Protein-arginine deiminase type-1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Streptonigrin	IC50	48300.0 [1]
	Cl-amidine (TFA)	Ki	62000.0 [1]
	F-Amidine	Ki	110000.0 [1]
	7-Amino-2-pyridin-2-ylquinoline-5,8-dione	IC50	950.0 [1]
	7-Bromo-6-methoxyquinoline-5,8-dione	IC50	4550.0 [1]
	6-(7-Amino-5,8-dioxo-5,8-dihydroquinolin-2-yl)picolinic acid	IC50	70.0 [1]
	7-Aminoquinoline-5,8-dione	IC50	960.0 [1]
	2-{[(2s)-1-Amino-5-{[(1z)-2-Fluoroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic Acid	Ki	9400.0 [1]
	5,5-Dimethyl-3-(piperazin-1-ylmethyl)imidazolidine-2,4-dione	Ki	445000.0 [1]
	N-[(2S)-1-(Benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]furan-2-carboxamide	Ki	1086000.0 [1]
	N-[(2S)-1-(Benzylamino)-4-imidazol-1-yl-1-oxobutan-2-yl]furan-2-carboxamide	Ki	10000000.0 [1]
	N-[(2S)-4-(4-Methylpiperazin-1-yl)-1-oxo-1-(propan-2-ylamino)butan-2-yl]morpholine-4-carboxamide	Ki	10000000.0 [1]
	N-[(2S)-1-(Benzylamino)-4-imidazol-1-yl-1-oxobutan-2-yl]-1-methylpyrrole-2-carboxamide	Ki	155000.0 [1]
	N-[(2S)-1-(Benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]-4-fluorobenzamide	Ki	10000000.0 [1]
	N-[(2S)-4-[4-(Cyanomethyl)imidazol-1-yl]-1-oxo-1-(propan-2-ylamino)butan-2-yl]furan-2-carboxamide	Ki	353000.0 [1]
	5,5-Dimethyl-3-[2-(2H-tetrazol-5-yl)ethyl]imidazolidine-2,4-dione	Ki	384000.0 [1]
	5,5-Dimethyl-3-[2-(2-methylimidazol-1-yl)ethyl]imidazolidine-2,4-dione	Ki	2417000.0 [1]
	N-[(2S)-1-(Benzylamino)-1-oxo-4-(triazol-1-yl)butan-2-yl]-1-methylpyrrole-2-carboxamide	Ki	112000.0 [1]
	N-[(2S)-4-Imidazol-1-yl-1-oxo-1-(propan-2-ylamino)butan-2-yl]furan-2-carboxamide	Ki	964000.0 [1]
	5,5-Dimethyl-3-(2-morpholin-4-ylethyl)imidazolidine-2,4-dione	Ki	602000.0 [1]
	7-Amino-6-bromoquinoline-5,8-dione	IC50	2270.0 [1]
	2-{[(2s)-1-Amino-5-{[(1z)-2-Chloroethanimidoyl]amino}-1-Oxopentan-2-Yl]carbamoyl}benzoic Acid	IC50	840.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 22 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Protein-arginine deiminase type-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/protein-arginine-deiminase-type-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ Protein-arginine deiminase type-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/protein-arginine-deiminase-type-1-inhibitors-ic50-ki.
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