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Prostate specific antigen Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Ahx-FSQn(boro)BpgKi75.0 [1]
[(1R)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutyl]boronic acidKi65.0 [1]
8-[(2R,3S)-5,7-Dihydroxy-2-(4-hydroxyphenyl)-4-oxo-2,3-dihydrochromen-3-yl]-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-2,3-dihydrochromen-4-oneIC5013000.0 [1]
Benzyl (2S,3S)-3-[(4-hydroxyphenyl)methyl]-4-oxo-1-[2-(3-phenylmethoxycarbonylphenyl)acetyl]azetidine-2-carboxylateIC50226.0 [1]
[(1R)-1-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]hexanoyl]amino]-3-methylbutyl]boronic acidKi48.4 [1]
[(1R)-1-[[(2S)-5-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]-5-oxopentanoyl]amino]-3-methylbutyl]boronic acidKi27.5 [1]
[(1R)-1-[[(2S)-5-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(morpholine-4-carbonylamino)propanoyl]amino]propanoyl]amino]-5-oxopentanoyl]amino]-3-methylbutyl]boronic acidKi25.3 [1]
[(1R)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]-methylamino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutyl]boronic acidKi2.5 [1]
[(1R)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]-methylamino]propanoyl]amino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutyl]boronic acidKi19.9 [1]
[(1R)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-[methyl(phenylmethoxycarbonyl)amino]propanoyl]amino]propanoyl]amino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutyl]boronic acidKi0.2 [1]
[(1R)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-[methyl(phenylmethoxycarbonyl)amino]propanoyl]amino]propanoyl]-methylamino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutyl]boronic acidKi5.6 [1]
[(1R)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-[methyl(phenylmethoxycarbonyl)amino]propanoyl]-methylamino]propanoyl]-methylamino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutyl]boronic acidKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi3.6 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi4.4 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi6.5 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi11.9 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-4-methylsulfinyl-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi12.8 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-3-(4-hydroxyphenyl)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi13.1 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi13.7 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-3-(1H-imidazol-2-yl)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi18.6 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-5-amino-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi21.8 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-4-hydroxy-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi29.4 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S,4S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi37.4 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-4-amino-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi41.9 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-(N-[2-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]anilino)-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2R)-3-tert-butylsulfanyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-6-amino-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[cyclohexyl-[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-3-hydroxy-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-3-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi50.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S,3R)-3-hydroxy-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi100.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi100.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-naphthalen-2-ylamino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi100.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-3-(4-bromophenyl)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi500.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[(2S)-2-[[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi500.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[2-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi1000.0 [1]
(3S)-3-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]hexanoyl]amino]-4-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acidKi1000.0 [1]
(4S)-4-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]hexanoyl]amino]-5-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentanoic acidKi1000.0 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi3.9 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S)-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi7.5 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S)-4-hydroxy-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi8.8 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[cyclohexyl-[(2S)-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi13.1 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-4-amino-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi18.2 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi19.9 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S)-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-4-methylsulfinyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi25.9 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S,3R)-3-hydroxy-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi43.8 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[(2S)-1-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi500.0 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[(2S)-2-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi1000.0 [1]
Benzyl N-[(2S)-3-hydroxy-1-[[(2S)-3-hydroxy-1-[[2-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]carbamateKi1000.0 [1]
(4S)-4-[[(2S)-3-Hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]-5-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-oxopentanoic acidKi1000.0 [1]
(3S)-3-[[(2S)-3-Hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]-4-[[(2S)-4-methyl-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-4-oxobutanoic acidKi1000.0 [1]
2-O-Benzyl 1-O-(3-phenylmethoxycarbonylphenyl) (2S,3S)-3-[(4-hydroxyphenyl)methyl]-4-oxoazetidine-1,2-dicarboxylateIC50226.0 [1]
(3,4-Dimethoxyphenyl)-(5-methyl-3-pyridin-3-yl-1,2,4-triazol-1-yl)methanoneKi500.0 [1]
[(1S)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]hexanoyl]amino]hexanoyl]amino]-2-phenylethyl]boronic acidKi164.5 [1]
[(1S)-1-[[(2S)-2-[[(2S)-6-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-3-hydroxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]hexanoyl]amino]hexanoyl]amino]-4-bromobutyl]boronic acidKi24.23 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(2S)-2-(6-aminohexanoylamino)-3-hydroxypropanoyl]amino]-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-3-methylbutyl]boronic acidKi43.05 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-(6-aminohexanoylamino)-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-2-phenylethyl]boronic acidKi22.01 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-(6-aminohexanoylamino)-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-4-bromobutyl]boronic acidKi302.1 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(2S)-2-(6-aminohexanoylamino)propanoyl]amino]-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-2-phenylethyl]boronic acidKi310.29 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(2S)-2-(6-aminohexanoylamino)propanoyl]amino]-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-4-bromobutyl]boronic acidKi52.11 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(2S)-2-(6-aminohexanoylamino)-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-2-phenylethyl]boronic acidKi61.48 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-(6-Aminohexanoylamino)-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]amino]-N-[(2S)-1-[[(1S)-4-bromo-1-[(1R,2S,6R,8R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]butyl]amino]-1-oxohexan-2-yl]pentanediamideKi73.33 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[6-[(4-iodobenzoyl)amino]hexanoylamino]-3-phenylpropanoyl]amino]propanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-4-bromobutyl]boronic acidKi64.41 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(3S)-3-(6-aminohexanoylamino)-4-naphthalen-2-ylbutanoyl]amino]-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-2-phenylethyl]boronic acidKi228.78 [1]
[(1S)-1-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-2-[[(3S)-3-(6-aminohexanoylamino)-4-naphthalen-2-ylbutanoyl]amino]-3-hydroxypropanoyl]amino]-5-oxopentanoyl]amino]hexanoyl]amino]-4-bromobutyl]boronic acidKi102.46 [1]
Benzyl N-[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[(2S,3R)-3-hydroxy-2-[[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamateKi500.0 [1]
(2S)-6-Amino-N-[(2S)-1-[[(2S)-5-amino-1,5-dioxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]-3-hydroxypropanoyl]amino]hexanamideKi45000.0 [1]
2-(2-Methyl-3-nitrophenyl)-4H-3,1-benzoxazin-4-oneKi300.0 [1]
Items per page: 1 - 10 of 68
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References

This online tool may be cited as follows

MLA

"Quest Database™ Prostate specific antigen Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/prostate-specific-antigen-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Prostate specific antigen Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/prostate-specific-antigen-inhibitors-ic50-ki.
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