfonylamino]pyrrolidine-1-carboxylateIC503600.0 [1]
4-(4-Acryloylamino-2-trifluoromethyl-benzenesulfonyl)-piperazine-1-carboxylic acid benzyl esterIC501400.0 [1]
Benzyl N-methyl-N-[2-[methyl-[4-(prop-2-enoylamino)phenyl]sulfonylamino]ethyl]carbamateIC508100.0 [1]
Benzyl 4-[[[4-(prop-2-enoylamino)phenyl]sulfonylamino]methyl]piperidine-1-carboxylateIC501800.0 [1]
Benzyl N-[[1-[4-(prop-2-enoylamino)phenyl]sulfonylpiperidin-4-yl]methyl]carbamateIC502900.0 [1]
[2-(Trifluoromethyl)phenyl]methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC508300.0 [1]
Benzyl N-[(3R)-1-[4-(prop-2-enoylamino)phenyl]sulfonylpyrrolidin-3-yl]carbamateIC5014000.0 [1]
N-(4-Piperazin-1-ylsulfonylphenyl)prop-2-enamideIC5045000.0 [1]
N-[4-(4-Pyridin-2-ylpiperazin-1-yl)sulfonylphenyl]prop-2-enamideIC504500.0 [1]
N-[4-[4-(3-Methylpyridin-2-yl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC501700.0 [1]
N-[4-[4-(6-Methylpyridin-2-yl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC504200.0 [1]
N-[4-[4-[3-(Trifluoromethyl)pyridin-2-yl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC505900.0 [1]
N-[4-[4-[5-(Trifluoromethyl)pyridin-2-yl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC5018000.0 [1]
N-[4-(4-Phenylpiperazin-1-yl)sulfonylphenyl]prop-2-enamideIC506100.0 [1]
N-[4-[4-[2-(Trifluoromethyl)phenyl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC5057000.0 [1]
Benzyl (3S)-3-[[4-(prop-2-enoylamino)phenyl]sulfonylamino]pyrrolidine-1-carboxylateIC502900.0 [1]
Benzyl N-[(3S)-1-[4-(prop-2-enoylamino)phenyl]sulfonylpyrrolidin-3-yl]carbamateIC5014000.0 [1]
(4-Fluorophenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC504100.0 [1]
(3,5-Difluorophenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC509800.0 [1]
(2-Methylphenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC505100.0 [1]
Naphthalen-1-ylmethyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC506800.0 [1]
Naphthalen-2-ylmethyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5076000.0 [1]
Methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC506900.0 [1]
N-[4-[4-(3,4,4a,5,6,7,8,8a-Octahydro-1H-isoquinoline-2-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC507200.0 [1]
N-[4-[4-(3,4,4a,5,6,7,8,8a-Octahydro-2H-quinoline-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC502600.0 [1]
N-[4-[4-(3-Phenylpropanoyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC5010000.0 [1]
N-[4-[4-[(1S,2S)-2-Phenylcyclopropanecarbonyl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC503100.0 [1]
N-[5-[4-(Cyclopropanecarbonyl)piperazin-1-yl]sulfonylpyridin-2-yl]prop-2-enamideIC503400.0 [1]
N-[5-[4-(Adamantane-1-carbonyl)piperazin-1-yl]sulfonylpyridin-2-yl]prop-2-enamideIC505600.0 [1]
Tert-butyl 4-[2-(prop-2-enoylamino)pyrimidin-5-yl]sulfonylpiperazine-1-carboxylateIC501800.0 [1]
Benzyl 4-[2-(prop-2-enoylamino)pyrimidin-5-yl]sulfonylpiperazine-1-carboxylateIC505100.0 [1]
N-[5-[4-(Adamantane-1-carbonyl)piperazin-1-yl]sulfonylpyrimidin-2-yl]prop-2-enamideIC503000.0 [1]
Tert-butyl 4-[4-(2-fluoroprop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-(2-methylprop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(Z)-but-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(E)-but-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(E)-2-methylbut-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(Z)-3-chloroprop-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC508800.0 [1]
4-[4-(1-Oxo-but-2-ynylamino)-benzenesulfonyl]-piperazine-1-carboxylic acid tert-butyl esterIC5080000.0 [1]
Benzyl 4-[4-[(E)-4-ethoxy-4-oxobut-2-enyl]phenyl]sulfonylpiperazine-1-carboxylateIC508900.0 [1]
Benzyl 4-[3-[methyl(2-methylpropyl)amino]-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5014000.0 [1]
Benzyl 4-[3-fluoro-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5020000.0 [1]
4-(4-Acryloylamino-2-methoxy-benzenesulfonyl)-piperazine-1-carboxylic acid tert-butyl esterIC5019000.0 [1]
Tert-butyl 4-[2-methyl-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC506500.0 [1]
Tert-butyl 4-[2-fluoro-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC502400.0 [1]
Tert-butyl 4-[2-chloro-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50950.0 [1]
Ethyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC505000.0 [1]
Methyl (2S)-2-[[(2S)-1-[(2S)-5-amino-2-[[(E,2S)-6-methylsulfonyl-2-(phenylmethoxycarbonylamino)hex-5-enoyl]amino]-5-oxopentanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoateIC50250.0 [1]
Tert-butyl 4-(4-cyanophenyl)sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 5-[4-(prop-2-enoylamino)phenyl]sulfonyl-2,5-diazabicyclo[2.2.1]heptane-2-carboxylateIC5014000.0 [1]
(2-Phenoxyphenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5010000.0 [1]
(4-Phenoxyphenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC507700.0 [1]
N-[[4-(Aminomethyl)phenyl]methyl]-3-[5-[[[(E)-2-phenylethenyl]sulfonyl-(pyridin-2-ylmethyl)amino]methyl]-1,2,4-oxadiazol-3-yl]benzamideIC5080000.0 [1]
[4-(4-Acryloylamino-piperidine-1-sulfonyl)-phenyl]carbamic acid benzyl esterIC50910.0 [1]
Tert-butyl 2-[[(2S)-2-(phenylmethoxycarbonylamino)-6-(prop-2-enoylamino)hexanoyl]amino]acetateIC5080000.0 [1]
Benzyl N-[(2S)-1-oxo-1-(4-phenylpiperidin-1-yl)-6-(prop-2-enoylamino)hexan-2-yl]carbamateIC509300.0 [1]
N-[2-(4-Methoxyphenyl)ethyl]-4-[4-(prop-2-enoylamino)piperidin-1-yl]sulfonylbenzamideIC501200.0 [1]
Benzyl 4-[4-(4-diazo-3-oxobutyl)phenyl]sulfonylpiperazine-1-carboxylateIC506400.0 [1]
1-[(5-Methyl-[1,3]thiazolo[2,3-b][1,3,4]thiadiazol-4-ium-2-yl)sulfanyl]propan-2-oneIC50250.0 [1]
Items per page: 1 - 10 of 91
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References

This online tool may be cited as follows

MLA

"Quest Database™ Protein-glutamine gamma-glutamyltransferase K Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/protein-glutamine-gamma-glutamyltransferase-k-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Protein-glutamine gamma-glutamyltransferase K Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-glutamine-gamma-glutamyltransferase-k-inhibitors-ic50-ki.
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