![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_bba0e8ca6afb314c59542be5b90d2370.svg) | Olaparib | IC50 | 46.0 [1], 230.0 [2], 320.0 [3] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_7de353ee3e6da7d439f1ec3aa8996b73.svg) | 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one | IC50 | 831.76 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_67f6ced2b72cac0cc2b4d65f0d199019.svg) | Niraparib | IC50 | 296.0 [1], 1300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_9d37a00818f71911ddc7ae7fb3af75a7.svg) | N~2~,N~2~-Dimethyl-N~1~-(6-oxo-5,6-dihydrophenanthridin-2-YL)glycinamide | IC50 | 1430.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_5bde39defdeb9b3639f2a3e58f77f3b5.svg) | Veliparib | IC50 | 2040.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_4ce1e392071f9a35d153ee0e21369703.svg) | Rucaparib | IC50 | 512.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_979b4880256c881f24510e2d72655f5e.svg) | Bmn-673 8R,9S | IC50 | 62.8 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_35aec792bbfc6c95d4c64c30a66ec983.svg) | 4-Methoxybenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_6f319471151e9109735392e9e66bb80c.svg) | 3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-Phenylethyl]propanamide | IC50 | 900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_028a11317906182ba0740511a9b10018.svg) | 4,4'-Oxydibenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_da759c45c4a5813431ec3296123568ca.svg) | 4-[[3-[(6S)-3-(1,1-Difluoroethyl)-6-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]-difluoromethyl]-2H-phthalazin-1-one | IC50 | 2800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_7260fe64bd7e1b45b18038522ee7fe7a.svg) | 5-(2-Oxo-2-phenylethoxy)isoquinolin-1(2H)-one | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_41feab3c9fd34f20ec15f681338460cd.svg) | 4-Quinazolinol, 5,6,7,8-tetrahydro-2-(4-methyl-1-piperazinyl)- | IC50 | 91000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_9f55c70eef839ae3878767dd7b8cd018.svg) | 2-(4-Tert-Butylphenyl)-2,3-dihydroquinazoline-4(1H)-one | IC50 | 34000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_aee167f244ed6999c4420a7616495cc6.svg) | 4-(4-Carbamoylphenoxy)benzoic acid | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_410af0ab6e7320aee9a24ec4c166c008.svg) | 4-[(2-Fluorophenyl)methoxy]benzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_c18e776e19bcb8483ae899b1f9dd2f26.svg) | 2-[4-[3-[(4-Oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]pyridine-3-carbonitrile | IC50 | 46.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_cc06a47ef1cd90f88c44822007ee39ab.svg) | N-{4-[(2-Chlorophenyl)(Pyrimidin-4-Yl)carbamoyl]phenyl}-4-Methoxybenzamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_fbc186dc6ed96f500ea5b572e86e159c.svg) | 1-[3-[4-(2-Chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxo-3H-benzimidazole-5-carbonitrile | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_2d7962cdae8647afd55af5b543f9687f.svg) | Pamiparib | IC50 | 185.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_930130505680794c2112dfd2eb766622.svg) | 3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-(Pyridin-2-Yl)ethyl]propanamide | IC50 | 1300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_049877b51ce1ec8a958c9166b8ffbe6f.svg) | 3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1r)-1-(Pyridin-2-Yl)ethyl]propanamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_a4f9318d3e76064ae440acfc7f000042.svg) | 3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)-N-[(1s)-1-Phenylpropyl]propanamide | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_eba93f51209f31881e26d898f45c9b64.svg) | N-[(2s)-1-Hydroxy-3-Phenylpropan-2-Yl]-3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanamide | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_fb083c629dd685768ce47d1c43659acf.svg) | N-[(2s)-1-Hydroxybutan-2-Yl]-3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanamide | IC50 | 9600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_402cca4728ec8019acf9bdc4b0f766e9.svg) | Methyl N-[3-(4-Oxo-3,4-Dihydroquinazolin-2-Yl)propanoyl]-L-Phenylalaninate | IC50 | 2200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_a08cd9b05982a7d9e21c6b0eafcb79a6.svg) | 2-(4-((Pyridin-4-Yl)methyl)piperazin-1-Yl)-3,4,5,6,7,8-Hexahydroquinazolin-4-One | IC50 | 13000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_2e14cc7d0095f864892bafb0383bb66b.svg) | 4-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 40000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_841732ebe8b3ab4c3c60886e582b565f.svg) | 4-[3-(8-Methyl-4-oxo-3H-quinazolin-2-yl)propanoylamino]-N-quinolin-8-ylbenzamide | IC50 | 45000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_79fb0066600a21901f09afb45bd4df0e.svg) | N-[1-(4-Imidazol-1-ylphenyl)ethyl]-3-(4-oxo-3H-quinazolin-2-yl)propanamide | IC50 | 13200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_fac52ba29959f1bc425676971d78205f.svg) | 3-(4-Oxo-3,4-dihydroquinazolin-2-yl)-N-[1-(4-sulfamoylphenyl)ethyl]propanamide | IC50 | 14400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_75ec9484ab919b4876096fee09d7c6ec.svg) | N-[(1R)-2,3-Dihydro-1H-inden-1-yl]-3-(4-oxo-3H-quinazolin-2-yl)propanamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_e048c1358d3b57e7358bce5c79d53592.svg) | N-[(1S)-2,3-Dihydro-1H-inden-1-yl]-3-(4-oxo-3H-quinazolin-2-yl)propanamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_0ed298f980fa1c484097f9195aea4e3d.svg) | 3-(4-Oxo-3H-quinazolin-2-yl)-N-[(1R)-1-phenylethyl]propanamide | IC50 | 15200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_64cf33b0235d070f10fc95ac922c3d6f.svg) | (2S)-2-[3-(4-Oxo-3H-quinazolin-2-yl)propanoylamino]-3-phenylpropanamide | IC50 | 3800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_344ddb68a40ca0113fbc145d12452b76.svg) | N-[(2S)-1-Hydroxypropan-2-yl]-3-(4-oxo-3H-quinazolin-2-yl)propanamide | IC50 | 11100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_e082074a4efae2c0d45f6a2dd0e4c08a.svg) | 2-(3-Pyrazin-2-ylpropanoyl)-2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-10-one | IC50 | 70.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_71e9ff8508013ed176658eb62261908f.svg) | 2-(2-Pyridin-3-ylacetyl)-2,11-diazatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-10-one | IC50 | 50.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_bf78858640441e659323229959dd3639.svg) | 4-(4-Formyl-phenoxy)-benzamide | IC50 | 86000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_4c5ea469a0ea7857d02dfcb671f92660.svg) | 1,2-Dihydro-2-(4-isopropylphenyl)-4(3H)-quinazolinone | IC50 | 50000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_64a36171129b71301828f12d468cff2f.svg) | 4-[(4s)-5,5-Dimethyl-2-Oxo-4-Phenyl-1,3-Oxazolidin-3-Yl]-N-(Quinolin-8-Yl)benzamide | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_34ae1521cd2fb0931e21c900ada104d2.svg) | 7-(2-Fluorophenyl)-4-Methylquinolin-2(1h)-One | IC50 | 10000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_329e6f978feb6d6e3d8d0bd501cd3c9d.svg) | N-[3-Chloranyl-4-[[4-(4-Methoxyphenyl)oxan-4-Yl]methylcarbamoyl]phenyl]furan-2-Carboxamide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_d02df27a332d3f58de88c96e4b5ad517.svg) | 6,7,16-Triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 199.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_7fef78a441b75afed083a6136c5694ed.svg) | 11-Fluoro-3,3-dimethyl-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 136.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_c10f0d9b6eacf1a6029100232f1a9180.svg) | 3-Propan-2-yl-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 760.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_ad6230eca03a66647ac4953a94df908b.svg) | 3-(Cyclopropanecarbonyl)-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 180.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_57c2b982008f1797fa61c7003ac06c8a.svg) | 3-(2,2-Dimethylpropanoyl)-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 660.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_9975f22b259a2f26d7a1c6c20abea9fc.svg) | 3-(2-Amino-2-methylpropanoyl)-3,6,7,16-tetrazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 18.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_ec4962732229d0f63ad373d9a6118c9f.svg) | 3,3-Dimethyl-16-(2-piperidin-1-ylethyl)-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_4667afb33041f15cbd9c1fab7acce276.svg) | 16-[2-(Diethylamino)ethyl]-3,3-dimethyl-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 11000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_b6579e335e5e9719c8d264ccd27c4d39.svg) | 3,3-Dimethyl-16-(oxiran-2-ylmethyl)-6,7,16-triazatetracyclo[11.2.1.05,15.09,14]hexadeca-1(15),5,9(14),10,12-pentaen-8-one | IC50 | 1000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/poly-adp-ribose-polymerase-3_00c2124fb9869b276d7ecf21eda38440.svg) | 4-[[4-Fluoro-3-[5-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl]phenyl]methyl]-2H-phthalazin-1-one | IC50 | 66.9 [1] |